BDBM82020 1-Methyl-3,9-dihydro-purine-2,6-dione(1-methyl xanthine)::1-Methylxanthine::CAS_80220::CHEMBL1250::NSC_80220
SMILES Cn1c(=O)[nH]c2nc[nH]c2c1=O
InChI Key InChIKey=SNXCZWZKBPOLIM-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 82020
Affinity DataKi: 1.15E+4nMAssay Description:Affinity against adenosine A1 receptor in the brain membranes by the displacement of [3H]-CPX.More data for this Ligand-Target Pair
Affinity DataKi: 6.71E+4nMAssay Description:Affinity against adenosine A2 receptor in the brain membranes measured by the displacement of [3H]-CPXMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University
Curated by ChEMBL
Hokuriku University
Curated by ChEMBL
Affinity DataKi: 1.63E+5nMAssay Description:Inhibition of c-AMP phosphodiesterase activity in guinea pig tracheal muscleMore data for this Ligand-Target Pair
Affinity DataEC50: 7.59E+4nMAssay Description:Relexant activity on the spontaneous tone of isolated guinea pig tracheal ring chains.More data for this Ligand-Target Pair