Compile Data Set for Download or QSAR
Report error Found 13922 Enz. Inhib. hit(s) with Target = 'Delta-type opioid receptor'
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM309406(US9656962, Compound 31 | (2R,3aS,4R,9bS)-12-(cyclo...)
Affinity DataEC50:  75.5nMAssay Description: Radioligand dose-displacement binding assays for μ-opioid receptors used 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, Conn.), with 5 mg me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM309413(US9656962, Compound 38 | (2S,3aS,4R,9bS)-12-(cyclo...)
Affinity DataEC50:  1.56nMAssay Description: Radioligand dose-displacement binding assays for μ-opioid receptors used 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, Conn.), with 5 mg me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM21008((4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)pr...)
Affinity DataKd:  0.450nM EC50:  1.60nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2008
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM21008((4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)pr...)
Affinity DataKd:  0.5nM EC50:  1.60nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM21008((4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)pr...)
Affinity DataKd:  0.5nM EC50:  1.60nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM393487(US9963460, 13)
Affinity DataEC50:  1.70nMAssay Description:In a [3SS] GTPγS binding test, the opioid receptor agonist activity of test compounds based on a GTP-GDP exchange reaction was evaluated. In the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM54821(N-[(2S)-1-[(3R,6R)-3-benzyl-6-[(4-hydroxyphenyl)me...)
Affinity DataEC50:  3.12E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics Source Affiliation: Sanford-Burnham Medical Research Institute Network: NIH Molecular Lib...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM54833(cid_3218102 | 4-ethoxy-N-[9-(phenylmethyl)-9-azabi...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM54816(cid_3218139 | MLS000709692 | 4-methyl-N-[9-[(4-met...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM54781(SMR000119685 | N-(3,4-Dimethoxy-benzyl)-2-(3-oxo-2...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62173(cid_653720 | MLS-0043215.0001 | N-[(4-methoxypheny...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62187((phenylmethyl) N-[2,2,2-tris(chloranyl)-1-[(2,4-di...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62188(benzyl N-[2,2,2-trichloro-1-[(2,5-dimethylphenyl)c...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM57352(benzyl N-[2,2,2-trichloro-1-[(3-chlorophenyl)carba...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM54805(MLS000561692 | cid_3091265 | {2,2,2-Trichloro-1-[3...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM54803(cid_3091267 | N-[2,2,2-trichloro-1-[[sulfanylidene...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM54836(4-[1-[2-(7-chloroquinolin-4-yl)hydrazinyl]propylid...)
Affinity DataEC50:  3.07E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM46582((4Z)-4-[[2-(7-chloroquinolin-4-yl)hydrazinyl]methy...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM54784(2-[5-[(4-tert-butylphenyl)methylsulfanyl]-4-(furan...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62189(cid_16294686 | MLS-0355913.0001 | N-[2-(dimethylam...)
Affinity DataEC50:  1.60E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62190(4-[[(4-ethanoylphenyl)sulfonylamino]methyl]-N-[2-[...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM54775(MLS000082434 | SMR000043634 | 2-[5-[(2,4-dichlorop...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM54788(N-butyl-N-[(6-methyl-2-oxo-1H-quinolin-3-yl)methyl...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM54783(Pyridine-2-carboxylic acid butyl-(2-hydroxy-quinol...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62174(MLS-0015756.0001 | cid_665086 | N-cyclohexyl-N-[(2...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62175(MLS-0015758.0001 | cid_665037 | N-[(7-methyl-2-oxi...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62176(N-butyl-N-[(6-methoxy-2-oxidanylidene-1H-quinolin-...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62177(cid_3440378 | N-[(6-methyl-2-oxidanylidene-1H-quin...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62178(MLS-0019234.0001 | cid_665054 | N-methyl-N-[(6-met...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM42469(SMR000044072 | MLS000082430 | 2-[5-[(4-bromophenyl...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM54774(N-(4-chloranyl-2-methoxy-5-methyl-phenyl)-2-[[4-(f...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM54773(MLS000082432 | SMR000042990 | 2-[5-[(3-chloropheny...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62179(1-(4-chlorophenyl)-2-[[4-(furan-2-ylmethyl)-5-pyri...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62180(MLS-0058733.0001 | 2-[5-[(2-chlorophenyl)methylsul...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62181(MLS-0046572.0001 | 2-[[4-(furan-2-ylmethyl)-5-pyri...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62182(2-[[4-(furan-2-ylmethyl)-5-pyridin-2-yl-1,2,4-tria...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62191(cid_9550286 | N-[[4-[4-(phenylmethyl)piperazin-1-y...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM54779(cid_1297443 | N-[1-[(2,6-dimethylphenyl)carbamoyl]...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM54778(SMR000078652 | 2-[4-(2-furanylmethyl)-5-[[(E)-3-ph...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62183([4-[(4-methoxyphenyl)methyl]-1-[[1-(3-methylphenyl...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62184(cid_44537711 | [1-[[1-(3-methylphenyl)imidazol-2-y...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62192((4Z)-4-[[(5-chloro-8-quinolinyl)amino]methylidene]...)
Affinity DataEC50:  1.48E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM40197(MLS000530291 | 2-[(8-quinolinylamino)methylene]-1-...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62193(N-[2,2,2-trichloro-1-[[(4-methylanilino)-sulfanyli...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62194((phenylmethyl) N-[2,2,2-tris(chloranyl)-1-[(2,4-di...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62195(cid_3091266 | (phenylmethyl) N-[2,2,2-tris(chloran...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62196((phenylmethyl) N-[1-[(4-bromophenyl)carbamothioyla...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62197(benzyl N-[1-[(3-bromophenyl)carbamothioylamino]-2,...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62198(cid_3091277 | N-[2,2,2-trichloro-1-[[(4-fluoroanil...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetDelta-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM62199(N-[1-[[anilino(sulfanylidene)methyl]amino]-2,2,2-t...)
Affinity DataEC50: >3.20E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
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