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Report error Found 538 Enz. Inhib. hit(s) with Target = 'Methionine aminopeptidase 1'
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558959(CHEMBL4740594)
Affinity DataKd:  1.5nMAssay Description:Binding affinity to human MetAP1 expressed in Escherichia coli BL21 (DE3) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558957(CHEMBL4755128)
Affinity DataKd:  3.5nMAssay Description:Binding affinity to human MetAP1 expressed in Escherichia coli BL21 (DE3) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558956(CHEMBL4743733)
Affinity DataKd:  3.60nMAssay Description:Binding affinity to human MetAP1 expressed in Escherichia coli BL21 (DE3) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558967(CHEMBL4759563)
Affinity DataKd:  8.5nMAssay Description:Binding affinity to human MetAP1 expressed in Escherichia coli BL21 (DE3) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50375165(CHEMBL271696)
Affinity DataKi:  10nMAssay Description:Inhibition of human methionine aminopeptidase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50435210(CHEMBL2392907)
Affinity DataEC50:  36nMAssay Description:Inhibition of human recombinant full-length cytosolic METAP1 expressed in Escherichia coli BL21(DE3) using Met-Pro-p-nitroanilide as substrate after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50433382(CHEMBL1329554)
Affinity DataEC50:  49nMAssay Description:Inhibition of human methionine aminopeptidase 1 in presence of Co2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50435211(CHEMBL2392906)
Affinity DataEC50:  49nMAssay Description:Inhibition of human recombinant full-length cytosolic METAP1 expressed in Escherichia coli BL21(DE3) using Met-Pro-p-nitroanilide as substrate after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50435184(CHEMBL2392932)
Affinity DataEC50:  63nMAssay Description:Inhibition of human recombinant full-length cytosolic METAP1 expressed in Escherichia coli BL21(DE3) using Met-Pro-p-nitroanilide as substrate after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50433386(CHEMBL2375615)
Affinity DataEC50:  73nMAssay Description:Inhibition of human methionine aminopeptidase 1 in presence of Co2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Baker's yeast)
Shanghai Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50170371(5-Piperidin-1-ylmethyl-thiazole-4-carboxylic acid ...)
Affinity DataIC50: 75nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50433393(CHEMBL2375622)
Affinity DataEC50:  81nMAssay Description:Inhibition of human methionine aminopeptidase 1 in presence of Co2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50433373(CHEMBL2375609)
Affinity DataEC50:  93nMAssay Description:Inhibition of human methionine aminopeptidase 1 in presence of Co2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50435202(CHEMBL2392914)
Affinity DataEC50:  93nMAssay Description:Inhibition of human recombinant full-length cytosolic METAP1 expressed in Escherichia coli BL21(DE3) using Met-Pro-p-nitroanilide as substrate after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50433391(CHEMBL2375620)
Affinity DataEC50:  94nMAssay Description:Inhibition of human methionine aminopeptidase 1 in presence of Co2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50433387(CHEMBL2375616)
Affinity DataEC50:  94nMAssay Description:Inhibition of human methionine aminopeptidase 1 in presence of Co2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50433395(CHEMBL2375624)
Affinity DataEC50:  100nMAssay Description:Inhibition of human methionine aminopeptidase 1 in presence of Co2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50267199(CHEMBL4079583)
Affinity DataIC50: 100nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50433392(CHEMBL2375621)
Affinity DataEC50:  110nMAssay Description:Inhibition of human methionine aminopeptidase 1 in presence of Co2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50433381(CHEMBL2375613)
Affinity DataEC50:  110nMAssay Description:Inhibition of human methionine aminopeptidase 1 in presence of Co2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50433380(CHEMBL2375612)
Affinity DataEC50:  120nMAssay Description:Inhibition of human methionine aminopeptidase 1 in presence of Co2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50433374(CHEMBL2375610)
Affinity DataEC50:  120nMAssay Description:Inhibition of human methionine aminopeptidase 1 in presence of Co2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Baker's yeast)
Shanghai Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50169672(5-(Cyclopentanecarbonyl-amino)-thiazole-4-carboxyl...)
Affinity DataIC50: 130nMAssay Description:Inhibitory concentration required against Saccharomyces cerevisiae MetAP1 (330 nM) More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50435207(CHEMBL2392910)
Affinity DataEC50:  140nMAssay Description:Inhibition of human recombinant full-length cytosolic METAP1 expressed in Escherichia coli BL21(DE3) using Met-Pro-p-nitroanilide as substrate after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Baker's yeast)
Shanghai Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50129648(3-(4-Methyl-pent-3-enoylamino)-pyridine-2-carboxyl...)
Affinity DataIC50: 140nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Baker's yeast)
Shanghai Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50170369(5-(2-Ethoxy-3-methyl-butyl)-thiazole-4-carboxylic ...)
Affinity DataIC50: 150nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50435201(CHEMBL2392915)
Affinity DataEC50:  160nMAssay Description:Inhibition of human recombinant full-length cytosolic METAP1 expressed in Escherichia coli BL21(DE3) using Met-Pro-p-nitroanilide as substrate after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50435183(CHEMBL2392933)
Affinity DataEC50:  160nMAssay Description:Inhibition of human recombinant full-length cytosolic METAP1 expressed in Escherichia coli BL21(DE3) using Met-Pro-p-nitroanilide as substrate after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50433389(CHEMBL2375618)
Affinity DataEC50:  180nMAssay Description:Inhibition of human methionine aminopeptidase 1 in presence of Co2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50433375(GNF-Pf-359 | CHEMBL472879)
Affinity DataEC50:  190nMAssay Description:Inhibition of human methionine aminopeptidase 1 in presence of Co2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Baker's yeast)
Shanghai Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50129642(Phenyl-acetic acid 2-(thiazol-2-ylcarbamoyl)-pyrid...)
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50435182(CHEMBL2392934)
Affinity DataEC50:  200nMAssay Description:Inhibition of human recombinant full-length cytosolic METAP1 expressed in Escherichia coli BL21(DE3) using Met-Pro-p-nitroanilide as substrate after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50435195(CHEMBL2392921)
Affinity DataEC50:  200nMAssay Description:Inhibition of human recombinant full-length cytosolic METAP1 expressed in Escherichia coli BL21(DE3) using Met-Pro-p-nitroanilide as substrate after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMethionine aminopeptidase 1(Baker's yeast)
Shanghai Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50169671(5-Propionylamino-thiazole-4-carboxylic acid thiazo...)
Affinity DataIC50: 220nMAssay Description:Inhibitory concentration required against Saccharomyces cerevisiae MetAP1 (330 nM) More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50435198(CHEMBL2392918)
Affinity DataEC50:  220nMAssay Description:Inhibition of human recombinant full-length cytosolic METAP1 expressed in Escherichia coli BL21(DE3) using Met-Pro-p-nitroanilide as substrate after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Baker's yeast)
Shanghai Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50170363(5-[2-(2-Chloro-phenyl)-2-methoxy-ethyl]-thiazole-4...)
Affinity DataIC50: 230nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50433399(CHEMBL2375608)
Affinity DataEC50:  250nMAssay Description:Inhibition of human methionine aminopeptidase 1 in presence of Co2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Baker's yeast)
Shanghai Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50169669(5-(Cyclobutanecarbonyl-amino)-thiazole-4-carboxyli...)
Affinity DataIC50: 250nMAssay Description:Inhibitory concentration required against Saccharomyces cerevisiae MetAP1 (330 nM) More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50435197(CHEMBL2392919)
Affinity DataEC50:  260nMAssay Description:Inhibition of human recombinant full-length cytosolic METAP1 expressed in Escherichia coli BL21(DE3) using Met-Pro-p-nitroanilide as substrate after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50435196(CHEMBL2392920)
Affinity DataEC50:  260nMAssay Description:Inhibition of human recombinant full-length cytosolic METAP1 expressed in Escherichia coli BL21(DE3) using Met-Pro-p-nitroanilide as substrate after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Baker's yeast)
Shanghai Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50170383(5-[2-(2-Fluoro-phenyl)-2-methoxy-ethyl]-thiazole-4...)
Affinity DataIC50: 270nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50435212(CHEMBL2392905)
Affinity DataEC50:  270nMAssay Description:Inhibition of human recombinant full-length cytosolic METAP1 expressed in Escherichia coli BL21(DE3) using Met-Pro-p-nitroanilide as substrate after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50433377(CHEMBL2375628)
Affinity DataEC50:  280nMAssay Description:Inhibition of human methionine aminopeptidase 1 in presence of Co2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50435208(CHEMBL2392909)
Affinity DataEC50:  300nMAssay Description:Inhibition of human recombinant full-length cytosolic METAP1 expressed in Escherichia coli BL21(DE3) using Met-Pro-p-nitroanilide as substrate after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Baker's yeast)
Shanghai Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50129669(3-(5-Methyl-hex-4-enoylamino)-pyridine-2-carboxyli...)
Affinity DataIC50: 310nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Baker's yeast)
Shanghai Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50170370(5-[2-Methoxy-2-(4-methoxy-phenyl)-ethyl]-thiazole-...)
Affinity DataIC50: 310nMAssay Description:Inhibitory concentration against ScMetAP1 enzyme activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Baker's yeast)
Shanghai Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50129649(Cyclohexanecarboxylic acid 2-(thiazol-2-ylcarbamoy...)
Affinity DataIC50: 320nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Baker's yeast)
Shanghai Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50129635(3-Formylamino-pyridine-2-carboxylic acid thiazol-2...)
Affinity DataIC50: 320nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50042874(2,2'-bipyridine | 2,2'-Bipyridin | 2,2'-bipyridyl ...)
Affinity DataEC50:  320nMAssay Description:Inhibition of human methionine aminopeptidase 1 in presence of Co2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50435188(CHEMBL2392928)
Affinity DataEC50:  330nMAssay Description:Inhibition of human recombinant full-length cytosolic METAP1 expressed in Escherichia coli BL21(DE3) using Met-Pro-p-nitroanilide as substrate after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
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