Report error Found 168 Enz. Inhib. hit(s) with Target = 'Protein Tat'
Affinity DataKd: 25nMAssay Description:Dissociation constant for TAR RNAMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of Tat peptide binding to HIV-1 TAR RNAMore data for this Ligand-Target Pair
Affinity DataKd: 30nMAssay Description:Dissociation constant for TAR RNAMore data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
Affinity DataKd: 290nMAssay Description:Dissociation constant for TAR RNAMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of Tat peptide binding to HIV-1 TAR RNAMore data for this Ligand-Target Pair
Affinity DataEC50: 800nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataEC50: 900nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Inhibition of Tat-mediated transcription of viral promoter in 293 T cells transfected with HIV1 tat by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataEC50: 1.30E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataEC50: 1.30E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataEC50: 1.70E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of Tat peptide binding to HIV-1 TAR RNAMore data for this Ligand-Target Pair
Affinity DataKd: 1.80E+3nMT: 2°CAssay Description:In vitro binding affinity towards Tat/TAR to determine interaction between TAR RNA and Tat peptide at room temperature using fluorescence spectrophot...More data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataEC50: 2.20E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataEC50: 2.60E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.60E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of HIV-1 nuclear regulatory protein TatMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of HIV-1 nuclear regulatory protein TatMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataEC50: 2.80E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataEC50: 2.90E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataEC50: 3.10E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
Affinity DataEC50: 3.10E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataEC50: 3.30E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+3nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.60E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataEC50: 3.60E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataEC50: 3.70E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataEC50: 3.70E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of HIV-1 nuclear regulatory protein TatMore data for this Ligand-Target Pair
Affinity DataEC50: 4.30E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+3nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.70E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair













































