BDBM84522 Sulindac analogue, 19

SMILES CC1=C(CC(O)=O)c2ccc(Br)cc2\C1=C/c1ccsc1

InChI Key InChIKey=ALAVELGECUJLKK-NSIKDUERSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 84522   

TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Max-Planck-Institut FÜR Molekulare Physiologie

LigandPNGBDBM84522(Sulindac analogue, 19)
Affinity DataIC50:  3.00E+3nMAssay Description:The kinase-catalyzed phosphorylation of poly(Glu4-Tyr) in the presence of varying concentrations of inhibitor was determined. The kinase were employ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Max-Planck-Institut FÜR Molekulare Physiologie

LigandPNGBDBM84522(Sulindac analogue, 19)
Affinity DataIC50:  4.00E+3nMAssay Description:The kinase-catalyzed phosphorylation of poly(Glu4-Tyr) in the presence of varying concentrations of inhibitor was determined. The kinase were employ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
Max-Planck-Institut FÜR Molekulare Physiologie

LigandPNGBDBM84522(Sulindac analogue, 19)
Affinity DataIC50:  1.00E+3nMAssay Description:The kinase-catalyzed phosphorylation of poly(Glu4-Tyr) in the presence of varying concentrations of inhibitor was determined. The kinase were employ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Max-Planck-Institut FÜR Molekulare Physiologie

LigandPNGBDBM84522(Sulindac analogue, 19)
Affinity DataIC50:  4.00E+3nMAssay Description:The kinase-catalyzed phosphorylation of poly(Glu4-Tyr) in the presence of varying concentrations of inhibitor was determined. The kinase were employ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Max-Planck-Institut FÜR Molekulare Physiologie

LigandPNGBDBM84522(Sulindac analogue, 19)
Affinity DataIC50:  2.30E+4nMAssay Description:The kinase-catalyzed phosphorylation of poly(Glu4-Tyr) in the presence of varying concentrations of inhibitor was determined. The kinase were employ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Max-Planck-Institut FÜR Molekulare Physiologie

LigandPNGBDBM84522(Sulindac analogue, 19)
Affinity DataIC50:  1.20E+4nMAssay Description:The kinase-catalyzed phosphorylation of poly(Glu4-Tyr) in the presence of varying concentrations of inhibitor was determined. The kinase were employ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed