Report error Found 1277 Enz. Inhib. hit(s) with Target = 'Nuclear factor erythroid 2-related factor 2'
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: 2.5nMAssay Description:Modulation of Keap1-Nrf2 protein-protein interaction in human U2OS cells assessed as inhibition of Keap1 by PathHunter assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: 2.90nMAssay Description:Modulation of Keap1-Nrf2 protein-protein interaction in human U2OS cells assessed as inhibition of Keap1 by PathHunter assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: 3.10nMAssay Description:Modulation of Keap1-Nrf2 protein-protein interaction in human U2OS cells assessed as inhibition of Keap1 by PathHunter assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: 3.20nMAssay Description:Modulation of Keap1-Nrf2 protein-protein interaction in human U2OS cells assessed as inhibition of Keap1 by PathHunter assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 3.70nMAssay Description:Inhibition of human Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3 pLysS cells/Nrf2 (unknown origin) protein-protein...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: 4.5nMAssay Description:Modulation of Keap1-Nrf2 protein-protein interaction in human U2OS cells assessed as inhibition of Keap1 by PathHunter assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataKd: 5nMAssay Description:Binding affinity to Keap1/Nrf2 complex (unknown origin) by ITC methodMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: 5.80nMAssay Description:Modulation of Keap1-Nrf2 protein-protein interaction in human U2OS cells assessed as inhibition of Keap1 by PathHunter assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataKi: 6.40nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 7.20nMAssay Description:Inhibition of recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)pLysS cells interaction with FITC-9m...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataKi: 7.60nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 8.90nMAssay Description:Inhibition of recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)pLysS cells interaction with FITC-9m...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataKi: 9.10nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: 9.20nMAssay Description:Activation of Nrf2 in human spinal cord astrocytes assessed as increase in glutathione level after 20 hrsMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: <10nMAssay Description:NAD(P)H:quinone oxidoreductase 1 (NQO1), also called DT diaphorase, is a homodimeric FAD-containing enzyme that catalyzes obligatory NAD(P)H-dependen...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: <10nMAssay Description:NAD(P)H:quinone oxidoreductase 1 (NQO1), also called DT diaphorase, is a homodimeric FAD-containing enzyme that catalyzes obligatory NAD(P)H-dependen...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of Keap1 kelch domain (unknow origin)/Nrf2-ETGE peptide (unknown origin) interaction by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: <10nMAssay Description:NAD(P)H:quinone oxidoreductase 1 (NQO1), also called DT diaphorase, is a homodimeric FAD-containing enzyme that catalyzes obligatory NAD(P)H-dependen...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of full length Flag/His-tagged Keap1 kelch domain (unknown origin)/full length Avi-tagged Nrf2 (unknown origin) interaction after 2.25 hrs...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of full length Flag/His-tagged Keap1 kelch domain (unknown origin)/full length Avi-tagged Nrf2 (unknown origin) interaction after 2.25 hrs...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human U2OS cells co-expressing Keap1 assessed as increase in Nrf2 nuclear translocation incubated fo...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Activation of Nrf2 in human BEAS2B cells assessed as increase in NQO1 enzymatic activity measured after 48 hrs by MTT assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)pLysS cells interaction with FITC-9m...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)pLysS cells interaction with FITC-9m...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Inhibition of KEAP1/NRF2 interaction in human BEAS2B cells assessed as induction of NQO1 specific activity incubated for 48 hrs measured on day 4 pos...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of Keap1 Kelch domain/FITC-9mer Nrf2 (unknown origin) interaction after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of Keap1 Kelch domain-Nrf2 ETGE (unknown origin) protein-protein interaction incubated for 30 mins by fluorescence polarization competitio...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: 16nMAssay Description:Inhibition of KEAP1/NRF2 interaction in human bronchial epithelial cells from COPD patient assessed as induction of HO-1 mRNA expression incubated fo...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of Keap1 Kelch domain/FITC-9mer Nrf2 (unknown origin) interaction after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of Keap1 Kelch domain-Nrf2 ETGE (unknown origin) protein-protein interaction incubated for 30 mins by fluorescence polarization competitio...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Activation of Nrf2 in human PathHunter U2OS Keap1-Nrf2 cells assessed as Nrf2 nuclear translocation by chemiluminescent assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of Keap1/Nrf2 (unknown origin) interaction assessed as displacement of FITC-betaAla-DEETGEF-OH from Keap1 Kelch domain after 1 hr by FITC-...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of NRF2 in human KYSE-70 cellsMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: 22nMAssay Description:Inhibition of KEAP1/NRF2 interaction in human bronchial epithelial cells from COPD patient assessed as induction of NQO1 mRNA expression incubated fo...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)pLysS cells interaction with FITC-9m...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of Keap1 Kelch domain (unknown origin) /Nrf2 (unknown origin) interaction using fluorescein-labeled 9-mer peptide containing NRF2 Neh2 dom...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: 26nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human U2OS cells co-expressing Keap1 assessed as increase in Nrf2 nuclear translocation incubated fo...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of human Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3 pLysS cells/Nrf2 (unknown origin) protein-protein...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: 27nMAssay Description:Inhibition of KEAP1/NRF2 interaction in human bronchial epithelial cells from COPD patient assessed as induction of TXNRD1 mRNA expression incubated ...More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataEC50: 29nMAssay Description:Inhibition of Keap1 (unknown origin) interaction to Nrf2More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of Keap1/Nrf2 complex (unknown origin)More data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey
Curated by ChEMBL
The State University of New Jersey
Curated by ChEMBL
Affinity DataKd: 29nMAssay Description:Binding affinity to Keap1/Nrf2 complex (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair


































