Compile Data Set for Download or QSAR
Report error Found 1092 Enz. Inhib. hit(s) with Target = 'Urotensin-2 receptor'
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048701(CHEMBL3315148)
Affinity DataEC50:  0.0126nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048697(CHEMBL3315144)
Affinity DataEC50:  0.0195nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50320472((3S,6S,9S,15S)-3-((4R,7S,10S,13S,16S,19R)-13-((1H-...)
Affinity DataKi:  0.0200nMAssay Description:Displacement of [125I]U2 from rat urotensin 2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50320463(H-Asp-Cys-Phe-Trp-Lys-Tyr-Cys-Val-OH | D[CFWKYC]V ...)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50089666(CHEMBL3577310)
Affinity DataEC50: <0.100nMAssay Description:Modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aortic ring assessed as human urotensin-2 EC50 for induction of aortic ring contrac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50320456(TAD[CFWKYC]V | CHEMBL1165734)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50302273((4R,7S,10S,13S,16S,19R)-13-((1H-indol-3-yl)methyl)...)
Affinity DataKi:  0.120nMAssay Description:Displacement of [125I]U2 from rat urotensin 2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50302273((4R,7S,10S,13S,16S,19R)-13-((1H-indol-3-yl)methyl)...)
Affinity DataKi:  0.120nMAssay Description:Displacement of [125I]urotensin 2 from rat urotensin 2 receptor expressed in CHOK1 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50320457(AD[CFWKYC]V | CHEMBL1163460)
Affinity DataEC50:  0.160nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50320454(AGTAD[CFWKYC]V | CHEMBL1163463)
Affinity DataEC50:  0.170nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50320454(AGTAD[CFWKYC]V | CHEMBL1163463)
Affinity DataKi:  0.190nMAssay Description:Displacement of [125I]U2 from rat urotensin 2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048691(CHEMBL3315139)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413761(CHEMBL390094)
Affinity DataKi:  0.200nMAssay Description:Binding affinity towards human Urotensin 2 receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413761(CHEMBL390094)
Affinity DataKi:  0.200nMAssay Description:Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413761(CHEMBL390094)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413761(CHEMBL390094)
Affinity DataEC50:  0.251nMAssay Description:Agonist activity at UT2 receptor in Albino rat aorta assessed as induction of aortic contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413760(CHEMBL426020)
Affinity DataKi:  0.251nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413760(CHEMBL426020)
Affinity DataKi:  0.251nMAssay Description:Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413760(CHEMBL426020)
Affinity DataKi:  0.251nMAssay Description:Binding affinity towards human Urotensin 2 receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50320463(H-Asp-Cys-Phe-Trp-Lys-Tyr-Cys-Val-OH | D[CFWKYC]V ...)
Affinity DataKi:  0.251nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413764(CHEMBL504097)
Affinity DataKi:  0.282nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50320455(GTAD[CFWKYC]V | CHEMBL1163467)
Affinity DataEC50:  0.290nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50244020(4'-[1-({2-[Cyanomethyl-(3,4-dichloro-phenyl)-amino...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to human urotensin-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50320472((3S,6S,9S,15S)-3-((4R,7S,10S,13S,16S,19R)-13-((1H-...)
Affinity DataEC50:  0.340nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048696(CHEMBL3315142)
Affinity DataKi:  0.398nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048691(CHEMBL3315139)
Affinity DataEC50:  0.398nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50320462(AD[CFWKYC]A | CHEMBL1165767)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50377218(CHEMBL257171)
Affinity DataKi:  0.400nMAssay Description:Displacement of [125I]hU-2 from human recombinant Urotensin 2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50377220(CHEMBL255509)
Affinity DataKi:  0.400nMAssay Description:Displacement of [125I]hU-2 from human recombinant Urotensin 2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50558696(CHEMBL4777970)
Affinity DataEC50:  0.450nMAssay Description:Agonist activity at human U-IIR expressed in HEK293-A cells by Fluo4-AM dye based intracellular calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50302273((4R,7S,10S,13S,16S,19R)-13-((1H-indol-3-yl)methyl)...)
Affinity DataEC50:  0.540nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50302273((4R,7S,10S,13S,16S,19R)-13-((1H-indol-3-yl)methyl)...)
Affinity DataEC50:  0.540nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50320458(AA[CFWKYC]V | CHEMBL1165735)
Affinity DataEC50:  0.600nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50377217(CHEMBL256989)
Affinity DataKi:  0.600nMAssay Description:Displacement of [125I]hU-2 from human recombinant Urotensin 2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048705(CHEMBL3315152)
Affinity DataEC50:  0.631nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413764(CHEMBL504097)
Affinity DataEC50:  0.661nMAssay Description:Agonist activity at UT2 receptor in Albino rat aorta assessed as induction of aortic contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048692(CHEMBL3315140)
Affinity DataEC50:  0.724nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048695(CHEMBL3315141)
Affinity DataKi:  0.724nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50320464([CFWKYC]V | CHEMBL1163473)
Affinity DataEC50:  0.760nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048701(CHEMBL3315148)
Affinity DataKi:  0.776nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413762(CHEMBL509604)
Affinity DataKi:  0.794nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataKi:  0.794nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataKi:  0.794nMAssay Description:Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataKi:  0.794nMAssay Description:Binding affinity towards human Urotensin 2 receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413784(UROTENSIN-II)
Affinity DataKi:  0.794nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048699(CHEMBL3315146)
Affinity DataEC50:  0.813nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50558700(CHEMBL4748168)
Affinity DataEC50:  0.830nMAssay Description:Agonist activity at human U-IIR expressed in HEK293-A cells by Fluo4-AM dye based intracellular calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataEC50:  0.832nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataEC50:  0.832nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413766(CHEMBL510618)
Affinity DataKi:  0.891nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
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