BDBM8813 3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}phenyl)-1-(3-methylphenyl)urea::CHEMBL371329::CHEMBL537435::KDR Kinase Inhibitor, 7::N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)-phenyl]-N -(3-methylphenyl)urea::Thienopyrimidine deriv. 11
SMILES Cc1sc2ncnc(N)c2c1-c1ccc(NC(=O)Nc2cccc(C)c2)cc1
InChI Key InChIKey=UKICZFWMZQMZGK-UHFFFAOYSA-N
Data 13 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 13 hits for monomerid = 8813
Affinity DataIC50: 6nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
Affinity DataIC50: 9nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
Affinity DataIC50: 110nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition assay using KDR.More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of c-Kit by HTRF methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of VEGFR-2 kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of Tie2 kinaseMore data for this Ligand-Target Pair