BDBM99012 US8497265, 468

SMILES OCC1CCN(CC1)c1ncc(C2=CCOCC2)c(OC2CN(C2)c2ccc3ccccc3n2)n1

InChI Key InChIKey=GYPKGKLLWMFEDT-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 99012   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Rattus norvegicus (rat))
Amgen

US Patent
LigandPNGBDBM99012(US8497265, 468)
Affinity DataIC50:  1.10nMAssay Description:Enzyme activity: An IMAP TR-FRET assay was used to analyze the enzyme activity (Molecular Devices Corp., Sunnyvale, Calif). More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent