BDBM82258 CAS_114798-26-4::Losartan::NSC_3961
SMILES CCCCc1nc(Cl)c(CO)n1Cc1ccc(cc1)-c1ccccc1-c1nnn[nH]1
InChI Key InChIKey=PSIFNNKUMBGKDQ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 82258
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
School Of Chemical Engineering & The Environment
Curated by ChEMBL
School Of Chemical Engineering & The Environment
Curated by ChEMBL
Affinity DataIC50: 16.2nMAssay Description:Displacement of [125I]Sar1Ile8-Ang2 from angiotensin AT1 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(RABBIT)
School Of Chemical Engineering & The Environment
Curated by ChEMBL
School Of Chemical Engineering & The Environment
Curated by ChEMBL
Affinity DataKd: 12.6nMAssay Description:Antagonist activity at AT1 receptor in Japanese white rabbit thoracic aorta assessed as inhibition of KCl-induced contraction incubated 30 mins post ...More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
School Of Chemical Engineering & The Environment
Curated by ChEMBL
School Of Chemical Engineering & The Environment
Curated by ChEMBL
Affinity DataIC50: 0.330nMAssay Description:Inhibition of angiotensin AT1 receptorMore data for this Ligand-Target Pair