Compound Name

SMILES String

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(NC(=O)NC3CC3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(NC(=O)NCc3nn[nH]n3)cc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(NC(=O)NC3CC3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(NC(=O)NC3(C)CC3)cc12 |r|

C[C@@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1cc(C(C)=O)c2cc(NC(=O)NC3CC3)ccc12)c1cccc(Cl)c1F |r|

CC(C)NC(=O)Nc1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)cc(C(C)=O)c2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(NC(=O)NCc3ccon3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(NC(=O)NCc3ncccn3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(NC(=O)N3CCCC3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(NC(=O)NC3CC3)cc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(NC(=O)NC3CC3)cc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(NC(=O)N3CCCC3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(NC(=O)N3CCC(F)(F)C3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(NC(=O)OC3CC3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(NC(=O)OCC3CC3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(NC(=O)N3CCCC(F)(F)C3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(NC(=O)N3CCCC(F)(F)C3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(NC(=O)N3CCCC(F)(F)C3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(NC(=O)Nc3ccon3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(n2)C(F)(F)F)c2ccc(NC(=O)N3CCCC(F)(F)C3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(NC(=O)NCC(F)(F)F)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(NC(=O)N3Cc4cncnc4C3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(NC(=O)Nc3cncnc3)cc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(NC(=O)N3CCCC(F)(F)C3)cc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(NC(=O)Nc3ccon3)cc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(NC(=O)N3CCCC(F)(F)C3)cc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(NC(=O)N3CCCC(F)(F)C3)cc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(NC(=O)N3CCCC(F)(F)C3)cc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ncccc2Cl)c2ccc(NC(=O)N3CCCC(F)(F)C3)cc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(NC(=O)N3CCC(F)(F)C3)cc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(NC(=O)N3CCC(F)(F)CC3)cc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(NC(=O)NCc3ncccn3)cc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(NC(=O)N3CCCC(F)(F)C3)cc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(NC(=O)N3CCCC(F)(F)C3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(NC(=O)C3CCC(F)(F)C3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(NC(=O)CC(F)(F)F)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(NC(=O)OC(C)(C)C)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C(=O)N1CCC(=CC1)B(O)O |r,c:42|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C(=O)N1CC2CCC1C2 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C(=O)N1CCCC(F)(F)C1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C(=O)NC1CC1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)C(=O)N1CCC(CN)C1 |r,w:38.42|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)C(=O)NS(C)(=O)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)C(=O)N[C@H]1CCN(C1)C(=O)OC(C)(C)C |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)C(=O)N[C@H]1CCNC1 |r|

CC(=O)N1CC[C@@H](C1)NC(=O)c1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)C(=O)NS(=O)(=O)C1CC1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)C(=O)NCC1CCNC1 |r,w:36.40|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)C(=O)NCC1CCN(C1)C(=O)OC(C)(C)C |r,w:36.40|

COC(=O)C1CCN(C1)C(=O)c1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r,w:4.3|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)C(=O)N1CCC(C1)C(O)=O |r,w:38.44|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)C(=O)NS(=O)(=O)c1ccccc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2cc(ccc12)C(=O)NS(=O)(=O)C1CC1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2ccn(CC(F)(F)F)n2)c2ccccc12

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2ccn(CC(F)(F)F)n2)c2cnccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2ccn(CC(F)(F)F)n2)c2cnccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2ccn(n2)C(F)(F)F)c2ccccc12

CC(C)n1ccc(NC(=O)[C@@H]2C[C@H]3C[C@H]3N2C(=O)Cn2nc(C(N)=O)c3ccccc23)n1

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)N(CC(=O)N1C[C@H](F)C[C@H]1C(=O)NCc1cccc(Cl)c1F)S(C)(=O)=O |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;$|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(NS(=O)(=O)C(F)(F)F)ccc12 |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(Nc3cncc(F)c3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)n2)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@H](CO)c2cccc(Cl)c2F)c2ccc(Nc3cncnc3)cc12 |r,$;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;;$|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@@H](CO)c2cccc(Cl)c2F)c2ccc(Nc3cncnc3)cc12 |r,$;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;;$|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(Nc3cccnn3)cc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(Nc3cncnc3)cc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)n2)c2ccc(Nc3cccnn3)cc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)n2)c2ccc(Nc3cncnc3)cc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(Nc3ncc(cn3)C#N)cc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(Nc3cnc(nc3)C(F)(F)F)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)N(COC(=O)C(C)(C)C)c1cncnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2nc3ccccc3s2)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2ccccn2)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cc(F)cc(Cl)c2)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2)c2ccc(Nc3cncnc3)cc12 |r|

CNC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1cc(C(C)=O)c2cc(Nc3cncnc3)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)c2)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Cl)c2)c2ccc(Nc3cncnc3)cc12 |r|

CCN1Cc2ccc(NC(=O)[C@@H]3C[C@@H](F)CN3C(=O)Cn3cc(C(C)=O)c4cc(Nc5cncnc5)ccc34)cc2C1=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc3CC(C)(C)Oc23)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc3cn[nH]c3c2)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc(F)c(c2)-c2nnc3CCCCCn23)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Cc2cccc3CN(Cc23)c2ccccn2)c2ccc(Nc3cncnc3)cc12 |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;$|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCCc3nc(sc23)-c2ccc(F)cc2)c2ccc(Nc3cncnc3)cc12 |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;$|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(ns2)-c2ccccc2Cl)c2ccc(Nc3cncnc3)cc12 |r,$;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;;;$|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccccc2-n2nccc2C)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccnc2)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccccc2-c2nc3ccccc3s2)c2ccc(Nc3cncnc3)cc12 |r,$;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;$|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Cl)n2)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nnc(s2)-c2ccccc2Cl)c2ccc(Nc3cncnc3)cc12 |r,$;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;;;$|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc3OC(F)(F)Oc3cc2F)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@H]2CCCC[C@@H]2O)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)c2-n2cncn2)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)C2C[C@H](F)C[C@H]2C(=O)Nc2ccc3[nH]c(C)c(C)c3c2)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(C(=O)CN2C[C@H](F)C[C@H]2C(=O)Nc2nnc(s2)-c2ccc(Cl)c(Cl)c2)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccccc2N2CCOC2=O)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(C)nc3nc(nn23)C(F)(F)F)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCCN(C2)c2cnn(C)c2)c2ccc(Nc3cncnc3)cc12 |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;$|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccnc2)c2ccc(Nc3cncnc3)cc12 |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;$|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ncc(Br)cn2)c2ccc(Nc3cncnc3)cc12 |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;$|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc(OCc3ccccc3)cn2)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc3ccccc3c2)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)C2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)c2C(F)(F)F)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(cs2)-c2c(C)nc3sccn23)c2ccc(Nc3cncnc3)cc12 |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;$|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(cs2)-c2ccc3CCCCc3c2)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCc3c2c(F)ccc3F)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)C2C[C@H](F)C[C@H]2C(=O)Nc2noc3cc(ccc23)C(F)(F)F)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc(CN)cc2)c2ccc(Nc3cncnc3)cc12 |r|

COc1cc(C)cc2C(CCOc12)NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1cc(C(C)=O)c2cc(Nc3cncnc3)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2c[nH]nc2-c2ccc(Cl)cc2Cl)c2ccc(Nc3cncnc3)cc12 |r,$;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;$|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc3ncsc3c2)c2ccc(Nc3cncnc3)cc12 |r,$;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;$|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(C)nn2-c2ccccc2F)c2ccc(Nc3cncnc3)cc12 |r,$;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;;;;$|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCCN(C2=O)c2ccccc2Cl)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2ccncc2)c2ccc(Nc3cncnc3)cc12 |r,$;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;$|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(ns2)-c2cccc(Cl)c2)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccccc2-c2nncn2C)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2noc(n2)-c2ccccc2Cl)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCCN(C2=O)c2cc(C)ccc2F)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCN(C2=O)c2ccn(C)n2)c2ccc(Nc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(O)n2)c2ccc(Nc3cncnc3)cc12 |r|

CCOP(=O)(OCC)c1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CCOP(O)(=O)c1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)P(O)(O)=O |r|

CC(C)OC(=O)OCOP(=O)(OCOC(=O)OC(C)C)c1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CCOP(=O)(OCC)c1ccc2c(cn(CC(=O)N3[C@@H]4CCC[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CCOP(=O)(OCOC(=O)OC(C)C)c1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3CCC[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)P(O)(O)=O |r|

CCOP(=O)(OCC)c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)cc(C(C)=O)c2c1 |r|

CCOP(O)(=O)c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)cc(C(C)=O)c2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)P(O)(O)=O |r|

CCOC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)P(=O)(OCC)OCC |r|

CCOP(=O)(OCC)c1ccc2c(nn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(O)=O |r|

CCOP(=O)(OCC)c1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(=O)OC |r|

COC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)P(O)(O)=O |r|

CCOP(=O)(OCC)c1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(N)=O |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)P(O)(O)=O |r|

CCOP(=O)(OCC)c1ccc2c(nn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(N)=O |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)P(O)(O)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)P(=O)(OCC(F)(F)F)OCC(F)(F)F |r|

CCCCOP(=O)(OCCCC)c1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CCCCOP(O)(=O)c1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CC(C)OC(=O)OCOP(O)(=O)c1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CCOP(=O)(c1ccccc1)c1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CCOP(=O)(CC)c1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)P(O)(=O)c1ccccc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)P(=O)(OCOC(=O)C(C)(C)C)OCOC(=O)C(C)(C)C |r|

CCP(O)(=O)c1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)P(O)(=O)OCOC(=O)C(C)(C)C |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)P(O)(=O)OCC(F)(F)F |r|

CCOP(=O)(OCC)c1cc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)cc(C(C)=O)c2cc1F |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(c(F)cc12)P(O)(O)=O |r|

OP(O)(=O)c1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(=O)C(F)(F)F |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)P(=O)(Oc1ccccc1)Oc1ccccc1 |r|

CC(=O)c1cn(CC(=O)Oc2ccc3n(CC(=O)N4C[C@H](F)C[C@H]4C(=O)NCc4cccc(Cl)c4F)cc(C(C)=O)c3c2)c2ccc(O)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OC(=O)NCc3cscn3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OC(=O)NCc3cscn3)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OC(=O)NCc3nn[nH]n3)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OC(=O)NCCc3nn[nH]n3)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OC(=O)NCCP(O)(O)=O)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OC(=O)NCc3ccc(cc3)B(O)O)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OC(=O)NC3CC3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OC(=O)NCc3cocn3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OC(=O)NCc3nnn[nH]3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)C(=O)CS(C)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OC(=O)N3CCOCC3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OC(=O)NCc3ncccn3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OC(=O)NCCc3nn[nH]n3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OC(=O)NCCc3c[nH]cn3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OC(=O)N3CCNCC3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCC3CC3)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OS(=O)(=O)C(F)(F)F)ccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCC3CC3)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2cc(OCC3CC3)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCCC3CC3)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCc3cc4CCc5ccc(CCc3cc4)cc5)ccc12 |r|

CCOP(=O)(COc1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O)OCC |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCP(O)(O)=O)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OS(=O)(=O)C(F)(F)F)cc12 |r|

CCOP(=O)(COc1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)cc(C(C)=O)c2c1)OCC |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OCP(O)(O)=O)cc12 |r|

CC(C)OC(=O)OCOP(=O)(COc1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O)OCOC(=O)OC(C)C |r|

CC(C)OC(=O)OCOP(O)(=O)COc1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CCOP(=O)(CC)COc1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCS(=O)(=O)NC(C)(C)C)ccc12 |r|

CCP(O)(=O)COc1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCS(N)(=O)=O)ccc12 |r|

CCOP(=O)(COc1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)N[C@H](C)c3cccc(Cl)c3F)c2c1)C(C)=O)OCC |r|

C[C@@H](NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1cc(C(C)=O)c2ccc(OCP(O)(O)=O)cc12)c1cccc(Cl)c1F |r|

CCCCCCCCCCCCCCCCOCCCOP(O)(=O)COc1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCP(=O)(OCOC(=O)C(C)(C)C)OCOC(=O)C(C)(C)C)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2CNS(=O)(=O)c2cccc(Cl)c2F)c2cc(OCP(O)(O)=O)ccc12 |r|

CCC(=O)OC(OP(=O)(COc1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O)OC(OC(=O)CC)C(C)C)C(C)C |r,w:5.57,45.54|

CC(C)OC(=O)[C@H](C)NP(=O)(COc1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O)N[C@@H](C)C(=O)OC(C)C |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc(OC(F)(F)F)c(F)c2)c2cc(OCP(O)(O)=O)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Oc3ccccc3)c2)c2cc(OCP(O)(O)=O)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2cc(OCP(O)(O)=O)ccc12 |r|

CC(C)(C)NS(=O)(=O)COc1ccc2c(nn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)c2c1)C(N)=O |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2cc(OCS(N)(=O)=O)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(Oc3ncccn3)ccc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(Oc3cncnc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2cc(Oc3ncccn3)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(Oc3ncc(Br)cn3)cc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(Oc3ncc(Br)cn3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(Oc3ncc(Br)cn3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(Oc3cnc(nc3)C#N)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(Oc3ncc(F)cn3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(Oc3ncccn3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(Oc3ncccn3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(Oc3ncc(C)cn3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(Oc3ncc(C)cn3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(Oc3ncc(cn3)C(F)(F)F)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(Oc3cnc(Cl)nc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H](C[C@@H]3CCCC[C@H]23)C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H](Cc3ccccc23)C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)n1cc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)n1cc(NC(=O)[C@@H]2C[C@H](F)CN2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)n1cc(NC(=O)[C@@H]2C[C@H](F)CN2C(=O)NCc2ccccc2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NS(=O)(=O)c2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NS(=O)(=O)c2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)n1cc(NC(=O)[C@H]2CC(F)(F)CN2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)n1cc(NC(=O)[C@H]2CCCN2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2c2ncc([nH]2)-c2cccc(Cl)c2)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2c2ncc([nH]2)-c2cccc(Cl)c2)c2ccccc12 |r|

CC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2c2ncc([nH]2)-c2cccc(Br)n2)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2c2ncc([nH]2)-c2cccc(Cl)n2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2c2nc3cc(Cl)ccc3[nH]2)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2c2nc3cc(Cl)ccc3[nH]2)c2ccccc12 |r|

CC(=O)n1cc(NC(=O)[C@H]2CCCN2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccccc12 |r|

CC(=O)n1cc(NC(=O)[C@H]2CC(F)(F)CN2C(=O)Cc2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2CC[C@@H](OCC3CC3)[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

COc1ccc2c(O[C@@H]3C[C@H](N(C3)C(=O)Nc3cn(C(C)=O)c4ccccc34)C(=O)NCc3cccc(Cl)c3F)cc(nc2c1)-c1ccccc1 |r|

CC(=O)n1cc(NC(=O)Nc2cn(C(C)=O)c3ccccc23)c2ccccc12

CC(=O)c1cn(CC(=O)N2C[C@H](F)[C@@H](OCC3CC3)[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(O)ccc12 |r|

Fc1c(Cl)cccc1CNC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1cc(C(=O)C2CC2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)[C@@H]2CCC[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

F[C@@H]1C[C@H](N(C1)C(=O)Cn1cc(C(=O)C2CC2)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

CC(=O)c1cn(CC(=O)N2CC(F)C(OCC3CC3)[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(O)ccc12 |r|

NC(=O)N1CC(NC(=O)[C@@H]2CCC[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r,w:6.5|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2Cn2cc(nn2)-c2ccc(F)cc2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2Cn2cc(nn2)-c2ccc(F)cc2)c2ccccc12 |r|

COc1ccc2c(O[C@@H]3C[C@H](N(C3)C(=O)Cn3cc(C(C)=O)c4ccccc34)C(=O)NCc3cccc(Cl)c3F)cc(nc2c1)-c1ccccc1 |r|

NC(=O)N1C[C@H](F)C[C@H]1Cn1cc(nn1)-c1ccc(F)c(Cl)c1 |r|

NC(=O)n1cc(NC(=O)C2=C(CCC2)C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |t:9|

CC(=NC#N)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r,w:2.2|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N2Cc3ccccc3C2)c2ccccc12 |r|

CN(Cc1cccc(Cl)c1F)C(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1cc(C(C)=O)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@H]3CCCC[C@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(O)ccc12 |r|

F[C@@H]1C[C@H](N(C1)C(=O)Cn1cc(C#N)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

F[C@@H]1C[C@H](N(C1)C(=O)Cn1c2CCCC(=O)c2c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

CC(C)(C)OC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1C[C@H](F)C[C@H]1C(=O)NCc1cccc(Cl)c1F |r|

N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1C[C@H](F)C[C@H]1C(=O)NCc1cccc(Cl)c1F |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2c2ncc([nH]2)-c2cccc(Br)n2)c2cc(O)ccc12 |r|

CC(=O)c1cn(CC(=O)N2CC3(C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)OCCO3)c2cc(O)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCc3ccccc23)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2Cc3ccccc3C2)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCc3c2cccc3Cl)c2ccccc12 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(SC(F)(F)F)c2)c2cnccc12 |r|

[O-][N+](=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)Nc1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(SC(F)(F)F)c2)c2cc(O)ccc12 |r|

F[C@@H]1C[C@H](N(C1)C(=O)CC1=Nc2ccccc2S(=O)(=O)N1)C(=O)NCc1cccc(Cl)c1F |r,t:10|

F[C@@H]1C[C@H](N(C1)C(=O)c1csc(n1)-c1cccnc1)C(=O)NCc1cccc(Cl)c1F |r|

CC(=O)Nc1ccc(cn1)C(=O)N1C[C@H](F)C[C@H]1C(=O)NCc1cccc(Cl)c1F |r|

F[C@@H]1C[C@H](N(C1)C(=O)Cn1nc(I)c2ccncc12)C(=O)NCc1cccc(Cl)c1F |r|

CCOP(=O)(OCC)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnccc12 |r|

F[C@@H]1C[C@H](N(C1)C(=O)Nc1cn(C(=O)C2CC2)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

CC(C(=O)N1C[C@H](F)C[C@H]1C(=O)NCc1cccc(Cl)c1F)n1cc(C(C)=O)c2ccccc12 |r,w:1.0|

CC(=O)c1cn(c2ccccc12)C(C)(C)C(=O)N1C[C@H](F)C[C@H]1C(=O)NCc1cccc(Cl)c1F |r|

OP(O)(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnccc12 |r|

CC(=O)c1ccc(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CCOP(=O)(OCC)c1cc(Cl)cc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2cc(C(C)=O)c3ccccc23)c1 |r|

CCOP(O)(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnccc12 |r|

CCOP(=O)(OCC)c1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2cc(C(C)=O)c3ccccc23)c1 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3CCC[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(O)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cc(cc(Cl)c2F)P(O)(O)=O)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@@]2(C[C@H]2C=C)C(=O)NS(=O)(=O)C2CC2)c2cc(O)ccc12 |r|

F[C@@H]1C[C@H](N(C1)C(=O)CN1C=NS(=O)(=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r,c:11|

CC(=O)c1cn(CC(=O)N2[C@@H]3CCCC[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(O)ccc12 |r|

CC(C)(C)OC(=O)N1CCc2c(C1)n(CC(=O)N1C[C@H](F)C[C@H]1C(=O)NCc1cccc(Cl)c1F)c1ccccc21 |r|

F[C@@H]1C[C@H](N(C1)C(=O)Cn1c2CNCCc2c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

CS(=O)(=O)N1CCc2c(C1)n(CC(=O)N1C[C@H](F)C[C@H]1C(=O)NCc1cccc(Cl)c1F)c1ccccc21 |r|

CCOC(=O)CC(=O)N1CCc2c(C1)n(CC(=O)N1C[C@H](F)C[C@H]1C(=O)NCc1cccc(Cl)c1F)c1ccccc21 |r|

CC(=O)n1cc(C(=O)C(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

OC(=O)CCC(=O)N1CCc2c(C1)n(CC(=O)N1C[C@H](F)C[C@H]1C(=O)NCc1cccc(Cl)c1F)c1ccccc21 |r|

F[C@@H]1C[C@H](N(C1)C(=O)Cn1nc(-c2cn[nH]c2)c2ccncc12)C(=O)NCc1cccc(Cl)c1F |r|

F[C@@H]1C[C@H](N(C1)C(=O)Cn1nc(C(F)=C)c2ccncc12)C(=O)NCc1cccc(Cl)c1F |r|

F[C@@H]1C[C@H](N(C1)C(=O)Cn1nc(-c2cnc[nH]2)c2ccncc12)C(=O)NCc1cccc(Cl)c1F |r|

NS(=O)(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)cc1Br |r|

NC(c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12)C(F)(F)F |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2c(cccc12)C#N |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2cc(F)c(F)cc2Cl)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)C1(CC1)N1C(=O)c2ccccc2C1=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2cc(F)c(F)cc2Cl)c2ccccc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2cc(F)c(F)cc2Cl)c2cnccc12 |r|

CC(=O)n1cc(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccsc12 |r|

CC(=O)Nc1cccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)cc(C(C)=O)c12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccc(F)c(F)c2Cl)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccc(F)c(F)c2Cl)c2ccccc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2cc(F)cc(F)c2Cl)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2cc(F)cc(F)c2Cl)c2ccccc12 |r|

COc1cccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)cc(C(C)=O)c12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2cccc(C#N)c12 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2sccc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccsc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(n2)-c2c(F)cc(F)cc2Cl)c2cnccc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2)-c2c(F)cc(F)cc2Cl)c2cnccc12 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccsc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2CCCCc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2C3=NC(=NC3C=Cc12)c1cccc(Cl)c1 |r,c:30,34,t:28|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccsc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccsc12 |r|

COc1ncc(cn1)-c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)nc1C(N)=O |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2c(cccc12)C#N |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2c(cccc12)-c1ccc(Cl)nc1 |r|

Cc1cc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)nc(C(N)=O)c2s1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2c(cccc12)-c1cn[nH]c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2c(cccc12)C1CC1 |r|

CC(=O)c1ccc(Cl)c(c1)-c1cccc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(N)=O)c3ccccc23)c1F |r|

Cc1cc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(N)=O)c2s1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)C1(CC1)NC(=O)c1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2cc(OC(F)(F)F)ccc2Cl)c2ccccc12 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2c2nc3cc(ccc3[nH]2)-c2ccccc2Cl)c2ccccc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccc3[nH]cnc3c2Cl)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)C1(CC1)NC(=O)OC(C)(C)C |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2c(cccc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnccc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnccc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cn[nH]c1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cncnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1ccc(cc1)N1CCOCC1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cncnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cncnc1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cncnc1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(cc12)-c1cncnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(cc12)-c1cncnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(nc1)N1CCCC1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(nc1)N1CCCC1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1ccc(F)nc1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1ccc(F)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cncnc1 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cncnc1 |r|

CC(=O)N1CCN(CC1)c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)cc(C(C)=O)c2c1 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cncnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnc(cc12)-c1cncnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2cnc(cc12)-c1cncnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1ccnnc1 |r|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)cc(C(C)=O)c2c1 |r|

CN1CCC(=CC1)c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(N)=O)c2c1 |r,c:4|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)n2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)n2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(nc1)N1CCCC1 |r|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)cc(C(C)=O)c2c1 |r|

CC(=O)N1CCC(=CC1)c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)cc(C(N)=O)c2c1 |r,c:6|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)cc(C(N)=O)c2c1 |r|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Cl)n3)nc(C(N)=O)c2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)N1CCN(CC1)c1ncccn1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)N1CCN(CC1)c1ncc(F)cn1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)N1CCN(CC1)S(C)(=O)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccccc2-c2nc3ccccc3s2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2nc3ccccc3s2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCc3c2c(F)ccc3F)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccnc2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2ccccn2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccnc2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2ccncc2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccccc2-c2nc3ccccc3s2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2noc3cc(ccc23)C(F)(F)F)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCc3c2c(F)ccc3F)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cc(F)cc(Cl)c2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccnc2)c2ccc(cc12)-c1ccnnc1 |r|

CCN1Cc2ccc(NC(=O)[C@@H]3C[C@@H](F)CN3C(=O)Cn3nc(C(N)=O)c4cc(ccc34)-c3ccnnc3)cc2C1=O |r|

CCN1Cc2ccc(NC(=O)[C@@H]3C[C@@H](F)CN3C(=O)Cn3cc(C(C)=O)c4cc(ccc34)-c3ccnnc3)cc2C1=O |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc3ncsc3c2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@@H]2CCCC2OCc2ccccc2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2nc3ccccc3s2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc3[nH]c(C)c(C)c3c2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(cs2)-c2ccc3CCCCc3c2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(cs2)-c2ccc3CCCCc3c2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc3ncsc3c2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(cs2)-c2c(C)nc3sccn23)c2ccc(cc12)-c1ccnnc1 |r|

Cc1nc2sccn2c1-c1csc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)CC2N=C(C(N)=O)c3cc(ccc23)-c2ccnnc2)n1 |r,t:29|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccnc2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2ccc(OCc3ccccc3)nc2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc(CNC(=O)OCC3c4ccccc4-c4ccccc34)cc2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cc(F)cc(Cl)c2)c2ccc(cc12)-c1ccnnc1 |r|

Cc1[nH]c2ccc(NC(=O)[C@@H]3C[C@@H](F)CN3C(=O)Cn3nc(C(N)=O)c4cc(ccc34)-c3ccnnc3)cc2c1C |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccccc2N2CCOC2=O)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccccc2N2CCOC2=O)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Cl)c2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Cl)c2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)c2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nnc(s2)-c2ccc(Cl)c(Cl)c2)c2ccc(cc12)-c1ccnnc1 |r|

NCc1ccc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(N)=O)c3cc(ccc23)-c2ccnnc2)cc1 |r|

Cc1ccnn1-c1ccccc1NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(N)=O)c2cc(ccc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccccc2-n2nccc2C)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OCc3ccccc3)n2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@H]2CCCC[C@@H]2OCc2ccccc2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc3CC(C)(C)Oc3c2)c2ccc(cc12)-c1ccnnc1 |r|

CC1(C)Cc2ccc(NC(=O)[C@@H]3C[C@@H](F)CN3C(=O)Cn3nc(C(N)=O)c4cc(ccc34)-c3ccnnc3)cc2O1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@H]2CCC[C@@H]2OCc2ccccc2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@H]2CCCC[C@@H]2OCc2ccccc2)c2ccc(cc12)-c1ccnnc1 |r|

CNC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(N)=O)c2cc(ccc12)-c1ccnnc1 |r|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)cc(C(C)=O)c2c1 |r|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(Br)n3)cc(C(C)=O)c2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(nc1)C#N |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(F)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc(CN)cc2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc3cn[nH]c3c2)c2ccc(cc12)-c1ccnnc1 |r|

CNC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1cc(C(C)=O)c2cc(ccc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Cl)n2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Cl)n2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc(F)c(c2)-c2nnc3CCCCCn23)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)c2C(F)(F)F)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2c[nH]nc2-c2ccc(Cl)cc2Cl)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)c2-n2cncn2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)c2-n2cncn2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(C)nc3nc(nn23)C(F)(F)F)c2ccc(cc12)-c1ccnnc1 |r|

CN1C=NCN1c1ccccc1NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(N)=O)c2cc(ccc12)-c1ccnnc1 |r,c:2|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(ns2)-c2ccccc2Cl)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1ccccc1Cl |r|

Cc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(N)=O)c2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

Cc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)nc(C(N)=O)c2c1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc3CN(Cc23)c2ccccn2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc3CN(Cc23)c2ccccn2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCCc3nc(sc23)-c2ccc(F)cc2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCCc3nc(sc23)-c2ccc(F)cc2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ncc(Br)cn2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ncc(Br)cn2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc3ccccc3c2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@H]2CCCC[C@@H]2O)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2noc3cc(ccc23)C(F)(F)F)c2ccc(cc12)-c1ccnnc1 |r|

Cc1cc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(N)=O)c3cc(ccc23)-c2ccnnc2)n2nc(nc2n1)C(F)(F)F |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(ns2)-c2ccccc2Cl)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nnc(s2)-c2ccccc2Cl)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nnc(s2)-c2ccccc2Cl)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nnc(s2)-c2ccc(Cl)c(Cl)c2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)Nc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)cc(C(C)=O)c2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cccc(Cl)c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1ccc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnnc(C)c1 |r|

COc1cc(C)cc2C(CCOc12)NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(N)=O)c2cc(ccc12)-c1ccnnc1 |r|

COc1cc(C)cc2C(CCOc12)NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1cc(C(C)=O)c2cc(ccc12)-c1ccnnc1 |r|

Cc1ccc(F)c(c1)N1CCCC(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(N)=O)c3cc(ccc23)-c2ccnnc2)C1=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCCN(C2=O)c2cc(C)ccc2F)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)c2C(F)(F)F)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc3OC(F)(F)Oc3cc2F)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc3OC(F)(F)Oc3cc2F)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc3ccccc3c2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)-c1cnc(C)nc1 |r|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)cc(C(C)=O)c2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)Nc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)cc(C(C)=O)c2c1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2ccccn2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCCN(C2)c2cnn(C)c2)c2ccc(cc12)-c1ccnnc1 |r|

Cn1cc(cn1)N1CCCC(C1)NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(N)=O)c2cc(ccc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc3cn[nH]c3c2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@@H]2CCC[C@H]2O)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(O)n2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@@H]2CCC[C@H]2O)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(ns2)-c2cccc(Cl)c2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(ns2)-c2cccc(Cl)c2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1ccc(C)nn1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2Cl)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2cc(F)c(F)cc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1ccc(C)nc1 |r|

CC1Oc2cccc(NC(=O)[C@@H]3C[C@@H](F)CN3C(=O)Cn3nc(C(N)=O)c4cc(ccc34)-c3ccnnc3)c2NC1=O |r|

CC1Oc2cccc(NC(=O)[C@@H]3C[C@@H](F)CN3C(=O)Cn3cc(C(C)=O)c4cc(ccc34)-c3ccnnc3)c2NC1=O |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(O)ccn2)c2ccc(cc12)-c1ccnnc1 |r|

Cn1ccc(n1)N1CCC(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(N)=O)c3cc(ccc23)-c2ccnnc2)C1=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2c[nH]nc2-c2ccc(Cl)cc2Cl)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2ccncc2)c2ccc(cc12)-c1ccnnc1 |r|

Cc1cc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(N)=O)c3cc(ccc23)-c2ccnnc2)n(n1)-c1ccccc1F |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCCN(C2=O)c2ccccc2Cl)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)C2C[C@H](F)C[C@H]2C(=O)Nc2cc(C)nn2-c2ccccc2F)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@@H](F)C[C@@H]2C(=O)NC2CCCN(C2=O)c2ccccc2Cl)c2ccc(cc12)-c1ccnnc1 |r|

CC(NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1cc(C(C)=O)c2cc(ccc12)-c1ccnnc1)c1oc2ccc(F)cc2c1C |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ncccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2noc(n2)-c2ccccc2Cl)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(O)nc1 |r|

COCCNc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)cc(C(C)=O)c2c1 |r|

CNc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)cc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2)c2ccccc12

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2)c2ccccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2)c2ccncc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H]2C[C@@H]2c2ccccc2)c2cnccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2)c2cnccc12 |r|

COc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)N[C@@H]3C[C@H]3c3ccccc3)c2cc1OC)C(N)=O |r|

COc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)N[C@H]3C[C@@H]3c3ccccc3)c2cc1OC)C(N)=O |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2)c2ncccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2)c2cnccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)N[C@@H]1C[C@H]1c1ccccc1)C(=O)Cn1nc(C(C)=O)c2ccccc12 |r|

COc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)N[C@@H]3C[C@H]3c3ccccc3)c2cc1OC)C(C)=O |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2)c2ccccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2)c2ncccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2)c2ccncc12 |r|

Cc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)N[C@@H]3C[C@H]3c3ccccc3)c2cn1)C(N)=O |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2)c2ccncc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2)c2ncccc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2)c2ccccc12 |r|

CCc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)N[C@@H]3C[C@H]3c3ccccc3)c2cn1)C(N)=O |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2)c2cc3OCCOc3cc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H]2C[C@@H]2c2ccccc2Cl)c2cnccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@]2(C)C[C@H]2c2ccccc2)c2cnccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@]2(C)C[C@@H]2c2ccccc2)c2cnccc12 |r|

C[C@@]1(C[C@@H]1c1ccccc1)NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1nc(C(N)=O)c2ccccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@@]2(F)c2ccccc2)c2cc(F)c(F)cc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@@]2(F)c2ccccc2)c2ccc(F)cc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@@]2(F)c2ccccc2)c2ccc(Cl)cc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(CO)C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2)c2ncccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(CO)C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2)c2cnccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(CO)C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2Cl)c2ccccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(CO)C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2Cl)c2cnccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC2CC2c2cccc(c2)C(F)F)c2cnccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC2CC2c2cccc(c2)C(F)(F)F)c2cnccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC2CC2c2ccc(C)c(C)c2)c2cnccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC2CC(C2)c2ccccc2)c2ncccc12 |r,wU:14.16,wD:12.11,10.10,(-5.83,-5.63,;-6.6,-4.29,;-8.14,-4.29,;-5.83,-2.96,;-6.31,-1.5,;-5.06,-.59,;-5.06,.95,;-3.73,1.72,;-2.4,.95,;-3.73,3.26,;-4.98,4.16,;-6.04,5.63,;-4.5,5.63,;-2.96,5.63,;-2.49,4.16,;-1,3.77,;-.6,2.28,;.09,4.85,;1.58,4.46,;2.35,3.12,;3.68,3.89,;2.91,5.23,;5.17,3.49,;5.57,2.01,;7.06,1.61,;8.14,2.7,;7.75,4.18,;6.26,4.58,;-3.82,-1.5,;-2.31,-1.18,;-1.28,-2.32,;-1.76,-3.79,;-3.26,-4.11,;-4.29,-2.96,)|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC2CC(C2)c2ccccc2F)c2ncccc12 |r,wU:14.16,wD:12.11,10.10,(-5.83,-5.85,;-6.6,-4.52,;-8.14,-4.52,;-5.83,-3.18,;-6.31,-1.72,;-5.06,-.81,;-5.06,.73,;-3.73,1.5,;-2.4,.73,;-3.73,3.04,;-4.98,3.94,;-6.04,5.41,;-4.5,5.41,;-2.96,5.41,;-2.49,3.94,;-1,3.54,;-.6,2.06,;.09,4.63,;1.58,4.23,;2.35,2.9,;3.68,3.67,;2.91,5,;5.17,3.27,;5.57,1.79,;7.06,1.39,;8.14,2.48,;7.75,3.96,;6.26,4.36,;5.86,5.85,;-3.82,-1.72,;-2.31,-1.4,;-1.28,-2.54,;-1.76,-4.01,;-3.26,-4.33,;-4.29,-3.18,)|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC2CCC(CC2)c2ccccc2)c2cnccc12 |r,wU:14.16,wD:12.11,10.10,(-6.27,-5.63,;-7.04,-4.29,;-8.58,-4.29,;-6.27,-2.96,;-6.75,-1.5,;-5.5,-.59,;-5.5,.95,;-4.17,1.72,;-2.83,.95,;-4.17,3.26,;-5.41,4.16,;-6.48,5.63,;-4.94,5.63,;-3.4,5.63,;-2.92,4.16,;-1.43,3.77,;-1.03,2.28,;-.34,4.85,;1.14,4.46,;1.54,2.97,;3.03,2.57,;4.12,3.66,;3.72,5.15,;2.23,5.54,;5.61,3.26,;6,1.77,;7.49,1.37,;8.58,2.46,;8.18,3.95,;6.69,4.35,;-4.25,-1.5,;-2.75,-1.18,;-1.72,-2.32,;-2.19,-3.79,;-3.7,-4.11,;-4.73,-2.96,)|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H]2C[C@]2(F)c2ccccc2)c2ccccc12

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@@]2(F)c2ccccc2)c2ccccc12

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2F)c2cnccc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@H]2C[C@@H]2c2ccccc2F)c2cnccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H]2C[C@]2(F)c2ccccc2)c2cnccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@@]2(F)c2ccccc2)c2cnccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@@]2(F)c2ccccc2)c2ncccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H]2C[C@]2(F)c2ccccc2)c2ncccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@@]2(F)c2ccccc2)c2cnccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H]2C[C@]2(F)c2ccccc2)c2cnccc12 |r|

Cc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)N[C@@H]3C[C@@]3(F)c3ccccc3)c2cn1)C(N)=O |r|

Cc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)N[C@H]3C[C@]3(F)c3ccccc3)c2cn1)C(N)=O |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC2CC2(F)c2ccccc2F)c2ccccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@H]2c2cccc(Cl)c2)c2ncccc12

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H]2C[C@@H]2c2cccc(Cl)c2)c2ncccc12

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@H]2c2cccc(Cl)c2F)c2ncccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H]2C[C@@H]2c2cccc(Cl)c2F)c2ncccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2Cl)c2ccccc12

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2)c2ccccc12 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@H]2C[C@@H]2c2ccccc2)c2ccccc12 |r|

CC(=O)c1nn(CC(=O)N2C[C@H]3C[C@H]3[C@H]2C(=O)N[C@H]2C[C@@H]2c2ccccc2)c2ccccc12 |r|

CC(=O)c1nn(CC(=O)N2C[C@H]3C[C@H]3[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2)c2ccccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2F)c2ncccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H]2C[C@@H]2c2ccccc2F)c2ncccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2Cl)c2cnccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2Cl)c2ncccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2Cl)c2cnccc12 |r|

CCc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)N[C@@H]3C[C@H]3c3ccccc3Cl)c2cn1)C(N)=O |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H]2C[C@@H]2c2ccccc2Cl)c2ccccc12 |r|

Cc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)N[C@@H]3C[C@H]3c3ccccc3F)c2cn1)C(N)=O |r|

Cc1cc2c(nn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)N[C@@H]3C[C@H]3c3ccccc3F)c2cn1)C(N)=O |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccc(Cl)cc2)c2cnccc12 |r|

Cc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)N[C@@H]3C[C@H]3c3ccccc3Cl)c2cn1)C(N)=O |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC2CC2c2ccc(F)cc2F)c2ccccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC2CCCC(C2)c2ccccc2)c2ccccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC2CCCC(C2)c2ccccc2)c2cnccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC2CC[C@@H](C2)c2ccccc2)c2cnccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC2CC[C@H](C2)c2ccccc2)c2cnccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2F)c2cc(ccc12)C(O)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)C#C |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)C#CC(O)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)C#C[Si](C)(C)C |r|

COC(=O)C#Cc1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)C#Cc1c[nH]c(=O)nc1N |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#CC(O)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1c[nH]c(=O)nc1N |r|

CCS(=O)(=O)NC(=O)C#Cc1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)cc(C(C)=O)c2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1ncccn1 |r|

CCS(=O)(=O)NC(=O)C#Cc1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

OC(=O)C#Cc1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(=O)C(F)(F)F |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1cccc(OC(F)(F)F)c1F |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1ncc(O)cn1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1ccccc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(C#C)c2F)c2cnccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1cncnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1ccncc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1cnsc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1ccccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1ncccn1 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1ccccn1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1c[nH]nc1C#N |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1ncccn1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1cnccn1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ncccc2Cl)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1cn[nH]c1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(-c3cccc(Cl)c3)c2F)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N2CCc3c(C2)[nH]c2ccccc32)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(n2)C(F)(F)F)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1ccc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1cccc(N)n1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1cccc(F)n1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)C#Cc1ncccn1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

CC1(C)CCCC(C1)NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(N)=O)c2cc(ccc12)C#Cc1ncccn1 |r,w:8.8|

[#6]\[#6](-[#6])=[#6](\F)-[#6]-[#7]-[#6](=O)-[#6@@H]-1-[#6]-[#6@@H](F)-[#6]-[#7]-1-[#6](=O)-[#6]-n1nc(-[#6](-[#7])=O)c2cc(ccc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(n2)-c2ccccc2Cl)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)C#Cc1ccccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccc(F)cc2Cl)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(n2)-c2cn[nH]c2)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3CC(F)(F)[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2CC[C@@H](O)[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(n2)C2CC2)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Cl)n2)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(n2)C#N)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)C#Cc1ccc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)C#Cc1ccc(cn1)C(F)(F)F |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)C#Cc1ccc(cn1)C#N |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)C#Cc1ncc(cn1)C(F)(F)F |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(F)n2)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2cc(F)c(F)cc2Cl)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2F)-c2ccc(F)cc2Cl)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)C#Cc1cc(F)ccn1 |r|

NC(=O)c1nn(CC(=O)N2CCS[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnc(cc12)C#Cc1ccccc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)c2)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(-c3cncnc3)c2F)c2ccc(cc12)C#Cc1ncccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(n2)C(F)(F)F)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc3cccc(Cl)c3n2)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2ccn(CC(F)(F)F)n2)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)C#Cc1cccnn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(cc(Cl)n2)C(F)(F)F)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)n2)c2ccc(cc12)C#Cc1cccnn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc(c(Cl)n2)C(F)(F)F)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Cl)n2)c2ccc(cc12)C#Cc1cccnn1 |r|

COc1nc(ncc1F)C#Cc1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)nc(C(N)=O)c2c1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)C#Cc1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)n2)c2ccc(cc12)C#Cc1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(Br)ccc2F)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)n2)c2ccc(cc12)C#Cc1cnccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)C#Cc1cnccn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(n2)-c2ccccc2Cl)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(n2)-c2c(F)cccc2Cl)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(n2)-c2cc(F)c(F)cc2Cl)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)n2)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)C#Cc1cnccn1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)C#Cc1ncc(F)cn1 |r|

Cc1cnc(nc1)C#Cc1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(N)=O)c2c1 |r|

COc1ncc(cn1)C#Cc1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(N)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(nc1)N1CCCC1 |r|

CC(=O)N1CCC(=CC1)c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)cc(C(C)=O)c2c1 |r,c:6|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)nc(C(N)=O)c2c1 |r|

CC(=O)c1cn(CC(=O)N2CC(F)CC2C(=O)Nc2ccccc2-c2cc3ccccc3s2)c2ccc(cc12)-c1ccnnc1

CC(=O)C1=NC(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2ccncc2)c2ccc(cc12)-c1ccnnc1 |r,t:3|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccccc2-c2nc3ccccc3s2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)C1CC(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2noc3cc(ccc23)C(F)(F)F)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccnc2)c2ccc(cc12)-c1ccnnc1 |r|

Cc1nc2sccn2c1-c1csc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(N)=O)c3cc(ccc23)-c2ccnnc2)n1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OCc3ccccc3)n2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)c2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc(F)c(c2)-c2nnc3CCCCCn23)c2ccc(cc12)-c1ccnnc1 |r|

Cn1cnnc1-c1ccccc1NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(N)=O)c2cc(ccc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)C2C[C@H](F)C[C@H]2C(=O)Nc2noc3cc(ccc23)C(F)(F)F)c2ccc(cc12)-c1ccnnc1 |r|

Cc1cc(NC(=O)[C@@H]2C[C@@H](F)CC2C(=O)Cn2nc(C(N)=O)c3cc(ccc23)-c2ccnnc2)n2nc(nc2n1)C(F)(F)F |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc3OC(F)(F)Oc3c2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc3OC(F)(F)Oc3c2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(C)nn2-c2ccccc2F)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccnc2Cl)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCN(C2=O)c2ccn(C)n2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(=O)[nH]n2C2CCCCC2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2n[nH]c(C)c2-c2ccccc2)c2ccc(cc12)-c1ccnnc1 |r|

Cc1[nH]nc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(N)=O)c3cc(ccc23)-c2ccnnc2)c1-c1ccccc1 |r|

CC1Cc2c(NC(=O)[C@@H]3C[C@@H](F)CN3C(=O)Cn3cc(C(C)=O)c4cc(ccc34)-c3ccnnc3)nn(C)c2NC1=O |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@H]2CCCC[C@@H]2O)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccnc(=O)n2C)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(O)n2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc(O)cn2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc(O)cn2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(O)ccn2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nccc(Cl)n2)c2ccc(cc12)-c1ccnnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ncc(I)cn2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nccc(Cl)n2)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccccc2-c2nncn2C)c2ccc(cc12)-c1ccnnc1 |r|

C[C@@H](NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(N)=O)c2cc(ccc12)-c1ccnnc1)c1oc2ccc(F)cc2c1C |r|

C[C@H](NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(N)=O)c2cc(ccc12)-c1ccnnc1)c1oc2ccc(F)cc2c1C |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccnc2Cl)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(nc1)C(F)(F)F |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2cc(ccc2Cl)C(C)=O)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(NCC(F)(F)F)nc1 |r|

CCOc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)cc(C(C)=O)c2c1 |r|

CC(C)Nc1ncc(cn1)-c1ccc2n(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccnc2O)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccnc2O)c2ccc(cc12)-c1ccnnc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2cc(ccc2Cl)C(N)=O)c2ccc(cc12)-c1cnc(C)nc1 |r|

COCCNc1ncc(cn1)-c1ccc2n(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(Br)n3)cc(C(C)=O)c2c1 |r|

COCCNc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)cc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnnc(C)c1 |r|

Cc1ncc(cn1)-c1ccc2n(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(N)=O)c2c1 |r|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](Cl)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)cc(C(C)=O)c2c1 |r|

COC(=O)c1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)cc(C(C)=O)c2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(nc1)C(O)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccncc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(C)c(Cl)c1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)cc1-c1ccsc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(nc1)C(N)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(nc1)S(C)(=O)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(nc1)C(=O)NC1CC1 |r|

COCCOCCNC(=O)c1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)cc(C(C)=O)c2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(nc1)C(N)=O |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccc3[nH]cnc3c2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(N)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(nc1)C1CC1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2ccnn2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(nc1)C(C)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(N)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2N=CCC2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |w:14.14,c:10|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2nccn2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)n2)c2ccc(cc12)-c1cnc2ccnn2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(cc12)-c1cnc2ccnn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2NCCC2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |w:14.14|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nccc(n2)-c2sccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(Cl)sc2C)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2CCC[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](O)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCN(CC2)C(=O)c2cc(Cl)c[nH]2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CCCCCC(=O)NC1CCC(CC1)NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1 |r,wU:17.17,wD:19.20,(9.55,1.2,;8.01,1.2,;7.24,2.54,;5.7,2.54,;4.93,3.87,;3.39,3.87,;2.62,2.54,;2.62,5.2,;1.08,5.2,;.31,6.54,;-1.23,6.54,;-2,5.2,;-1.23,3.87,;.31,3.87,;-3.54,5.2,;-4.31,3.87,;-3.54,2.54,;-5.85,3.87,;-6.75,5.12,;-8.22,4.64,;-9.55,5.41,;-8.22,3.1,;-6.75,2.62,;-6.35,1.14,;-4.87,.74,;-7.44,.05,;-7.05,-1.44,;-7.95,-2.69,;-7.05,-3.93,;-7.44,-5.42,;-6.35,-6.51,;-8.93,-5.82,;-5.58,-3.46,;-4.25,-4.23,;-2.91,-3.46,;-2.91,-1.92,;-4.25,-1.15,;-5.58,-1.92,;-1.58,-4.23,;-1.58,-5.77,;-.25,-6.54,;1.09,-5.77,;2.42,-6.54,;1.09,-4.23,;-.25,-3.46,)|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2ccnn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(cc12)-c1cnc2ccnn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)-c1cnc2ccnn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc2ccnn2c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2ccnn2c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(cc12)-c1cnc2ccnn2c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)-c1cnc2ccnn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2n(C)cnc2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1ccn2nccc2n1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)N1CCn2c(C1)nnc2C(F)(F)F |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2ncccn12 |r|

CSc1cccc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc(C)nc2)n1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(F)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1ccc2ncnn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@@H](O)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2CC(=O)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1[nH]nnc1-c1cncnc1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1[nH]nnc1-c1ncccn1 |r|

CC(=O)c1nn(CC(=O)N2C[C@@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

COCCN(C)CCN1CC(CC1=O)NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2CC(F)(F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(Cl)cs2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(nc1)C1CC1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(N)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCN(CC2)C(=O)c2cn[nH]c2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2c(C#N)c(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2c(cnn2c1)C#N |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(n2)C(F)(F)F)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(n2)C#N)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1C |r|

CCc1cn(CC(=O)N2NCCC2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |w:13.13|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2c(C)cnn2c1 |r|

COCCNc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2CC[C@@H](N)[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H](CCC2=O)C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2c(F)c(F)c(F)c(F)c2F)c2ccc(cc12)-c1cnc(C)nc1 |r,wU:14.15,wD:11.11,(-7.77,-5.45,;-6.28,-5.06,;-5.19,-6.14,;-5.88,-3.57,;-6.78,-2.32,;-5.88,-1.08,;-6.28,.41,;-5.19,1.5,;-3.7,1.1,;-5.19,3.04,;-6.65,3.52,;-6.65,5.06,;-7.99,5.83,;-5.19,5.53,;-4.28,4.29,;-2.8,4.68,;-2.4,6.17,;-1.31,4.29,;-.54,2.95,;-.94,1.46,;.15,.38,;1.64,.77,;2.04,2.26,;.95,3.35,;1.35,4.84,;3.53,2.66,;4.61,1.57,;4.22,.08,;6.1,1.97,;7.19,.88,;6.5,3.46,;7.99,3.86,;5.41,4.55,;5.81,6.03,;3.92,4.15,;2.83,5.24,;-4.42,-1.55,;-3.08,-.78,;-1.75,-1.55,;-1.75,-3.09,;-3.08,-3.86,;-4.42,-3.09,;-.41,-3.86,;-.41,-5.4,;.92,-6.17,;2.25,-5.4,;3.59,-6.17,;2.25,-3.86,;.92,-3.09,)|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)c2F)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(C)c1cc2ncc(cn2n1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r|

COc1cccc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc3cc(C)nn3c2)c1F |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

Cc1ncc(cn1)-c1cc2c(nn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)c2cn1)C(N)=O |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cc(C=C)cc(Cl)c2F)c2ccc(cc12)-c1cnc(NCCCCCCCCCC=C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)c2C#N)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)F)c2F)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)F)c2F)c2ccc(cc12)-c1cnc2ccnn2c1 |r|

Cc1cc2ncc(cn2n1)-c1cc2c(nn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(OC(F)(F)F)c3F)c2cn1)C(N)=O |r|

Cc1cc2ncc(cn2n1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(N)=O)c2c1 |r|

Cc1cc2ncc(cn2n1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(OC(F)(F)F)c3F)nc(C(N)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2CC=C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r,c:11|

CCOC(=O)c1cc2ncc(cn2n1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2cc(nn2c1)C(N)=O |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2cc(nn2c1)C(O)=O |r|

COCCOCCNC(=O)c1cc2ncc(cn2n1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1n[nH]c2ccsc12 |r|

CC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2CC=C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r,c:11|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(-c3cccc(c3)S(C)(=O)=O)c2F)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1nc2CCCCc2s1 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(n2)C(F)(F)F)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2cccnn12 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1ccc2nccn2n1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnn2ccnc2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2cc(F)ccc2S(C)(=O)=O)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

Cc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)cc(C(N)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2CCS[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2CCCCn12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1ccc2nc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2CSC[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(n2)C(F)(F)F)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

Cc1ncc(cn1)-c1cc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)nc(C(N)=O)c2s1 |r|

CC(=O)c1nn(CC(=O)N2CC[C@@H](O)[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

COCCOCCOCCOCCOCCOc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

COc1cc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)cc(C(C)=O)c2cc1-c1cnc(C)nc1 |r|

COc1cc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)cc(C(C)=O)c2cc1-c1cnc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2cc(O)c(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2nc(C)ccn12 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1cnc2ccnn2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1cnc2ccnn2c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1ccc2nc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(-c3sccc3Cl)c2F)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2cc(O)c(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2CSC(C)(C)[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)n2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(C)cc(Br)n2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(O[C@@H]2CO[C@@H]3[C@H](O)CO[C@H]23)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(O[C@@H]2CO[C@@H]3[C@H](O)CO[C@H]23)nc1 |r|

CO[C@@H]1CO[C@@H]2[C@@H](CO[C@H]12)Oc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(c3F)-c3ccccc3Cl)cc(C(C)=O)c2c1 |r|

Cc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(CC(N)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2cc(ccc2Cl)S(N)(=O)=O)c2ccc(cc12)-c1cnc(C)nc1 |r|

CNS(=O)(=O)c1ccc(Cl)c(c1)-c1cccc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc(C)nc2)c1F |r|

CN(C)S(=O)(=O)c1ccc(Cl)c(c1)-c1cccc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc(C)nc2)c1F |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(C)cc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)[C@@H](O)[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cnc(C)c(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

COc1cc(Br)nc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc(C)nc2)c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1cnc(N)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1cnc(N)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1cnc(nc1)C1CC1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(CC(F)(F)F)cs2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccn(CC(F)(F)F)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)c2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(Cl)cc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CN(C)C(=O)c1cc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2cc1-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2ccn(CC(F)(F)F)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(N)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cnc(C)c(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

COc1cc(Br)nc(NC(=O)[C@@H]2C[C@H]3C[C@H]3N2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc(C)nc2)c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(NC2CC2)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Cl)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2CC3CC3C2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(cc(Br)n2)C(F)(F)F)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@@H]3C[C@@H]3[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(C)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

COc1cc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2cc1-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(CO)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cncc(Cl)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccnc(OCC(F)(F)F)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ncn(CC(F)(F)F)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CNc1ncc(cn1)-c1ccc2n(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cncc(Br)n3)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1cnc(NC2CC2)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(Br)n(C)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@H]3C[C@@]3(C)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@H]3C[C@@]3(CO)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cncc(Br)n3)nc(C(C)=O)c2c1 |r|

COc1ccc(Br)nc1NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1 |r|

CN(C)Cc1cc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2cc1-c1cnc(C)nc1 |r|

CCc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cncc(Br)n3)nc(C(C)=O)c2c1 |r|

CC(C)c1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cncc(Br)n3)nc(C(C)=O)c2c1 |r|

CNc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(CC#N)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(CO)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)Nc1cccc(Br)n1)C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1 |r|

COc1ccc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc(C)nc2)nc1Br |r|

CC(=O)c1nn(CC(=O)N2C[C@@](F)(CN)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

COC(=O)c1cc(Cl)nc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc(C)nc2)c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc(C)c(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1cnc(CO)nc1 |r|

CC(=O)c1nn(CC(=O)N2CC(F)(CN)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@@](F)(CO)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccn(CC(F)F)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(CNC(=O)OC(C)(C)C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(CN)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(Br)ccc2C)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)NCc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc(F)cn2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ncc(F)cc2Br)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(O)c1nn(CC(=O)N2C3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn([C@H](F)C(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn([C@@H](F)C(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H]3C[C@H]3[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@@H]3C[C@@H]3[C@@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@@](F)(CF)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

COC[C@]12C[C@H]1N([C@@H](C2)C(=O)Nc1cccc(Br)n1)C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1 |r|

COC[C@@]12C[C@@H]1N([C@@H](C2)C(=O)Nc1cccc(Br)n1)C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2CC(C)(C)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

COC[C@@]1(F)C[C@H](N(C1)C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1)C(=O)Nc1cccc(Br)n1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nn(CC(F)(F)F)cc2Br)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2nc(Br)ccc2C)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nn(CC(F)(F)F)cc2C)c2ccc(cc12)-c1cnc(C)nc1 |r|

CNC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

C[C@H](O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

C[C@@H](O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)[C@@H](N)[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@@H](N)[C@H](F)[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(C)n(CC(F)(F)F)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nn(CC(F)(F)F)cc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

COc1cc(Br)nc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc(OC)nc2)c1 |r|

COc1cc(Br)nc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc(N)nc2)c1 |r|

COc1cc(Br)nc(NC(=O)[C@@H]2C[C@H]3C[C@H]3N2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc(OC)nc2)c1 |r|

COc1cc(Br)nc(NC(=O)[C@@H]2C[C@H]3C[C@H]3N2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc(N)nc2)c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(Br)ccc2C)c2ccc(cc12)-c1cnc(N)nc1 |r|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3nc(Br)ccc3C)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccn(CCC(F)(F)F)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(F)ncc2Br)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nn(C)c3ncccc23)c2ccc(cc12)-c1cnc(C)nc1 |r|

Cc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(=O)CO)c2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2ccccc2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCCc2ccccc2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCCCc2ccccc2)c2ccc(cc12)-c1cnc(C)nc1 |r|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3nc(Br)ccc3C)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2nc(Br)ccc2C)c2ccc(cc12)-c1cnc(N)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2ccc(F)c(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(Br)cs2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(Br)c(C)s2)c2ccc(cc12)-c1cnc(C)nc1 |r|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3ccc(F)c(Br)n3)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc(F)c(Br)n2)c2ccc(cc12)-c1cnc(N)nc1 |r|

CC(=O)O[C@@H]1[C@@H](F)CN([C@@H]1C(=O)Nc1cccc(Br)n1)C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(cs2)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C3CC3(CN)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

Cc1cccc(CC(O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2cc(C(N)=O)c3cc(ccc23)-c2cnc(C)nc2)n1 |r|

CC(F)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3ccc(F)c(Br)n3)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2ccc(F)c(Br)n2)c2ccc(cc12)-c1cnc(N)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCC2CC2(Cl)Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2C[C@H]2c2ccccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r,w:17.18|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCCCCc2ccccc2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2CC3CC2(C3)C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |(-3.1,-5.84,;-4.19,-4.75,;-5.68,-5.15,;-3.79,-3.27,;-4.7,-2.02,;-3.79,-.77,;-4.19,.71,;-3.1,1.8,;-1.61,1.4,;-3.5,3.29,;-4.96,3.77,;-4.96,5.31,;-3.5,5.78,;-2.59,4.54,;-3.87,4.22,;-1.05,4.54,;-.28,5.87,;-.28,3.2,;1.26,3.2,;2.03,1.87,;3.57,1.87,;4.34,3.2,;3.57,4.54,;4.34,5.87,;2.03,4.54,;-2.33,-1.25,;-.99,-.48,;.34,-1.25,;.34,-2.79,;-.99,-3.56,;-2.33,-2.79,;1.68,-3.56,;1.68,-5.1,;3.01,-5.87,;4.34,-5.1,;5.68,-5.87,;4.34,-3.56,;3.01,-2.79,)|

CCn1ccc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc(C)nc2)n1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCCC(C)(C)C2)c2ccc(cc12)-c1cnc(C)nc1 |r,w:17.18|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)cn1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(Br)ccc2C)c2ccc(cc12)-c1cnc(C)cn1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(Br)ccc2C)c2ccc(cc12)-c1ccnc(C)n1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2c2nc(c[nH]2)-c2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(Br)ccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

Cc1cccc(NC(=O)[C@@H]2C3CCC(C3)N2C(=O)Cn2cc(C(N)=O)c3cc(ccc23)-c2cnc(C)nc2)n1 |r,TLB:16:15:12.11:14,THB:7:9:12.11:14|

[#6]\[#6](-[#6])=[#6](\F)-[#6]-[#7]-[#6](=O)-[#6@@H]-1-[#6]-[#6@@H](F)-[#6]-[#7]-1-[#6](=O)-[#6]-n1nc(-[#6](-[#6])=O)c2cc(ccc12)-c1cnc(-[#6])nc1 |r|

CC(=O)c1nn(CC(=O)N2C3CCC(C3)[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r,TLB:16:15:11.12:14,THB:7:9:11.12:14|

CC(=O)c1nn(CC(=O)N2C[C@H](F)CC2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H]3C[C@H]3C2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccn(n2)-c2ccc(F)cn2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(C)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(N)nc1 |r|

CC(=O)c1cn(CC(=O)N2CC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

[#6]\[#6](-[#6])=[#6](\F)-[#6]-[#7]-[#6](=O)-[#6@@H]-1-[#6]-[#6@H]-2-[#6]-[#6@H]-2-[#7]-1-[#6](=O)-[#6]-n1nc(-[#6](-[#6])=O)c2cc(ccc12)-c1cnc(-[#6])nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2CNCc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

COc1cc(Br)nc(NC(=O)[C@@H]2C[C@@]3(C)C[C@H]3N2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc(C)nc2)c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(C)C[C@H]2C(=O)Nc2nc(Br)ccc2C)c2ccc(cc12)-c1cnc(C)nc1 |r|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3[C@@H]4C[C@]4(C)C[C@H]3C(=O)Nc3cncc(Br)n3)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H]3C[C@H]3[C@H]2C(=O)Nc2nc(Br)ccc2C)c2ccc(cc12)-c1cnc(C)nc1 |r|

Cc1cccc(NC(=O)[C@@H]2C3CCC(C3)N2C(=O)Cn2cc(C(N)=O)c3cc(ccc23)-c2ccc3ccccc3c2)n1 |r,TLB:16:15:12.11:14,THB:7:9:12.11:14|

Cc1ccc(cn1)-c1ccc2n(CC(=O)N3C4CCC(C4)[C@H]3C(=O)Nc3cccc(C)n3)cc(C(N)=O)c2c1 |r,TLB:13:15:17.18:20,THB:22:21:17.18:20|

Cc1ncc(cn1)-c1ccc2n(CC(=O)N3C4CCC(C4)[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(N)=O)c2c1 |r,TLB:13:15:17.18:20,THB:22:21:17.18:20|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC[C@H]2CC2(Cl)Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC[C@@H]2CC2(Cl)Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

COc1ccc(cn1)-c1ccc2n(CC(=O)N3C4CCC(C4)[C@H]3C(=O)Nc3cccc(C)n3)cc(C(N)=O)c2c1 |r,TLB:14:16:18.19:21,THB:23:22:18.19:21|

Cc1cccc(NC(=O)[C@@H]2C3CCC(C3)N2C(=O)Cn2cc(C(N)=O)c3cc(ccc23)-c2cccc(c2)C#N)n1 |r,TLB:16:15:12.11:14,THB:7:9:12.11:14|

Cc1cccc(NC(=O)[C@@H]2C3CCC(C3)N2C(=O)Cn2cc(C(N)=O)c3cc(ccc23)-c2ccc(N)nc2)n1 |r,TLB:16:15:12.11:14,THB:7:9:12.11:14|

Cc1cccc(NC(=O)[C@@H]2C3CCC(C3)N2C(=O)Cn2cc(C(N)=O)c3cc(ccc23)-c2ccc3cccnc3c2)n1 |r,TLB:16:15:12.11:14,THB:7:9:12.11:14|

Cc1cccc(NC(=O)[C@@H]2C3CCC(C3)N2C(=O)Cn2cc(C(N)=O)c3cc(ccc23)-c2cccnc2)n1 |r,TLB:16:15:12.11:14,THB:7:9:12.11:14|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC\C(F)=C(\C)c2cccc(Cl)c2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1ccc2ncncc2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(OCC(F)(F)F)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC\C(F)=C(\C)c2cccc(Cl)c2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)c2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)c2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc(F)c(Br)c2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2CCNS(=O)(=O)c2ccccc2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@@](F)(CF)C[C@H]2C(=O)Nc2nc(Br)ccc2C)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)N[C@@H]1[C@@H](F)CN([C@@H]1C(=O)Nc1cccc(Br)n1)C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1 |r|

CC(=O)N[C@@H]1CN([C@@H]([C@H]1F)C(=O)Nc1cccc(Br)n1)C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[Si](C)(C)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

Cc1cccc(NC(=O)[C@@H]2C3CCC(C3)N2C(=O)Cn2cc(C(N)=O)c3cc(ccc23)-c2ccc3CCCCc3c2)n1 |r,TLB:16:15:12.11:14,THB:7:9:12.11:14|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC\C(F)=C(/C)c2cccc(Cl)c2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@@H](F)C[C@@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2CCc2cccc(C)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(Br)c(F)cc2C)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(nc1)S(C)(=O)=O |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(nc1)-n1cccn1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC\C(F)=C(\C)c2ccccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc(F)c(Br)c2F)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2CCC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1cccnc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@H]2C[C@@H]2c2ccccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@@H]2C[C@H]2c2ccccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC\C(F)=C(/C)c2ccccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

COC(=O)Cc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r|

C[C@H]1CC[C@H](N1C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1)C(=O)Nc1cccc(Br)n1 |r|

CSc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(CC(N)=O)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(CC(O)=O)nc1 |r|

CCc1ccc(Br)nc1NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1 |r|

Cc1cccc(NC(=O)[C@@H]2C3CCC(C3)N2C(=O)Cn2cc(C(N)=O)c3cc(ccc23)-c2cnc3CCCc3c2)n1 |r,TLB:16:15:12.11:14,THB:7:9:12.11:14|

Cc1cccc(NC(=O)[C@@H]2C3CCC(C3)N2C(=O)Cn2cc(C(N)=O)c3cc(ccc23)-c2ccc3CCc3c2)n1 |r,TLB:16:15:12.11:14,THB:7:9:12.11:14|

CCOC(=O)Cc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(Br)ccc2C2CC2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CCOC(=O)Cc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3ccc(F)c(Br)n3)nc(C(C)=O)c2c1 |r|

CCOC(=O)Cc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3nc(Br)ccc3C)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC\C(F)=C(\C)c2ccccc2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2CC[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

COc1ccc(cn1)-c1ccc2n(CC(=O)N3CCC[C@H]3C(=O)Nc3cccc(C)n3)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2CCC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1cccc(c1)C#N |r|

CC(=O)c1nn(CC(=O)N2CCC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1ccc(F)nc1 |r|

COc1ccc(cn1)-c1ccc2n(CC(=O)N3CC[C@H]3C(=O)Nc3cccc(C)n3)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2CC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1cccc(c1)C#N |r|

CC(=O)c1nn(CC(=O)N2CC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1cccnc1 |r|

CC(=O)c1nn(CC(=O)N2CC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1ccc(F)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCC2CCN(CC(F)(F)F)C2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCC(F)=C(C)C2CC2)c2ccc(cc12)-c1cnc(C)nc1 |r,w:21.23,21.24|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(Oc2ccncc2)nc1 |r|

CN(C)C(=O)OCc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(NS(C)(=O)=O)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC\C(F)=C(/C)c2ccccc2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccn(CC(F)(F)F)n2)c2ccc(cc12)-c1cnc(N)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)n2)c2ccc(cc12)-c1cnc(N)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(n2)C(F)(F)F)c2ccc(cc12)-c1cnc(N)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(n2)C(F)(F)F)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(cc12)-c1cnc(N)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccnc(C)c2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CCc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r|

CC(C)c1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r|

CN1CC[C@@H](CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc(C)nc2)C1 |r|

CN1CC[C@H](CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc(C)nc2)C1 |r|

C[C@@H](NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1)[C@H]1CC1(Cl)Cl |r|

CC(=O)c1nn(CC(=O)N2CCC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1ccc2CCCc2c1 |r|

CC(=O)c1nn(CC(=O)N2CC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1ccc2CCCc2c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2nc(Br)ccc2CO)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC\C(F)=C/c2ccccc2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(n2)C2CC2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CN(C)C[C@]12C[C@H]1N([C@H](C2)C(=O)Nc1cccc(Br)n1)C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1 |r|

CN(C)C[C@@]12C[C@@H]1N([C@H](C2)C(=O)Nc1cccc(Br)n1)C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@@](F)(CF)C[C@@H]2C(=O)Nc2nc(Br)ccc2C)c2ccc(cc12)-c1cnc(N)nc1 |r|

COc1cccc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc(C)nc2)n1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(n2)C(F)(F)F)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(F)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(n2)C(C)=O)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2CCC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1ccc2ccccc2c1 |r|

CC(=O)c1nn(CC(=O)N2CCC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1ccc(C)cc1 |r|

CC(=O)c1nn(CC(=O)N2CC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1ccc2ccccc2c1 |r|

CC(=O)c1nn(CC(=O)N2CC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1ccc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2CCC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1ccc2cccnc2c1 |r|

CC(=O)c1nn(CC(=O)N2CC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1ccc2cccnc2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(OC2CS(=O)(=O)C2)nc1 |r|

CC(=O)c1nn(CC(=O)N2CCCC[C@@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2CCCC[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1cn(CCN2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(cc12)-c1cnc(C)nc1 |r|

COC(=O)c1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r|

CC(=O)Nc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(nc1)C(O)=O |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(nc1)C(N)=O |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(n2)-c2ncco2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(OCC(F)(F)F)ccc2C)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(ccc2C)C(C)(F)F)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2nc(Br)ccc2C2CC2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(O)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@@H]3C[C@@H]3[C@H]2C(=O)Nc2nc(Br)ccc2C)c2ccc(cc12)-c1cnc(C)nc1 |r|

COCc1ccc(Br)nc1NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1 |r|

COC(=O)c1ccc(Br)nc1NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2c(C)cc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2cc(C)c(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCN(CC(F)(F)F)C2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC2CCN(CC(F)(F)F)C2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCC23CC4CC(CC(C4)C2)C3)c2ccc(cc12)-c1cnc(C)nc1 |r,TLB:22:23:27:20.21.26,26:21:28:27.25.24,26:25:28:20.22.21,THB:22:21:27:28.23.24|

[#6]-[#6@@H](-[#7]-[#6](=O)-[#6@@H]-1-[#6]-[#6@@H](F)-[#6]-[#7]-1-[#6](=O)-[#6]-n1nc(-[#6](-[#6])=O)c2cc(ccc12)-c1cnc(-[#6])nc1)-[#6](\F)=[#6](\[#6])-[#6] |r|

[#6]-[#6@H](-[#7]-[#6](=O)-[#6@@H]-1-[#6]-[#6@@H](F)-[#6]-[#7]-1-[#6](=O)-[#6]-n1nc(-[#6](-[#6])=O)c2cc(ccc12)-c1cnc(-[#6])nc1)-[#6](\F)=[#6](\[#6])-[#6] |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2nc(Br)ccc2C(O)=O)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(C)C[C@H]2C(=O)Nc2nc(Br)ccc2C2CC2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C3CCC(C3)[C@H]2C(=O)Nc2nc(Br)ccc2C)c2ccc(cc12)-c1cnc(C)nc1 |r,TLB:16:15:11.12:14,THB:7:9:11.12:14|

CN(C)C(=O)c1cccc(CC[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc(C)nc2)n1 |r|

CNC(=O)c1cccc(CC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc(C)nc2)n1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(C)C[C@H]2C(=O)Nc2nc(Br)ccc2C)c2ccc(cc12)-c1cnc(N)nc1 |r|

[#6]\[#6](-[#6])=[#6](/F)-[#6]-[#7]-[#6](=O)-[#6@@H]-1-[#6][C@@]2([#6])[#6]-[#6@H]2-[#7]-1-[#6](=O)-[#6]-n1nc(-[#6](-[#6])=O)c2cc(ccc12)-c1cnc(-[#6])nc1 |r|

[#6]-[#6@H](-[#7]-[#6](=O)-[#6@@H]-1-[#6][C@@]2([#6])[#6]-[#6@H]2-[#7]-1-[#6](=O)-[#6]-n1nc(-[#6](-[#6])=O)c2cc(ccc12)-c1cnc(-[#6])nc1)-[#6](\F)=[#6](\[#6])-[#6] |r|

[#6]-[#6@@H](-[#7]-[#6](=O)-[#6@@H]-1-[#6][C@@]2([#6])[#6]-[#6@H]2-[#7]-1-[#6](=O)-[#6]-n1nc(-[#6](-[#6])=O)c2cc(ccc12)-c1cnc(-[#6])nc1)-[#6](\F)=[#6](\[#6])-[#6] |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(C)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(C)C[C@H]2C(=O)Nc2ccn(CC(F)(F)F)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(C)C[C@H]2C(=O)NCc2cccc(Cl)c2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(C)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(C)C[C@H]2C(=O)NCC2CC2(Cl)Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(C)C[C@H]2C(=O)NC[C@H]2CC2(Cl)Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(C)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(C)C[C@H]2C(=O)Nc2cccc(n2)C(F)(F)F)c2ccc(cc12)-c1cnc(C)nc1 |r|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3[C@@H]4C[C@]4(C)C[C@H]3C(=O)Nc3nc(Br)ccc3C)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2cnc(cc12)-c1cnc(C)nc1 |r|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H]4C[C@H]4[C@H]3C(=O)Nc3nc(Br)ccc3C)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H]3C[C@H]3[C@H]2C(=O)Nc2nc(Br)ccc2C)c2ccc(cc12)-c1cnc(N)nc1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(C)C[C@H]2C(=O)Nc2nc(Br)ccc2C)c2c(C)cc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H]3C[C@H]3[C@H]2C(=O)Nc2nc(Br)ccc2C2CC2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H]3C[C@H]3[C@H]2C(=O)Nc2ccn(CC(F)(F)F)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CN(C)C[C@@]1(F)C[C@H](N(C1)C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1)C(=O)Nc1cccc(Br)n1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(C)C[C@H]2C(=O)Nc2cncc(n2)C(F)(F)F)c2c(C)cc(cc12)-c1cnc(C)nc1 |r|

COc1ncc(cn1)-c1ccc2n(CC(=O)N3C[C@H]4C[C@H]4[C@H]3C(=O)Nc3nc(Br)ccc3C3CC3)nc(C(C)=O)c2c1 |r|

C[C@H]1C[C@H](N(C1)C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1)C(=O)Nc1nc(Br)ccc1C |r|

C[C@@H]1C[C@H](N(C1)C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1)C(=O)Nc1nc(Br)ccc1C |r|

CN(C)C[C@@]1(F)C[C@H](N(C1)C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1)C(=O)Nc1nc(Br)ccc1C |r|

C[C@H]1CC[C@H](N1C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1)C(=O)Nc1nc(Br)ccc1C |r|

CC(=O)c1nn(CC(=O)N2[C@H]3C[C@H]3C[C@H]2C(=O)Nc2nc(Br)ccc2C)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)CC2C(=O)Nc2nc(Br)ccc2C(O)=O)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(nc1)S(C)=O |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(Cl)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1ccc2nc(C)cn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1ccc2cc(nn2c1)C1CC1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)F)n2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1ccc2nc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1ccn2nc(C)nc2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cnc(C)c(Br)n2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cnc(C)c(Br)n2)c2ccc(cc12)-c1ccc2nc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1cnc2ccnn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cnc(C)c(Br)n2)c2ccc(cc12)-c1cnc2ccnn2c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cnc(C)c(Br)n2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cnc(C)c(Br)n2)c2ccc(cc12)-c1cnc2ccnn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(OC(F)(F)F)n2)c2ccc(cc12)-c1cnc2ccnn2c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccc(cc12)-c1cnc2cc(nn2c1)C1CC1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)n2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)n2)c2ccc(cc12)-c1cnc2ccnn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)n2)c2ccc(cc12)-c1cnc2cc(nn2c1)C1CC1 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2cc(nn2c1)C1CC1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2cc(nn2c1)C1CC1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cnc(C)c(Br)n2)c2ccc(cc12)-c1cnc2cc(nn2c1)C1CC1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(Cl)cc(Br)n2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccnn2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccn(CC(F)(F)F)n2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

COC(=O)Cc1cccc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc3cc(C)nn3c2)n1 |r|

CC(C)c1cccc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(C)=O)c3cc(ccc23)-c2cnc3cc(C)nn3c2)n1 |r|

CCc1cc2ncc(cn2n1)-c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2cc(nn2c1)C(C)(C)C |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2cc(F)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2cc(nn2c1)C(F)(F)F |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2ccccc2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCCc2ccccc2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCCCc2ccccc2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCCCCc2ccccc2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2CC3C[C@]2(C3)C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r,wU:13.16,(-4.39,-5.84,;-5.48,-4.75,;-6.96,-5.15,;-5.08,-3.27,;-5.98,-2.02,;-5.08,-.77,;-5.48,.71,;-4.39,1.8,;-2.9,1.4,;-4.79,3.29,;-6.25,3.77,;-6.25,5.31,;-4.79,5.78,;-3.88,4.54,;-5.16,4.22,;-2.34,4.54,;-1.57,5.87,;-1.57,3.2,;-.03,3.2,;.74,1.87,;2.28,1.87,;3.05,3.2,;2.28,4.54,;3.05,5.87,;.74,4.54,;-3.61,-1.25,;-2.28,-.48,;-.95,-1.25,;-.95,-2.79,;-2.28,-3.56,;-3.61,-2.79,;.39,-3.56,;.39,-5.1,;1.72,-5.87,;3.05,-5.1,;4.52,-5.58,;5.42,-4.33,;6.96,-4.33,;4.52,-3.08,;3.05,-3.56,;1.72,-2.79,)|

Cc1cc2ncc(cn2n1)-c1ccc2n(CC(=O)N3C4CCC(C4)C3C(=O)Nc3cccc(C)n3)cc(C(N)=O)c2c1 |TLB:16:18:20.21:23,THB:25:24:20.21:23|

CC(=O)c1cn(CC(=O)N2CC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnn2CCCc12 |r|

Cc1cccc(NC(=O)[C@@H]2C3CCC(C3)N2C(=O)Cn2cc(C(N)=O)c3cc(ccc23)-c2cnc3ncccn23)n1 |r,TLB:16:15:12.11:14,THB:7:9:12.11:14|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnn(c1)-c1ncccn1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2CCNS(=O)(=O)c2ccccc2)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

Cc1cccc(NC(=O)C2C3CCC(C3)N2C(=O)Cn2cc(C(N)=O)c3cc(ccc23)-c2cnc3CCCCn23)n1 |TLB:16:15:12.11:14,THB:7:9:12.11:14|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnn(c1)-c1ncc(F)cn1 |r|

CC(=O)c1nn(CC(=O)N2CCC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1cnc2CCCCn12 |r|

CC(=O)c1cn(CCN2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(=O)n(C)c1 |r|

Cc1cccc(NC(=O)[C@@H]2C3CCC(C3)N2C(=O)Cn2cc(C(N)=O)c3cc(ccc23)-c2c[nH]c3ccsc23)n1 |r,TLB:16:15:12.11:14,THB:7:9:12.11:14|

CC(=O)c1nn(CC(=O)N2CC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1cnc2CCCCn12 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnn(c1)C1CC1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cn[nH]c1 |r|

CC(=O)c1nn(CC(=O)N2CCC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1cnc2ncccn12 |r|

CC(=O)c1nn(CC(=O)N2CC[C@H]2C(=O)Nc2cccc(C)n2)c2ccc(cc12)-c1cnc2ncccn12 |r|

CC(=O)n1cc(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)n1cc(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

Cc1cc2ncc(cn2n1)-c1nc2n(CC(=O)N3CCC[C@H]3C(=O)Nc3cccc(C)n3)nc(C(N)=O)c2s1 |r|

Cc1cccc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2nc(C(N)=O)c3sc(nc23)-c2cnc(C)nc2)n1 |r|

CC(=O)c1ccc(Cl)c(c1)-c1cccc(NC(=O)[C@@H]2C[C@H]3C[C@H]3N2C(=O)Cn2nc(C(N)=O)c3sc(nc23)-c2cnc3cc(C)nn3c2)c1F |r|

CC(=O)c1ccc(Cl)c(c1)-c1cccc(NC(=O)[C@@H]2C[C@H]3C[C@H]3N2C(=O)Cn2nc(C(N)=O)c3sc(nc23)-c2cnc(C)nc2)c1F |r|

COc1ccc(cc1)N1C[C@@H]2CC[C@H]1C=C2c1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(Br)n3)nc(C(C)=O)c2c1 |r,c:16,THB:5:8:15.14:11.12|

CNc1ncc2cc(ccc2n1)-c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)nc1C(N)=O |r|

Cc1cc2ncc(cn2n1)-c1nc2n(CC(=O)C3CCC[C@H]3C(=O)Nc3cccc(C)n3)nc(C(N)=O)c2s1 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)cc1-c1cnn(c1)C1CC1 |r|

CC(=O)N1CCC(=CC1)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)nc1C(N)=O |r,c:6|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)cc1-c1cnn(c1)-c1ncc(F)cn1 |r|

C[C@@H]1CC[C@H](N1C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1)C(=O)Nc1nc(Br)ccc1C |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1ccc(cc1)S(C)(=N)=O |r|

CN(C)C[C@@]1(F)C[C@H](N(C1)C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(C)nc1)C(=O)Nc1nc(Br)ccc1C1CC1 |r|

CC(=O)c1nn(CC(=O)N2C3CCC(CC3)[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r,wU:16.18,TLB:17:16:15.14:12.11,THB:7:9:15.14:12.11,(-2.74,-7.21,;-3.83,-6.12,;-5.31,-6.52,;-3.43,-4.63,;-4.33,-3.39,;-3.43,-2.14,;-3.83,-.65,;-2.74,.43,;-1.25,.04,;-3.14,1.92,;-4.46,2.52,;-4.46,4.52,;-3.6,5.67,;-3.6,3.96,;-5.23,3.24,;-6.04,2.02,;-2.33,3.24,;-.79,3.24,;-.02,1.9,;-.02,4.57,;1.52,4.57,;2.29,3.24,;3.83,3.24,;4.6,4.57,;3.83,5.9,;4.6,7.24,;2.29,5.9,;-1.96,-2.62,;-.63,-1.85,;.71,-2.62,;.71,-4.16,;-.63,-4.93,;-1.96,-4.16,;2.04,-4.93,;2.04,-6.47,;3.37,-7.24,;4.71,-6.47,;6.04,-7.24,;4.71,-4.93,;3.37,-4.16,)|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1nc2ccccc2[nH]1 |r|

CN(C(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(C)=O)c2cc(ccc12)-c1cnc(CO)nc1)c1cccc(Br)n1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2C#N)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2(CC2)C#N)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(N)[n+]([O-])c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)[n+]([O-])c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)[n+]2[O-])c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)[n+]2[O-])c2ccc(cc12)-c1cnc(C)[n+]([O-])c1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)-c2cc(ccc2Cl)S(=O)(=O)NC2CC2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2CCOC[C@@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2CCOC[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C3CC3(CN3CCOCC3)C[C@H]2C(=O)Nc2nc(Br)ccc2C)c2ccc(cc12)-c1cnc(C)nc1 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2)S(=O)(=O)C(F)(F)F)c2ccc(cc12)-c1cnc2cc(C)nn2c1 |r|

CC(=O)c1nn(CC(=O)N2C3CC3(CN3CCCC3)C[C@H]2C(=O)Nc2nc(Br)ccc2C)c2ccc(cc12)-c1cnc(C)nc1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

NC(=O)c1cc(NC(=O)N2CCC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccn12 |r|

c1ccc2c(c1)c(cn2C(=O)N)NC(=O)N3CCC[C@H]3C(=O)Nc4cccc(c4)OC(F)(F)F

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2ccccc2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccnc2)c2ccccc12 |r|

COCCN(C)Cc1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@H](CO)c2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2ccncc2)c2ccccc12 |r|

CN1CCN(CC1)c1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(O)c2)c2ccccc12 |r|

CN1CCN(Cc2cc(Cl)c(F)c(CNC(=O)[C@@H]3C[C@@H](F)CN3C(=O)Nc3cn(C(N)=O)c4ccccc34)c2)CC1 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2ccc(Cl)s2)c2ccccc12 |r|

CCN(CC)Cc1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@H](CO)c2ccccc2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(F)c2F)c2ccccc12 |r|

CC[C@H](C)[C@H](NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)OC(C)(C)C |r|

COC1CCN(CC1)c1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

CN(C)CCN(C)Cc1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cc(CN3CCOCC3)cc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cc(cc(Cl)c2F)N2CCOCC2)c2ccccc12 |r|

COC1CCN(Cc2cc(Cl)c(F)c(CNC(=O)[C@@H]3C[C@@H](F)CN3C(=O)Nc3cn(C(N)=O)c4ccccc34)c2)CC1 |r|

COCCN(C)c1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

CN(C)CCNCc1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2ccccc2C(O)=O)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(c2)C(O)=O)c2ccccc12 |r|

CC[C@H](C)[C@H](NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12)C(O)=O |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)Nc1ccccc1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1ccccc1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1 |r|

Cc1cccc(CNC(=O)[C@@H]2C[C@H](N)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(c1)C(F)(F)F |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(F)c1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(c1)C#N |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Br)c1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(O)c1 |r|

COc1cccc(CNC(=O)[C@@H]2C[C@H](N)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(OC(F)(F)F)c1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Oc2ccccc2)c1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(c1)-c1ccccc1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(c1)-n1cccc1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(c1)-c1ccc(Cl)s1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1ccc(s1)-c1ccc(Cl)s1 |r|

Cc1ccc(CNC(=O)[C@@H]2C[C@H](N)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)cc1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1ccc(Cl)cc1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1ccc(cc1)C(F)(F)F |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1ccc(OC(F)(F)F)cc1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1ccc(O)cc1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1ccccc1O |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1ccccc1F |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1ccccc1Cl |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1ccccc1-c1ccccc1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(F)c1F |r|

COc1ccc(Cl)cc1CNC(=O)[C@@H]1C[C@H](N)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

COc1ccc(CNC(=O)[C@@H]2C[C@H](N)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)cc1Cl |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cc(Cl)ccc1F |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1ccc(F)c(Cl)c1 |r|

Cc1c(Cl)cccc1CNC(=O)[C@@H]1C[C@H](N)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

Cc1ccc(Cl)cc1CNC(=O)[C@@H]1C[C@H](N)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

Cc1ccc(CNC(=O)[C@@H]2C[C@H](N)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)cc1Cl |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cc(Cl)cc(Cl)c1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1ccc(Cl)c(Cl)c1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1c(F)ccc(Cl)c1F |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1ccc2ccccc2c1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc2ccccc12 |r|

Cc1cnc(CNC(=O)[C@@H]2C[C@H](N)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)s1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1ccc(Cl)s1 |r|

Cc1ccnc(CNC(=O)[C@@H]2C[C@H](N)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

C[C@H](NC(=O)[C@@H]1C[C@H](N)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12)c1cccc(Cl)c1 |r|

C[C@@H](NC(=O)[C@@H]1C[C@H](N)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12)c1cccc(Cl)c1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NC(CO)c1cc(Cl)cc(Cl)c1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NC(CCO)c1cccc(Cl)c1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NC1(CC1)c1ccccc1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NC(c1ccccc1)c1ccccc1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCC1CCCCC1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NC[C@H]1CCCC[C@@H]1O |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NC[C@@H]1CCCC[C@@H]1O |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NC1CCCCC1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NC1CCCN(C1)c1ccccn1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NC1CCc2ccc(Cl)cc12 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NC1CCOc2ccc(Cl)cc12 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCCc1ccccc1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCC(O)c1ccccc1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)N[C@@H]1C[C@H]1c1ccccc1 |r|

C[C@@H](CNC(=O)[C@@H]1C[C@H](N)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12)c1ccccc1 |r|

C[C@H](CNC(=O)[C@@H]1C[C@H](N)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12)c1ccccc1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCCc1cccc(Cl)c1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCCc1ccccc1Cl |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCCc1ccccc1F |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCCc1cccc(F)c1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCCc1cc(F)cc(Cl)c1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCCCOc1ccccc1 |r|

CC[C@H](C)[C@H](NC(=O)[C@@H]1C[C@H](N)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)OC |r|

CCC[C@H](NC(=O)[C@@H]1C[C@H](N)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)OC |r|

COC(=O)[C@@H](NC(=O)[C@@H]1C[C@H](N)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12)C(C)C |r|

COC(=O)[C@H](CC(C)C)NC(=O)[C@@H]1C[C@H](N)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

COC(=O)[C@H](COC(C)(C)C)NC(=O)[C@@H]1C[C@H](N)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

COC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1C[C@H](N)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

COC(=O)[C@@H](NC(=O)[C@@H]1C[C@H](N)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12)c1ccccc1 |r|

CC[C@H](C)[C@H](NC(=O)[C@@H]1C[C@H](N)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12)C(N)=O |r|

CCc1cccc(CNC(=O)[C@@H]2C[C@H](N)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

CC[C@H](C)[C@@H](CO)NC(=O)[C@@H]1C[C@H](N)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

CC(C)c1cccc(NC(=O)[C@@H]2C[C@H](N)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)Nc1cccc(c1)-c1ccccc1 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2CNS(=O)(=O)c2ccccc2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2CNS(=O)(=O)c2ccccc2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2CNS(=O)(=O)c2cccc(F)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2CNS(=O)(=O)c2cccc(Cl)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2CNS(=O)(=O)c2cccc(Br)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2CNS(=O)(=O)c2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2CNS(=O)(=O)c2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2CNS(=O)(=O)c2ccc(Cl)s2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CCC[C@H]2CNS(=O)(=O)c2cccc(Cl)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2CNC(=O)Cc2ccccc2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2CNC(=O)Oc2ccccc2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2CNC(=O)Oc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2CNCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CCC[C@H]2CNc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

NC(=O)c1cn(CC(=O)N2CCC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12

CC(=O)n1cc(CC(=O)N2CCC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12

CC(=O)n1cc(C(N)C(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(C(=O)N1C[C@H](F)C[C@H]1C(=O)Nc1cccc(OC(F)(F)F)c1)c1cc(C(N)=O)n2ccccc12 |r|

NC(=O)c1cc(NC(=O)N2CCC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)n2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)C#N)c2ccccc12 |r|

C[C@@H]1CCN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

CC(C)(C)OC(=O)Cc1ccc2c(NC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)cn(C(N)=O)c2c1 |r|

CO[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)Nc1cccc(OC(F)(F)F)c1 |r|

CC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H](CO)c2cccc(Cl)c2F)c2ccccc12 |r|

CNC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](O)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

COCCOc1ccc2n(cc(NC(=O)N3C[C@](C)(F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(N)=O |r|

COC(=O)COc1ccc2n(cc(NC(=O)N3C4CC4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(N)=O |r|

NC(=O)n1cc(NC(=O)N2[C@H]3CC3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CC3CC3[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CC3C[C@]2(C3)C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r,wU:13.16,(-4.44,-5.63,;-5.21,-4.29,;-6.75,-4.29,;-4.44,-2.96,;-4.91,-1.5,;-3.67,-.59,;-3.67,.95,;-2.33,1.72,;-1,.95,;-2.33,3.26,;-3.58,4.16,;-3.1,5.63,;-1.56,5.63,;-1.09,4.16,;-2.63,4.16,;.4,3.77,;.8,2.28,;1.49,4.85,;2.98,4.46,;3.37,2.97,;2.29,1.88,;2.68,.39,;4.17,-.01,;5.26,1.08,;6.75,.68,;4.86,2.57,;5.95,3.66,;-2.42,-1.5,;-.92,-1.18,;.11,-2.32,;-.36,-3.79,;-1.87,-4.11,;-2.9,-2.96,)|

C[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)Nc1cccc(OC(F)(F)F)c1 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Br)c2F)c2ccccc12 |r|

CC(=O)NC[C@H]1CC[C@H](N1C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)Nc1cccc(OC(F)(F)F)c1 |r|

NC(=O)n1cc(NC(=O)N2CCC[C@@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CC3CC3[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CCS[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccccc12 |r|

COC(=O)c1cc(Cl)cc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cc(cc(Cl)c2F)C(O)=O)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CC=C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r,c:11|

NC(=O)n1cc(NC(=O)N2CC3O[C@@H]3[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](C[C@H]2C(=O)NCc2cccc(Cl)c2F)C(F)(F)F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)Nc2cccc(Br)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CC[C@@H]3C[C@]23C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)c2)c2ccccc12 |r|

CC1(C)SC[C@H](N1C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)Nc1cccc(OC(F)(F)F)c1 |r|

NC(=O)n1cc(NC(=O)N2CCC[C@H]2C(=O)Nc2cccc(c2)-c2ccc(cc2)C#N)c2ccccc12 |r|

COC(=O)c1cc(Br)cc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

CN(C)CCNC(=O)c1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)NCc2ccc(Cl)s2)c2ccccc12 |r|

COC(=O)c1ccc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)cc1Br |r|

C[C@@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)Nc1cccc(OC(F)(F)F)c1 |r|

CCc1cccc(NC(=O)[C@@H]2CC3CC3N2C(=O)Nc2cn(C(N)=O)c3ccccc23)n1 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(Br)cc(c2)C(O)=O)c2ccccc12 |r|

CC(C)(C)c1csc(NC(=O)[C@@H]2CCCN2C(=O)Nc2cn(C(N)=O)c3ccccc23)n1 |r|

NC(=O)n1cc(NC(=O)N2CSC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

COCCOc1ccc2n(cc(NC(=O)N3C4CC4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(N)=O |r|

CCc1cccc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)n1 |r|

C[C@]1(O)C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

Cc1ncc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)cc1Br |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H]3C[C@H]3[C@H]2C(=O)NCc2cccc(Cl)c2)c2ccccc12 |r|

Cc1ncc(Br)cc1NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CCS[C@H]2C(=O)NCc2cccc(F)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CCC[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cncc(Br)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2ncccc2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2ccccc2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CCS[C@H]2C(=O)NCc2cccc(Cl)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)Nc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CC[C@@H](O)[C@H]2C(=O)NCc2cccc(Cl)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CCS[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H](CN=[N+]=[N-])CC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CC3(CC3)C[C@H]2C(=O)NCc2cccc(Cl)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@@](F)(CO)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

C[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)NCc2cccc(Cl)c2)c2ccccc12 |r|

COC[C@]12C[C@H]1N([C@@H](C2)C(=O)NCc1cccc(Cl)c1F)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)Nc2ccncc2F)c2ccccc12 |r|

CO[C@@H]1CCN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CCCC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)C#N)c2ccccc12 |r|

CN(C)[C@@H]1CN([C@@H]([C@H]1F)C(=O)NCc1cccc(Cl)c1F)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CC[C@@H](F)[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

c1ccc2c(c1)c(cn2C(=O)N)NC(=O)N3C[C@@H](C[C@H]3C(=O)Nc4cccc(c4)OC(F)(F)F)F

C[C@]1(CCCN1C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)Nc1cccc(OC(F)(F)F)c1 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Cl)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cncc(Br)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(F)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@@](O)(CO)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H]3OC3[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

COC(=O)c1cc(Br)cc(NC(=O)[C@@H]2SCCN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

Cn1nc(cc1NC(=O)[C@@H]1CCCN1C(=O)Nc1cn(C(N)=O)c2ccccc12)-c1ccccc1 |r|

COC(=O)[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

NC(=O)n1cc(NC(=O)N2N=CCC2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |c:10|

NC(=O)n1cc(NC(=O)N2C[C@](O)(CO)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H](CO)c2cccc(Cl)c2F)c2ccccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

C[C@@]1(F)C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

CC(=O)N[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@@H]3C[C@@H]3[C@H]2C(=O)N[C@H](CO)c2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CC[C@H](F)[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@](F)(CN3CCOCC3)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H]3C[C@H]3[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)N[C@@H]1CN([C@@H]([C@H]1F)C(=O)NCc1cccc(Cl)c1F)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H]3C[C@H]3[C@H]2C(=O)N[C@H](CO)c2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CC[C@@H](O)[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

COC[C@@]12C[C@@H]1N([C@@H](C2)C(=O)NCc1cccc(Cl)c1F)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cncc(F)c2)c2ccccc12 |r|

COc1ccc2c(NC(=O)N3C4CC4C[C@H]3C(=O)NCc3cccc(Cl)c3F)cn(C(N)=O)c2c1 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H](CO)c2cccc(Br)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3CC3C[C@H]2C(=O)Nc2cccc(c2F)C(F)(F)F)c2ccccc12 |r|

COC(=O)c1cccc(NC(=O)[C@@H]2CCCN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2CCCC[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)NC[C@@]1(F)C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(c2F)C(F)(F)F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H](CCO)c2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

COc1ccc(CNC(=O)[C@@H]2SCCN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c(F)c1F |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccnc2)c2ccccc12 |r|

C[C@H]1CCN([C@@H]1C(=O)Nc1cccc(OC(F)(F)F)c1)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)NCc2cncc(Cl)c2)c2ccccc12 |r|

C[C@@]1(F)C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)N[C@H](CCO)c1cccc(Cl)c1F |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2ccncc2F)c2ccccc12 |r|

COC[C@@H](NC(=O)[C@@H]1[C@@H]2C[C@@H]2CN1C(=O)Nc1cn(C(N)=O)c2ccccc12)c1cccc(Cl)c1F |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2ccnc(c2F)C(F)(F)F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CCC[C@H]2C(=O)Nc2cccc(c2)S(N)(=O)=O)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)Nc2cccc(OC(F)F)c2)c2ccccc12 |r|

COc1cc(F)c(F)c(CNC(=O)[C@@H]2SCCN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

COC[C@@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Nc1cn(C(N)=O)c2ccccc12)c1cccc(Cl)c1F |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cncc(Cl)c2)c2ccccc12 |r|

CCc1cccc(NC(=O)[C@@H]2CCCN2C(=O)Nc2cn(C(N)=O)c3ccccc23)n1 |r|

C[C@@]1(F)C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)N[C@H](CO)c1cccc(Cl)c1F |r|

CNC(=O)c1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2C[C@](F)(CF)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)NCc2ncccc2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@@](F)(CN3CCOCC3)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

COC(=O)c1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

COC[C@@H](NC(=O)[C@@H]1[C@H]2C[C@H]2CN1C(=O)Nc1cn(C(N)=O)c2ccccc12)c1cccc(Cl)c1F |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NC(C(O)=O)c2cccc(Cl)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cncc(Cl)c2)c2ccccc12 |r|

CN(C)C[C@@H](NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Nc1cn(C(N)=O)c2ccccc12)c1cccc(Cl)c1F |r|

NC(=O)n1cc(NC(=O)N2C[C@@H](O)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cc(cc(Cl)c2F)C(=O)N2CCOCC2)c2ccccc12 |r|

COc1cccc(NC(=O)[C@@H]2CC3CC3N2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

CCN(CC)c1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2CCS[C@H]2C(=O)N[C@H](CO)c2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)Nc2cccc(Cl)c2)c2ccccc12 |r|

COC1CN(C1)C(=O)c1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2C[C@@H](C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)C#N)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CC[C@H](O)[C@H]2C(=O)NCc2cccc(Cl)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2ccccc2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CC[C@@H](O)[C@H]2C(=O)NCc2ccc(Cl)s2)c2ccccc12 |r|

CC(=O)n1cc(NC(=O)N2C[C@@H](CO)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)NCc2cccc(c2F)C(F)(F)F)c2ccccc12 |r|

COc1ccc(F)c(F)c1CNC(=O)[C@@H]1SCCN1C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CCS[C@H]2C(=O)NCc2cnc(Cl)s2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CCS[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(F)ccc12 |r|

CNC(=O)n1cc(NC(=O)N2[C@@H]3C[C@]3(CO)S[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CC(=C)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CCS[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCC=C)ccc12 |r|

Cc1ccc2c(NC(=O)N3CCC[C@H]3C(=O)Nc3cccc(OC(F)(F)F)c3)cn(C(N)=O)c2c1 |r|

CNC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H](COC)c2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)n1cc(NC(=O)N2CCC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

COC(=O)c1cc(Br)cc(NC(=O)[C@@H]2C[C@H]3C[C@H]3N2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2[C@@H](CC[C@@H]2c2ccccc2)C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccccc12 |r|

CC(=O)n1cc(NC(=O)N2[C@@H]3C[C@]3(CO)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

COC(=O)COc1ccc2c(NC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(OC(F)(F)F)c3)cn(C(N)=O)c2c1 |r|

CN(C)C(=O)c1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccc(C(O)=O)c(Br)c2)c2ccccc12 |r|

Cn1nc(cc1NC(=O)[C@@H]1CCCN1C(=O)Nc1cn(C(N)=O)c2ccccc12)C(C)(C)C |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OCC=C)cc12 |r|

CN(C)C[C@@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Nc1cn(C(C)=O)c2ccccc12)c1cccc(Cl)c1F |r|

CNC(=O)n1cc(NC(=O)N2CCC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CC[C@@H](O)[C@H]2C(=O)NCc2cnc(Cl)s2)c2ccccc12 |r|

CNC(=O)n1cc(NC(=O)N2[C@@H]3C[C@]3(COC)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CC(C)c1cccc(NC(=O)[C@@H]2C[C@H]3C[C@H]3N2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2CCC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccc(Br)cc12 |r|

CNC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H](CO)c2cccc(Cl)c2F)c2ccccc12 |r|

CCc1ccc2c(NC(=O)N3CCC[C@H]3C(=O)Nc3cccc(OC(F)(F)F)c3)cn(C(N)=O)c2c1 |r|

CNC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H](CN(C)C)c2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CCC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccc(cc12)C(F)(F)F |r|

NC(=O)n1cc(NC(=O)N2CCC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccc(Cl)cc12 |r|

COc1ccc2n(cc(NC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(N)=O |r|

NC(=O)n1cc(NC(=O)N2CCS[C@H]2C(=O)NCc2ccc(Cl)s2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(F)ccc12 |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)NCc2cnc(Cl)s2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@@H](c2cccc(Cl)c2)C(F)(F)F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccc(F)cc12 |r|

COc1ccc2n(cc(NC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(OC(F)(F)F)c3F)c2c1)C(N)=O |r|

NC(=O)n1cc(NC(=O)N2CC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

COc1ccc2n(cc(NC(=O)N3C4CC4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(N)=O |r|

NC(=O)n1cc(NC(=O)N2CC(F)(F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CC1(C)CC[C@H](N1C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

COCCOc1ccc2n(cc(NC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(N)=O |r|

Cc1ccnc(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1F |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cncc(c2)C(F)(F)F)c2ccccc12 |r|

CCOC(=O)Cc1ccc2n(cc(NC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(N)=O |r|

NC(=O)n1cc(NC(=O)N2CCC3C[C@]23C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OC(F)F)cc12 |r|

COc1cc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)ccn1 |r|

NC(=O)n1cc(NC(=O)N2CCS[C@H]2C(=O)Nc2cncc(Cl)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OCC=C)cc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@@H](CO)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CCC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccc(OCc3ccccc3)cc12 |r|

CN(C)C[C@@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Nc1cn(C(N)=O)c2ccccc12)c1cccc(Cl)c1F |r|

CCOC(=O)Cc1ccc2c(NC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)cn(C(N)=O)c2c1 |r|

CO[C@@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)Nc1cccc(OC(F)(F)F)c1 |r|

CC(C)(C)c1cc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)ccn1 |r|

COC(=O)COc1ccc2n(cc(NC(=O)N3C[C@](C)(F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(N)=O |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@H](c2cccc(Cl)c2)C(F)(F)F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H](CO)c2cccc(Cl)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CCS[C@H]2C(=O)Nc2cncc(Br)c2)c2ccccc12 |r|

CN1CCN(CC1)C(=O)c1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ccncc2F)c2ccccc12 |r|

NC(=O)c1cccc(NC(=O)[C@@H]2CCCN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

CS(=O)(=O)c1cccc(NC(=O)[C@@H]2CCCN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NC2CCOc3ccc(Cl)cc23)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2ncccc2F)c2ccccc12 |r|

CN(C)C[C@@]1(F)C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

CN(C)CCN(C)c1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

CC(C)(C)c1cccc(NC(=O)[C@@H]2CC3CC3N2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2C[C@@H](O)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CC(F)(F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

CCOC(=O)c1cc(Br)c(F)c(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CCC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2cc(OCC=C)ccc12 |r|

C[C@@H]1CC[C@H](N1C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)Nc1cccc(OC(F)(F)F)c1 |r|

C[C@H]1CC[C@H](N1C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)Nc1cccc(OC(F)(F)F)c1 |r|

CC[C@@H]1CC[C@H](N1C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)Nc1cccc(OC(F)(F)F)c1 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(Cl)cc(c2)C(O)=O)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cc(Br)cc(c2)C(O)=O)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CCS[C@H]2C(=O)Nc2cc(Br)cc(c2)C(O)=O)c2ccccc12 |r|

COc1ccc2n(cc(NC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cc(Br)cc(c3)C(O)=O)c2c1)C(N)=O |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cc(cc(Br)c2F)C(O)=O)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cc(Br)cc(c2)-c2nnn[nH]2)c2ccccc12 |r|

CC(C)(C)n1nnnc1-c1cc(Br)cc(NC(=O)[C@@H]2C[C@H]3C[C@H]3N2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cc(cc(Cl)c2F)-c2nnn[nH]2)c2ccccc12 |r|

CC(C)(C)n1nnnc1-c1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC(=O)n1cc(NC(=O)N2CC[C@H](F)[C@H]2C(=O)NCc2cccc(Cl)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2CC[C@@H](F)[C@H]2C(=O)NCc2cccc(Cl)c2)c2ccccc12 |r|

C[C@@H]1CC[C@H](N1C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

CC[C@@H]1CC[C@H](N1C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

NC(=O)n1cc(NC(=O)N2C[C@H](CO)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

COC(=O)[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1c(F)ccc(Cl)c1F |r|

NC(=O)n1cc(NC(=O)N2C[C@H](C[C@H]2C(=O)NCc2c(F)ccc(Cl)c2F)C(O)=O)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@@H](CO)C[C@H]2C(=O)NCc2cccc(Br)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@](F)(CO)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@H]3C[C@@]3(CO)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@]3(CO)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](C[C@H]2C(=O)NCc2cccc(Cl)c2F)C(F)F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H](CO)CC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2N=CCC2C(=O)NCc2cccc(Cl)c2)c2ccccc12 |c:10|

NC(=O)n1cc(NC(=O)N2N=CC[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r,c:10|

NC(=O)n1cc(NC(=O)N2N=CC[C@@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r,c:10|

C[C@@H](NC(=O)[C@@H]1[C@H](O)CCN1C(=O)Nc1cn(C(N)=O)c2ccccc12)c1cccc(Cl)c1F |r|

C[C@H](NC(=O)[C@@H]1[C@H](O)CCN1C(=O)Nc1cn(C(N)=O)c2ccccc12)c1cccc(Cl)c1F |r|

OCC(=O)n1cc(NC(=O)N2CCC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12 |r|

CC(=O)n1cc(NC(=O)N2CCC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccc(cc12)C#N |r|

CC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OC(F)F)cc12 |r|

NC(=O)n1cc(NC(=O)N2CCC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccc(O)cc12 |r|

NC(=O)n1cc(NC(=O)N2CCC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2cc(O)ccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(O)ccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2ccccc2F)c2cc(O)ccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCC#N)ccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCC(O)=O)ccc12 |r|

C[C@@]1(F)C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccc(OCC(O)=O)cc12)C(=O)NCc1cccc(Cl)c1F |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OCC(O)=O)cc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(CC(O)=O)ccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(CC(O)=O)cc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCCO)ccc12 |r|

NC(=O)n1cc(NC(=O)N2CCS[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCCO)ccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2cc(OCCO)ccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@@H]3C[C@@H]3[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCCO)ccc12 |r|

C[C@@]1(F)C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccc(OCCO)cc12)C(=O)NCc1cccc(Cl)c1F |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(CCO)cc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(CCO)ccc12 |r|

CC(C)(O)COc1ccc2n(cc(NC(=O)N3C4CC4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(N)=O |r|

CN(C)CCOc1ccc2n(cc(NC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(N)=O |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCCN3CCCC3)ccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCCn3ccnc3)ccc12 |r|

CC(C)(C)OC(=O)COc1ccc2n(cc(NC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3ccccc3F)c2c1)C(N)=O |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)NCc2ccccc2F)c2cc(OCC(O)=O)ccc12 |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(O)cc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(O)cc12 |r|

COC(=O)COc1ccc2c(NC(=O)N3C4CC4C[C@H]3C(=O)NCc3cccc(Cl)c3F)cn(C(N)=O)c2c1 |r|

NC(=O)n1cc(NC(=O)N2C3CC3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OCCO)cc12 |r|

c1ccc2c(c1)c(cn2C(=O)N)NC(=O)N3C[C@H](C[C@H]3C(=O)Nc4cccc(c4)OC(F)(F)F)N

CO[C@H]1[C@H](N)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

N[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2cc(OCc3ccccc3)ccc12)C(=O)Nc1cccc(OC(F)(F)F)c1 |r|

NC(=O)n1cc(NC(=O)N2CCNC[C@H]2C(=O)NCc2cccc(Cl)c2)c2ccccc12 |r|

NCc1ccc(cc1)-c1cccc(NC(=O)[C@@H]2CCCN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NCc1ccc(c(F)c1)-c1cccc(NC(=O)[C@@H]2CCCN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

NC[C@H]1CC[C@H](N1C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)Nc1cccc(OC(F)(F)F)c1 |r|

NC[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)Nc1cccc(OC(F)(F)F)c1 |r|

NC[C@@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)Nc1cccc(OC(F)(F)F)c1 |r|

NC[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

CN(C)C[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

NC[C@@]1(O)C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

NC[C@]1(F)C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

NC[C@@]1(F)C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

NC(=O)n1cc(NC(=O)N2C[C@@](F)(CNC=O)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC[C@@]1(F)C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1c(F)ccc(Cl)c1F |r|

CC(=O)n1cc(NC(=O)N2C[C@@](F)(CN)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC[C@@]1(F)C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)N[C@H](CF)c1cccc(Br)c1 |r|

NC[C@@]1(F)C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)Nc1cccc(OC(F)(F)F)c1 |r|

N[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

N[C@H]1CN([C@@H]([C@@H]1O)C(=O)NCc1cccc(Cl)c1F)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

N[C@@H]1CCN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

CC(=O)n1cc(NC(=O)N2CC[C@@H](N)[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

N[C@@H]1CCN([C@@H]1C(=O)N[C@@H](c1cccc(Cl)c1F)C(F)(F)F)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

N[C@H]1CCN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

N[C@H]1CCN([C@@H]1C(=O)NCc1cccc(Cl)c1)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

CC(=O)N[C@@H]1CCN([C@@H]1C(=O)NCc1cccc(Cl)c1)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

COCCN[C@@H]1CCN([C@@H]1C(=O)NCc1cccc(Cl)c1)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

CNC[C@@]1(F)C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

CN[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

COCCN[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

CN(C)[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

COC1(C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F)OC |r|

N[C@@H]1CN([C@@H]([C@H]1O)C(=O)NCc1cccc(Cl)c1F)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

N[C@@H]1CN([C@@H]([C@H]1F)C(=O)NCc1cccc(Cl)c1F)C(=O)Nc1cn(C(N)=O)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2NCC[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2NCC[C@@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2NCCC2C(=O)NCc2cccc(Cl)c2)c2ccccc12

COC(=O)[C@H]1C[C@H](N(C1)C(=O)Nc1cn(C(N)=O)c2ccccc12)C(=O)Nc1cccc(OC(F)(F)F)c1F |r|

NC(=O)n1cc(NC(=O)N2C[C@@H](CO)C[C@H]2C(=O)NCc2c(F)ccc(Cl)c2F)c2ccccc12 |r|

NC(=O)c1cc(Br)cc(NC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

COCCNC(=O)c1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Nc2cn(C(N)=O)c3ccccc23)c1 |r|

CC(C)c1cc(NC(=O)[C@@H]2CCCN2C(=O)Nc2cn(C(N)=O)c3ccccc23)on1 |r|

NC(=O)n1cc(NC(=O)N2CCC[C@H]2C(=O)Nc2cc(no2)-c2ccccc2)c2ccccc12 |r|

NC(=O)n1cc(CC(=O)N2CCC[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ccccc12

NC(=O)n1cc(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccccc12 |r|

NC(=O)n1cc(CC(=O)N2C[C@@H]3C[C@@H]3[C@H]2C(=O)N[C@H](CO)c2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(CC(=O)N2CC[C@@H](O)[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CN(C)C[C@@]1(F)C[C@H](N(C1)C(=O)Cc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

NC(=O)n1cc(CC(=O)N2C3CC3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

C[C@@]1(F)C[C@H](N(C1)C(=O)Cc1cn(C(N)=O)c2ccccc12)C(=O)N[C@H](CCO)c1cccc(Cl)c1F |r|

NC(=O)n1cc(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H](CO)c2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(CC(=O)N2CCS[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(CC(=O)N2C[C@@](F)(CO)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

COc1ccc2n(cc(CC(=O)N3C4CC4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(N)=O |r|

NC(=O)n1cc(CC(=O)N2C3CC3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCCO)ccc12 |r|

COC[C@]12C[C@H]1N([C@@H](C2)C(=O)NCc1cccc(Cl)c1F)C(=O)Cc1cn(C(N)=O)c2ccccc12 |r|

NC(=O)n1cc(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2cc(OCCO)ccc12 |r|

NC(=O)n1cc(CC(=O)N2C3CC3C[C@H]2C(=O)NCc2ccc(Cl)s2)c2ccccc12 |r|

NC(=O)n1cc(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H](CCO)c2cccc(Cl)c2F)c2ccccc12 |r|

CN(C)C[C@@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cc1cn(C(N)=O)c2ccccc12)c1cccc(Cl)c1F |r|

C[C@@]1(F)C[C@H](N(C1)C(=O)Cc1cn(C(N)=O)c2ccc(OCCO)cc12)C(=O)NCc1cccc(Cl)c1F |r|

NC(=O)n1cc(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(F)ccc12 |r|

Cc1c(CC(=O)N2C3CC3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc2n1C(N)=O |r|

NC(=O)n1cc(CC(=O)N2CCS[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCCO)ccc12 |r|

NC(=O)n1cc(CC(=O)N2C[C@H]3C[C@H]3[C@H]2C(=O)N[C@H](CO)c2cccc(Cl)c2F)c2ccccc12 |r|

COC[C@@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cc1cn(C(N)=O)c2ccccc12)c1cccc(Cl)c1F |r|

NC(=O)n1cc(CC(=O)N2C[C@@H]3C[C@@H]3[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCCO)ccc12 |r|

N[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cc1cn(C(N)=O)c2ccccc12 |r|

NC(=O)n1cc(CC(=O)N2[C@@H]3C[C@]3(CO)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)n1cc(CC(=O)N2NCCC2C(=O)NCc2cccc(Cl)c2)c2ccccc12

NC[C@@]1(F)C[C@H](N(C1)C(=O)Cc1cn(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

NC[C@@]1(F)C[C@H](N(C1)C(=O)Cc1cn(C(N)=O)c2ccccc12)C(=O)NCc1c(F)ccc(Cl)c1F |r|

CN(C)CCOc1ccc2n(cc(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(N)=O |r|

NC(=O)n1cc(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(CC(O)=O)cc12 |r|

NC(=O)n1cc(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(CCO)cc12 |r|

NC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

COc1cccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c12)C(N)=O |r|

CC(=O)c1cn(CC(=O)N2CCCC[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(Br)c(F)cc12 |r|

COC(=O)c1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@H]3C[C@H]3N2C(=O)Cn2cc(C(N)=O)c3ccccc23)c1 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Br)c2F)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@](C)(F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ncccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2ccc(Cl)s2)c2ncccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1cc(C(C)=O)c2cc(OC)ccc12 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Cl)c2F)c2ccccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1cc(C(C)=O)c2ccc(OC)cc12 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(Cl)cc12 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2c(Cl)cccc12 |r|

COC[C@]12C[C@H]1N([C@@H](C2)C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1cc(C(C)=O)c2cccnc12 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(Cl)ccc12 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(F)c(F)cc12 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OC(F)(F)F)ccc12 |r|

COc1cnc2n(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)cc(C(C)=O)c2c1 |r|

Fc1c(Cl)cccc1CNC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1cc(C(=O)C(F)(F)F)c2ccccc12 |r|

C[C@@]1(F)C[C@H](N(C1)C(=O)Cn1cc(C(N)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

COc1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)cc(C(N)=O)c2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cc(cc(Cl)c2F)C#N)c2ccccc12 |r|

COc1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(N)=O |r|

COc1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

COc1ccc2n(CC(=O)N3CCCC[C@H]3C(=O)NCc3cccc(Cl)c3F)cc(C(C)=O)c2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@](C)(F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccncc12 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OCc3ccccc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H](CCO)c2cccc(Cl)c2F)c2ccccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1cc(C(C)=O)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H]3C[C@H]3[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OCc3ccccc3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OC(F)(F)F)ccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@](C)(F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3CC[C@@H](C3)[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2CCS[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ncccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cc(Br)cc(c2)-c2nnn[nH]2)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Br)c2F)c2ccccc12 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(c2F)C(F)(F)F)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@H](CO)c2cccc(Cl)c2F)c2ccccc12 |r|

CNC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1cc(C(C)=O)c2cccnc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cc(cc(Cl)c2F)-c2nnn[nH]2)c2ccccc12 |r|

CN(C)C[C@@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1cc(C(C)=O)c2ccccc12)c1cccc(Cl)c1F |r|

COC(=O)c1cc(Cl)c(F)c(CNC(=O)[C@@H]2C[C@@H](F)CN2C(=O)Cn2cc(C(C)=O)c3ccccc23)c1 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccncc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cc(cc(Cl)c2F)-c2nnn[nH]2)c2ccccc12 |r|

COC(=O)c1ccc2c(cn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cc(cc(Cl)c2F)C#N)c2ccccc12 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OC(F)F)ccc12 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCc3ccccc3)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@](C)(F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ncccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(Cl)ccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2nc(ccc12)C#N |r|

COC[C@@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1cc(C(C)=O)c2cccnc12)c1cccc(Cl)c1F |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCc3ccccc3)ccc12 |r|

COC[C@@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1cc(C(C)=O)c2ccncc12)c1cccc(Cl)c1F |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCc3ccccc3)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H]3C[C@H]3[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccncc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H]3C[C@H]3[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ncccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OC(F)(F)F)cc12 |r|

COC(=O)c1ccc2n(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)cc(C(C)=O)c2c1 |r|

COC(=O)c1cccc2c(cn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c12)C(C)=O |r|

COC(=O)c1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

C[C@@]1(F)C[C@H](N(C1)C(=O)Cn1cc(C(=O)CO)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

CC(=O)c1cn(CC(=O)N2C[C@@H]3C[C@@H]3[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnccc12 |r|

COC(=O)Cc1ccc2c(cn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

F[C@@H]1C[C@H](N(C1)C(=O)Cn1cc(C(=O)C(F)(F)F)c2ccccc12)C(=O)NCc1cccc(Br)c1F |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ncccc12 |r|

COC(=O)c1ccc2c(cn(CC(=O)N3C[C@](C)(F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

COC(=O)Cc1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnccc12 |r|

OCC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)N[C@H](CF)c2cccc(Br)c2)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cccnc12 |r|

C[C@@]1(F)C[C@H](N(C1)C(=O)Cn1cc(C(=O)C(F)(F)F)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

CN(C)[C@@H]1CN([C@@H]([C@H]1F)C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1cc(C(C)=O)c2ccccc12 |r|

OCC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H](CCO)c2cccc(Cl)c2F)c2ncccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2)c2ncccc12 |r|

FC(F)(F)Oc1cccc(NC(=O)[C@@H]2CCCN2C(=O)Cn2cc(C=O)c3cccnc23)c1 |r|

COc1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)cc(C=O)c2c1 |r|

F[C@@H]1C[C@H](N(C1)C(=O)Cn1cc(C(=O)C(F)(F)F)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ncccc12 |r|

OCC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

OCC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Br)c2F)c2ccccc12 |r|

COCC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)c1cn(CC(=O)N2C[C@@](F)(CO)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)c1cn(CC(=O)N2CCS[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

COC[C@@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1cc(C(C)=O)c2ccccc12)c1cccc(Cl)c1F |r|

CCO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1cc(C(C)=O)c2ccccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)N[C@H](C)c1cccc(Cl)c1F)C(=O)Cn1cc(C(C)=O)c2ccccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)N[C@@H](C)c1cccc(Cl)c1F)C(=O)Cn1cc(C(C)=O)c2ccccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NC1(CC1)c1cccc(Cl)c1)C(=O)Cn1cc(C(C)=O)c2ccccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NC1(CC1)c1ccc(Cl)cc1)C(=O)Cn1cc(C(C)=O)c2ccccc12 |r|

N[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1cc(C(N)=O)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)[C@@H](N)[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@@H](N)[C@H](F)[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(O)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(O)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(O)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@](C)(F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(O)cc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3CC3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(O)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@](C)(F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(O)ccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3CC3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(O)ccc12 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCc3nn[nH]n3)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCc3nn[nH]n3)ccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3CC3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCc3nn[nH]n3)ccc12 |r|

COc1ccc2n(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)cc(C(C)=O)c2c1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OCc3ccccn3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OCc3ncccn3)cc12 |r|

COCCOc1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(N)=O |r|

COC(=O)COc1ccc2c(cn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(N)=O |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCC(O)=O)ccc12 |r|

NC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCCO)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(CC(O)=O)ccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3CC3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(CC(O)=O)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)C(O)=O |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3CC3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)C(O)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@](C)(F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)C(O)=O |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1cc(C(C)=O)c2ccc(cc12)C(O)=O |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3CC3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2c(cccc12)C(O)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(OCc3ccc(cc3)C(O)=O)ccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3CC3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(cc12)C(O)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(CO)ccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cc(cc(Cl)c2F)C(O)=O)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3CC3C[C@H]2C(=O)NCc2cc(cc(Cl)c2F)C(O)=O)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@@](F)(CN)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CN[C@H]1C[C@H](N(C1)C(=O)Cn1cc(C(C)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

COCCN[C@H]1C[C@H](N(C1)C(=O)Cn1cc(C(C)=O)c2ccccc12)C(=O)NCc1cccc(Cl)c1F |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@]3(CO)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ncccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@]3(CO)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@@H]3C[C@@H]3[C@H]2C(=O)N[C@H](CO)c2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H](CO)c2cccc(Cl)c2F)c2ncccc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@](C)(F)C[C@H]2C(=O)N[C@H](CO)c2cccc(Cl)c2F)c2ncccc12 |r|

CN(C)C(=N)c1ccc2n(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)cc(C(C)=O)c2c1 |r|

CN(C)C(=N)c1ccc2c(cn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)-c1nnn[nH]1 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3CC3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)-c1nnn[nH]1 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)[C@@H](O)[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

CC(=O)c1nc(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)n2ccccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3CC3C[C@H]2CNC(=O)Oc2cccc(Cl)c2F)c2ccccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)N[C@H](C)c1cccc(Cl)c1F)C(=O)Cn1nc(C(C)=O)c2cccnc12 |r|

CC(=O)c1nn(CC(=O)N2C[C@@H]3C[C@@H]3[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnc(C)cc12 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnc(C)cc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)Nc1cccc(OC(F)(F)F)c1F)C(=O)Cn1nc(C(N)=O)c2ccccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)Nc1cccc(OC(F)(F)F)c1F)C(=O)Cn1nc(C(N)=O)c2ccncc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1nc(C(C)=O)c2cnccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NC1(CC1)c1cccc(Cl)c1F)C(=O)Cn1nc(C(C)=O)c2ccncc12 |r|

COC(=O)c1ccc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c1)C(C)=O |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NC2(COC2)c2cccc(Cl)c2F)c2ncccc12 |r|

CN(C)CCO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1cc(C(C)=O)c2ccccc12 |r|

CC(=O)c1nn(CC(=O)N2C[C@H](F)[C@@H](O)[C@H]2C(=O)NC2(CC2)c2cccc(Cl)c2F)c2cnccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)Nc1cccc(OC(F)(F)F)c1F)C(=O)Cn1nc(C(N)=O)c2cc(C)ncc12 |r|

CCc1cc2c(nn(CC(=O)N3C[C@H](F)[C@@H](OC)[C@H]3C(=O)Nc3cccc(OC(F)(F)F)c3F)c2cn1)C(N)=O |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)Nc1cccc(OC(F)(F)F)c1F)C(=O)Cn1nc(C(C)=O)c2cc(OCc3ncccn3)ccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cc(ccc12)C(O)=O |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1nc(C(C)=O)c2ccc(cc12)C(O)=O |r|

C[C@@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1cc(C(C)=O)c2ccncc12)c1cccc(Cl)c1F

CN(C)CC[C@@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1nc(C(C)=O)c2ccccc12)c1cccc(Cl)c1F |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)N[C@H](C)c1cccc(Cl)c1F)C(=O)Cn1nc(C(N)=O)c2cccnc12 |r|

CC(=O)c1nc(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H](CO)c2cccc(Cl)c2F)n2ccccc12 |r|

CCC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnc(C)cc12 |r|

COc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2cc1OC)C(C)=O |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnc(C)cc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ncncc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccncc12 |r|

Cc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2cn1)C(N)=O |r|

OCC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

Cc1cc2n(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)nc(C(N)=O)c2cn1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ncccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2nnccc12 |r|

NC(=O)c1nn(CC(=O)N2CCCC[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnccc12 |r|

NC(=O)c1nn(CC(=O)N2CCS[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1cc(C(C)=O)c2cc(C)ncc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NC1(CC1)c1cccc(Cl)c1F)C(=O)Cn1nc(C(N)=O)c2cccnc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NC1(CC1)c1cccc(Cl)c1F)C(=O)Cn1nc(C(N)=O)c2cnccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1nc(C(N)=O)c2cc(C)ncc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1nc(C(N)=O)c2ccncc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1nc(C(N)=O)c2cnccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)N[C@H](C)c1cccc(Cl)c1F)C(=O)Cn1nc(C(N)=O)c2ccncc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)N[C@H](C)c1cccc(Cl)c1F)C(=O)Cn1nc(C(N)=O)c2cnccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccc(OCc3ncccn3)cc12 |r|

CCO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1cc(C(C)=O)c2cc(C)ncc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)c2F)c2cnccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)c2F)c2ccccc12 |r|

Cc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(Br)c3F)c2cn1)C(N)=O |r|

CCc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(Br)c3F)c2cn1)C(N)=O |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(n2)C2CC2)c2ccccc12 |r|

CC(C)c1cccc(NC(=O)[C@@H]2C[C@H]3C[C@H]3N2C(=O)Cn2nc(C(N)=O)c3ccncc23)n1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(C3CC3)c2F)c2ccccc12 |r|

C[C@]12C[C@H]1N([C@@H](C2)C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1nc(C(N)=O)c2ccncc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2nc(N)ccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H](CO)c2cccc(Cl)c2F)c2ncccc12 |r|

COC[C@@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cc1nc(C(C)=O)c2ccccn12)c1cccc(Cl)c1F |r|

CC(=O)c1nc(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)N[C@H](CC#N)c2cccc(Cl)c2F)n2ccccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1nc(C(C)=O)c2ccccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1cc(C(C)=O)c2ccncc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCc1cccc(Cl)c1F)C(=O)Cn1nc(C(C)=O)c2ccncc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2)S(F)(F)(F)(F)F)c2ccc(OCc3ncccn3)cc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2F)c2cnccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2F)-c2ccccc2Cl)c2cnccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2F)-c2ncccc2F)c2ccccc12 |r|

Cc1cccnc1-c1cccc(NC(=O)[C@@H]2C[C@H]3C[C@H]3N2C(=O)Cn2nc(C(N)=O)c3ccncc23)c1F |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2F)-c2ncccc2Cl)c2cnccc12 |r|

COC(=O)c1ccc2c(cn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2n1)C(C)=O |r|

C[C@@H](NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(N)=O)c2ccncc12)c1cccc(Cl)c1F |r|

C[C@@H](NC(=O)[C@@H]1C[C@@H](F)CN1C(=O)Cn1nc(C(N)=O)c2cc(C)ncc12)c1cccc(Cl)c1F |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12 |r|

C[C@@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1nc(C(N)=O)c2ccnc(C)c12)c1cccc(Cl)c1F |r|

Cc1nccc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c12)C(N)=O |r|

Cc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)NCc3cccc(Cl)c3F)c2c(C)n1)C(N)=O |r|

C[C@@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1nc(C(N)=O)c2cc(C)nc(C)c12)c1cccc(Cl)c1F |r|

CCc1cc2c(nn(CC(=O)N3C[C@H](F)[C@@H](OC)[C@H]3C(=O)NCc3cccc(Cl)c3F)c2cn1)C(N)=O |r|

C[C@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1nc(C(N)=O)c2ccncc12)c1cccc(Cl)c1F |r|

C[C@@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1nc(C(N)=O)c2cc(ncc12)C(F)(F)F)c1cccc(Cl)c1F |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2cnc(cc12)C1CC1 |r|

C[C@@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1nc(C(N)=O)c2cc(ncc12)C1CC1)c1cccc(Cl)c1F |r|

C[C@H](c1cccc(c1F)Cl)NC(=O)[C@@H]2C[C@H]3C[C@H]3N2C(=O)Cn4c5cnccc5c(n4)C(=O)N

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2nc(ccc12)C(O)=O |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCc2cccc(Cl)c2F)c2c[n+]([O-])ccc12 |r|

C[C@@H](NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1nc(C(N)=O)c2cc[n+]([O-])cc12)c1cccc(Cl)c1F |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccccc12

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccncc12 |r|

COC(=O)c1ccc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(OC(F)(F)F)c3F)c2c1)C(C)=O |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ncccc12 |r|

CCc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(OC(F)(F)F)c3F)c2cn1)C(N)=O |r|

Cc1cc2n(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(OC(F)(F)F)c3F)nc(C(N)=O)c2cn1 |r|

COc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(OC(F)(F)F)c3F)c2cn1)C(N)=O |r|

CCc1cc2c(nn(CC(=O)N3C[C@H](F)C[C@H]3C(=O)Nc3cccc(OC(F)(F)F)c3F)c2cn1)C(N)=O |r|

Cc1nccc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(OC(F)(F)F)c3F)c12)C(N)=O |r|

Cc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(OC(F)(F)F)c3F)c2c(C)n1)C(N)=O |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(OCc3ncccn3)cc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2cnc(cc12)C1CC1 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2nnccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(n2)-c2c(F)cccc2F)c2cnccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2)-c2c(F)cccc2Cl)c2cnccc12 |r|

Cc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(OC(F)(F)F)c3F)c2cn1)C(N)=O |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2cnccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2cc(ccc12)C(O)=O |r|

Cc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(OC(F)(F)F)c3F)c2c[n+]1[O-])C(N)=O |r|

c1ccc2c(c1)c(nn2CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc5cccc(n5)Br)C(=O)N

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2cnccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)F)c2F)c2ccccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)F)c2F)c2cnccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Cl)c2F)c2ccccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(n2)C(F)(F)F)c2cnccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(n2)C(F)(F)F)c2cnccc12 |r|

Cc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(Br)n3)c2cn1)C(N)=O |r|

CCc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(Br)n3)c2cn1)C(N)=O |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2cnccc12 |r|

C[C@]12C[C@H]1N([C@@H](C2)C(=O)Nc1cccc(OC(F)(F)F)c1F)C(=O)Cn1nc(C(N)=O)c2ccccc12 |r|

C[C@]12C[C@H]1N([C@@H](C2)C(=O)Nc1cccc(OC(F)(F)F)c1F)C(=O)Cn1nc(C(N)=O)c2ccncc12 |r|

NC(=O)c1nn(CC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccncc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cncc(Br)n2)c2ccccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2nc(Br)cs2)c2ccccc12 |r|

Cc1cc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(Br)n3)c2c(C)n1)C(N)=O |r|

C[C@]12C[C@H]1N([C@@H](C2)C(=O)Nc1cccc(Br)n1)C(=O)Cn1nc(C(N)=O)c2ccccc12 |r|

Cc1cc2c(nn(CC(=O)N3[C@@H]4C[C@]4(C)C[C@H]3C(=O)Nc3cccc(Br)n3)c2cn1)C(N)=O |r|

NC(=O)c1nn(CC(=O)N2C[C@H]3C[C@H]3[C@H]2C(=O)Nc2cccc(Br)n2)c2ccccc12 |r|

Cc1nccc2c(nn(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(Br)n3)c12)C(N)=O |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccc(OCc3ncccn3)cc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2cc(Cl)ccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ncccc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccncc12 |r|

CC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2nnccc12 |r|

NC(=O)c1cn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)Nc1cccc(Br)n1)C(=O)Cn1nc(C(N)=O)c2ccccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)Nc1cccc(Br)c1F)C(=O)Cn1nc(C(N)=O)c2ccccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)Nc1cccc(Br)n1)C(=O)Cn1nc(C(C)=O)c2ccccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(CO)C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(CO)C[C@H]2C(=O)Nc2cccc(Br)c2F)c2ccccc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@]3(CO)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccccc12 |r|

CC(=O)c1nc(CC(=O)N2[C@@H]3C[C@]3(CO)C[C@H]2C(=O)NCc2cccc(Cl)c2F)n2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H]3C[C@H]3[C@H]2C(=O)Nc2cccc(Br)n2)c2ccccc12 |r|

NC(=O)n1cc(NC(=O)N2C[C@H](F)C[C@H]2C(=O)Nc2cccc(Br)n2)c2ccccc12 |r|

CCOC(=O)[C@H](CC1CCCCC1)NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1nc(C(C)=O)c2cccnc12 |r|

COC(=O)[C@H](CC(C)C)NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1nc(C(C)=O)c2cccnc12 |r|

COC(=O)C(CCC(F)(F)F)NC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1nc(C(C)=O)c2cccnc12 |r|

NC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(c2)S(F)(F)(F)(F)F)c2ccccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2nccc(n2)C(F)(F)F)c2ncccc12 |r|

COCCOc1ccc2n(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(OC(F)(F)F)c3F)nc(C(C)=O)c2c1

CC(Oc1ccc2n(CC(=O)N3[C@@H]4C[C@@H]4C[C@H]3C(=O)Nc3cccc(OC(F)(F)F)c3F)nc(C(C)=O)c2c1)C#N |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)Nc2cccc(OC(F)(F)F)c2F)c2ccc(OCC3CCCO3)cc12 |r|

CC(=O)c1cn(CC(=O)N2C[C@H](F)[C@@H](F)[C@H]2C(=O)NCc2cccc(Cl)c2F)c2ccccc12

CC(C)(C)CCNC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1nc(C(N)=O)c2ccccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCCCOC(F)(F)F)c2ccccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCCC(C)(C)C)C(=O)Cn1nc(C(N)=O)c2ccccc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCCC(C)(C)C)C(=O)Cn1nc(C(N)=O)c2cc(C)ncc12 |r|

CO[C@@H]1[C@@H](F)CN([C@@H]1C(=O)NCCC(C)(C)C)C(=O)Cn1nc(C(C)=O)c2ccccc12 |r|

CC(C)(C)CCNC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1nc(C(N)=O)c2ccncc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCCC(C)(C)C)c2cnccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCCC(C)(C)C)c2ccc(OCc3ncccn3)cc12 |r|

C[Si](C)(C)CCNC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1nc(C(N)=O)c2ccncc12 |r|

CC(C)(O)CCNC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1nc(C(N)=O)c2ccncc12 |r|

CO[C@@H]1CN([C@@H]([C@H]1F)C(=O)NCCC(C)(C)C)C(=O)Cn1nc(C(N)=O)c2ccccc12 |r|

CCNC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1nc(C(N)=O)c2ccncc12 |r|

CCNC(=O)[C@@H]1C[C@H]2C[C@H]2N1C(=O)Cn1nc(C(C)=O)c2cc(OCc3ncccn3)ccc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCCCOC(F)(F)F)c2ccc(OCc3ncccn3)cc12 |r|

CC(=O)c1nn(CC(=O)N2[C@@H]3C[C@@H]3C[C@H]2C(=O)NCCOC(F)(F)F)c2ccc(OCc3ncccn3)cc12 |r|