Compile Data Set for Download or QSAR
Report error Found 221 Enz. Inhib. hit(s) with Target = 'Dipeptidase 1'
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50292408(5S-hydroxy-6R-(S-cysteinylglycinyl)-7E,9E,11E,14Z-...)
Affinity DataKi:  0.490nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2011
Entry Details
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50297387((5S-(5R*,6S*(S*),7E,9E,11Z,14Z))-6-((2-Amino-2-car...)
Affinity DataKi:  1.53nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2011
Entry Details
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM81801(CAS_5283121 | NSC_5283121 | LTC4)
Affinity DataKi:  3.58nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2011
Entry Details
PubMed
TargetDipeptidase 1(Human)
The Sidney Kimmel Comprehensive Cancer Center At Johns Hopkins

Curated by ChEMBL
LigandPNGBDBM50148534(2-[(1-Amino-2-cyclohexyl-ethyl)-hydroxy-phosphinoy...)
Affinity DataIC50: 5nMAssay Description:Concentration required to inhibit renal dipeptidase (RDP) by 50% in crude lysates prepared from human colon cancerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidase 1(Human)
The Sidney Kimmel Comprehensive Cancer Center At Johns Hopkins

Curated by ChEMBL
LigandPNGBDBM50148543(2-[(1-Amino-2-cyclohexyl-ethyl)-hydroxy-phosphinoy...)
Affinity DataIC50: 6nMAssay Description:Concentration required to inhibit renal dipeptidase (RDP) by 50% in crude lysates prepared from human colon cancerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidase 1(Human)
The Sidney Kimmel Comprehensive Cancer Center At Johns Hopkins

Curated by ChEMBL
LigandPNGBDBM50148531(CHEMBL326292 | CHEMBL334279 | 2-[(1-Amino-2-cycloh...)
Affinity DataIC50: 8nMAssay Description:Concentration required to inhibit renal dipeptidase (RDP) by 50% in crude lysates prepared from human colon cancerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidase 1(Human)
The Sidney Kimmel Comprehensive Cancer Center At Johns Hopkins

Curated by ChEMBL
LigandPNGBDBM50148532(CHEMBL420537 | CHEMBL333841 | 2-[(1-Amino-2-cycloh...)
Affinity DataIC50: 10nMAssay Description:Concentration required to inhibit renal dipeptidase (RDP) by 50% in crude lysates prepared from human colon cancerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidase 1(Human)
The Sidney Kimmel Comprehensive Cancer Center At Johns Hopkins

Curated by ChEMBL
LigandPNGBDBM50148534(2-[(1-Amino-2-cyclohexyl-ethyl)-hydroxy-phosphinoy...)
Affinity DataIC50: 15nMAssay Description:Concentration required to inhibit renal dipeptidase (RDP) by 50% in crude lysates prepared from human colon cancerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023962(2-[(2,2-Dibromo-cyclopropanecarbonyl)-amino]-hex-2...)
Affinity DataKi:  15nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Human)
The Sidney Kimmel Comprehensive Cancer Center At Johns Hopkins

Curated by ChEMBL
LigandPNGBDBM50148533(CHEMBL119118 | CHEMBL332970 | 2-[(1-Amino-2-cycloh...)
Affinity DataIC50: 20nMAssay Description:Concentration required to inhibit renal dipeptidase (RDP) by 50% in crude lysates prepared from human colon cancerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023979(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-7-(3...)
Affinity DataKi:  20nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Human)
The Sidney Kimmel Comprehensive Cancer Center At Johns Hopkins

Curated by ChEMBL
LigandPNGBDBM50148531(CHEMBL326292 | CHEMBL334279 | 2-[(1-Amino-2-cycloh...)
Affinity DataIC50: 25nMAssay Description:Concentration required to inhibit renal dipeptidase (RDP) by 50% in crude lysates prepared from human colon cancerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024024(2-[(2,2-Dibromo-cyclopropanecarbonyl)-amino]-but-2...)
Affinity DataKi:  30nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Human)
The Sidney Kimmel Comprehensive Cancer Center At Johns Hopkins

Curated by ChEMBL
LigandPNGBDBM50148543(2-[(1-Amino-2-cyclohexyl-ethyl)-hydroxy-phosphinoy...)
Affinity DataIC50: 30nMAssay Description:Concentration required to inhibit renal dipeptidase (RDP) by 50% in crude lysates prepared from human colon cancerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidase 1(Human)
The Sidney Kimmel Comprehensive Cancer Center At Johns Hopkins

Curated by ChEMBL
LigandPNGBDBM50148530(CHEMBL119392 | CHEMBL334143 | 2-[(1-Amino-2-cycloh...)
Affinity DataIC50: 30nMAssay Description:Concentration required to inhibit renal dipeptidase (RDP) by 50% in crude lysates prepared from human colon cancerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidase 1(Human)
The Sidney Kimmel Comprehensive Cancer Center At Johns Hopkins

Curated by ChEMBL
LigandPNGBDBM50148528(CHEMBL332290 | 2-[(1-Amino-2-cyclohexyl-ethyl)-hyd...)
Affinity DataIC50: 40nMAssay Description:Concentration required to inhibit renal dipeptidase (RDP) by 50% in crude lysates prepared from human colon cancerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023951(2-{6-Carboxy-6-[(2,2-dimethyl-cyclopropanecarbonyl...)
Affinity DataKi:  40nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024072(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-8-et...)
Affinity DataKi:  44nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Human)
The Sidney Kimmel Comprehensive Cancer Center At Johns Hopkins

Curated by ChEMBL
LigandPNGBDBM50148541(2-[(1-Amino-2-cyclohexyl-ethyl)-hydroxy-phosphinoy...)
Affinity DataIC50: 45nMAssay Description:Concentration required to inhibit renal dipeptidase (RDP) by 50% in crude lysates prepared from human colon cancerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023999(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-hept...)
Affinity DataKi:  48nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024019(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-oct-...)
Affinity DataKi:  58nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50367508(CHEMBL1907817)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024071(2-[(2,2-Dichloro-cyclopropanecarbonyl)-amino]-oct-...)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Human)
The Sidney Kimmel Comprehensive Cancer Center At Johns Hopkins

Curated by ChEMBL
LigandPNGBDBM50148536(2-[(1-Amino-2-cyclohexyl-ethyl)-hydroxy-phosphinoy...)
Affinity DataIC50: 70nMAssay Description:Concentration required to inhibit renal dipeptidase (RDP) by 50% in crude lysates prepared from human colon cancerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023983(2-[(2,2-Dichloro-cyclopropanecarbonyl)-amino]-but-...)
Affinity DataKi:  80nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50367506(CHEMBL1907823)
Affinity DataKi:  80nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023933(8-Cyano-2-[(2,2-dimethyl-cyclopropanecarbonyl)-ami...)
Affinity DataKi:  82nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024023(Sodium; 6-carboxy-6-[(2,2-dimethyl-cyclopropanecar...)
Affinity DataKi:  87nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024055(2-{6-Carboxy-6-[(2,2-dimethyl-cyclopropanecarbonyl...)
Affinity DataKi:  90nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023947(2,11-Bis-[(2,2-dimethyl-cyclopropanecarbonyl)-amin...)
Affinity DataKi:  92nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024044(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-dec-...)
Affinity DataKi:  96nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Human)
The Sidney Kimmel Comprehensive Cancer Center At Johns Hopkins

Curated by ChEMBL
LigandPNGBDBM50148529(2-[(1-Amino-2-cyclohexyl-ethyl)-hydroxy-phosphinoy...)
Affinity DataIC50: 100nMAssay Description:Concentration required to inhibit renal dipeptidase (RDP) by 50% in crude lysates prepared from human colon cancerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023992(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-7-ph...)
Affinity DataKi:  100nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Human)
The Sidney Kimmel Comprehensive Cancer Center At Johns Hopkins

Curated by ChEMBL
LigandPNGBDBM50148529(2-[(1-Amino-2-cyclohexyl-ethyl)-hydroxy-phosphinoy...)
Affinity DataIC50: 100nMAssay Description:Concentration required to inhibit renal dipeptidase (RDP) by 50% in crude lysates prepared from human colon cancerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024042(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-unde...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023995(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-dode...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50367502(CILASTATIN)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023990(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-hept...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024045(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-hex-...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023942(10-Bromo-2-[(2,2-dimethyl-cyclopropanecarbonyl)-am...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024036(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-5-me...)
Affinity DataKi:  120nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024069(7-Carboxymethylsulfanyl-2-[(2,2-dimethyl-cycloprop...)
Affinity DataKi:  130nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024003(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-6-(3...)
Affinity DataKi:  130nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024078(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-trid...)
Affinity DataKi:  140nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023971(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-hex-...)
Affinity DataKi:  140nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50367507(CHEMBL1237318)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024012(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-8-me...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023963(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-6-me...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024059(7-Bromo-2-[(2,2-dimethyl-cyclopropanecarbonyl)-ami...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetDipeptidase 1(Pig)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023946(4-Cyclohexyl-2-[(2,2-dimethyl-cyclopropanecarbonyl...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
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