Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Urotensin-2 receptor' and Ligand = 'BDBM50413766'
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50413766(CHEMBL510618)
Affinity DataKi:  0.891nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50413766(CHEMBL510618)
Affinity DataEC50:  1.38nMAssay Description:Agonist activity at UT2 receptor in Albino rat aorta assessed as induction of aortic contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed