Report error Found 405 Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, kainate 2'
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]kianic acid from recombinant GluK2 kainate receptor (unknown origin) expressed in HEK293 cell membranes measured after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of [3H](2S, 4R)-4-MeGlu (SYM-2081) from GluK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 6.04nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR6More data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity against human ionotropic glutamate receptor ionotropic kainate 2 in HEK293 cells using [3H]kainate as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 11.9nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 12.7nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR6More data for this Ligand-Target Pair
Affinity DataKi: 12.7nMAssay Description:Displacement of [3H]kainic acid from rat recombinant iGluR6(V,C,R) receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR6More data for this Ligand-Target Pair
Affinity DataKi: 18.3nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 18.5nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]KA from rat recombinant GluR6 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 23.3nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 29.8nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 31.7nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity against human ionotropic glutamate receptor ionotropic kainate 2 in HEK293 cells using [3H]kainate as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Compound was tested for agonistic activity at Glutamate receptor 6 using HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 38.4nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKd: 39nMAssay Description:Displacement of [3H]kainate from rat GLUK6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Displacement of [3H]KA from rat recombinant GluR6 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 41.1nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Compound was tested for binding affinity against human Ionotropic glutamate receptor ionotropic kainate 2 in HEK293 cells using [3H]-kainate as radio...More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Displacement of [3H]-kainate from human recombinant GluK2 receptor expressed in HEK293 cell membranes after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 54.3nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 57.4nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Binding affinity against human ionotropic glutamate receptor ionotropic kainate 2 in HEK293 cells using [3H]kainate as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Binding affinity against human ionotropic glutamate receptor ionotropic kainate 2 in HEK293 cells using [3H]kainate as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 82.2nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 90.6nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair

































3D Structure (crystal)