Compile Data Set for Download or QSAR
Report error Found 223 Enz. Inhib. hit(s) with Target = 'Microtubule-associated protein 2'
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50088527(CHEMBL3527358)
Affinity DataEC50:  0.0950nMAssay Description:Inhibition of MetAP2 activity in HUVEC assessed as inhibition of cell proliferation by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2016
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50088526(CHEMBL3527591)
Affinity DataEC50:  0.300nMAssay Description:Inhibition of MetAP2 activity in HUVEC assessed as inhibition of cell proliferation by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2016
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50088525(CHEMBL3526173)
Affinity DataEC50:  1.30nMAssay Description:Inhibition of MetAP2 activity in HUVEC assessed as inhibition of cell proliferation by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2016
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50547191(CHEMBL4746468)
Affinity DataIC50: 2nMAssay Description:Inhibition of MetAP2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167916(CHEMBL3798615)
Affinity DataIC50: 3nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50547190(CHEMBL4762949)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of MetAP2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167926(CHEMBL3798871)
Affinity DataIC50: 4nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167915(CHEMBL3798727)
Affinity DataIC50: 4nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167922(CHEMBL3797286)
Affinity DataIC50: 5nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167274(CHEMBL3797399)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167275(CHEMBL3798249)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167959(CHEMBL3799242)
Affinity DataIC50: 5nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167960(CHEMBL3799512)
Affinity DataIC50: 5nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50547180(CHEMBL4796852)
Affinity DataIC50: 5nMAssay Description:Inhibition of MetAP2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167929(CHEMBL3798702)
Affinity DataIC50: 5nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167961(CHEMBL3800596)
Affinity DataIC50: 6nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167917(CHEMBL3797663)
Affinity DataIC50: 6nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167279(CHEMBL3799090)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167280(CHEMBL3797259)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50547179(CHEMBL4743507)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of MetAP2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50088524(CHEMBL3527328)
Affinity DataEC50:  6.5nMAssay Description:Inhibition of MetAP2 activity in HUVEC assessed as inhibition of cell proliferation by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2016
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50088523(CHEMBL3527383)
Affinity DataEC50:  7.10nMAssay Description:Inhibition of MetAP2 activity in HUVEC assessed as inhibition of cell proliferation by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2016
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167278(CHEMBL3800236)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167276(CHEMBL3798844)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167919(CHEMBL3799449)
Affinity DataIC50: 8nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167920(CHEMBL3800546)
Affinity DataIC50: 8nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167921(CHEMBL3800534)
Affinity DataIC50: 8nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50088522(CHEMBL3527218)
Affinity DataEC50:  8.80nMAssay Description:Inhibition of MetAP2 activity in HUVEC assessed as inhibition of cell proliferation by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2016
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167918(CHEMBL3799467)
Affinity DataIC50: 9nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167923(CHEMBL3797707)
Affinity DataIC50: 10nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167281(CHEMBL3799796)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167285(CHEMBL3797780)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167914(CHEMBL3798034)
Affinity DataIC50: 11nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167927(CHEMBL3800090)
Affinity DataIC50: 11nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50088521(CHEMBL3527219)
Affinity DataEC50:  12nMAssay Description:Inhibition of MetAP2 activity in HUVEC assessed as inhibition of cell proliferation by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2016
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167274(CHEMBL3797399)
Affinity DataEC50:  13nMAssay Description:Inhibition of human MetAP2 in HUVEC cells assessed as accumulation of N-Met 14-3-3gamma after 24 hrs by western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167925(CHEMBL3798047)
Affinity DataIC50: 13nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167277(CHEMBL3797386)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167924(CHEMBL3798381)
Affinity DataIC50: 15nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167960(CHEMBL3799512)
Affinity DataEC50:  15nMAssay Description:Inhibition of MetAP2 in HUVEC assessed as accumulation of N-Met-14-3-3gamma after 24 hrs by Western blot methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167909(CHEMBL3798509)
Affinity DataIC50: 20nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167279(CHEMBL3799090)
Affinity DataEC50:  20nMAssay Description:Inhibition of human MetAP2 in HUVEC cells assessed as accumulation of N-Met 14-3-3gamma after 24 hrs by western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167928(CHEMBL3797699)
Affinity DataIC50: 21nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50547187(CHEMBL4791887)
Affinity DataIC50: 25nMAssay Description:Inhibition of MetAP2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167281(CHEMBL3799796)
Affinity DataEC50:  25nMAssay Description:Inhibition of human MetAP2 in HUVEC cells assessed as accumulation of N-Met 14-3-3gamma after 24 hrs by western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50547178(CHEMBL4800438)
Affinity DataIC50: 25nMAssay Description:Inhibition of MetAP2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167278(CHEMBL3800236)
Affinity DataEC50:  32nMAssay Description:Inhibition of human MetAP2 in HUVEC cells assessed as accumulation of N-Met 14-3-3gamma after 24 hrs by western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167925(CHEMBL3798047)
Affinity DataEC50:  37nMAssay Description:Inhibition of MetAP2 in HUVEC assessed as accumulation of N-Met-14-3-3gamma after 24 hrs by Western blot methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50167929(CHEMBL3798702)
Affinity DataEC50:  38nMAssay Description:Inhibition of MetAP2 in HUVEC assessed as accumulation of N-Met-14-3-3gamma after 24 hrs by Western blot methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50234032(CHEMBL4060668)
Affinity DataIC50: 38nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed
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