Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with Target = 'Isoform C of Bromodomain-containing protein 4 (Short)'
TargetIsoform C of Bromodomain-containing protein 4 (Short)(Human)
Dana-Farber Cancer Institute

LigandPNGBDBM205429( (R)-JQ1 (3) | US9320741, (R)-JQ1 | US10407441, Co...)
Affinity DataKd:  11nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetIsoform C of Bromodomain-containing protein 4 (Short)(Human)
Dana-Farber Cancer Institute

LigandPNGBDBM205431((6S+2S)-PEG1 (7))
Affinity DataKd:  0.0130nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetIsoform C of Bromodomain-containing protein 4 (Short)(Human)
Dana-Farber Cancer Institute

LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataKd:  3.80E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
Go to US Patent

TargetIsoform C of Bromodomain-containing protein 4 (Short)(Human)
Dana-Farber Cancer Institute

LigandPNGBDBM298346(US10124009, Compound 1)
Affinity DataKd:  1.50E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
Go to US Patent

TargetIsoform C of Bromodomain-containing protein 4 (Short)(Human)
Dana-Farber Cancer Institute

LigandPNGBDBM298347(US10124009, Compound 2)
Affinity DataKd:  1.90E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
Go to US Patent

TargetIsoform C of Bromodomain-containing protein 4 (Short)(Human)
Dana-Farber Cancer Institute

LigandPNGBDBM298348(US10124009, Compound 3)
Affinity DataKd:  1.20E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
Go to US Patent

TargetIsoform C of Bromodomain-containing protein 4 (Short)(Human)
Dana-Farber Cancer Institute

LigandPNGBDBM298349(US10124009, Compound 4)
Affinity DataKd:  1.30E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
Go to US Patent

TargetIsoform C of Bromodomain-containing protein 4 (Short)(Human)
Dana-Farber Cancer Institute

LigandPNGBDBM298350(US10124009, Compound 5)
Affinity DataKd:  400nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
Go to US Patent

TargetIsoform C of Bromodomain-containing protein 4 (Short)(Human)
Dana-Farber Cancer Institute

LigandPNGBDBM298351(US10124009, Compound 7)
Affinity DataKd:  2.10E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
Go to US Patent

TargetIsoform C of Bromodomain-containing protein 4 (Short)(Human)
Dana-Farber Cancer Institute

LigandPNGBDBM50380682(CHEMBL2017291 | I-BET151 (16))
Affinity DataIC50: 29.4nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetIsoform C of Bromodomain-containing protein 4 (Short)(Human)
Dana-Farber Cancer Institute

LigandPNGBDBM205429( (R)-JQ1 (3) | US9320741, (R)-JQ1 | US10407441, Co...)
Affinity DataIC50: 7.76E+3nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetIsoform C of Bromodomain-containing protein 4 (Short)(Human)
Dana-Farber Cancer Institute

LigandPNGBDBM205431((6S+2S)-PEG1 (7))
Affinity DataKi:  0.00780nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetIsoform C of Bromodomain-containing protein 4 (Short)(Human)
Dana-Farber Cancer Institute

LigandPNGBDBM205453(MTI (35))
Affinity DataKi:  0.0620nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed