Compile Data Set for Download or QSAR
Report error Found 143 Enz. Inhib. hit(s) with Target = 'Relaxin-3 receptor 1'
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50534453(CHEMBL4557279)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human RXFP3 receptor expressed in CHOK1 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by alphascreen surefire ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581017(CHEMBL5081158)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581020(CHEMBL5094669)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581018(CHEMBL5084331)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581019(CHEMBL5089949)
Affinity DataEC50:  3.10nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50534453(CHEMBL4557279)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at human RXFP3 receptor expressed in CHOK1 cells cotransfected with beta-galactosidase assessed as inhibition of forskolin-stimulate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50534454(CHEMBL4540069)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at human RXFP3 receptor expressed in CHOK1 cells cotransfected with beta-galactosidase assessed as inhibition of forskolin-stimulate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50382991(CHEMBL2030700)
Affinity DataIC50: 4.27nMAssay Description:Agonist activity at RXFP3 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 6 hrs by beta galactosidase r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50561919(CHEMBL4781389)
Affinity DataEC50:  4.40nMAssay Description:Agonist activity at RXFP3 (unknown origin) stably expressed in CHO-K1 cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50534445(CHEMBL4476408)
Affinity DataEC50:  4.5nMAssay Description:Agonist activity at human RXFP3 receptor expressed in CHOK1 cells cotransfected with beta-galactosidase assessed as inhibition of forskolin-stimulate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50534448(CHEMBL4435599)
Affinity DataEC50:  4.5nMAssay Description:Agonist activity at human RXFP3 receptor expressed in CHOK1 cells cotransfected with beta-galactosidase assessed as inhibition of forskolin-stimulate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50382992(CHEMBL2030701)
Affinity DataIC50: 5.13nMAssay Description:Agonist activity at RXFP3 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 6 hrs by beta galactosidase r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50534442(CHEMBL4438620)
Affinity DataEC50:  5.20nMAssay Description:Agonist activity at human RXFP3 receptor expressed in CHOK1 cells cotransfected with beta-galactosidase assessed as inhibition of forskolin-stimulate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581016(CHEMBL5083969)
Affinity DataEC50:  5.60nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50561920(CHEMBL4764969)
Affinity DataEC50:  6.20nMAssay Description:Agonist activity at RXFP3 (unknown origin) stably expressed in CHO-K1 cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50561918(CHEMBL4761849)
Affinity DataEC50:  6.20nMAssay Description:Agonist activity at RXFP3 (unknown origin) stably expressed in CHO-K1 cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581010(CHEMBL5072593)
Affinity DataEC50:  7.70nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581017(CHEMBL5081158)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as beta arrestin-2 recruitment measured after 4 hrs by beta-galactosidase ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50605987(CHEMBL5185575)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]R3/I5 from human RXFP3 expressed in CHO-K1 cells membrane assessed as inhibition constant incubated for 1 hr by microplate scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581012(CHEMBL5077251)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50534443(CHEMBL4447532)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human RXFP3 receptor expressed in CHOK1 cells cotransfected with beta-galactosidase assessed as inhibition of forskolin-stimulate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581019(CHEMBL5089949)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as beta arrestin-2 recruitment measured after 4 hrs by beta-galactosidase ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50382993(CHEMBL2030702)
Affinity DataIC50: 12.6nMAssay Description:Agonist activity at RXFP3 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 6 hrs by beta galactosidase r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50561921(CHEMBL4778498)
Affinity DataEC50:  13nMAssay Description:Agonist activity at RXFP3 (unknown origin) stably expressed in CHO-K1 cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581009(CHEMBL5094670)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581008(CHEMBL5078386)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50561922(CHEMBL4799017)
Affinity DataEC50:  16nMAssay Description:Agonist activity at RXFP3 (unknown origin) stably expressed in CHO-K1 cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50526409(CHEMBL4522365)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50580994(CHEMBL5080438)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50526409(CHEMBL4522365)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as beta arrestin-2 recruitment measured after 4 hrs by beta-galactosidase ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50561918(CHEMBL4761849)
Affinity DataKi:  46nMAssay Description:Displacement of Eu-labeled H3B1-22R from RXFP3 (unknown origin) stably expressed in CHO-K1 cells by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581002(CHEMBL5078678)
Affinity DataEC50:  52nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581015(CHEMBL5094396)
Affinity DataEC50:  53nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581006(CHEMBL5076246)
Affinity DataEC50:  56nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581004(CHEMBL5075697)
Affinity DataEC50:  67nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581019(CHEMBL5089949)
Affinity DataKi:  69nMAssay Description:Displacement of [125I]R3/I5 from human RXFP3 expressed in human CHO-K1 cells incubated for 1 hr by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581003(CHEMBL5084431)
Affinity DataEC50:  70nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581014(CHEMBL5078074)
Affinity DataEC50:  73nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50526406(CHEMBL4546426)
Affinity DataEC50:  75nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50526409(CHEMBL4522365)
Affinity DataEC50:  82nMAssay Description:Agonist activity at human RXFP3 expressed in CHOK1 cells assessed as inhibition of forskolin-stimulated intracellular cAMP accumulation preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50580993(CHEMBL5078324)
Affinity DataEC50:  82nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50534445(CHEMBL4476408)
Affinity DataKi:  93nMAssay Description:Displacement of Eu-H3/15 from human RXFP3 receptor expressed in CHOK1 cells by time-resolved fluorescent whole cell binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50581007(CHEMBL5082272)
Affinity DataEC50:  98nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50534442(CHEMBL4438620)
Affinity DataKi:  107nMAssay Description:Displacement of Eu-H3/15 from human RXFP3 receptor expressed in CHOK1 cells by time-resolved fluorescent whole cell binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50382993(CHEMBL2030702)
Affinity DataKi:  110nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50561920(CHEMBL4764969)
Affinity DataKi:  110nMAssay Description:Displacement of Eu-labeled H3B1-22R from RXFP3 (unknown origin) stably expressed in CHO-K1 cells by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50534454(CHEMBL4540069)
Affinity DataKi:  110nMAssay Description:Displacement of Eu-H3/15 from human RXFP3 receptor expressed in CHOK1 cells by time-resolved fluorescent whole cell binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50382991(CHEMBL2030700)
Affinity DataKi:  112nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50382992(CHEMBL2030701)
Affinity DataKi:  112nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50526409(CHEMBL4522365)
Affinity DataEC50:  119nMAssay Description:Agonist activity at human RXFP3 expressed in CHOK1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding after 3 hrs by scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
Displayed 1 to 50 (of 143 total ) | Next | Last >>
Jump to: