Compile Data Set for Download or QSAR
Report error Found 150 Enz. Inhib. hit(s) with Target = 'Follicle-stimulating hormone receptor'
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50403050(CHEMBL2216803)
Affinity DataEC50:  1nMAssay Description:Allosteric activation of human FSH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142662(1-Butyl-1-[4'-((2S,5S)-1,5-dimethyl-4-octyl-3,6-di...)
Affinity DataEC50:  1.20nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142654(2-{(S)-3-[3'-(1-Butyl-3-methyl-ureidomethyl)-biphe...)
Affinity DataEC50:  1.70nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142669([4'-((2S,5S)-1,5-Dimethyl-4-octyl-3,6-dioxo-pipera...)
Affinity DataEC50:  1.80nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142672(Butyl-[4'-((2S,5S)-1,5-dimethyl-4-octyl-3,6-dioxo-...)
Affinity DataEC50:  2.70nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142651(N-Hexyl-2-[(S)-4-methyl-2,5-dioxo-3-(3',4',5'-trim...)
Affinity DataEC50:  3nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142670(1-[4'-((2S,5S)-1,5-Dimethyl-4-octyl-3,6-dioxo-pipe...)
Affinity DataEC50:  3.60nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50410306(CHEMBL436481)
Affinity DataIC50: 5nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50410307(CHEMBL360981)
Affinity DataIC50: 5nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50410303(CHEMBL361847)
Affinity DataIC50: 7nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142675(1-Butyl-1-[4'-((2S,5S)-4-hexyl-1,5-dimethyl-3,6-di...)
Affinity DataEC50:  7.20nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142662(1-Butyl-1-[4'-((2S,5S)-1,5-dimethyl-4-octyl-3,6-di...)
Affinity DataEC50:  7.90nMAssay Description:Agonistic activity in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142656(Butyl-[4'-((2S,5S)-4-hexyl-1,5-dimethyl-3,6-dioxo-...)
Affinity DataEC50:  8.90nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50410309(CHEMBL365545)
Affinity DataIC50: 9nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142675(1-Butyl-1-[4'-((2S,5S)-4-hexyl-1,5-dimethyl-3,6-di...)
Affinity DataEC50:  9.5nMAssay Description:Agonistic activity in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142680(N-[4'-((2S,5S)-1,5-Dimethyl-4-octyl-3,6-dioxo-pipe...)
Affinity DataEC50:  9.70nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50162936(Biphenyl-4-carboxylic acid (1-acetyl-2,2,4-trimeth...)
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of maximum response evoked by cAMP on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142676((3S,6S)-1,3-Dimethyl-4-octyl-6-(3',4',5'-trimethox...)
Affinity DataEC50:  13nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142661(N-Butyl-N-[4'-((2S,5S)-1,5-dimethyl-4-octyl-3,6-di...)
Affinity DataEC50:  14nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50614128(CHEMBL5281228)
Affinity DataIC50: 17nMAssay Description:Allosteric antagonist activity at human FSHR expressed in CHO cells assessed as inhibition of FSH-induced activity incubated for 4 hrs by CRE-lucifer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50649628(CHEMBL5618086)
Affinity DataIC50: 17nMAssay Description:Inhibition of human FSH receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50410304(CHEMBL195469)
Affinity DataIC50: 25nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142657((3S,6S)-1-Heptyl-4,6-dimethyl-3-(3',4',5'-trimetho...)
Affinity DataEC50:  25nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50410302(CHEMBL361167)
Affinity DataIC50: 27nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50162936(Biphenyl-4-carboxylic acid (1-acetyl-2,2,4-trimeth...)
Affinity DataIC50: 28nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50162936(Biphenyl-4-carboxylic acid (1-acetyl-2,2,4-trimeth...)
Affinity DataIC50: 28nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50410308(CHEMBL192868)
Affinity DataIC50: 30nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142672(Butyl-[4'-((2S,5S)-1,5-dimethyl-4-octyl-3,6-dioxo-...)
Affinity DataEC50:  31nMAssay Description:Agonistic activity in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50410298(CHEMBL178980)
Affinity DataIC50: 31nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142676((3S,6S)-1,3-Dimethyl-4-octyl-6-(3',4',5'-trimethox...)
Affinity DataEC50:  32nMAssay Description:Agonistic activity in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142657((3S,6S)-1-Heptyl-4,6-dimethyl-3-(3',4',5'-trimetho...)
Affinity DataEC50:  32nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142661(N-Butyl-N-[4'-((2S,5S)-1,5-dimethyl-4-octyl-3,6-di...)
Affinity DataEC50:  35nMAssay Description:Agonistic activity in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50335479((R)-N-(1-acetyl-2,2,4-trimethyl-4-(4-(prop-2-ynylo...)
Affinity DataIC50: 39nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142656(Butyl-[4'-((2S,5S)-4-hexyl-1,5-dimethyl-3,6-dioxo-...)
Affinity DataEC50:  48nMAssay Description:Agonistic activity in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142656(Butyl-[4'-((2S,5S)-4-hexyl-1,5-dimethyl-3,6-dioxo-...)
Affinity DataEC50:  48nMAssay Description:Agonistic activity in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50410294(CHEMBL195347)
Affinity DataIC50: 50nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50403051(CHEMBL2216804)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human FSH receptor by aromatase-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50410292(CHEMBL192334)
Affinity DataIC50: 54nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50614109(CHEMBL5285685)
Affinity DataIC50: 64nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142674((3S,6R)-1,3-Dimethyl-4-octyl-6-(3',4',5'-trimethox...)
Affinity DataEC50:  68nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50410300(CHEMBL179505)
Affinity DataIC50: 76nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50403051(CHEMBL2216804)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human FSH receptor by cAMP-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50012105(CHEMBL3263667)
Affinity DataEC50:  100nMAssay Description:Positive allosteric modulation of human FSHR expressed in rat granulocytes assessed as FSH-induced estradiol production after 72 hrs by radioimmunoss...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2017
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50012120(CHEMBL3263691)
Affinity DataEC50:  100nMAssay Description:Positive allosteric modulation of human FSHR expressed in rat granulocytes assessed as FSH-induced estradiol production after 72 hrs by radioimmunoss...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2017
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50173579(CHEMBL3809148)
Affinity DataEC50:  100nMAssay Description:Positive allosteric modulation of human FSHR expressed in rat granulocytes assessed as FSH-induced estradiol production after 72 hrs by radioimmunoss...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2017
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50173578(CHEMBL3263694)
Affinity DataEC50: <100nMAssay Description:Positive allosteric modulation of FSHR (unknown origin) expressed in CHO cells assessed as FSH-induced cAMP accumulation incubated for 1 hr by HTRF a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2017
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50173579(CHEMBL3809148)
Affinity DataEC50:  100nMAssay Description:Positive allosteric modulation of FSHR (unknown origin) expressed in CHO cells assessed as FSH-induced cAMP accumulation incubated for 1 hr by HTRF a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2017
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50142665((3S,6S)-1-Hexyl-4,6-dimethyl-3-(3',4',5'-trimethox...)
Affinity DataEC50:  100nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50173580(CHEMBL3808949)
Affinity DataEC50: <100nMAssay Description:Positive allosteric modulation of FSHR (unknown origin) expressed in CHO cells assessed as FSH-induced cAMP accumulation incubated for 1 hr by HTRF a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2017
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50173581(CHEMBL3809644)
Affinity DataEC50: <100nMAssay Description:Positive allosteric modulation of FSHR (unknown origin) expressed in CHO cells assessed as FSH-induced cAMP accumulation incubated for 1 hr by HTRF a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2017
Entry Details Article
PubMed
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