Compile Data Set for Download or QSAR
Report error Found 872 Enz. Inhib. hit(s) with Target = 'Neuropeptide Y receptor type 4'
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50630037(CHEMBL5395013)
Affinity DataKd:  0.00200nMAssay Description:Binding affinity to human Y4R expressed in CHO cells co-expressing Gqi5-mtAEQ assessed as dissociation constant under sodium free buffer conditionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Rat)
Uppsala University

Curated by PDSP Ki Database
LigandPNGBDBM82300(NSC_41735 | CAS_59763-91-6 | PP, rat)
Affinity DataKi:  0.00270nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Rat)
Uppsala University

Curated by PDSP Ki Database
LigandPNGBDBM82286(CAS_59763-91-6 | PP,SALMON | PP, human)
Affinity DataKi:  0.00300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Rat)
Uppsala University

Curated by PDSP Ki Database
LigandPNGBDBM82297(CAS_59763-91-6 | PP, BOVINE)
Affinity DataKi:  0.00600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Rat)
Uppsala University

Curated by PDSP Ki Database
LigandPNGBDBM85378(PP, guinea pig)
Affinity DataKi:  0.00700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50466554(CHEMBL4286615)
Affinity DataKi:  0.0100nMAssay Description:Displacement of [125I]-PP from human Y4R expressed in CHO-K1 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50466554(CHEMBL4286615)
Affinity DataKi:  0.0100nMAssay Description:Displacement of [125I]-PP from human Y4R expressed in CHO-K1 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50630036(CHEMBL5423253)
Affinity DataKi:  0.0100nMAssay Description:Displacement of [3H]-(9S,12S,15S,19R,E)-4-amino-N-((S)-1-(((S)-1-(((S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl)amino)-5-guanidino-1-oxopentan-2-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50466543(CHEMBL4276961)
Affinity DataKi:  0.0100nMAssay Description:Displacement of [125I]-PP from human Y4R expressed in CHO-K1 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50466543(CHEMBL4276961)
Affinity DataKi:  0.0100nMAssay Description:Displacement of [125I]-PP from human Y4R expressed in CHO-K1 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50578262(CHEMBL4873376)
Affinity DataKi:  0.0110nMAssay Description:Displacement of [3H]-(9S,12S,15S,19R,E)-4-amino-N-((S)-1-(((S)-1-(((S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl)amino)-5-guanidino-1-oxopentan-2-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50630037(CHEMBL5395013)
Affinity DataKd:  0.0120nMAssay Description:Binding affinity to human Y4R expressed in CHO cells co-expressing Gqi5-mtAEQ under sodium free buffer conditionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50630037(CHEMBL5395013)
Affinity DataKd:  0.0140nMAssay Description:Binding affinity to human Y4R expressed in CHO cells co-expressing Gqi5-mtAEQ assessed as dissociation constant preincubated for 20 mins under DPBS c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50528183(CHEMBL4540843)
Affinity DataKi:  0.0230nMAssay Description:Binding affinity to human Y4R under hypotonic sodium free conditionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50630027(CHEMBL5437701)
Affinity DataKi:  0.0260nMAssay Description:Displacement of [3H]UR-KK200 from human Y4R expressed in CHO cells co-expressing Gqi5-mtAEQMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50240829(CHEMBL3559801)
Affinity DataEC50:  0.0300nMAssay Description:Positive allosteric modulation of human NY4 receptor expressed in African green monkey COS7 cells co-expressing delta6Galphaqi4-myr assessed as poten...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM82297(CAS_59763-91-6 | PP, BOVINE)
Affinity DataKi:  0.0310nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50630026(CHEMBL5422869)
Affinity DataKi:  0.0310nMAssay Description:Displacement of [3H]UR-KK200 from human Y4R expressed in CHO cells co-expressing Gqi5-mtAEQMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50578268(CHEMBL4856311)
Affinity DataKi:  0.0330nMAssay Description:Displacement of [3H]UR-KK200 from human neuropeptide Y Y4 receptor expressed in CHO-mtAEQ cells co-expressing Gqi5 measured after 90 mins by scintill...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50578268(CHEMBL4856311)
Affinity DataKi:  0.0330nMAssay Description:Displacement of [3H]UR-KK200 from human Y4 receptor expressed in CHO-Gqi5-mtAQE cells measured after 90 mins by MicroBeta plate counter based competi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50630036(CHEMBL5423253)
Affinity DataKi:  0.0360nMAssay Description:Displacement of [3H]UR-KK200 from human Y4R expressed in CHO cells co-expressing Gqi5-mtAEQMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50528183(CHEMBL4540843)
Affinity DataKi:  0.0370nMAssay Description:Displacement of [3H]-(9S,12S,15S,19R,E)-4-amino-N-((S)-1-(((S)-1-(((S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl)amino)-5-guanidino-1-oxopentan-2-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM82286(CAS_59763-91-6 | PP,SALMON | PP, human)
Affinity DataKi:  0.0390nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50240829(CHEMBL3559801)
Affinity DataEC50:  0.0398nMAssay Description:Positive allosteric modulation of human NY4 receptor expressed in African green monkey COS7 cells co-expressing delta6Galphaqi4-myr assessed as poten...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50630028(CHEMBL5435492)
Affinity DataKi:  0.0410nMAssay Description:Displacement of [3H]UR-KK200 from human Y4R expressed in CHO cells co-expressing Gqi5-mtAEQMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50578262(CHEMBL4873376)
Affinity DataKi:  0.0480nMAssay Description:Displacement of [3H]UR-KK200 from human Y4 receptor expressed in CHO-Gqi5-mtAQE cells measured after 90 mins by MicroBeta plate counter based competi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50578262(CHEMBL4873376)
Affinity DataKi:  0.0480nMAssay Description:Displacement of [3H]UR-KK200 from human neuropeptide Y Y4 receptor expressed in CHO-mtAEQ cells co-expressing Gqi5 measured after 90 mins by scintill...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM82286(CAS_59763-91-6 | PP,SALMON | PP, human)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2011
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50185364(Sub[-Tyr-Arg-Leu-Arg-Tyr-NH2]2 | CHEMBL415187 | CH...)
Affinity DataKi:  0.0500nMAssay Description:Agonist activity at human NPY4 receptor in HEK293 cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM85378(PP, guinea pig)
Affinity DataKi:  0.0600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM85679(CAS_59763-91-6 | PP, human)
Affinity DataKi:  0.0600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50240829(CHEMBL3559801)
Affinity DataKi:  0.0631nMAssay Description:Effect on pancreatic polypeptide-mediated displacement of 125I-pancreatic polypeptide from human C-terminal eYFP-tagged NY4 receptor expressed in HEK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50630034(CHEMBL5437695)
Affinity DataKi:  0.0660nMAssay Description:Displacement of [3H]UR-KK200 from human Y4R expressed in CHO cells co-expressing Gqi5-mtAEQMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM82297(CAS_59763-91-6 | PP, BOVINE)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2011
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Mouse)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50620388(CHEMBL5420881)
Affinity DataEC50:  0.0700nMAssay Description:Positive allosteric modulation of mouse Y4 receptor transfected with COS-7 cells assessed as activation of G-protein signaling measured after 24 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM82286(CAS_59763-91-6 | PP,SALMON | PP, human)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM82300(NSC_41735 | CAS_59763-91-6 | PP, rat)
Affinity DataKi:  0.0710nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50578262(CHEMBL4873376)
Affinity DataKi:  0.0760nMAssay Description:Displacement of [3H]-(9S,12S,15S,19R,E)-4-amino-N-((S)-1-(((S)-1-(((S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl)amino)-5-guanidino-1-oxopentan-2-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM82294(PP2-36, HUMAN)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2011
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50099198(Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly-Glu-Asp-Ala-Pr...)
Affinity DataKi:  0.0800nMAssay Description:Affinity for cloned Y4 receptor using [125I]PP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50630036(CHEMBL5423253)
Affinity DataKi:  0.0880nMAssay Description:Displacement of [3H]-(9S,12S,15S,19R,E)-4-amino-N-((S)-1-(((S)-1-(((S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl)amino)-5-guanidino-1-oxopentan-2-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM82289(I31,G34-PP,human)
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2011
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50630037(CHEMBL5395013)
Affinity DataKd:  0.0900nMAssay Description:Binding affinity to human Y4R expressed in CHO cells co-expressing Gqi5-mtAEQ assessed as dissociation constant preincubated for 2 hrs under DPBS con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50630030(CHEMBL5421880)
Affinity DataKi:  0.0930nMAssay Description:Displacement of [3H]UR-KK200 from human Y4R expressed in CHO cells co-expressing Gqi5-mtAEQMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50528183(CHEMBL4540843)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]UR-KK200 from human Y4R expressed in CHO cells co-expressing Gqi5-mtAEQMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Mouse)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466543(CHEMBL4276961)
Affinity DataEC50:  0.100nMAssay Description:Displacement of [125I]-PYY(1 to 36 residues) from mouse Y4R expressed in HEK293 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50466547(CHEMBL4278700)
Affinity DataKi:  0.100nMAssay Description:Displacement of [125I]-PP from human Y4R expressed in CHO-K1 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Mouse)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466543(CHEMBL4276961)
Affinity DataEC50:  0.100nMAssay Description:Displacement of [125I]-PYY(1 to 36 residues) from mouse Y4R expressed in HEK293 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50466547(CHEMBL4278700)
Affinity DataKi:  0.100nMAssay Description:Displacement of [125I]-PP from human Y4R expressed in CHO-K1 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM82291(P34-PYY,human)
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2011
Entry Details Article
PubMed
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