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Report error Found 121 Enz. Inhib. hit(s) with Target = 'Chymotrypsin-like elastase family member 1'
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014738(CHEMBL130253 | N-(Adamantyl-sulfonyl)-N-(methoxy s...)
Affinity DataKi:  0.580nMAssay Description:Binding affinity against human Elastase for more active diasteriomerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014735(CHEMBL336171 | (1-{1-Methyl-2-oxo-2-[2-(3,3,3-trif...)
Affinity DataKi:  1nMAssay Description:Binding affinity against human Elastase for more active diasteriomerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014738(CHEMBL130253 | N-(Adamantyl-sulfonyl)-N-(methoxy s...)
Affinity DataKi:  15nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014747(CHEMBL131780 | 3-[(1-{2-[(1-Acetyl-pyrrolidine-2-c...)
Affinity DataKi:  29nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50326056((1S,3aR,6aS)-2-((S)-2-((S)-2-cyclohexyl-2-(pyrazin...)
Affinity DataIC50: 30nMAssay Description:Inhibition of human Pancreatic elastase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM50312532(molassamide | CHEMBL1077010)
Affinity DataIC50: 32nMAssay Description:Inhibition of pig pancreatic elastase preincubated for 15 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014736(CHEMBL337396 | (1-{1-Methyl-2-oxo-2-[2-(3,3,3-trif...)
Affinity DataKi:  32nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014730(CHEMBL130271 | N-(1-{1-Methyl-2-oxo-2-[2-(3,3,3-tr...)
Affinity DataKi:  33nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014736(CHEMBL337396 | (1-{1-Methyl-2-oxo-2-[2-(3,3,3-trif...)
Affinity DataKi:  44nMAssay Description:Binding affinity against human Elastase for more active diasteriomerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50038879(JTP-4819 | CHEMBL79993 | (S)-2-(2-Formyl-pyrrolidi...)
Affinity DataIC50: 51.6nMAssay Description:Inhibition of Flavobacterium meningosepticum PEPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50071966((R)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)...)
Affinity DataIC50: 60nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50071968((S)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)...)
Affinity DataIC50: 60nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50071973((S)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)...)
Affinity DataIC50: 60nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014732(CHEMBL339870 | 1-{2-[2-(5-Dimethylamino-naphthalen...)
Affinity DataKi:  88nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014730(CHEMBL130271 | N-(1-{1-Methyl-2-oxo-2-[2-(3,3,3-tr...)
Affinity DataKi:  92nMAssay Description:Binding affinity against human elastase for less active diasteriomerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014745(CHEMBL131188 | 3-{2-[2-(2-Benzyloxycarbonylamino-p...)
Affinity DataKi:  140nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014742(CHEMBL130128 | Acetyl-Ala-Ala-Pro-Ala-triflurometh...)
Affinity DataKi:  150nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014737(CHEMBL446422 | {1-Benzyl-2-oxo-2-[2-(3,3,3-trifluo...)
Affinity DataKi:  160nMAssay Description:Binding affinity against human Elastase for more active diasteriomerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50071983(CHEMBL310738 | (S)-3-((S)-2-Acetylamino-3-carboxy-...)
Affinity DataIC50: 190nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014748(CHEMBL436383 | 3-[(1-{2-[2-(3-Methoxycarbonyl-prop...)
Affinity DataKi:  200nMAssay Description:Binding affinity against human Elastase for more active diasteriomerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014740(CHEMBL130718 | Acetyl-Pro-Ala-Pro-Ala-trifluoro me...)
Affinity DataKi:  240nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50269564(5,6,5',6'-tetrahydroxy[3,3']bibenzofuranyl-2,2'-di...)
Affinity DataKi:  290nMAssay Description:Inhibition of Flavobacterium meningosepticum PEPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014745(CHEMBL131188 | 3-{2-[2-(2-Benzyloxycarbonylamino-p...)
Affinity DataKi:  300nMAssay Description:Binding affinity against human Elastase for more active diasteriomerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50015856(CHEMBL313754 | 3-Acetoxymethyl-7-formyloxy-5,5,8-t...)
Affinity DataIC50: 400nMAssay Description:Inhibitory concentration which is required to cause 50% inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014734(CHEMBL132768 | N-{1-Benzyl-2-oxo-2-[2-(3,3,3-trifl...)
Affinity DataKi:  660nMAssay Description:Binding affinity against human Elastase for more active diasteriomerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014748(CHEMBL436383 | 3-[(1-{2-[2-(3-Methoxycarbonyl-prop...)
Affinity DataKi:  680nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014744(CHEMBL335981 | 3-[(1-{2-[(1-Acetyl-pyrrolidine-2-c...)
Affinity DataKi:  690nMAssay Description:Binding affinity against porcine pancreatic ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50228470(CHEMBL2370693)
Affinity DataKi:  800nMAssay Description:Binding affinity against porcine pancreatic ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014747(CHEMBL131780 | 3-[(1-{2-[(1-Acetyl-pyrrolidine-2-c...)
Affinity DataKi:  850nMAssay Description:Binding affinity against human Elastase for more active diasteriomerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Bovine)
University of Helsinki

LigandPNGBDBM65489(MdnA7)
Affinity DataIC50: 1.05E+3nMT: 2°CAssay Description:The inhibition assays were performed in 96-well microtiter plates as follows: 30 uL of the enzyme solution (trypsin [100 ug/mL] or elastase [1.5 U/mL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2018
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50269565(propeptin | CHEMBL500199)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Flavobacterium meningosepticum PEPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50269564(5,6,5',6'-tetrahydroxy[3,3']bibenzofuranyl-2,2'-di...)
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of Flavobacterium meningosepticum PEPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50269567(Kynapcin-12 | CHEMBL515528)
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of Flavobacterium meningosepticum PEPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014737(CHEMBL446422 | {1-Benzyl-2-oxo-2-[2-(3,3,3-trifluo...)
Affinity DataKi:  1.80E+3nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50015876(CHEMBL84768 | 7-Acetoxy-3-acetoxymethyl-5,5,8-trio...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory concentration which is required to cause 50% inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50071965((S)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)...)
Affinity DataIC50: 2.20E+3nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50226399(CHEMBL3143932)
Affinity DataKi:  2.40E+3nMAssay Description:Compound is evaluated for the inhibition of porcine pancreatic (PP) elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50429202(LYNGBYASTATIN 7)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of pig pancreatic elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50479189(CHEBI:66142 | KEMPOPEPTIN A)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of pig pancreatic elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50269566(polyozellin | CHEMBL458248)
Affinity DataIC50: 2.72E+3nMAssay Description:Inhibition of Flavobacterium meningosepticum PEPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50479190(SOMAMIDE B)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of pig pancreatic elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014733(CHEMBL340062 | 2,2-Difluoro-4-[(1-{2-[2-(3-methoxy...)
Affinity DataKi:  4.30E+3nMAssay Description:Binding affinity against human Elastase for more active diasteriomerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM50405198(CHEMBL52356)
Affinity DataKi:  8.13E+3nMAssay Description:Inhibitory activity against porcine pancreatic elastase (PP elastase) expressed as inhibitory constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014733(CHEMBL340062 | 2,2-Difluoro-4-[(1-{2-[2-(3-methoxy...)
Affinity DataKi:  9.90E+3nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50326055((1R,21S,24S)-21-tert-Butyl-N-((1R,2R)-1-{[(cyclopr...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human Pancreatic elastase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50310584(CHEMBL1078049 | N-(5-Chloro-pyridin-2-yl)-2-(4-{N-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM50302107(Grassystatin A | CHEMBL567893)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of porcine pancreatic elastase after 10 to 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Human)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM12311(SCH 503034 | (1R,5S)-N-[3-Amino-1-(cyclobutylmethy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human Pancreatic elastase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM50405207(CHEMBL53936)
Affinity DataKi:  1.51E+4nMAssay Description:Inhibitory activity against porcine pancreatic elastase (PP elastase) expressed as inhibitory constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50226400(CHEMBL3143923)
Affinity DataKi:  1.95E+4nMAssay Description:Compound is evaluated for the inhibition of porcine pancreatic (PP) elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details Article
PubMed
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