Compound Name

SMILES String

COc1ccc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc1

COc1cccc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1

COc1ccccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CCOc1ccc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc1

CCOc1cccc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1

CCOc1ccccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

COc1cccc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1Cl

COc1ccc(F)cc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

COc1cc(Cl)ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

COc1c(Cl)cccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(OCCN3CCCCC3)c2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(OCCN3CCCC3)c2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(OCCN3CCOCC3)c2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(OCCN3CCOCC3)cc2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(OCCN3CCCCC3)c(Cl)c2)CC1)C(F)(F)F

CN(C)C(=O)C1CCN(CC1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(Cl)cc3N3CCCC3)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3c(cccc3C(F)(F)F)N3CC4COCC4C3)C2)CC1)C(F)(F)F

FCCN1CCN(CC1)c1cc(Cl)ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FCCN1CCN(CC1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(Cl)cc3N3CCOCC3)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(cc3N3CCOCC3)C(F)(F)F)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(cc3N3CCCCC3)C(F)(F)F)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(Cl)cc3N3CCCCC3)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(Cl)cc3N3CC4COCC4C3)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(cc3N3CC4COCC4C3)C(F)(F)F)C2)CC1)C(F)(F)F

FCCOc1cccc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1

FCCOc1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc1Cl

FCCOc1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc1F

FCCOc1cc(Cl)ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FCCOc1ccc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc1

CCOc1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc1Cl

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(Cl)cc(c2)N2CCOCC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(Cl)cc(c2)N2CCCC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(cc(c2)C(F)(F)F)N2CCOCC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(cc(c2)C(F)(F)F)N2CCCC2)CC1)C(F)(F)F

FC(F)(F)Oc1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)N1CCOCC1

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(Cl)cc(c2)N2CC3COCC3C2)CC1)C(F)(F)F

FC1CCN(CC1)c1cc(Cl)cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1

CS(=O)(=O)N1CCN(CC1)c1cc(Cl)cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(cc(c2)C(F)(F)F)N2CCN(CC2)C2CC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(cc(c2)C(F)(F)F)N2CCS(=O)(=O)CC2)CC1)C(F)(F)F

CS(=O)(=O)N1CCN(CC1)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(cc(c2)C(F)(F)F)N2CCC(CC2)C(F)(F)F)CC1)C(F)(F)F

FC1CCN(CC1)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(cc(c2)C(F)(F)F)N2CC3COCC3C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(cc(c2)C(F)(F)F)N2CCC2)CC1)C(F)(F)F

CC1(C)CC2(CN1Cc1ccc(Cl)cc1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

COc1cc(Cl)ccc1CN1CC2(CC1(C)C)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(C)CC2(CN1Cc1ccc(Cl)cc1N1CCOCC1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(C)CC2(CN1Cc1ccc(cc1N1CCOCC1)C(F)(F)F)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(C)CC2(CN1Cc1ccc(cc1N1CCC3(C1)CCOCC3)C(F)(F)F)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

COC(=O)C1CCN(CC1)c1cc(ccc1CN1CC2(CC1(C)C)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

CC1(C)CC2(CN1Cc1cccc(Cl)c1N1CCOCC1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(C)CC2(CN1Cc1ccc(cc1N1CC3COCC3C1)C(F)(F)F)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(C)CC2(CN1Cc1c(cccc1C(F)(F)F)N1CCC3(C1)CCOCC3)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(C)CC2(CN1Cc1c(cccc1C(F)(F)F)N1CC3COCC3C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3cccc(c3)N3CCCC3)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3c(cccc3C(F)(F)F)N3CCCC3)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccccc2Cl)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(Cl)c2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(Cl)cc2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccccc2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3cccc(Cl)c3N3CCC(F)(F)CC3)C2)CC1)C(F)(F)F

FC1CCN(CC1)c1c(Cl)cccc1CN1CCC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2N2CCCC2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2N2CCOCC2)C(F)(F)F)CC1)C(F)(F)F

CN1CCCc2ccc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc12

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(c2)N2CCOCC2)CC1)C(F)(F)F

COC(=O)N1CCCc2cccc(CN3CCC4(C3)CCN(CC4)C(=O)OC(C(F)(F)F)C(F)(F)F)c12

CCN1CCCc2cccc(CN3CCC4(C3)CCN(CC4)C(=O)OC(C(F)(F)F)C(F)(F)F)c12

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(cc3N3CCCC3)C(F)(F)F)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2N2CC3CCC(C2)O3)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(Cl)cc2N2CCCCC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(Cl)cc2N2CC3CCC(C2)O3)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(Cl)cc2N2CCCC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(Cl)cc2N2CCOCC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2N2CCCCC2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(N3CCOCC3)c2Cl)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(N3CCCCC3)c2Cl)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(N3CCCC3)c2Cl)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(N3CC4CCC(C3)O4)c2Cl)CC1)C(F)(F)F

Cc1c(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cccc1N1CCOCC1

Cc1c(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cccc1N1CCCCC1

Cc1c(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cccc1N1CCCC1

Cc1c(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cccc1N1CC2CCC(C1)O2

CCN1CCN(CC1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

CC(=O)N1CCN(CC1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

CC(C)(C)c1ccc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(c1)N1CCN(CC1)S(C)(=O)=O

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2N2CCC(F)(F)CC2)C(F)(F)F)CC1)C(F)(F)F

FC1CCN(CC1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2N2CCS(=O)(=O)CC2)C(F)(F)F)CC1)C(F)(F)F

CC(=O)NC1CCN(CC1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

CS(=O)(=O)NC1CCN(CC1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2N2CCCCCC2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2N2CCC2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2N2CC3COCC3C2)C(F)(F)F)CC1)C(F)(F)F

CCN1CCN(CC1)c1cc(Cl)ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC(=O)N1CCN(CC1)c1cc(Cl)ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CS(=O)(=O)N1CCN(CC1)c1cc(Cl)ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(Cl)cc2N2CCC(F)(F)CC2)CC1)C(F)(F)F

FC1CCN(CC1)c1cc(Cl)ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(Cl)cc2N2CCS(=O)(=O)CC2)CC1)C(F)(F)F

CC(=O)NC1CCN(CC1)c1cc(Cl)ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CS(=O)(=O)NC1CCN(CC1)c1cc(Cl)ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(Cl)cc2N2CCCCCC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(Cl)cc2N2CCC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(Cl)cc2N2CC3COCC3C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(N3C4CCC3COC4)c2Cl)CC1)C(F)(F)F

FC1CCN(CC1)c1cccc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1Cl

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(N3CCC(F)(F)CC3)c2Cl)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(N3CC4COCC4C3)c2Cl)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(N3CCN(CS(=O)=O)CC3)c2Cl)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(N3CCN(CC=O)CC3)c2Cl)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(N3CCN(CC3)C3CC3)c2Cl)CC1)C(F)(F)F

CCN1CCN(CC1)c1cccc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1Cl

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(N3CCC4(C3)CCOCC4)c2Cl)CC1)C(F)(F)F

OC(=O)C1CCN(CC1)c1cc(Cl)ccc1CN1CCC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

OC(=O)C1CCN(CC1)c1cc(ccc1CN1CCC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)C1CCN(CC1)c1cc(Cl)ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

OC(=O)C1CCN(CC1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)C1CCN(CC1)c1cc(Cl)cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1

OC(=O)C1CCN(CC1)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

Cc1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc1Cl

Cc1ccc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc1Cl

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc3OCCOc3c2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(N3CCOCC3)c(Cl)c2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(N3CCCC3)c(Cl)c2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(N3CCOCC3)c(c2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(N3CCCC3)c(c2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(Cl)c(c2)N2CCOCC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(Cl)c(c2)N2CCCC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(c(c2)N2CCOCC2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(c(c2)N2CCCC2)C(F)(F)F)CC1)C(F)(F)F

Cc1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc1Cl

Cc1ccc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc1Cl

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc4OCCOc4c3)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(N4CCOCC4)c(Cl)c3)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(N4CCCC4)c(Cl)c3)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(N4CCOCC4)c(c3)C(F)(F)F)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(N4CCCC4)c(c3)C(F)(F)F)C2)CC1)C(F)(F)F

CC(=O)N1CCCc2cccc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)c12

CS(=O)(=O)N1CCCc2cccc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)c12

CCN1CCc2cccc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)c2C1

CC(=O)N1CCc2cccc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)c2C1

CS(=O)(=O)N1CCc2cccc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)c2C1

CC(C)N1CCc2cccc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)c2C1

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc3CCN(Cc23)C2CC2)CC1)C(F)(F)F

CC(C)CN1CCc2cccc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)c2C1

CCc1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc1F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc3COCc3c2)CC1)C(F)(F)F

CCc1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc1F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc4COCc4c3)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(Cl)c(c3)N3CCOCC3)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(Cl)c(c3)N3CCCC3)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(c(c3)N3CCOCC3)C(F)(F)F)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(c(c3)N3CCCC3)C(F)(F)F)C2)CC1)C(F)(F)F

CCN1CCCc2cccc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)c12

CCN1CCc2cccc(CN3CCC4(C3)CCN(CC4)C(=O)OC(C(F)(F)F)C(F)(F)F)c2C1

CC(=O)N1CCc2cccc(CN3CCC4(C3)CCN(CC4)C(=O)OC(C(F)(F)F)C(F)(F)F)c2C1

CS(=O)(=O)N1CCc2cccc(CN3CCC4(C3)CCN(CC4)C(=O)OC(C(F)(F)F)C(F)(F)F)c2C1

CC(C)N1CCc2cccc(CN3CCC4(C3)CCN(CC4)C(=O)OC(C(F)(F)F)C(F)(F)F)c2C1

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3cccc4CCN(Cc34)C3CC3)C2)CC1)C(F)(F)F

CC(C)CN1CCc2cccc(CN3CCC4(C3)CCN(CC4)C(=O)OC(C(F)(F)F)C(F)(F)F)c2C1

CN1CCC(CC1)Oc1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

CN1CCC(CC1)Oc1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2OCC(=O)N2CCCC2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(OCC(=O)N3CCCC3)cc(c2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2OC2CCOCC2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(OC3CCOCC3)cc(c2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2Oc2nc3ccccc3s2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(Oc3nc4ccccc4s3)cc(c2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2Oc2cccnc2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(Oc3cccnc3)cc(c2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2OC2CCS(=O)(=O)CC2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(OC3CCS(=O)(=O)CC3)cc(c2)C(F)(F)F)CC1)C(F)(F)F

Cc1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc1C(F)(F)F

NC(=O)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc1C(F)(F)F

OC(=O)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc1C(F)(F)F

Cc1ccc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc1C(F)(F)F

NC(=O)c1ccc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc1C(F)(F)F

OC(=O)c1ccc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc1C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(c(Cl)c2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(Cl)c(c2)C(F)(F)F)CC1)C(F)(F)F

CC1(C)CC2(CN1Cc1cccc(N3CCOCC3)c1Cl)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(C)CC2(CN1Cc1cc(Cl)cc(c1)N1CCOCC1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(C)CC2(CN1Cc1cc(Cl)ccc1N1CCOCC1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(C)CC2(CN1Cc1cc(cc(c1)C(F)(F)F)N1CCOCC1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

CN1CCN(CC1)c1c(Cl)cccc1CN1CC2(CC1(C)C)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(C)CC2(CN1Cc1cccc(OC(F)(F)F)c1N1CCOCC1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(C)CC2(CN1Cc1cccc(CN3CCOCC3)c1F)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(C)CC2(CN1Cc1cc(CN3CCOCC3)ccc1OC(F)(F)F)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

CS(=O)(=O)C1CCN(C1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)C1CCN(Cc2cc(Cl)cc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)c2)CC1

CC1(CN(CCO1)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F)C(O)=O

OC(=O)[C@@H]1CCCCN1c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F |r|

OC(=O)C1CN(CCO1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)C1CCN(CC1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C#C

OC(=O)C1CCN(C1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)C1COCCN1c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

OC(=O)C1CCN(C1)c1cc(ccc1CN1CCC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)C1CCN(C1)c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

OC(=O)C1CCN(C1)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

OC(=O)C1CN(CCO1)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(cc(c2)C(F)(F)F)-c2nnn[nH]2)CC1)C(F)(F)F

OC(=O)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

OC(=O)C1CN(CCO1)c1cc(ccc1CN1CCC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)C1CCN(CC1)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C#N

OC(=O)[C@@H]1CCCN(C1)c1cc(ccc1CN1CCC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F |r|

OC(=O)[C@@H]1CCCN(C1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F |r|

CC1(CCCN(C1)c1cc(ccc1CN1CCC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)C(O)=O

OC(=O)[C@H]1CCCN(C1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F |r|

CC1(CCCN(C1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)C(O)=O

CC1(CCN(C1)c1cc(ccc1CN1CCC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)C(O)=O

CC1(CCCN(C1)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F)C(O)=O

OC(=O)C1CCN(CC1)c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

CC1(CCCN(C1)c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F)C(O)=O

OC(=O)C1CCCCN1c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

OC(=O)C1CCCCN1c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(O)=O

OC(=O)C1CCN(CC1)c1ccc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc1C(F)(F)F

CC1(CCN(C1)c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F)C(O)=O

CC1(CCN(C1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)C(O)=O

CC1(CCN(C1)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(O)=O)C(O)=O

OC(=O)C1CCN(CC1)c1cc(Cl)cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)c1

OC(=O)C1CCN(CC1)c1cc(F)cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)c1

OC(=O)C1CCN(CC1)c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc1C(F)(F)F

CC(=O)C1CCC(CC1)c1cc(ccc1CN1CCC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F |(-1.85,9.48,;-3.25,8.85,;-4.5,9.76,;-3.42,7.32,;-2.17,6.41,;-2.33,4.88,;-3.74,4.26,;-4.98,5.16,;-4.82,6.69,;-3.9,2.72,;-5.31,2.1,;-5.47,.57,;-4.22,-.34,;-2.81,.29,;-2.65,1.82,;-1.25,2.45,;,1.54,;;1.46,-.48,;2.37,.77,;1.46,2.02,;3.14,-.56,;4.68,-.56,;5.45,.77,;4.68,2.1,;3.14,2.1,;6.99,.77,;7.76,-.56,;7.76,2.1,;9.3,2.1,;10.07,3.44,;10.84,4.77,;8.74,4.21,;11.4,2.67,;10.07,.77,;10.84,-.56,;8.74,,;11.4,1.54,;-6.87,-.06,;-8.28,-.69,;-7.5,1.35,;-6.25,-1.47,)|

OC(=O)C1CCN(CC1)c1cc(F)cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1

OC(=O)C1CCN(CC1)c1cc(F)ccc1CN1CCC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

OC(=O)C1CCN(Cc2cc(ccc2CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)CC1

OC(=O)C1CCN(Cc2cc(ccc2CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)CC1

OC(=O)C1CCN(CC1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)S(F)(F)(F)(F)F

OC(=O)C1CCN(CC1)c1cc(ccc1CN1CCC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)S(F)(F)(F)(F)F

Cc1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(O)=O

OC(=O)C1CCN(Cc2cc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c2)C(F)(F)F)CC1

OC(=O)C1CCN(Cc2cc(CN3CCC4(C3)CCN(CC4)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c2)C(F)(F)F)CC1

OC(=O)C1CCN(Cc2cc(CN3CCC4(C3)CCN(CC4)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc2Cl)CC1

OC(=O)C1CCN(Cc2ccc(CN3CCC4(C3)CCN(CC4)C(=O)OC(C(F)(F)F)C(F)(F)F)cc2C(F)(F)F)CC1

OC(=O)C1CCN(CC1)c1cc(OC(F)(F)F)ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

OC(=O)C1CCN(CC1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C#N

CC1(CN(CCO1)c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F)C(O)=O

OC(=O)C1CCN(Cc2cc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c2)C(F)(F)F)C1

OC(=O)c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc1C(F)(F)F

CC1(CN(CCO1)c1cc(ccc1CN1CCC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)C(O)=O

OC(=O)c1ccc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc1C(F)(F)F

CC1(CN(CCO1)c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc1C(F)(F)F)C(O)=O

OC(=O)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)C1CCN(Cc2cc(ccc2CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)C1

OC(=O)C1CCN(CC1)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)S(F)(F)(F)(F)F

OC(=O)C1CCN(CC1)c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)S(F)(F)(F)(F)F

OC(=O)c1ccc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(c1)C(F)(F)F

OC(=O)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc1Cl

CS(=O)(=O)C1CCN(CC1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

CS(=O)(=O)C1CN(C1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)C1CCN(Cc2cc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(OC(F)(F)F)c2)CC1

OC(=O)C1CCN(Cc2cc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(OC(F)(F)F)c2)C1

OC(=O)C1CCN(CC1)C(=O)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(O)=O

OC(=O)C1CCN(Cc2cc(Cl)cc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)c2)C1

OC(=O)[C@H]1CCCCN1c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F |r|

NC(=O)C1CCN(Cc2cc(ccc2CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)CC1

NC(=O)C1CCN(CC1)C(=O)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)C1CN(CCO1)c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

OC(=O)C1COCCN1c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2)C#C)CC1)C(F)(F)F

OC(=O)C1CCN(CC1)C(=O)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

CCOC(=O)CCCNc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

CC(C)(C)OC(=O)CCCNc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)CCCOc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)CCCOc1cc(Cl)ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CCOC(=O)OC(C)OC(=O)CCCNc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

CC(C)OC(=O)OC(C)OC(=O)CCCNc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

CC(C)(C)C(=O)OCOC(=O)CCCNc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

CC(C)C(=O)OC(C)OC(=O)CCCNc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)COCCNc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)COCCNc1ccc(Cl)cc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

OC(=O)COCCNc1c(F)cccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CN(CCNc1cc(Cl)ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)CC(O)=O

OC(=O)COc1cc(Cl)ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

OC(=O)COc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)CCCCc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)C1(CC1)Oc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCN(Cc2cc(COC=O)cc(c2)C(F)(F)F)CC1)C(F)(F)F

CC(C)(OC=O)C#Cc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCN(Cc2cc(OC3(CC3)OC=O)cc(c2)C(F)(F)F)CC1)C(F)(F)F

Cc1ccc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(OCC(=O)NS(C)(=O)=O)c1F

Cc1ccc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(OCC(=O)NS(=O)(=O)C2CC2)c1F

OC(=O)C1(CC1)Oc1c(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cccc1C(F)(F)F

Cc1ccc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(OCC2(CC2)C(O)=O)c1Cl

Cc1ccc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(C#CC(C)(C)C(O)=O)c1F

CC(C)(C#Cc1c(F)cccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(O)=O

OC(=O)C1(COc2c(CN3CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(F)cc2C#N)CC1

OC(=O)C1(COc2cc(ccc2CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)CC1

OC(=O)C1(COc2cc(CN3CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c2)C(F)(F)F)CC1

Cc1ccc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(OCC2(CC2)C(O)=O)c1F

OC(=O)C1(COc2c(CN3CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cccc2C(F)(F)F)CC1

Cc3ccc(CN1CCN(C(=O)OC(C(F)(F)F)C(F)(F)F)CC1)c(OCC2(C(=O)NS(C)(=O)=O)CC2)c3F

Cc1ccc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(OCC2(CCCC2)C(O)=O)c1F

OC(=O)C1(COc2c(CN3CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc(F)c2F)CC1

OC(=O)C1(COc2cc(F)c(F)cc2CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)CC1

OC(=O)C1(COc2cc(ccc2CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C#N)CC1

OC(=O)C1(COc2c(CN3CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cccc2C#N)CC1

OC(=O)C1(COc2c(CN3CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc(F)c2F)CCCC1

Cc1c(F)ccc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1OCC1(CC1)C(O)=O

Cc1cc(F)cc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1OCC1(CC1)C(O)=O

Cc1cc(F)cc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1OCC1(CCCC1)C(O)=O

OC(=O)C1(COc2c(F)cccc2CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)CCCC1

OC(=O)C1(COc2cc(F)ccc2CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)CCCC1

OC(=O)C1(COc2cc(ccc2CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C#N)CCCC1

OC(=O)[C@@H]1C[C@@H](C1)Oc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F |r,wU:5.7,3.2,(-9.61,-3.62,;-8.28,-4.39,;-8.28,-5.93,;-6.94,-3.62,;-5.46,-4.02,;-5.06,-2.54,;-6.55,-2.14,;-3.72,-1.77,;-3.72,-.23,;-5.06,.54,;-5.06,2.08,;-3.72,2.85,;-2.39,2.08,;-2.39,.54,;-1.06,-.23,;.28,.54,;1.61,-.23,;2.94,.54,;2.94,2.08,;1.61,2.85,;.28,2.08,;4.28,2.85,;4.28,4.39,;5.61,2.08,;6.94,2.85,;8.28,2.08,;9.61,1.31,;7.51,.75,;9.05,3.42,;6.94,4.39,;8.48,4.39,;5.4,4.39,;6.94,5.93,;-6.39,2.85,;-7.73,2.08,;-6.39,4.39,;-6.39,1.31,)|

OC(=O)[C@H]1CC[C@H](C1)Oc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F |r|

OC(=O)[C@@H]1CC[C@H](C1)Oc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F |r|

OC(=O)[C@H]1C[C@@H](C1)Oc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F |r,wU:3.2,wD:5.7,(-9.61,-3.62,;-8.28,-4.39,;-8.28,-5.93,;-6.94,-3.62,;-6.55,-2.14,;-5.06,-2.54,;-5.46,-4.02,;-3.72,-1.77,;-3.72,-.23,;-5.06,.54,;-5.06,2.08,;-3.72,2.85,;-2.39,2.08,;-2.39,.54,;-1.06,-.23,;.28,.54,;1.61,-.23,;2.94,.54,;2.94,2.08,;1.61,2.85,;.28,2.08,;4.28,2.85,;4.28,4.39,;5.61,2.08,;6.94,2.85,;8.28,2.08,;9.61,1.31,;7.51,.75,;9.05,3.42,;6.94,4.39,;8.48,4.39,;5.4,4.39,;6.94,5.93,;-6.39,2.85,;-7.73,2.08,;-6.39,4.39,;-6.39,1.31,)|

CC(C)(C#Cc1cc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F)C(O)=O

Cc1ccc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(OCC(O)=O)c1Cl

Cc1ccc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(OCC(=O)NS(C)(=O)=O)c1Cl

Cc1ccc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(OCC(=O)NS(=O)(=O)C2CC2)c1Cl

CS(=O)(=O)NC(=O)COc1cc(Cl)ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

Cc3ccc(CN1CCN(C(=O)OC(C(F)(F)F)C(F)(F)F)CC1)c(OCC2(C(=O)NS(C)(=O)=O)CC2)c3Cl

Cc1ccc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(OCC(O)=O)c1F

CS(=O)(=O)NC(=O)C1(COc2cc(ccc2CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)CC1

CC(C)(C#Cc1c(Cl)cccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(O)=O

CCOC(=O)c1cccc(c1)B(O)O

OB(O)c1cccc(c1)C(F)(F)F

OB(O)c1cccc(c1)C#N

OB(O)c1cccc(c1)-c1ccccc1

COc1cccc(c1)B(O)O

OB(O)c1ccc(F)cc1

OB(O)c1ccc(cc1)C(F)(F)F

B(c1ccc(cc1)[N+](=O)[O-])(O)O

OB(O)c1ccc(cc1)C#N

OB(O)c1ccc(cc1)-c1ccccc1

COc1ccc(cc1)B(O)O

CCCCCCCCCc1ccc(cc1)B(O)O

OB(O)c1ccccc1F

OB(O)c1ccccc1C(F)(F)F

OB(O)c1ccccc1-c1ccccc1

COc1ccccc1B(O)O

B(c1cc2ccccc2s1)(O)O

OB(O)c1cc2ccccc2o1

OB(O)c1ccc(F)nc1

B(CCc1ccccc1)(O)O

OB(O)\C=C\c1ccc(cc1)-c1ccccc1

CN(C)C(=O)n1nnnc1Cc1ccc(cc1)-c1ccccc1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3ccc(Cl)c(Cl)c3)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3ccc(cc3)C(F)(F)F)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3ccc(cc3Cl)N3CCOCC3)C2)C1

CS(=O)(=O)Nc1cnn(c1)C(=O)N1CC2CN(Cc3ccccc3Cl)CC2C1

CS(=O)(=O)Nc1cnn(c1)C(=O)N1CC2CN(Cc3cccc(Cl)c3)CC2C1

CS(=O)(=O)Nc1cnn(c1)C(=O)N1CC2CN(Cc3ccc(Cl)cc3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccccc3Cl)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cccc(Cl)c3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(Cl)cc3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(Cl)c(Cl)c3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(cc3)N3CCCC3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(cc3)C(F)(F)F)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(cc3Cl)N3CCOCC3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2(C1)CCN(Cc1ccc(cc1Cl)N1CCOCC1)CC2

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CN(Cc3ccc(Cl)c(Cl)c3)C2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CN(Cc3ccc(cc3)C(F)(F)F)C2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CN(Cc3cccc(Cl)c3)C2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CN(Cc3cccc(c3)C(F)(F)F)C2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CN(Cc3ccccc3Cl)C2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CN(Cc3ccccc3C(F)(F)F)C2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3c(Cl)cccc3Cl)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3ccccc3Cl)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3ccc(Cl)cc3Cl)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3cc(Cl)cc(Cl)c3)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3ccc(C)cc3Cl)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3cccc(Cl)c3C)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3ccccc3C(F)(F)F)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3cccc(Cl)c3Cl)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3ccc(c(c3)N3CCOCC3)C(F)(F)F)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3cccc(c3)C(F)(F)F)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3cccc(c3)C(F)(F)F)C2)C1 |w:30.32|

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3ccc(N4CCCC4)c(Cl)c3)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3cc(cc(c3)C(F)(F)F)N3CCOCC3)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3cc(Cl)ccc3C(F)(F)F)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3cccc(Cl)c3)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(C)cc3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cccc(C)c3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(cc3C)N3CCCC3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccccc3C)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccccc3C(F)(F)F)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(Cl)c(c3)C(F)(F)F)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(F)c(c3)N3CCCC3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cccc(Cl)c3C)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cc(Cl)cc(Cl)c3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cccc(Cl)c3Cl)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cc(C)cc(C)c3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cc(Cl)ccc3Cl)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cc(Cl)cc(c3)N3CCCC3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3c(Cl)cccc3Cl)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cc(cc(c3)C(F)(F)F)N3CCCC3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(Cl)cc3Cl)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cc(cc(c3)C(F)(F)F)N3CCOCC3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(C)cc3Cl)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cccc(c3)C(F)(F)F)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cc(Cl)cc(c3)C3CC4COCC4C3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cccc(c3)N3CCCC3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cc(Cl)cc(c3)N3CCN(CC3)C3CC3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(F)c(Cl)c3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(N4CCCC4)c(Cl)c3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(c(c3)N3CCOCC3)C(F)(F)F)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cc(Cl)cc(c3)N3CCOCC3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(c(c3)N3CCCC3)C(F)(F)F)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(cc3C(F)(F)F)N3CCOCC3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)NCc1ccccc1Cl |r|

CN(C(C)=O)c1cnn(c1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)NCc1cccc(Cl)c1 |r|

CN(Cc1ccccc1Cl)[C@H]1C[C@H]2CN(C[C@H]2C1)C(=O)n1cc(cn1)N(C)C(C)=O |r|

CN(Cc1cccc(Cl)c1)[C@H]1C[C@H]2CN(C[C@H]2C1)C(=O)n1cc(cn1)N(C)C(C)=O |r|

CN(Cc1ccc(Cl)cc1)[C@H]1C[C@H]2CN(C[C@H]2C1)C(=O)n1cc(cn1)N(C)C(C)=O |r|

CN(Cc1ccccc1Cl)[C@@H]1C[C@H]2CN(C[C@H]2C1)C(=O)n1cc(cn1)N(C)C(C)=O |r|

CN(Cc1cccc(Cl)c1)[C@@H]1C[C@H]2CN(C[C@H]2C1)C(=O)n1cc(cn1)N(C)C(C)=O |r|

CN(Cc1ccc(Cl)cc1)[C@@H]1C[C@H]2CN(C[C@H]2C1)C(=O)n1cc(cn1)N(C)C(C)=O |r|

CN(Cc1ccc(N2C3CCC2COC3)c(c1)C(F)(F)F)[C@H]1C[C@H]2CN(C[C@H]2C1)C(=O)n1cc(cn1)N(C)C(C)=O |r|

CN(Cc1cc(cc(c1)C(F)(F)F)N1C2CCC1COC2)[C@H]1C[C@H]2CN(C[C@H]2C1)C(=O)n1cc(cn1)N(C)C(C)=O |r|

CN(Cc1ccc(N2C3CCC2COC3)c(c1)C(F)(F)F)[C@@H]1C[C@H]2CN(C[C@H]2C1)C(=O)n1cc(cn1)N(C)C(C)=O |r|

CN(Cc1cc(Cl)ccc1C(F)(F)F)[C@H]1C[C@H]2CN(C[C@H]2C1)C(=O)n1cc(cn1)N(C)C(C)=O |r|

CN(Cc1cc(Cl)ccc1C(F)(F)F)[C@@H]1C[C@H]2CN(C[C@H]2C1)C(=O)n1cc(cn1)N(C)C(C)=O |r|

CN(C(C)=O)c1cnn(c1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)N(Cc1ccccc1Cl)C(C)=O |r|

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3cc(Cl)ccc3Cl)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3cc(Cl)ccc3Cl)C2)C1 |w:28.30|

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(F)cc3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cccc(F)c3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cccc(CO)c3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccccc3F)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3ccccc3Cl)C2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3cccc(Cl)c3)C2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3ccc(Cl)cc3)C2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(OCC(=O)N4CCCC4)cc3Cl)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2cc(cc(c2)C(F)(F)F)N2CCCC2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2ccc(cc2N2CCCC2)C(F)(F)F)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2ccccc2Cl)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2cccc(Cl)c2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2ccc(Cl)cc2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2ccc(cc2N2C3CCC2COC3)C(F)(F)F)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2ccc(Cl)c(Cl)c2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2ccc(cc2)N2CCCC2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2ccc(cc2)C(F)(F)F)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2ccc(cc2C)-c2ccccc2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2cccc(Oc3ccccc3)c2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2ccc(cc2Cl)N2CCOCC2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2ccc(cc2C)N2CCOCC2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2cccc(F)c2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2cccc(C)c2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2cccc(c2)N2CCCC2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2cccc(c2)C(F)(F)F)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2ccccc2C)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCN(Cc2ccccc2C(F)(F)F)CC1

CC(=O)Nc1cnn(c1)C(=O)N1CCN(Cc2ccc(cc2N2CCCC2)C(F)(F)F)CC1

CN(c1cnn(c1)C(=O)N1CCN(Cc2ccc(cc2N2CCCC2)C(F)(F)F)CC1)S(C)(=O)=O

Cc1cc(ccc1CN1CCN(CC1)C(=O)n1cc(NS(C)(=O)=O)cn1)-c1ccccc1

COc1cc(ccc1CN1CCN(CC1)C(=O)n1cc(NS(C)(=O)=O)cn1)-c1ccccc1

CS(=O)(=O)Nc1cnn(c1)C(=O)N1CCN(Cc2ccc(cc2Cl)-c2ccccc2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(cc3C)-c3ccccc3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CN(Cc3ccc(cc3C)-c3ccccc3)C2)CC1

CC(=O)Nc1cnn(c1)C(=O)N1CCN(Cc2cc(C)cc(c2)N2CCCC2)CC1

CC(=O)Nc1cnn(c1)C(=O)N1CCN(Cc2ccc(cc2N2C3CCC2COC3)C(F)(F)F)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2(C1)CCN(Cc1cccc(Oc3ccccc3)c1)CC2

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3ccc(cc3C)-c3ccccc3)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cccc(Oc4ccccc4)c3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CN(Cc3cccc(Oc4ccccc4)c3)C2)CC1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3cccc(Oc4ccccc4)c3)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cccc(Oc4ccc(Cl)cc4)c3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cccc(Oc4ccccn4)c3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cccc(OCc4ccccc4)c3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cccc(Oc4ccccc4Cl)c3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(Oc4ccccc4)cc3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc4OC(F)(F)Oc4c3)CC2C1

COc1ccc(Oc2cccc(CN3CC4CN(CC4C3)C(=O)n3cc(cn3)N(C)C(C)=O)c2)cc1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cccc(Oc4cccc(Cl)c4)c3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(Oc4ccc(Cl)cc4)cc3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cc(F)c(F)cc3F)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cc(Cl)cc(c3)N3CCC4(C3)CCOCC4)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(OCc4ccccc4)cc3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3cc(Cl)cc(OCc4ccccc4)c3)CC2C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CCC2(CCN(Cc3ccc(cc3Cl)-c3ccncn3)C2)C1

CN(C(C)=O)c1cnn(c1)C(=O)N1CC2CN(Cc3ccc(Oc4cncnc4)cc3Cl)CC2C1

CS(=O)(=O)Nc1cnn(c1)C(=O)N1CC2CN(Cc3cc(Cl)ccc3C(F)(F)F)CC2C1

CS(=O)(=O)Nc1cnn(c1)C(=O)N1CCC2(CN(Cc3cc(Cl)ccc3C(F)(F)F)C2)CC1

CS(=O)(=O)Nc1cnn(c1)C(=O)N1CC2CN(Cc3ccc(cc3C(F)(F)F)N3CCCC3)CC2C1

CS(=O)(=O)Nc1cnn(c1)C(=O)N1CCN(Cc2ccc(cc2C(F)(F)F)N2CCCC2)CC1

CS(=O)(=O)Nc1cnn(c1)C(=O)N1CCN(Cc2cc(Cl)ccc2C(F)(F)F)CC1

CS(=O)(=O)Nc1cnn(c1)C(=O)N1CCC2(CCN(Cc3cc(Cl)cc(c3)C(F)(F)F)C2)CC1

CS(=O)(=O)Nc1cnn(c1)C(=O)N1CCN(Cc2ccc(cc2C(F)(F)F)-c2ncco2)CC1

O=C(Nc1cccc(c1)-c1ccccc1)OC1CCCCC1

O=C(NCCCCCc1ccccc1)OC1CCCCC1

O=C(Nc1ccccc1)OC1CCCCC1

O=C(Nc1cccc(c1)-c1ccccc1)OCCCCCc1ccccc1

Cc1cccc(c1)-c1cccc(NC(=O)OC2CCCCC2)c1

FC(F)(F)c1cccc(c1)-c1cccc(NC(=O)OC2CCCCC2)c1

O=C(Nc1cccc(Oc2cccc(c2)-c2ccccc2)c1)OC1CCCCC1

O=C(Nc1ccccc1-c1ccccc1)OC1CCCCC1

OCC(O)COC(=O)Nc1cccc(c1)-c1ccccc1

CC1(C)OCC(CO1)OC(=O)Nc1cccc(c1)-c1ccccc1

O=C(Nc1cccc(c1)-c1ccccc1)Oc1cccc(c1)-c1ccccc1

O=C(Nc1ccc(cc1)-c1ccccc1)OC1CCCCC1

O=C(Nc1cccc(c1)-c1ccccc1)Oc1ccccc1

Cc1cccc(c1)-c1cccc(NC(=O)OC(CO)CO)c1

OCC(CO)OC(=O)Nc1cccc(c1)-c1ccccc1

CN(C(=O)OC1CCCCC1)c1cccc(c1)-c1ccccc1

O=C(NC1CCCCC1)Nc1cccc(c1)-c1ccccc1

O=C(CC1CCCCC1)Nc1cccc(c1)-c1ccccc1

O=C(Nc1cccc(c1)-c1ccccc1)SC1CCCCC1

COC(=O)[C@]1(C)CC[C@]2(C)CC[C@]3(C)C4=CC=c5c(cc(O)c(O)c5=C)[C@]4(C)CC[C@@]3(C)C2C1 |r,c:16,t:14|

C[C@]12CC[C@](C)(C[C@H]1[C@]1(C)CC[C@]3(C)C(=CC=c4c3cc(O)c(O)c4=C)[C@@]1(C)CC2)C(O)=O |r,c:15,17|

COC(=O)[C@]1(C)CC[C@]2(C)CC[C@]3(C)C4=CCc5c(C)c(O)c(O)cc5[C@]4(C)CC[C@@]3(C)C2C1 |r,t:14|

Cc1c(O)c(O)cc2c1CC=C1[C@@]2(C)CC[C@@]2(C)C3C[C@@](C)(CC[C@]3(C)CC[C@]12C)C(O)=O |r,c:11|

CC(=O)Oc1cc2c(CC=C3[C@@]2(C)CC[C@@]2(C)[C@@H]4C[C@@](C)(CC[C@]4(C)CC[C@]32C)C(O)=O)c(C)c1OC(C)=O |r,c:9|

Fc1ccc(cc1)-n1ccc2cc(ccc12)C(=O)N1CC(C1)N1CCN(CC1)C(=O)c1nccs1

FC(F)(F)C(OC(=O)N1CCc2ccccc2C1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCc2ccccc2[C@H]1c1ccccc1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCc2ccccc2[C@@H]1c1ccccc1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCc2cccc(Br)c2C1)C(F)(F)F

FCC(CF)OC(=O)N1CCc2c(Br)cccc2C1

CC1N(CCc2ccccc12)C(=O)OC(C(F)(F)F)C(F)(F)F

CCC1N(CCc2ccccc12)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1Cc2ccc(Br)cc2C1)C(F)(F)F

Oc1ccc2CN(Cc2c1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCc2cc(Br)ccc12)C(F)(F)F

FC(F)(F)C(OC(=O)N1Cc2cc(Br)cnc2C1)C(F)(F)F

FC(F)(F)C(OC(=O)N1Cc2cccc(Br)c2C1)C(F)(F)F

CC1Cc2ccccc2CN1C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1Cc2ccc(Cl)nc2C1)C(F)(F)F

CC1N(Cc2cc(Br)ccc12)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCc2c(Br)cccc2C1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCc2cc(Br)ccc2C1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCc2ccc(Br)cc2C1)C(F)(F)F

COc1cccc2CN(Cc12)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1CN(Cc2ccccc12)C(=O)OC(C(F)(F)F)C(F)(F)F

COc1cc2CN(Cc2cc1OC)C(=O)OC(C(F)(F)F)C(F)(F)F

COc1cccc2CN(CCc12)C(=O)OC(C(F)(F)F)C(F)(F)F

COc1ccc2CN(CCc2c1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCCc2ccccc2C1)C(F)(F)F

FC(F)(F)C(OC(=O)N1Cc2ccc(cc2C1)-c1ccccc1)C(F)(F)F

COc1ccc(cc1F)-c1ccc2CN(Cc2c1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCc2cccc(-c3ccccc3)c2C1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCc2c(C1)cccc2-c1ccccc1)C(F)(F)F

FC(F)(F)C(OC(=O)N1Cc2ccc(cc2C1)N1CCNCC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1Cc2ccc(cc2C1)N1CCCC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1Cc2ccc(cc2C1)N1CCS(=O)(=O)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1Cc2ccc(cc2C1)N1CCOCC1)C(F)(F)F

CC1(C)C2C1C(=O)N(OC(=O)N1CCc3c(Br)cccc3C1)C2=O

Brc1cccc2CN(CCc12)ON1C(=O)C2CC2C1=O

CC1(C)C2C1C(=O)N(OC(=O)N1Cc3ccc(O)cc3C1)C2=O

CC1(C)C2C1C(=O)N(OC(=O)N1Cc3ccc(cc3C1)N1CCOCC1)C2=O

OC[C@@H](OC(=O)N1CCc2c(Br)cccc2C1)C(F)(F)F

FCCCOc1cccc2CN(CCc12)C(=O)OC(C(F)(F)F)C(F)(F)F

FCCCOc1ccc2CN(Cc2c1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1Cc2ccc(OCC3CC3)cc2C1)C(F)(F)F

FC(F)(F)C(OC(=O)N1Cc2ccc(OCCN3CCOCC3)cc2C1)C(F)(F)F

FC(F)COc1ccc2CN(Cc2c1)C(=O)OC(C(F)(F)F)C(F)(F)F

CN(C)CCOc1ccc2CN(Cc2c1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1Cc2ccc(NCCN3CCOCC3)cc2C1)C(F)(F)F

FC(F)(F)C(OC(=O)N1Cc2ccc(OCCN3CCCCC3)cc2C1)C(F)(F)F

FC(F)(F)C(OC(=O)N1Cc2ccc(OCCN3CCCC3)cc2C1)C(F)(F)F

FC(F)(F)C(OC(=O)N1Cc2ccc(OCC(=O)N3CCOCC3)cc2C1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CC2(CC(C2)Oc2cccc(c2)C(F)(F)F)C1)C(F)(F)F

Fc1cccc(OC2CC3(C2)CN(C3)C(=O)OC(C(F)(F)F)C(F)(F)F)c1

FC(F)(F)Oc1cccc(OC2CC3(C2)CN(C3)C(=O)OC(C(F)(F)F)C(F)(F)F)c1

Fc1cccc(OC2C[C@@]3(C2)CCN(C3)C(=O)OC(C(F)(F)F)C(F)(F)F)c1 |r,wU:9.9,(-17.05,-2.89,;-15.52,-3.05,;-14.89,-4.46,;-13.36,-4.62,;-12.46,-3.38,;-13.08,-1.97,;-12.18,-.72,;-10.65,-.88,;-9.68,-2.08,;-8.48,-1.11,;-9.45,.08,;-7.71,-2.45,;-6.2,-2.13,;-6.04,-.59,;-7.45,.03,;-4.71,.18,;-3.38,-.59,;-4.71,1.72,;-3.38,2.49,;-3.38,4.03,;-3.38,5.57,;-1.84,4.03,;-4.92,4.03,;-2.04,1.72,;-2.81,.38,;-1.27,3.05,;-.71,.95,;-14.62,-1.81,)|

Fc1cccc(OC2CCC3(CN(C3)C(=O)OC(C(F)(F)F)C(F)(F)F)C2)c1

Fc1cncc(OC2CC3(C2)CN(C3)C(=O)OC(C(F)(F)F)C(F)(F)F)c1

CC1(C)C2C1C(=O)N(OC(=O)N1CC3(CC(C3)Oc3cccc(c3)C(F)(F)F)C1)C2=O

CC1(C)C2C1C(=O)N(OC(=O)N1CC3(C1)CCC(C3)Oc1cncc(F)c1)C2=O

Fc1ccc(cc1)C(OC1CC2(C1)CCN(C2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1ccc(F)cc1 |(-8.79,-.56,;-7.25,-.56,;-6.48,-1.9,;-4.94,-1.9,;-4.17,-.56,;-4.94,.77,;-6.48,.77,;-2.63,-.56,;-1.86,.77,;-.32,.77,;.77,-.32,;1.86,.77,;.77,1.86,;2.76,2.02,;4.23,1.54,;4.23,,;2.76,-.48,;5.47,-.91,;5.31,-2.44,;6.88,-.28,;8.13,-1.18,;9.53,-.56,;10.94,.07,;8.91,.85,;10.16,-1.96,;7.97,-2.72,;7.81,-4.25,;6.43,-2.55,;9.5,-2.88,;-1.86,-1.9,;-.32,-1.9,;.45,-3.23,;-.32,-4.56,;.45,-5.9,;-1.86,-4.56,;-2.63,-3.23,)|

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3c(cccc3C(F)(F)F)C3CC4COCC4C3)C2)CC1)C(F)(F)F

CC(=O)N1CCCc2cccc(CN3CCC4(C3)CCN(CC4)C(=O)OC(C(F)(F)F)C(F)(F)F)c12

CS(=O)(=O)N1CCN(CC1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

CC1(CN(CCO1)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F)OC=O

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2N2CCOC(C2)OC=O)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3cc(cc(c3)C(F)(F)F)N3CCCC3)C2)CC1)C(F)(F)F

CC1CCCN(C1)c1cc(ccc1CN1CCC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

CC1CCN(C1)c1cc(ccc1CN1CCC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

CC1CCCN(C1)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3cc(cc(c3)C(F)(F)F)N3CCCCC3)C2)CC1)C(F)(F)F

OC(=O)C1CCCCN1c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(N4CCCCC4)c(c3)C(F)(F)F)C2)CC1)C(F)(F)F

CC1CCN(C1)c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

CC1CCN(C1)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3cc(Cl)cc(c3)N3CCCCC3)C2)CC1)C(F)(F)F

Fc1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)N1CCCCC1

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(c(c3)N3CCCCC3)C(F)(F)F)C2)CC1)C(F)(F)F

OC(=O)C1CCN(CC1)c1cc(F)ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

Fc1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)N1CCCCC1

Fc1ccc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)c(c1)N1CCCCC1

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2CN2CCCCC2)C(F)(F)F)CC1)C(F)(F)F

OC(=O)C1CCN(Cc2cc(F)ccc2CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)CC1

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(cc3N3CCCCC3)S(F)(F)(F)(F)F)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(CN3CCCCC3)cc(c2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3cc(CN4CCCCC4)cc(c3)C(F)(F)F)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(Cl)c(CN4CCCCC4)c3)C2)CC1)C(F)(F)F

CC1CN(CCO1)c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(cc3)C(F)(F)F)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3cccc(c3)C(F)(F)F)C2)CC1)C(F)(F)F

CC1(CN(CCO1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)C(O)=O

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2CN2CCCC2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(cc(c2)S(F)(F)(F)(F)F)N2CCCCC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccccc2C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)Oc1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(CN2CCCCC2)c1

FC(F)(F)Oc1cc(CN2CCCC2)cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1

FC(F)(F)Oc1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(=O)N1CCCCC1

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3cc(cc(c3)C(F)(F)F)N3CCOCC3)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CC1)CN(CCO2)S(=O)(=O)c1ccccc1)C(F)(F)F

Fc1ccc(cc1)S(=O)(=O)N1CCOC2(CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C1

FC(F)(F)C(OC(=O)N1CCC2(CC1)CN(CC1CCCOC1)CCO2)C(F)(F)F

Fc1ccc(cc1)S(=O)(=O)N1CCOC2(CCN(CC2)C(=O)ON2C(=O)CCC2=O)C1

O=C(ON1C(=O)CCC1=O)N1CCC2(CC1)CN(Cc1ccccc1)CCO2

CN([C@H]1COC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1 |r|

CN([C@H]1COC2(C1)CCN(CC2)C(=O)ON1C(=O)CCC1=O)S(=O)(=O)c1ccccc1 |r|

FC(F)(F)C(OC(=O)N1CCC2(CCN(C2)C(=O)c2ccccc2)CC1)C(F)(F)F

O=C(ON1C(=O)CCC1=O)N1CCC2(CCN(C2)C(=O)c2ccccc2)CC1

O=C(ON1C(=O)CCC1=O)N1CCC2(CC(CO2)c2ccc(cc2)C#N)CC1

FC(F)(F)C(OC(=O)N1CCC2(CC(CO2)c2ccc(cc2)C#N)CC1)C(F)(F)F

Fc1cnn(c1)[C@H]1COC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F |r|

Fc1cnn(c1)[C@H]1COC2(C1)CCN(CC2)C(=O)ON1C(=O)CCC1=O |r|

FC(F)c1ccc(OC2CC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cn1

FC(F)(F)C(OC(=O)N1CCC2(CC1)CN(Cc1ccccc1)CCO2)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CC1)CN(Cc1ccc(nc1)C(F)(F)F)CCO2)C(F)(F)F

Fc1ccc(CN2CCOC3(CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)C2)cc1

FC(F)(F)C(OC(=O)N1CCC2(CC1)CN(Cc1cccnc1C#N)CCO2)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CC1)CN(Cc1nccs1)CCO2)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CC1)CN(Cc1cnccn1)CCO2)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CC1)CN(Cc1ccccn1)CCO2)C(F)(F)F

CC[C@H]1C[C@H]1S(=O)(=O)N1CCOC2(CCN(CC2)C(=O)ON2C(=O)CCC2=O)C1 |r|

FC(F)(F)C(OC(=O)N1CCC2(CC1)CN(CC1CCOC1)CCO2)C(F)(F)F

CC(C)CN1CCOC2(CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C1

Fc1ccc(CN2CCOC3(CCN(CC3)C(=O)ON3C(=O)CCC3=O)C2)cc1

O=C(ON1C(=O)CCC1=O)N1CCC2(CC1)CN(Cc1cnccn1)CCO2

CC[C@H]1C[C@H]1S(=O)(=O)N1CCOC2(CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C1 |r|

FC(F)(F)C(OC(=O)N1CCC2(CC1)CN(CCO2)S(=O)(=O)CC1CCCCO1)C(F)(F)F

O=C(ON1C(=O)CCC1=O)N1CCC2(CC1)CN(CCO2)S(=O)(=O)CC1CCCCO1

O=C(ON1C(=O)CCC1=O)N1CCC2(CC1)CN(CCO2)S(=O)(=O)c1cnccn1

FC(F)(F)C(OC(=O)N1CCC2(CC1)CN(CCO2)S(=O)(=O)c1cnccn1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(C[C@H](CO2)NS(=O)(=O)c2ccccc2)CC1)C(F)(F)F |r|

FC(F)(F)C(OC(=O)N1CCC2(C[C@@H](CO2)NS(=O)(=O)c2ccccc2)CC1)C(F)(F)F |r|

O=C(ON1C(=O)CCC1=O)N1CCC2(CC(CO2)NS(=O)(=O)c2ccccc2)CC1

CN([C@H]1COC2(C1)CCN(CC2)C(=O)ON1C(=O)CCC1=O)S(=O)(=O)CC1CC1 |r|

CN([C@H]1COC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)S(=O)(=O)CC1CC1 |r|

CN(C1COC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)S(=O)(=O)C1CCC1

CC(C)CS(=O)(=O)N(C)C1COC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

CN(C1COC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)S(=O)(=O)C1CC1

CN(C1COC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1nccs1

CN(C1COC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)S(=O)(=O)CC1CCC1

CN(C1COC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)S(=O)(=O)Cc1ccccc1

CN(C1COC2(C1)CCN(CC2)C(=O)ON1C(=O)CCC1=O)S(=O)(=O)C1CC1

CC(C)CS(=O)(=O)N(C)C1COC2(C1)CCN(CC2)C(=O)ON1C(=O)CCC1=O

CN(C1COC2(C1)CCN(CC2)C(=O)ON1C(=O)CCC1=O)S(=O)(=O)c1nccs1

CN(C1COC2(C1)CCN(CC2)C(=O)ON1C(=O)CCC1=O)S(=O)(=O)CC1CCC1

CN(C1COC2(C1)CCN(CC2)C(=O)ON1C(=O)CCC1=O)S(=O)(=O)Cc1ccccc1

CN(C1COC2(C1)CCN(CC2)C(=O)ON1C(=O)CCC1=O)S(=O)(=O)C1CCC1

FC(F)(F)Oc1cccc(c1)C1COC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)Oc1cccc(c1)C1COC2(C1)CCN(CC2)C(=O)ON1C(=O)CCC1=O

CN(C1COC2(C1)CCN(CC2)C(=O)ON1C(=O)CCC1=O)C(=O)C(C)(C)C

CN(C1COC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(=O)C(C)(C)C

FC(F)c1ccc(OC2CC3(C2)CCN(CC3)C(=O)ON2C(=O)CCC2=O)cn1

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2ccc(cc2N2CCOCC2)C(F)(F)F)CC1

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)OCc1ccccc1Cl |r|

Cc1cc(ccc1CN1CCN(CC1)C(=O)n1ccc(n1)C(O)=O)-c1ccccc1

NC(=O)c1ccn(n1)C(=O)N1CC2CN(Cc3ccc(cc3C(F)(F)F)N3CCOCC3)CC2C1

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cc(Cl)cc(Oc3ccc(Cl)cc3)c2)CC1

OC(=O)c1nn(cc1Cl)C(=O)N1CC2CN(Cc3ccc(cc3C(F)(F)F)-c3cnc4ccccn34)CC2C1

NC(=O)c1ccn(n1)C(=O)N1CCC2(CCCN2Cc2cc3ccc(cc3s2)C(F)(F)F)CC1

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cccc(c1)-c1ncco1 |r|

OC(=O)c1nn(cc1Cl)C(=O)N1CCC2(CCN(Cc3cccc(Cl)c3C(F)(F)F)C2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCC(CC1)OCc1cc(Cl)cc(Oc2ccc(Cl)cc2)c1

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1ccccc1-n1cccn1 |r|

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCCN2Cc2cc(cc(c2)C(F)(F)F)-n2cccn2)CC1

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)OCc1cccc(c1)C1CCCC1 |r|

NC(=O)c1ccn(n1)C(=O)N1CC2CN(Cc3ccc(cc3C(F)(F)F)C3(CCOCC3)C(O)=O)CC2C1

CC(C)(O)CN(Cc1cccc(c1)C(F)(F)F)C1CCN(CC1)C(=O)n1ccc(n1)C(N)=O

CC(C)(O)COc1cccc(CN2CCN(CC2)C(=O)n2ccc(n2)C(N)=O)c1Cl

CC(C)(O)COc1cccc(CO[C@@H]2C[C@H]3CN(C[C@H]3C2)C(=O)n2ccc(n2)C(O)=O)c1Cl |r|

OC(=O)c1ccn(n1)C(=O)N1CCC(CC1)OCc1cc(F)cc(Cl)c1

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cc(Cl)ccc3C(F)(F)F)C2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2ccc(Oc3ccc(Cl)cc3)cc2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cccc(Oc3ccc(F)cc3)c2)CC1

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)OCc1cc(F)cc(Cl)c1 |r|

CN(CC1CCN(CC1)C(=O)n1cc(Cl)c(n1)C(O)=O)Cc1cc(Cl)ccc1C(F)(F)F

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)OCc1ccc(Oc2ccc(Cl)cc2)cc1 |r|

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cccc(Oc3cc(ccn3)C(F)(F)F)c2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cccc(Oc3ccc(cn3)C(F)(F)F)c2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cc(Cl)cc(c3)C(F)(F)F)C2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3ccc(cc3Cl)C(F)(F)F)C2)CC1

CN(Cc1cc(Cl)ccc1C(F)(F)F)C1CCN(CC1)C(=O)n1ccc(n1)C(O)=O

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2ccc(cc2N2CCCC2)C(F)(F)F)CC1

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cccc(Oc3cccc(Cl)c3)c2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cccc(Oc3ccccc3Cl)c2)CC1

CC1CN(Cc2ccc(cc2C)-c2ccccc2)CCN1C(=O)n1ccc(n1)C(O)=O

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2ccc(cc2N2CC[C@H](F)C2)C(F)(F)F)CC1 |r|

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCCN2Cc2ccc(cc2N2CCCC2)C(F)(F)F)CC1

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cccc(Oc3ccc(Cl)cc3)c2)CC1

NC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cc(Cl)ccc3C(F)(F)F)C2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2ccc(cc2N2CCCCC2)C(F)(F)F)CC1

CN(Cc1cc(Cl)ccc1C(F)(F)F)C1CCN(CC1)C(=O)n1cc(Cl)c(n1)C(O)=O

OC(=O)c1ccn(n1)C(=O)N1CC2CN(Cc3cccc(Oc4ccc(Cl)cc4)c3)CC2C1

OC(=O)c1ccn(n1)C(=O)N1CC2CN(Cc3cc(Cl)cc(c3)C(F)(F)F)CC2C1

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cccc(c1)-c1ccccc1 |r|

CN(Cc1ccccc1Cl)[C@@H]1C[C@H]2CN(C[C@H]2C1)C(=O)n1cc(Cl)c(n1)C(N)=O |r|

Cc1cn(nc1C(O)=O)C(=O)N1CCN(Cc2cccc(Oc3ccc(Cl)cc3)c2)CC1

Cc1cn(nc1C(O)=O)C(=O)N1CCC2(CCN(Cc3cc(Cl)ccc3C(F)(F)F)C2)CC1

Cc1cn(nc1C(O)=O)C(=O)N1CCC2(CN(Cc3cc(Cl)ccc3C(F)(F)F)C2)CC1

OC(=O)c1nn(cc1Cl)C(=O)N1CCN(Cc2cccc(Oc3ccc(Cl)cc3)c2)CC1

OC(=O)c1nn(cc1Cl)C(=O)N1CCC2(CCN(Cc3cc(Cl)ccc3C(F)(F)F)C2)CC1

OC(=O)c1nn(cc1Cl)C(=O)N1CCC2(CN(Cc3cc(Cl)ccc3C(F)(F)F)C2)CC1

OC(=O)c1nn(cc1Cl)C(=O)N1CC2CN(Cc3cc(Cl)ccc3Cl)CC2C1

OC(=O)c1nn(cc1Cl)C(=O)N1CC2CN(Cc3cccc(Oc4ccc(Cl)cc4)c3)CC2C1

OC(=O)c1nn(cc1Cl)C(=O)N1CCC2(CCN(Cc3ccc(cc3C(F)(F)F)N3CCCC3)C2)CC1

OC(=O)c1nn(cc1Cl)C(=O)N1CCC2(CCCN2Cc2cc3ccc(cc3s2)C(F)(F)F)CC1

OC(=O)c1nn(cc1Cl)C(=O)N1CC2CN(Cc3ccc(cc3C(F)(F)F)N3CCCC3)CC2C1

OC(=O)c1nn(cc1C(F)(F)F)C(=O)N1CC2CC(CC2C1)OCc1ccccc1Cl

NC(=O)c1ccn(n1)C(=O)N1CCN(Cc2ccc(cc2)C#C)CC1

OC(=O)c1nn(cc1C(F)(F)F)C(=O)N1CCC2(CCN(Cc3cc(Cl)ccc3C(F)(F)F)C2)CC1

OC(=O)c1nn(cc1C(F)(F)F)C(=O)N1CCC2(CCCN2Cc2cc3ccc(cc3s2)C(F)(F)F)CC1

Cc1cc(CN2CCC3(C2)CCN(CC3)C(=O)n2ccc(n2)C(O)=O)ccc1C(F)(F)F

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)OCc1cccc(c1)C(F)(F)F |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)OCc1cccc(Oc2ccc(Cl)cc2)c1 |r|

Cc1c(CO[C@@H]2C[C@H]3CN(C[C@H]3C2)C(=O)n2ccc(n2)C(O)=O)cccc1C(F)(F)F |r|

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cc(F)cc(Oc3ccc(Cl)cc3)c2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cc(Cl)cc(Cl)c3)C2)CC1

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@@H](C[C@@H]2C1)Oc1cccc(c1)-c1ccccc1 |r|

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2ccc(cc2C(F)(F)F)N2CCCC2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3ccc(cc3C(F)(F)F)-c3ccccc3)C2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3ccc(Cl)cc3N3CCCC3)C2)CC1

Cc1cc(CO[C@@H]2C[C@H]3CN(C[C@H]3C2)C(=O)n2ccc(n2)C(O)=O)ccc1C(F)(F)F |r|

NC(=O)c1ccn(n1)C(=O)N1CCN(Cc2ccc(cc2N2CCCC2)C(F)(F)F)CC1

NC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cnccc2C(F)(F)F)CC1

CN(Cc1cccc(c1)C(F)(F)F)C1CCN(CC1)C(=O)n1ccc(n1)C(N)=O

NC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3ccc(cc3C(F)(F)F)N3CCCC3)C2)CC1

NC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cc(Cl)cc(c3)C(F)(F)F)C2)CC1

NC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3ccc(cc3Cl)N3CCOCC3)C2)CC1

NC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cccc(c2N2CCOCC2)C(F)(F)F)CC1

CN(Cc1ccccc1Cl)[C@@H]1C[C@H]2CN(C[C@H]2C1)C(=O)n1ccc(n1)C(N)=O |r|

NC(=O)c1ccn(n1)C(=O)N1CC2CN(Cc3cc(Cl)cc(c3)C(F)(F)F)CC2C1

NC(=O)c1ccn(n1)C(=O)N1CC2CN(Cc3cc(Cl)ccc3Cl)CC2C1

CN(Cc1ccccc1C(F)(F)F)[C@H]1C[C@H]2CN(C[C@H]2C1)C(=O)n1ccc(n1)C(N)=O |r|

CN(Cc1ccc(cc1)C(F)(F)F)[C@H]1C[C@H]2CN(C[C@H]2C1)C(=O)n1ccc(n1)C(N)=O |r|

CN(Cc1ccccc1Cl)[C@H]1C[C@H]2CN(C[C@H]2C1)C(=O)n1ccc(n1)C(N)=O |r|

NC(=O)c1ccn(n1)C(=O)N1CC2CN(Cc3cccc(c3)C(F)(F)F)CC2C1

CN(CC1CCN(CC1)C(=O)n1ccc(n1)C(O)=O)Cc1cc(Cl)ccc1C(F)(F)F

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cccc(Oc4ccc(Cl)cc4)c3)C2)CC1

CC(C)(O)COc1cccc(CN2CCN(CC2)C(=O)n2ccc(n2)C(O)=O)c1Cl

C[C@H]1CN(Cc2cccc(OCC(C)(C)O)c2Cl)CCN1C(=O)n1ccc(n1)C(O)=O |r|

C[C@@H]1CN(Cc2cccc(OCC(C)(C)O)c2Cl)CCN1C(=O)n1ccc(n1)C(N)=O |r|

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cc(Cl)ccc3C(F)(F)F)CC2)CC1

Cc1cccc(O[C@@H]2C[C@H]3CN(C[C@H]3C2)C(=O)n2ccc(n2)C(O)=O)c1 |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cccc(c1)C1CC1 |r|

CC(C)c1cccc(O[C@@H]2C[C@H]3CN(C[C@H]3C2)C(=O)n2ccc(n2)C(O)=O)c1 |r|

CC(C)c1ccccc1O[C@@H]1C[C@H]2CN(C[C@H]2C1)C(=O)n1ccc(n1)C(O)=O |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cc(F)cc(Cl)c1 |r|

OC(=O)c1ccn(n1)C(=O)N1CCC(CC1)OCc1cccc(c1)C(F)(F)F

C[C@@H]1CN(Cc2ccc(cc2)-c2ccccc2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cc(Cl)cc(Cl)c1 |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cccc(c1)C(F)(F)F |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cccc(c1)C1CCCC1 |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cnccc1C(F)(F)F |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cccc(c1)N1CCCC1 |r|

Cc1c(COC2CCN(CC2)C(=O)n2ccc(n2)C(O)=O)cccc1C(F)(F)F

Cc1ccc(COC2CCN(CC2)C(=O)n2ccc(n2)C(O)=O)cc1C(F)(F)F

Cc1ccc(Cl)cc1CN1CCC2(C1)CCN(CC2)C(=O)n1ccc(n1)C(O)=O

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1ccccc1-c1ccccc1 |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1ccc(cc1)-c1ccccc1 |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cccc(c1)-c1cccnc1 |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cccc(c1)-c1ccccn1 |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cccc(c1)-c1ccncc1 |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1ccccc1-c1cccnc1 |r|

C[C@@H]1CN(Cc2ccc(cc2C)-c2ccccc2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

C[C@H]1CN(Cc2ccc(cc2C)-c2ccccc2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

C[C@@H]1CN(Cc2ccc(c(C)c2)-c2ccccc2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cccc(c1)-c1ncccn1 |r|

C[C@@H]1CN(Cc2ccc(cc2C)-c2ccccn2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

Cc1ccc(Oc2cccc(CN3CCN(CC3)C(=O)n3ccc(n3)C(O)=O)c2)cc1

Cc1cn(nc1C(O)=O)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)OCc1cc(F)cc(Cl)c1 |r|

C[C@@H]1CN(Cc2ccc(cc2F)-c2ccccc2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

Cc1cc(O[C@@H]2C[C@H]3CN(C[C@H]3C2)C(=O)n2ccc(n2)C(O)=O)ccc1C(F)(F)F |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@@H](C[C@@H]2C1)OCc1cccc(c1)C(F)(F)F |r|

Cc1c(O[C@@H]2C[C@H]3CN(C[C@H]3C2)C(=O)n2ccc(n2)C(O)=O)cccc1C(F)(F)F |r|

C[C@@H]1C[C@@H](CCN1C(=O)n1ccc(n1)C(N)=O)N(C)Cc1cccc(c1)C(F)(F)F |r|

CN(Cc1cccc(c1)C(F)(F)F)C1(C)CCN(CC1)C(=O)n1ccc(n1)C(N)=O

C[C@H]1C[C@@H](CCN1C(=O)n1ccc(n1)C(N)=O)N(C)Cc1cccc(c1)C(F)(F)F |r|

C[C@@H]1C[C@H](CCN1C(=O)n1ccc(n1)C(N)=O)N(C)Cc1cccc(c1)C(F)(F)F |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cccc(c1)-c1nccs1 |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cccc(c1)-c1cncs1 |r|

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cccc(Oc3cncc(F)c3)c2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cccc(Oc3ccc(F)cn3)c2)CC1

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cccc(c1)C1CCOCC1 |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1ccccc1C1CCOCC1 |r|

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cc(Cl)cc(c2)-c2cncnc2)CC1

C[C@H]1CN(Cc2cc(Cl)cc(c2)C(F)(F)F)CCN1C(=O)n1ccc(n1)C(N)=O |r|

C[C@@H]1CN(Cc2cc(Cl)cc(c2)C(F)(F)F)CCN1C(=O)n1ccc(n1)C(N)=O |r|

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2ccc(Cl)c(c2)-c2nccs2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCC(CC1)OCc1cc(Cl)cc(c1)C(F)(F)F

OC(=O)c1ccn(n1)C(=O)N1CCC(CC1)OCc1ccc(Cl)c(c1)C(F)(F)F

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)OCc1cccc(c1)-c1ccccc1 |r|

Cc1cn(nc1C(O)=O)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cccc(c1)-c1ccccc1 |r|

COc1cc(ccc1CN1CCN([C@H](C)C1)C(=O)n1ccc(n1)C(O)=O)-c1ccccc1 |r|

NC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cccc(c3)C(F)(F)F)C2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cc(Cl)ccc3Cl)C2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cccc(Cl)c3Cl)C2)CC1

COc1ccccc1Oc1cccc(CN2CCN(CC2)C(=O)n2ccc(n2)C(O)=O)c1

Cc1c(CO[C@H]2C[C@H]3CN(C[C@H]3C2)C(=O)n2ccc(n2)C(O)=O)cccc1C(F)(F)F |r|

Cc1cn(nc1C(O)=O)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)OCc1cccc(c1)C(F)(F)F |r|

C[C@@H]1CN(Cc2ccc(cc2Cl)-c2ccccc2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

C[C@@H]1CN(Cc2cccc(Oc3ccc(F)cc3)c2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

C[C@H]1CN(Cc2cccc(Oc3ccc(F)cc3)c2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

OC(=O)c1nn(cc1Cl)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)OCc1cc(F)cc(Cl)c1 |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cc(Cl)ccc1C(F)(F)F |r|

C[C@@H]1CN(Cc2ccc(Cl)c(c2)-c2nccs2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

Cc1cc(CN2CCCC22CCN(CC2)C(=O)n2ccc(n2)C(O)=O)cc(c1)C(F)(F)F

OC(=O)c1nn(cc1Cl)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1cccc(c1)-c1ccccc1 |r|

Cc1cn(nc1C(O)=O)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)OCc1cccc(c1C)C(F)(F)F |r|

OC(=O)c1ccn(n1)C(=O)N1CCC(CC1)Oc1ccc(cc1N1CCCC1)C(F)(F)F

OC(=O)c1ccn(n1)C(=O)N1CCC(CC1)Oc1cc(cc(c1)C(F)(F)F)N1CCCC1

NC(=O)c1ccn(n1)C(=O)N1CCC(CC1)N(CC(O)=O)Cc1cccc(c1)C(F)(F)F

C[C@H]1CN(Cc2cccc(Oc3ccc(Cl)cc3)c2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

C[C@@H]1CN(Cc2cccc(Oc3ccccc3Cl)c2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

OC(=O)c1ccn(n1)C(=O)N1CCC2(CN(Cc3cc(Cl)ccc3C(F)(F)F)C2)CC1

OC(=O)c1nn(cc1Cl)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)OCc1cccc(c1)C(F)(F)F |r|

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)Oc1ccc(Cl)c(c1)-c1nccs1 |r|

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cc(F)cc(Oc3ccccc3Cl)c2)CC1

OC(=O)c1nn(cc1Cl)C(=O)N1CCN(Cc2cccc(Oc3ccc(F)cc3)c2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cc(F)cc(Oc3cccc(Cl)c3)c2)CC1

OC(=O)c1nn(cc1Cl)C(=O)N1CCN(Cc2cc(Cl)cc(c2)-c2cncnc2)CC1

C[C@@H]1CN(Cc2ccc(cc2N2CCCC2)C(F)(F)F)CCN1C(=O)n1ccc(n1)C(N)=O |r|

C[C@@H]1CN(Cc2ccc(cc2N2CCCC2)C(F)(F)F)CCN1C(=O)n1ccc(n1)C(O)=O |r|

C[C@H]1CN(Cc2ccc(cc2C(F)(F)F)N2CCCC2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

C[C@@H]1CN(Cc2ccc(cc2C(F)(F)F)N2CCCC2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

OC(=O)c1ccn(n1)C(=O)N1CCC(CC1)OCc1cc(cc(c1)C(F)(F)F)N1CCCC1

O[C@@H]1CCN(C1)c1cc(ccc1CN1CCN(CC1)C(=O)n1ccc(n1)C(O)=O)C(F)(F)F |r|

C[C@H]1C[C@@H](CCN1C(=O)n1ccc(n1)C(O)=O)OCc1cccc(Oc2ccc(Cl)cc2)c1 |r|

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cc(Cl)cc(Cl)c3Cl)C2)CC1

OC(=O)c1nn(cc1Cl)C(=O)N1CCC2(CCN(Cc3cc(Cl)cc(Cl)c3)C2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cccc(c3Cl)C(F)(F)F)C2)CC1

Cc1c(CO[C@@H]2C[C@H]3CN(C[C@H]3C2)C(=O)n2cc(Cl)c(n2)C(O)=O)cccc1C(F)(F)F |r|

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cc(Cl)ccc3N3CCCC3)C2)CC1

OC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)OCc1ccc(Cl)c(c1)-c1nccs1 |r|

Cc1cn(nc1C(O)=O)C(=O)N1CCN(Cc2cc(F)cc(Oc3ccc(Cl)cc3)c2)CC1

C[C@H]1CN(Cc2cc(F)cc(Oc3ccc(Cl)cc3)c2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

C[C@@H]1CN(Cc2cc(F)cc(Oc3ccc(Cl)cc3)c2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

C[C@H]1CN(Cc2cc(F)cc(Oc3ccccc3Cl)c2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

C[C@@H]1CN(Cc2ccc(cc2C(F)(F)F)-c2ccccc2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cccc(Oc3cnccc3C(F)(F)F)c2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cccc(Oc3cccc(n3)C(F)(F)F)c2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cccc(Oc3ccnc(c3)C(F)(F)F)c2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cccc(Oc3ccncc3C(F)(F)F)c2)CC1

OC(=O)c1nn(cc1Cl)C(=O)N1CC2CN(Cc3cc(Cl)cc(c3)C(F)(F)F)CC2C1

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cccc(c3Cl)-c3ccccc3)C2)CC1

C[C@@H]1CC[C@@H](C)N1c1cc(ccc1CN1CCN(CC1)C(=O)n1ccc(n1)C(O)=O)C(F)(F)F |r|

C[C@H]1CC[C@H](C)N1c1cc(ccc1CN1CCN(CC1)C(=O)n1ccc(n1)C(O)=O)C(F)(F)F |r|

C[C@@H]1CN(Cc2ccc(cc2N2CC[C@H](F)C2)C(F)(F)F)CCN1C(=O)n1ccc(n1)C(O)=O |r|

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3ccc(Cl)c(c3)-c3nccs3)C2)CC1

OC(=O)c1nn(cc1Cl)C(=O)N1CCN(Cc2ccc(cc2C(F)(F)F)N2CCCC2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCCN2Cc2ccc(Cl)cc2N2CCCCC2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cc(Cl)ccc3OC(F)(F)F)C2)CC1

C[C@H]1CN(Cc2cccc(Oc3cc(ccn3)C(F)(F)F)c2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

C[C@@H]1CN(Cc2cccc(Oc3cc(ccn3)C(F)(F)F)c2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

C[C@H]1CN(Cc2cccc(Oc3ccc(cn3)C(F)(F)F)c2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

C[C@@H]1CN(Cc2cccc(Oc3ccc(cn3)C(F)(F)F)c2)CCN1C(=O)n1ccc(n1)C(O)=O |r|

OC(=O)c1nn(cc1Cl)C(=O)N1CCN(Cc2cc(F)cc(Oc3ccc(Cl)cc3)c2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2ccc(cc2N2CC3CCC(C2)O3)C(F)(F)F)CC1

CN(Cc1cc(cc(c1)C(F)(F)F)N1CCCC1)C1(C)CCN(CC1)C(=O)n1ccc(n1)C(O)=O

CN(Cc1cc(ccc1N1CCCC1)C(F)(F)F)C1(C)CCN(CC1)C(=O)n1ccc(n1)C(O)=O

CN(Cc1ccc(c(c1)N1CCCC1)C(F)(F)F)C1(C)CCN(CC1)C(=O)n1ccc(n1)C(O)=O

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCCN2Cc2ccc(Cl)cc2N2CCC(F)CC2)CC1

OC(=O)c1nn(cc1Cl)C(=O)N1CCC2(CCN(Cc3cc(Cl)cc(c3)C(F)(F)F)C2)CC1

NC(=O)c1ccn(n1)C(=O)N1CCC2(CCCN2C(=O)c2cc3ccc(cc3s2)C(F)(F)F)CC1

NC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(C2)C(=O)c2cc3ccc(cc3s2)C(F)(F)F)CC1

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cc(ccc3C(F)(F)F)N3CCCC3)C2)CC1

C[C@@H]1CN(Cc2ccc(cc2N2CC3COCC3C2)C(F)(F)F)CCN1C(=O)n1ccc(n1)C(O)=O |r|

NC(=O)c1ccn(n1)C(=O)N1CC2CN(Cc3ccc(cc3C(F)(F)F)C3(O)CCOCC3)CC2C1

CN(Cc1ccc(cc1N1CCCCC1)C(F)(F)F)C1(C)CCN(CC1)C(=O)n1ccc(n1)C(O)=O

CN(Cc1ccc(cc1N1CCCC1)C(F)(F)F)C1(C)CCN(CC1)C(=O)n1cc(C)c(n1)C(O)=O

OC(=O)c1nn(cc1Cl)C(=O)N1CCN(Cc2cccc(Oc3cc(ccn3)C(F)(F)F)c2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCCN2Cc2cc(cc(c2)C(F)(F)F)-c2cncnc2)CC1

C[C@@H]1CC[C@@H](C)N1c1cc(ccc1CN(C)C1(C)CCN(CC1)C(=O)n1ccc(n1)C(O)=O)C(F)(F)F |r|

C[C@H]1CC[C@H](C)N1c1cc(ccc1CN(C)C1(C)CCN(CC1)C(=O)n1ccc(n1)C(O)=O)C(F)(F)F |r|

OC(=O)c1nn(cc1C(F)(F)F)C(=O)N1CCN(Cc2cccc(Oc3cc(ccn3)C(F)(F)F)c2)CC1

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCCN2Cc2ccc(cc2N2CC3CCC(C2)O3)C(F)(F)F)CC1

OC(=O)c1ccn(n1)C(=O)N1CCC2(CCCN2Cc2cc(cc(c2)C(F)(F)F)N2CCC3(C2)CCOCC3)CC1

CNC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3ccc(Cl)cc3)C2)C1

CNC(=O)c1ccn(n1)C(=O)N1CC2CN(Cc3ccc(Cl)cc3)CC2C1

NC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cc(Cl)ccc3Cl)C2)C1

CNC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@@H](C[C@@H]2C1)N(C)Cc1ccccc1Cl |r|

CNC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cc(Cl)ccc3Cl)C2)C1

NC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cccc(c3)C(F)(F)F)C2)C1

CNC(=O)c1ccn(n1)C(=O)N1CC2CN(Cc3cc(Cl)ccc3Cl)CC2C1

CNC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@H](C[C@@H]2C1)N(C)Cc1ccccc1Cl |r|

CNC(=O)c1ccn(n1)C(=O)N1CC2CN(Cc3cccc(c3)C(F)(F)F)CC2C1

NC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cc(Cl)cc(c3)C(F)(F)F)C2)C1

CNC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@@H](C[C@@H]2C1)N(C)Cc1ccccc1C(F)(F)F |r|

CNC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3cc(Cl)cc(c3)C(F)(F)F)C2)C1

NC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3ccc(cc3C(F)(F)F)N3CCOCC3)C2)C1

CNC(=O)c1ccn(n1)C(=O)N1CC2CN(Cc3cc(Cl)cc(c3)C(F)(F)F)CC2C1

CNC(=O)c1ccn(n1)C(=O)N1CCC2(CCN(Cc3ccc(cc3C(F)(F)F)N3CCOCC3)C2)C1

CNC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@@H](C[C@@H]2C1)N(C)Cc1ccc(cc1)C(F)(F)F |r|

CNC(=O)c1ccn(n1)C(=O)N1CC2CN(Cc3ccc(cc3C(F)(F)F)N3CCOCC3)CC2C1

CN(C)C(=O)c1ccn(n1)C(=O)N1CCN(Cc2ccc(cc2N2CCOCC2)C(F)(F)F)CC1

C[C@H]1CN(Cc2cccc(Oc3ccc(Cl)cc3)c2)CCN1C(=O)n1cc(C)c(n1)C(O)=O |r|

OC(=O)c1nn(cc1Cl)C(=O)N1CCN(Cc2ccc(cc2N2CCCC2)C(F)(F)F)CC1

C[C@H]1CN(Cc2cccc(Oc3ccc(Cl)cc3)c2)CCN1C(=O)n1cc(c(n1)C(O)=O)C(F)(F)F |r|

CC(C)COc1cccc(O[C@@H]2C[C@H]3CN(C[C@H]3C2)C(=O)n2ccc(n2)C(O)=O)c1Cl |r|

C[C@H]1CN(Cc2cccc(OCC(C)(C)O)c2Cl)CCN1C(=O)n1ccc(n1)C(N)=O |r|

CC(C)(O)COc1cccc(O[C@@H]2C[C@H]3CN(C[C@H]3C2)C(=O)n2ccc(n2)C(O)=O)c1Cl |r|

OC(=O)c1ccn(n1)C(=O)N1CCN(Cc2cccc(c2N2CCOCC2)C(F)(F)F)CC1

OC(=O)CCCNc1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)CCCNc1cc(ccc1CN1CCC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)CCCNc1cc(ccc1CN1CC2CN(CC2C1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)CCCNc1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

OC(=O)CCCNc1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

OC(=O)CCCOc1cc(Cl)ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

OC(=O)COc1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)COc1cc(Cl)ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

OC(=O)CCCOc1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)CNc1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

CC(C)(CCNc1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)C(O)=O

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(Cl)cc(NCCOC=O)c2)CC1)C(F)(F)F

C[C@H](Nc1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)C(O)=O |r|

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(OC3CCC(CC3)OC=O)cc(c2)C(F)(F)F)CC1)C(F)(F)F |(9.77,3.53,;9.77,1.99,;11.31,1.99,;8.23,1.99,;9.77,.45,;8.44,-.32,;7.1,.45,;7.1,1.99,;5.77,-.32,;5.77,-1.86,;4.44,-2.63,;3.1,-1.86,;3.1,-3.4,;1.64,-3.88,;.73,-2.63,;1.64,-1.38,;1.24,.1,;-.25,.5,;-1.34,-.59,;-2.82,-.19,;-3.91,-1.28,;-5.4,-.88,;-5.8,.61,;-7.29,1.01,;-8.43,-.07,;-7.98,-1.57,;-6.49,-1.97,;-9.92,.33,;-11.01,-.76,;-12.49,-.36,;-3.22,1.3,;-2.13,2.39,;-.65,1.99,;-2.53,3.88,;-1.44,4.96,;-4.02,4.27,;-2.93,5.36,;3.1,-.32,;4.44,.45,;11.11,-.32,;12.44,-1.09,;11.88,1.01,;10.34,-1.65,)|

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2OC2CCC(CC2)OC=O)C(F)(F)F)CC1)C(F)(F)F |(8.57,-4.61,;7.24,-3.84,;6.47,-5.17,;8.01,-2.51,;5.91,-3.07,;4.57,-3.84,;3.24,-3.07,;3.24,-1.53,;1.91,-3.84,;1.91,-5.38,;.57,-6.15,;-.76,-5.38,;-.76,-6.92,;-2.23,-7.4,;-3.13,-6.15,;-2.23,-4.9,;-2.62,-3.42,;-4.11,-3.02,;-5.2,-4.11,;-6.69,-3.71,;-7.09,-2.22,;-6,-1.13,;-4.51,-1.53,;-3.42,-.44,;-3.82,1.05,;-2.73,2.14,;-3.13,3.62,;-4.63,4.08,;-5.71,2.93,;-5.31,1.45,;-5.03,5.56,;-6.52,5.96,;-6.92,7.45,;-8.57,-1.82,;-8.97,-.33,;-9.66,-2.91,;-10.06,-1.42,;-.76,-3.84,;.57,-3.07,;5.91,-1.53,;5.91,.01,;7.45,-1.53,;4.37,-1.53,)|

CS(=O)(=O)NC(=O)CCCNc1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(Cl)cc(OCCCOC=O)c2)CC1)C(F)(F)F

CS(=O)(=O)NC(=O)CCCOc1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

OC(=O)C1(CC1)Oc1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(Cl)cc2OCC2(CC2)OC=O)CC1)C(F)(F)F

OC(=O)CCNc1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F

OC(=O)C1(COc2cc(ccc2CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)CC1

OC(=O)C1(COc2ccc(F)cc2CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)CC1

OC(=O)C1(COc2cc(F)ccc2CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)CC1

OC(=O)C1(COc2c(F)cccc2CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)CC1

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cn3CCNCc3n2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cn3CCN(Cc3n2)C2CC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2c(nc3cccnn23)C2CC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cnc(s2)N2CCNCC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cncnc2N2CCCC2)CC1)C(F)(F)F

CC(C)n1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)c(n1)-c1ccccc1

CCc1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)n(n1)C1CCOCC1

CC(C)n1cc(C(=O)N2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(n1)-c1cccc(c1)N1CCCC1

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cn3CCN(Cc3n2)C2CCOC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc3c(Cl)cc(Cl)cc3[nH]2)CC1)C(F)(F)F

Cc1ccc2[nH]c(cc2c1)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cc3cc(Cl)cc(Cl)c3[nH]2)CC1)C(F)(F)F

Cc1ccc2sc(cc2c1)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CN(C(=O)c1cn2CCN(Cc2n1)C1CC1)C1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CN(C(=O)c1nnc2CN(CCn12)C1CC1)C1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC(C)(O)CN1CCn2cc(nc2C1)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC(C)N1CCn2cc(nc2C1)C(=O)N(C)C1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CN(C(=O)c1cn2CCN(Cc2n1)C1CCC1)C1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CN(C(=O)c1cn2CCN(CC(C)(C)O)Cc2n1)C1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)NC(=O)c1cn2CCN(Cc2n1)S(C)(=O)=O

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)C2(CC2)c2ncc(Cl)cn2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)C(F)(F)c2ncccn2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)C2(CC2)c2ncc(cn2)C2CC2)CC1)C(F)(F)F

CC(C)N1CCn2c(C1)nnc2C(=O)NC1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC(C)C(=O)N1CCn2cc(nc2C1)C(=O)NC1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)C2(CC2)c2cnc(nc2)C2CC2)CC1)C(F)(F)F

Fc1ccc(cc1)-c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)no1

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc3cc(Cl)ccc3s2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc3cc(ccc3s2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2sc3ccccc3c2Cl)CC1)C(F)(F)F

Cc1c(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)sc2ccccc12

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc3c(Cl)cccc3s2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2c[nH]c3cccc(Cl)c23)CC1)C(F)(F)F

COc1ccc(cc1)-c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)no1

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(on2)-c2ccc(Cl)cc2)CC1)C(F)(F)F

Cc1c(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)[nH]c2ccc(Cl)cc12

Cc1ccc2nc(Cl)c(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc2c1

CN(Cc1sc2ccccc2c1C)C1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3cc4cc(Cl)ccc4s3)C2)CC1)C(F)(F)F

Fc1ccc2[nH]c(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc2c1

COc1cccc2cc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)[nH]c12

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc3ccccc3n2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc3cc(Cl)ccc3n2)CC1)C(F)(F)F

Fc1ccc2nc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc2c1

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc3cccc(Cl)c3n2)CC1)C(F)(F)F

Cc1c(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)[nH]c2ccc(F)cc12

Cc1ccc2cc(sc2c1)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cc3ccc(Cl)cc3s2)CC1)C(F)(F)F

Cc1ccc2sc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc2c1

CN(Cc1cc2cc(Cl)ccc2s1)C1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

Cc1c([nH]c2c(C)cc(C)cc12)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3cccnc3)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3nccs3)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3cncnc3)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cn3ccccc3n2)CC1)C(F)(F)F

Cn1cc(cn1)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC(C)n1cc(cn1)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cnn(c2)-c2ccccc2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccccn3)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccncn3)C2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2nc3ccccc3s2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cc3ccccc3[nH]2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2ccc3occc3c2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cnn(c2)-c2ccc(Cl)cc2)CC1)C(F)(F)F

Cn1ccc(n1)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cc3ccccc3s2)CC1)C(F)(F)F

CC(C)n1ccc(n1)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2ccn(n2)-c2ccccc2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cc3ccccc3o2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2nc3ccccc3o2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2ccc3nccn3c2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2ccc3scnc3c2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2ccc3ocnc3c2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cnn(Cc3ccccc3)c2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2ccc3[nH]ccc3c2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2ccc3sccc3c2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2ccn(Cc3ccccc3)n2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2ccn(n2)-c2ccc(Cl)cc2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cc3cc(Cl)ccc3[nH]2)CC1)C(F)(F)F

Cc1c(sc2ccccc12)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cc3cc(Cl)ccc3s2)CC1)C(F)(F)F

Fc1cccc2cc(sc12)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cc3cccc(c3s2)C(F)(F)F)CC1)C(F)(F)F

Fc1ccc2sc(cc2c1)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cc3ccc(cc3s2)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cc3cc(ccc3s2)C(F)(F)F)CC1)C(F)(F)F

Fc1ccc2cc(sc2c1)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

Cc1c([nH]c2ccc(F)cc12)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cc3cccc(Cl)c3s2)CC1)C(F)(F)F

Fc1ccc2[nH]c(cc2c1)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

Cc1cccc2cc([nH]c12)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

Cc1c([nH]c2ccc(Cl)cc12)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc3cc(Cl)cc(Cl)c3[nH]2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cc3cc(Cl)c(Cl)cc3[nH]2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc3cc(Cl)c(Cl)cc3[nH]2)CC1)C(F)(F)F

CC(C)n1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(n1)-c1cccc(c1)C(O)=O

Cc1cc(Cl)c2nc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cn2c1

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cnc(Cl)nc2N2CCCC2)CC1)C(F)(F)F

OC(=O)Cn1cc(C(=O)N2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(n1)-c1cccc(Cl)c1

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cc(nc(Cl)n2)N2CCCC2)CC1)C(F)(F)F

Cn1cc(Cl)c(n1)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

Cc1cc(n2nc(C(=O)N3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)c(Cl)c2n1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cncnc2C(F)(F)F)CC1)C(F)(F)F

OC(=O)C1CCN(CC1)c1nc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F

Cc1c(C(=O)N2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(Cl)nn1C

Cn1cc(C(=O)N2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(Cl)n1

Cc1nc(C)c(o1)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

Cc1nc(C(=O)N2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(C)o1

Cc1ncoc1C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

Cc1c(Cl)c(nn1C)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cnc(s2)N2CCN(CC2)C2CC2)CC1)C(F)(F)F

Cn1cc(Cl)c(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)n1

Cc1nc2ccccn2c1C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cncnc2N2CCOCC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cnc3CNCCn23)CC1)C(F)(F)F

COc1ncc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)s1

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2c(nc3CCCCn23)C(F)(F)F)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cnc3ccccn23)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cnc3ncccn23)CC1)C(F)(F)F

Cc1nc2ccc(Cl)nn2c1C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

Cc1nc2cccnn2c1C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cnn3cccnc23)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cnn3ccc(Cl)nc23)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cnn3CCCNc23)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cnn3CCCCc23)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cnn3CCCOc23)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cc3ncccn3n2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cc3CNCCc3s2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2nc3NCCCn3n2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cn3CCN(CC4CC4)Cc3n2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cc3CN(CCn3n2)C2CC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cc3CN(CC4CC4)CCn3n2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cn3ccncc3n2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2nc3ncccn3n2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cn3CCN(Cc3n2)C2COC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)c2cn3CCN(Cc3n2)C2CCOCC2)CC1)C(F)(F)F

CN(C(=O)c1cnc2cccnn12)C1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

COCC(C)N1CCn2cc(nc2C1)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(CN2CCn3cc(nc3C2)C(=O)N2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)COC1

Cc1nn2cccnc2c1C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

Cc1nn2c(C)cc(C)nc2c1C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)NC(=O)c1cn2CCN(Cc2n1)C1CC1

CN(C(=O)C1(CC1)c1cnccn1)C1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)C2(CC2)c2cccnn2)CC1)C(F)(F)F

Fc1cnc(nc1)C1(CC1)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)NC(=O)c1cn2CCNCc2n1

CC(C)N1CCn2cc(nc2C1)C(=O)NC1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)NC(=O)c1cn2CCN(Cc2n1)C1CCC1

CC1(CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)NC(=O)c1cn2CCN(Cc2n1)C1COC1

CN(C(=O)c1cn2CCN(Cc2n1)C1COC1)C1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CN(C(=O)c1cn2CCNCc2n1)C1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC(C)C(=O)N1CCn2cc(nc2C1)C(=O)N(C)C1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CN(C(=O)c1cn2CCN(Cc2n1)C(=O)C1CC1)C1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC(=O)N1CCn2cc(nc2C1)C(=O)NC1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(CC1)C(=O)N1CCn2cc(nc2C1)C(=O)NC1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC(C)(C)C(=O)N1CCn2cc(nc2C1)C(=O)NC1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)NC(=O)c1cn2CCN(Cc2n1)C(=O)C1(F)CC1

CCC(C)(C)C(=O)N1CCn2cc(nc2C1)C(=O)NC1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC(C)Oc1cnc(nc1)C1(CC1)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

COc1cnc(cn1)C(F)(F)C(=O)N(C)C1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

COc1nccc(n1)C1(CC1)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)C2(CC2)c2ccnc(n2)C2CC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2C(=O)C2(CC2)c2nccc(n2)C(F)(F)F)CC1)C(F)(F)F

COc1ccnc(n1)C1(CC1)C(=O)N1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)NC(=O)c1nnc2CN(CCn12)C1CC1

CC1(CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)NC(=O)c1nnc2CN(CCn12)C1CCC1

CC(C)(O)CN1CCn2c(C1)nnc2C(=O)NC1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC1(CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)NC(=O)c1nnc2CN(CCn12)C1COC1

CC1(CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)NC(=O)c1nnc2CN(CCn12)C1CCOC1

CC1(CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)NC(=O)c1nnc2CN(CCn12)C1CCOCC1

CC1(CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)NC(=O)c1nnc2CNCCn12

COCCN(C(=O)C1(CC1)c1ncccn1)C1(C)CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

CC(C)(C)c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)n(n1)C1CCOCC1

CC(C)c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)n(n1)C1CCOCC1

CCc1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)n(n1)-c1ccccc1Cl

CC(C)c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)n(n1)-c1ccccc1Cl

CC(C)(C)c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)n(n1)-c1ccccc1Cl

CC(C)n1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)c(n1)-c1cccc(Cl)c1

CC(C)n1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(n1)-c1cccc(Cl)c1

CC(C)n1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(n1)-c1ccccc1F

CC(C)n1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(n1)-c1ccccc1Cl

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc3ccccc3s2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc3cc(Cl)ccc3[nH]2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cnc(s2)N2CCCC2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2csc(n2)-c2ccccc2)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cnc3ccccn23)CC1)C(F)(F)F

FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cnc3ccc(Cl)cn23)CC1)C(F)(F)F

FC(F)(F)c1cccc(OC2CC3(C2)CCN(CC3)C(=O)Oc2cncc(c2)C(F)(F)F)c1

FC(F)(F)c1cncc(OC(=O)N2CCC3(CN(Cc4ccc(Oc5cccc(Cl)c5)cc4)C3)CC2)c1

NC(=O)c1cncc(OC(=O)N2CCC3(CCN(Cc4cc(Cl)cc(c4)C(F)(F)F)C3)CC2)c1

NC(=O)c1cncc(OC(=O)N2CCC3(CCN(Cc4cc(Cl)ccc4C(F)(F)F)C3)CC2)c1

NC(=O)c1cncc(OC(=O)N2CCC3(CN(Cc4cccc(Oc5ccc(Cl)cc5)c4)C3)CC2)c1

CC(C)Oc1cc(CN2CCN(CC2)C(=O)Oc2cncc(N)c2)ccc1Cl

FC(F)(F)c1cncc(OC(=O)N2CCC3(CN(Cc4cccc(Oc5nc6ccccc6s5)c4)C3)CC2)c1

FC(F)(F)c1cncc(OC(=O)N2CCC3(CN(Cc4ccc(Oc5ccccc5Cl)cc4)C3)CC2)c1

FC(F)(F)c1cncc(OC(=O)N2CCC3(CN(Cc4cccc(Oc5ccccc5Cl)c4)C3)CC2)c1

FC(F)(F)c1cncc(OC(=O)N2CCC3(CN(Cc4cccc(Oc5cccc(Cl)c5)c4)C3)CC2)c1

FC(F)(F)c1cncc(OC(=O)N2CCC3(CN(Cc4cccc(Oc5cncnc5)c4)C3)CC2)c1

CC(C)Oc1cc(CN2CCN(CC2)C(=O)Oc2cncc(NS(C)(=O)=O)c2)ccc1Cl

CC1CCCN1c1ccc(CN2CCN(CC2)C(=O)Oc2cncc(c2)C(N)=O)c(OC(F)(F)F)c1

CC(C)Oc1ccc(CN2CCN(CC2)C(=O)Oc2cncc(c2)C(N)=O)c(OC(F)(F)F)c1

C[C@@H]1CN(Cc2cnccc2C(F)(F)F)CCN1C(=O)Oc1cncc(c1)C#N |r|

C[C@@H]1CN(Cc2cc(F)cc(c2)C(F)(F)F)CCN1C(=O)Oc1cncc(c1)C(N)=O |r|

C[C@@H]1CN(Cc2cccc(c2C)C(F)(F)F)CCN1C(=O)Oc1cc(cnc1C)C#N |r|

FC(F)(F)c1cncc(OC(=O)N2CCC3(CN(Cc4cc(Cl)cc(Oc5nc6ccccc6s5)c4)C3)CC2)c1

FC(F)(F)c1cncc(OC(=O)N2CCC3(CC(C3)Oc3cc(Cl)cc(Cl)c3)CC2)c1

FC(F)(F)c1cncc(OC(=O)N2CCC3(CC(C3)Oc3cccc(c3)C(=O)N3CCCC3)CC2)c1

FC(F)(F)c1cncc(OC(=O)N2CCC3(CC(C3)Oc3cc(Cl)ccc3Cl)CC2)c1

FC(F)(F)c1cncc(OC(=O)N2CCC3(CC(C3)Oc3ccc(cc3)-c3ccccc3)CC2)c1

FC(F)(F)c1cncc(OC(=O)N2CCC3(CC(C3)Oc3cccc(COc4ccc(Cl)cc4)c3)CC2)c1

FC(F)(F)c1cncc(OC(=O)N2CCC3(CN(Cc4ccc(Oc5ccc(Cl)cc5)cc4)C3)CC2)c1

FC(F)(F)c1cncc(OC(=O)N2CCC3(CN(Cc4cccc(Oc5ccc(Cl)cc5)c4)C3)CC2)c1

FC(F)(F)c1cncc(OC(=O)N2CCC3(CN(Cc4ccc(Oc5cncnc5)cc4)C3)CC2)c1

NC(=O)c1cncc(OC(=O)N2CCC3(CCN(Cc4ccc(Cl)c(Cl)c4)C3)CC2)c1

FC(F)(F)c1cncc(OC(=O)N2CCC3(CN(Cc4cccc(Oc5cncc(c5)C(F)(F)F)c4)C3)CC2)c1

FC(F)(F)c1cncc(OC(=O)N2CCC3(CN(Cc4cccc(Oc5ccc(nc5)C(F)(F)F)c4)C3)CC2)c1

FC(F)(F)c1cncc(OC(=O)N2CCC3(CN(Cc4cccc(Oc5cccc(Cl)c5)c4Cl)C3)CC2)c1

Fc1cncc(OC(=O)N2CCN(Cc3cc(Cl)ccc3C(F)(F)F)CC2)c1

FC(F)(F)c1ccc(Cl)cc1CN1CCN(CC1)C(=O)Oc1cncc(c1)C#N

FC(F)(F)c1cncc(OC(=O)N2CCN(Cc3cc(Cl)ccc3C(F)(F)F)CC2)c1

COc1ccc(CN2CCN(CC2)C(=O)Oc2cncc(F)c2)cc1C(F)(F)F

Fc1cncc(OC(=O)N2CCN(Cc3cnccc3C(F)(F)F)CC2)c1

CC(C)Oc1ccc(CN2CCN(CC2)C(=O)Oc2cncc(F)c2)c(C)c1

O=C(Oc1cncc(c1)C#N)N1CCN(Cc2cccc(Oc3ncccn3)c2)CC1

NC(=O)c1cncc(OC(=O)N2CCN(Cc3cc(Cl)cc(c3)C(N)=O)CC2)c1

CC(C)Oc1cc(CN2CCN(CC2)C(=O)Oc2cncc(NC(C)=O)c2)ccc1Cl

CC(C)Oc1cc(CN2CCN(CC2)C(=O)Oc2cncc(c2)C(N)=O)ccc1Cl

CC(C)Oc1cc(CN2CCN([C@H](C)C2)C(=O)Oc2cncc(c2)C(N)=O)ccc1Cl |r|

C[C@@H]1CN(Cc2cccc(c2C)C(F)(F)F)CCN1C(=O)Oc1cncc(c1)C(N)=O |r|

CC(C)Oc1cc(CN2CCN([C@H](C)C2)C(=O)Oc2cncc(N)c2)ccc1Cl |r|

CCOc1cc(OC2CCN(CC2)C(=O)Oc2cncc(c2)C(N)=O)ccc1Cl

C[C@@H]1CN(Cc2cc(Cl)cc(c2)C(F)(F)F)CCN1C(=O)Oc1cncc(c1)C(N)=O |r|

C[C@@H]1CN(Cc2cccc(c2Cl)C(F)(F)F)CCN1C(=O)Oc1cncc(c1)C(N)=O |r|

C[C@@H]1CN(Cc2cc(Cl)ccc2C(F)(F)F)CCN1C(=O)Oc1cncc(c1)C#N |r|

C[C@@H]1CN(Cc2cccc(c2C)C(F)(F)F)CCN1C(=O)Oc1cncc(c1)C#N |r|

C[C@@H]1CN(Cc2cccc(c2C)C(F)(F)F)CCN1C(=O)Oc1cncc(F)c1 |r|

Cc1c(F)cncc1OC(=O)N1CCN(Cc2cc(Cl)ccc2C(F)(F)F)CC1

Cc1c(OC(=O)N2CCN(Cc3cc(Cl)ccc3C(F)(F)F)CC2)cncc1C#N

C[C@@H]1CN(Cc2cccc(OC(F)(F)F)c2)CCN1C(=O)Oc1cncc(c1)C(N)=O |r|

C[C@@H]1CN(Cc2cccc(OC(F)(F)F)c2)CCN1C(=O)Oc1cncc(c1)C#N |r|

C[C@@H]1CN(Cc2cccc(OC(F)(F)F)c2)CCN1C(=O)Oc1cncc(F)c1 |r|

C[C@@H]1CN(Cc2cc(F)cc(c2)C(F)(F)F)CCN1C(=O)Oc1cncc(c1)C#N |r|

C[C@@H]1CN(Cc2cc(F)cc(c2)C(F)(F)F)CCN1C(=O)Oc1cncc(F)c1 |r|

C[C@@H]1CN(Cc2cccc(c2C)C(F)(F)F)CCN1C(=O)Oc1cncc(C#N)c1C |r|

C[C@@H]1CN(Cc2cccc(Oc3ncccn3)c2)CCN1C(=O)Oc1cncc(c1)C#N |r|

C[C@@H]1CN(Cc2cccc(c2)C(F)(F)F)CCN1C(=O)Oc1cncc(c1)C(N)=O |r|

C[C@@H]1CN(Cc2cc(F)cc(Cl)c2)CCN1C(=O)Oc1cncc(c1)C(N)=O |r|

C[C@H](N1CCN(CC1)C(=O)n1ccc(NS(C)(=O)=O)n1)c1ccc(Cl)c(c1)N1CCC(F)CC1 |r|

CC(=O)Nc1ccn(n1)C(=O)N1CCC2(CCCN2Cc2cc3cc(Cl)cc(Cl)c3[nH]2)CC1

CC(=O)Nc1ccn(n1)C(=O)N1CCC2(CCCN2Cc2cc3cc(ccc3[nH]2)C(N)=O)CC1

CC(=O)Nc1ccn(n1)C(=O)N1CC2CN(Cc3cccc(Oc4ccccc4Cl)c3)CC2C1

CC(=O)Nc1ccn(n1)C(=O)N1CCC2(CCCN2C(=O)c2ccc(Cl)c(c2)C2CC2)CC1

CC(=O)Nc1ccn(n1)C(=O)N1CCN(Cc2ccc(cc2C(F)(F)F)N2CC3COCC3C2)CC1

CC(=O)Nc1ccn(n1)C(=O)N1CCC2(CCN(Cc3ccc(cc3C(F)(F)F)N3CCCC3)C2)CC1

CC(=O)Nc1ccn(n1)C(=O)N1CCC2(CCN(Cc3cc(cc(c3)C3(CCCC3)C(O)=O)C(F)(F)F)C2)CC1

CC(C)(O)COc1cccc(CN2CCN(CC2)C(=O)n2ccc(NS(C)(=O)=O)n2)c1Cl

CC(=O)Nc1ccn(n1)C(=O)N1CCC2(CCCN2Cc2cc3cc(Cl)ccc3[nH]2)CC1

CC(=O)Nc1ccn(n1)C(=O)N1CCC2(CCCN2Cc2cc3cc(Cl)ccc3s2)CC1

CC(=O)Nc1ccn(n1)C(=O)N1CCC2(CCCN2Cc2cc3cc(Cl)c(Cl)cc3[nH]2)CC1

CN(Cc1cc(Cl)ccc1C(F)(F)F)[C@@H]1C[C@H]2CN(C[C@H]2C1)C(=O)n1ccc(NS(C)(=O)=O)n1 |r|

CS(=O)(=O)Nc1ccn(n1)C(=O)N1CCN(Cc2cc3ccc(cc3s2)C(F)(F)F)CC1

CS(=O)(=O)Nc1ccn(n1)C(=O)N1CCC2(CCN(Cc3ccc(Cl)cc3N3CCCC3)C2)CC1

CS(=O)(=O)Nc1ccn(n1)C(=O)N1CCC2(CCN(Cc3ccc(cc3N3C4CCC3COC4)C(F)(F)F)C2)CC1

CC(=O)Nc1ccn(n1)C(=O)N1CC2CN(Cc3ccc(cc3C(F)(F)F)N3CCCC3)CC2C1

CC(=O)Nc1ccn(n1)C(=O)N1CCN(Cc2ccc(cc2C)-c2ccccc2)CC1

CN(Cc1cc(cc(c1)C1(CCCC1)C(O)=O)C(F)(F)F)C1(C)CCN(CC1)C(=O)n1ccc(NC(C)=O)n1

C[C@@H](N1CCN(CC1)C(=O)n1ccc(NS(C)(=O)=O)n1)c1ccc(Cl)c(c1)N1CCC(F)CC1 |r|

CC(=O)Nc1ccn(n1)C(=O)N1CC2CN(Cc3cc(F)cc(Cl)c3)CC2C1

CC(=O)Nc1ccn(n1)C(=O)N1CC2CN(Cc3cc(Cl)cc(c3)C(F)(F)F)CC2C1

CS(=O)(=O)Nc1ccn(n1)C(=O)N1CCN(Cc2cccc(Oc3ccc(Cl)cc3)c2)CC1

CC(=O)Nc1ccn(n1)C(=O)N1CC2CN(Cc3ccc(Cl)c(c3)C(C)(C)O)CC2C1

CC(=O)Nc1ccn(n1)C(=O)N1CCC2(CCN(C2)C(=O)c2cc3ccc(cc3s2)C(F)(F)F)CC1

CC(=O)Nc1ccn(n1)C(=O)N1CC2CN(Cc3cc(Cl)cc(c3)N3CCCC3)CC2C1

CC(=O)Nc1ccn(n1)C(=O)N1CC2CN(Cc3cccc(Oc4ccccc4)c3)CC2C1

CC(=O)Nc1ccn(n1)C(=O)N1CCC2(CCN(Cc3cccc(c3)C(F)(F)F)C2)CC1

CC(=O)Nc1ccn(n1)C(=O)N1CCC2(CCN(Cc3cc(F)cc(Cl)c3)C2)CC1

C[C@H]1CN(Cc2ccc(c(c2)N2CC3COCC3C2)C(F)(F)F)CCN1C(=O)n1ccc(NS(C)(=O)=O)n1 |r|

C[C@H]1CN(CCN1Cc1ccc(c(c1)N1CC2COCC2C1)C(F)(F)F)C(=O)n1ccc(NS(C)(=O)=O)n1 |r|

C[C@@H]1CN(Cc2ccc(c(c2)N2CC3COCC3C2)C(F)(F)F)CCN1C(=O)n1ccc(NS(C)(=O)=O)n1 |r|

CS(=O)(=O)Nc1ccn(n1)C(=O)N1CCN(Cc2ccc(c(c2)N2CC3COCC3C2)C(F)(F)F)CC1

C[C@@H]1CN(CCN1Cc1ccc(c(c1)N1CC2COCC2C1)C(F)(F)F)C(=O)n1ccc(NS(C)(=O)=O)n1 |r|

CN(CC1CCN(CC1)C(=O)n1ccc(NS(C)(=O)=O)n1)Cc1cc(Cl)ccc1C(F)(F)F

C[C@H]1CN(CCN1Cc1ccc(c(c1)N1CCC(F)CC1)C(F)(F)F)C(=O)n1ccc(NS(C)(=O)=O)n1 |r|

C[C@@H]1CN(Cc2ccc(cc2C)-c2ccccc2)CCN1C(=O)n1ccc(NC(C)=O)n1 |r|

CC(C)(Oc1cc(Cl)ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(O)=O

CC(C)(Oc1c(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cccc1C(F)(F)F)C(O)=O

CC(C)(Oc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)C(O)=O

CC(C)(COc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)C(O)=O

CC(C)(COc1cc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F)C(O)=O

CC(C)(Oc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)C(=O)NS(=O)(=O)C1CC1

CC(C)(Oc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C1CC1)C(O)=O

CC(C)(Oc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C1(F)COC1)C(O)=O

CC(C)(Oc1cc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C#N)C(O)=O

CC(C)(Oc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)-c1ncco1)C(O)=O

Cc1ccc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(OC(C)(C)C(O)=O)c1F

CC(C)(Oc1c(F)cccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(O)=O

CC(C)(Oc1c(Cl)cccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(O)=O

Cc1ccc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(OC(C)(C)C(O)=O)c1Cl

Cc1ccc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(OC(C)(C)C(O)=O)c1

CC(C)(Oc1cc(F)ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(O)=O

CC(C)(Oc1ccccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(O)=O

Cc1cccc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1OC(C)(C)C(O)=O

CC(C)(Oc1c(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc(F)c1F)C(O)=O

CC(C)(Oc1cc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C1CC1)C(O)=O

CC(C)(Oc1ccc(cc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C1CC1)C(O)=O

CC(C)(Oc1cc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C1(F)COC1)C(O)=O

CC(C)(Oc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C#N)C(O)=O

CC(C)(Oc1ccc(C#N)c(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1)C(O)=O

COc1ccc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(OC(C)(C)C(O)=O)c1

CC(C)(Oc1cc(OC(F)(F)F)ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(O)=O

COc1cc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(OC(C)(C)C(O)=O)c1

CC(C)(Oc1cc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(OC(F)(F)F)c1)C(O)=O

CC(C)(Oc1cc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)-c1ncco1)C(O)=O

CC(C)(Oc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)-c1cnccn1)C(O)=O

CC(C)(Oc1cc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)-c1cnccn1)C(O)=O

CC(C)(Oc1ccc(OC(F)(F)F)c(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1)C(O)=O

CC(C)(Oc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)-c1ccccn1)C(O)=O

CC(C)(Oc1cc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)-c1ccccn1)C(O)=O

CC(C)(Oc1ccc(c(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1)-c1ccccn1)C(O)=O

C[C@@H](Oc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)C(O)=O |r|

C[C@H](Oc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)C(O)=O |r|

OC(=O)COc1cc(F)ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F

OC(=O)COc1cc(ccc1CN1CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C#N

OC(=O)COc1cc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(OC(F)(F)F)c1

CC(C)(Oc1cc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F)C(O)=O

Cc1ccc(CN2CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c(OCC(C)(C)C(O)=O)c1F

CC(=O)N(CCc1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)Cc1cccc(c1)C(F)(F)F

Fc1cccc(\C=C\c2ccc(cc2)C(=O)N2CCN(CC2)c2nc3ccccc3c(=O)[nH]2)c1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(Oc2ccccc2)cc1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1cccc(Oc2ccccc2)c1

FC(F)(F)Oc1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC(F)(F)Oc1cccc(c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2oc(nc2c1)-c1ccccc1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2nc(oc2c1)-c1ccccc1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2[nH]ccc2c1

Fc1ccc(cc1)-n1ccc2cc(ccc12)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)N1CCCC1

Ic1ccccc1CNc1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1cccc(OCc2ccccc2)c1

FC(F)(F)Oc1ccccc1CNc1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1cccc(OCC2CCCC2)c1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)-c1ccccc1

FC(F)(F)c1cccc(c1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Cc1nc(no1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1cc(no1)-c1ccccc1

Clc1cc(ccc1N1CCCC1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC(=O)N(CCc1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)Cc1ccccc1

FC(F)(F)c1cccc(c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2[nH]c(cc2c1)-c1ccccc1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)[C@@H]1C[C@@H]1c1ccccc1 |r|

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)[C@H]1C[C@@H]1c1ccccc1 |r|

FC(F)(F)Oc1cc(Br)cc(c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

C=CCOc1cccc(c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC(C)Cc1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC(C)c1nc(no1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Cc1nc2cc(ccc2n1-c1ccccc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC(F)(F)c1cc(cc(c1)C(F)(F)F)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC(F)(F)c1cccc(COCCc2ccc(cc2)C(=O)N2CCN(CC2)c2nc3ccccc3c(=O)[nH]2)c1

COc1cc(ccc1C(C)(C)C)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FS(F)(F)(F)(F)c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Fc1ccc(cc1)-n1ncc2cc(ccc12)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Cc1ccc(C)n1-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2cccnc2c1

FC(F)(F)Oc1ccc(cc1Br)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(Cn2cnc3ccccc23)cc1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)-c1nccs1

Cc1cnn(c1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Cc1ccn(n1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

COc1ccc2cc(oc2c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(COc2ccc3CCCc3c2)o1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1cc(-c2ccccc2)n(n1)-c1ccccc1

Clc1cccc(COc2ccc(cc2)C(=O)N2CCN(CC2)c2nc3ccccc3c(=O)[nH]2)c1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2[nH]c(nc2c1)-c1ccccc1

Fc1cccc(c1)-c1cc2cc(ccc2[nH]1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC(F)(F)c1cccc(c1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2cnccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2cnccc2c(=O)[nH]1)c1ccc2nc(oc2c1)-c1ccccc1

Fc1ccc(cc1)-n1ccc2cc(cnc12)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)N1CCCCC1

Fc1ccc(cc1)-n1cnc2cc(ccc12)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2nc(oc2c1)N1CCCCC1

Cn1c(nc2ccccc2c1=O)N1CCN(CC1)C(=O)c1ccc2nc(oc2c1)-c1ccccc1

FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC(F)(F)c1cnn(c1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC(F)(F)c1ccn(n1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)-c1noc(n1)C1CC1

Fc1cccc(c1)-c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Clc1cccc(c1)-c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC(F)(F)c1cccc(c1)-c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(OCc2ccccc2)cc1

CCN(CC)c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Clc1cccc(COc2cccc(c2)C(=O)N2CCN(CC2)c2nc3ccccc3c(=O)[nH]2)c1

Clc1cccc(COc2ccc(cc2Cl)C(=O)N2CCN(CC2)c2nc3ccccc3c(=O)[nH]2)c1

CC(C)(C)Cc1nc(no1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CN(c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)C(C)(C)C

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)N1CCc2ccccc12

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)N1CCC1

Clc1cc(ccc1C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)N1CCCC1

FC(F)(F)c1cc(ccc1OCc1cccc(Cl)c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Cc1cc(ccc1OCc1cccc(Cl)c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1cccc(c1)N1CCCC1

CC(C)(C)c1nc(no1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Clc1cccc(COc2ccc(cc2-c2ncc[nH]2)C(=O)N2CCN(CC2)c2nc3ccccc3c(=O)[nH]2)c1

Clc1cccc(COc2ccc(cc2C#N)C(=O)N2CCN(CC2)c2nc3ccccc3c(=O)[nH]2)c1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)C1CCCCC1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2nc(oc2c1)C1CCCCC1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)-c1ccccc1C#N

CCCCn1c(C)nc2cc(ccc12)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC(F)(F)c1cc(cc(c1)C(F)(F)F)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC(F)(F)Oc1cccc(c1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC(C)n1c(nc2cc(ccc12)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)C(F)(F)F

FC(F)(F)c1cccc(c1)-c1cncc(c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Fc1ccc(cc1F)-c1ccc(C(=O)N2CCN(CC2)c2nc3ccccc3c(=O)[nH]2)c(F)c1

COc1ccc(C)cc1-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Cc1c(oc2ccccc12)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

OCc1ccccc1-c1cccc(c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

OCc1cccc(c1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC(C)Oc1cc(Br)cc(c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

OCc1ccc(cc1)-c1cc(Cl)cc(c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC(C)COc1cc(ccc1Cl)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CCOc1cc(Br)cc(c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

OCc1ccccc1-c1cc(ccc1F)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Fc1cc(ccc1-c1cccc(c1)C(F)(F)F)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC(F)(F)Oc1ccccc1-c1cccc(c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC(F)(F)c1ccc2ncc(cc2c1)C(=O)N1CCN(CC1)c1nc2ccncc2c(=O)[nH]1

Cc1cc(C)c2cc([nH]c2c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CN(C)C(=O)c1ccc(cc1)-c1ccc(cc1C)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC(C)(C)c1ccc(cc1)-c1cc(ccn1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Clc1ccccc1Oc1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC(C)(C)c1cc(Cl)cc(c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)-c1cccc(OCc2ccccc2)c1

Cc1cccc(OCc2ccccc2)c1-c1cccc(c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

COc1ccc(cc1C(F)(F)F)-c1ccc(cc1C)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1c[nH]c2c(OCc3ccccc3)cccc12

Fc1cccc(F)c1-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2n(cnc2c1)C1CC1

CC(C)(C)c1ccc2cc([nH]c2c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CCOc1cc(ccc1Cl)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC1(C)CCN(CC1)c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC(F)(F)c1cccc2nc(cn12)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CN(C)C(=O)c1ccc(cc1)-c1cc(ccc1F)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Fc1cc(F)cc(c1)-c1cccc(c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Clc1ccc(cc1Cl)-c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Clc1ccc(cc1)-c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)N1CC2CCC1C2

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)N1CC2(CCC2)C1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)N1CCCCCC1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1cnc2nc(oc2c1)-c1ccccc1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)-c1nc(n[nH]1)C1CC1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)-c1nc(no1)C1CC1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1cc(C#N)c2nc(oc2c1)-c1ccccc1

Clc1ccc(cc1Cl)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(nc1)N1CCCC1

CC(C)(C)Cc1nc(no1)-c1cccc(c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)N1CC2(C1)CCCC2

CCc1nc(no1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Cc1nc(cs1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Fc1ccc(cc1F)-c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC(F)(F)c1ccc(cc1)-c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Fc1cc(ccc1C(F)(F)F)-c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Fc1ccc(cc1)-c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Fc1ccc2nc([nH]c(=O)c2c1)N1CCN(CC1)C(=O)c1ccc2nc(oc2c1)-c1ccccc1

Fc1ccc2c(c1)nc([nH]c2=O)N1CCN(CC1)C(=O)c1ccc2nc(oc2c1)-c1ccccc1

Fc1cc(ccc1Br)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cn1)N1CCCC1

Fc1cc(ccc1-c1cncc(c1)C(F)(F)F)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Cc1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC(F)(F)c1cc(cc2oc(nc12)-c1ccccc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Cc1cc(ccc1Br)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2nc(oc2c1)N1CCOCC1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)N1CCc2cccnc12

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)N1CCCC1c1ccccc1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2nc(oc2c1)-c1ccccn1

FC(F)(F)Cc1nc(no1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)N1CC2(COC2)C1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)-c1cccc(CC#N)c1

Fc1cc(ccc1-c1cccc(OC(F)(F)F)c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Cc1cc(ccc1-c1cccc(OC(F)(F)F)c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CCOc1cccc(c1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Clc1ccc2nc([nH]c(=O)c2c1)N1CCN(CC1)C(=O)c1ccc2nc(oc2c1)-c1ccccc1

FC(F)(F)c1cccc(CNCCc2ccc(cc2)C(=O)N2CCN(CC2)c2nc3ccccc3c(=O)[nH]2)c1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)C1(CCCC1)C#N

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1cc(N2CCOCC2)c2nc(oc2c1)-c1ccccc1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2nc(oc2c1)N1CC2(C1)CCCC2

FC1(F)CCC11CN(C1)c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CCCN(C)c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2nc(oc2c1)C1CCOCC1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2nc(oc2c1)-c1ccncc1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2nc(oc2c1)-c1cccnc1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2nc(oc2c1)-c1cccc(c1)C#N

CSc1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2nc(oc2c1)N1CCCC1

COC1CCN(CC1)c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

OC1CCN(CC1)c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC1CCN(C1)c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)N1CCC2(CCC2)C1

FC1(F)CCN(C1)c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC(O)C1CCN(C1)c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC(F)(F)C1CCN(CC1)c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc(cc1)N1CCC2(CC2)C1

Clc1ccnc(COc2ccc(cc2Cl)C(=O)N2CCN(CC2)c2nc3ccccc3c(=O)[nH]2)c1

Clc1cc(COc2ccc(cc2Cl)C(=O)N2CCN(CC2)c2nc3ccccc3c(=O)[nH]2)ccn1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1cccc(c1)-c1ccccc1

Clc1cccc(COc2ccc(cc2Cl)C(=O)N2CCN(CC2)c2nc3ccccc3c(=O)[nH]2)n1

FC(F)(F)c1cccc(c1)-c1cccc(c1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC(F)(F)c1cccc(Oc2ccc(cc2)C(=O)N2CCN(CC2)c2nc3ccccc3c(=O)[nH]2)c1

FC(F)(F)Cc1noc(n1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC1CCC(C)N1c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC1(F)CCN(CC1)c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Clc1cccc(OCc2ccc(cc2Cl)C(=O)N2CCN(CC2)c2nc3ccccc3c(=O)[nH]2)c1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2nc(sc2c1)-c1ccccc1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2nc(oc2c1)C1CCCO1

COCC1CCN(C1)c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC(F)(F)Cc1nc2cc(ccc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Cc1nc2c(OCc3cn[nH]c3)cc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC1(CC1)c1nc(no1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC(C)(CF)c1nc(no1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Clc1cc(ccc1C#N)-c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC(C)(C)c1noc(n1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC(C)(C)c1noc(n1)C12CC(C1)(C2)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Clc1cccc(c1)S(=O)(=O)N1CCC2(CCN(CC2)C(=O)N2CCN(CC2)c2nc3ccccc3c(=O)[nH]2)CC1

CC(C)(C)c1nc(no1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccc(Cl)cc2c(=O)[nH]1

CC1(C)CCN(C1)c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Cn1ccc(c1)-c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC(C)(CO)c1nc(no1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2nc(oc2c1)N1CCC2(C1)CCOCC2

COC1CCN(C1)c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

FC1(F)CC2(CN(C2)c2nc3ccc(cc3o2)C(=O)N2CCN(CC2)c2nc3ccccc3c(=O)[nH]2)C1

Cn1c(nc2ccccc2c1=O)N1CCN(CC1)C(=O)c1ccc2nc(oc2c1)N1CC2(C1)CCCC2

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2nc(oc2c1)N1CC2(CCC2)C1

OC1CC2(C1)CN(C2)c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC1(O)CCN(C1)c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC1(F)CCN(C1)c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC(C)(O)C1CCN(C1)c1nc2ccc(cc2o1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Cn1c(nc2ccccc2c1=O)N1CCN(CC1)C(=O)c1ccc2nc(oc2c1)N1CCC2(CCC2)C1

O=C(N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1)c1ccc2nc(oc2c1)N1CCC2(CCC2)C1

CC(C)(COCc1ccccc1)c1nc(no1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CC(C)(O)C#Cc1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

CCC1(CC)CCN(C1)c1ccc(cc1)C(=O)N1CCN(CC1)c1nc2ccccc2c(=O)[nH]1

Clc1ccc(cc1)S(=O)(=O)N1CCC2(CCN(C2)C(=O)N2CCN(CC2)c2nc3ccccc3c(=O)[nH]2)C1

Clc1cccc(c1)S(=O)(=O)N1CCC2(CCN(C2)C(=O)N2CCN(CC2)c2nc3ccccc3c(=O)[nH]2)C1

Clc1cccc(CN2CCC3(CCN(C3)C(=O)N3CCN(CC3)c3nc4ccccc4c(=O)[nH]3)C2)c1

O=C([C@H]1C[C@@]2(C1)COC(=O)N2)N1CCC2(CC(C2)c2ccccc2)CC1 |r,wU:2.1,wD:4.4,(-1.41,4.01,;-1.41,2.47,;-2.74,1.7,;-3.14,.21,;-4.63,.61,;-4.23,2.1,;-4.63,-.93,;-6.09,-1.41,;-7,-.16,;-8.48,.24,;-6.09,1.09,;-.07,1.7,;-.07,.16,;1.26,-.61,;2.6,.16,;2.99,-1.33,;4.48,-.93,;4.08,.56,;5.82,-1.7,;5.82,-3.24,;7.15,-4.01,;8.48,-3.24,;8.48,-1.7,;7.15,-.93,;2.6,1.7,;1.26,2.47,)|

CC(C)(C)c1cccc(c1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:21.23,wD:23.26,(9.82,-.16,;8.48,-.93,;8.48,.61,;9.82,-1.7,;7.15,-1.7,;7.15,-3.24,;5.82,-4.01,;4.48,-3.24,;4.48,-1.7,;5.82,-.93,;3.15,-.93,;1.66,-1.33,;1.26,.16,;2.75,.56,;-.07,-.61,;-1.41,.16,;-1.41,1.7,;-.07,2.47,;1.26,1.7,;-2.74,2.47,;-2.74,4.01,;-4.07,1.7,;-4.47,.21,;-5.96,.61,;-5.56,2.1,;-5.96,-.93,;-7.42,-1.41,;-8.33,-.16,;-9.82,.24,;-7.42,1.09,)|

Cc1ccc(cc1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.20,wD:20.23,(9.15,-4.01,;7.82,-3.24,;6.48,-4.01,;5.15,-3.24,;5.15,-1.7,;6.48,-.93,;7.82,-1.7,;3.81,-.93,;2.33,-1.33,;1.93,.16,;3.42,.56,;.59,-.61,;-.74,.16,;-.74,1.7,;.59,2.47,;1.93,1.7,;-2.07,2.47,;-2.07,4.01,;-3.41,1.7,;-3.8,.21,;-5.29,.61,;-4.89,2.1,;-5.29,-.93,;-6.76,-1.41,;-7.66,-.16,;-9.15,.24,;-6.76,1.09,)|

Cc1ccccc1C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.20,wD:20.23,(7.15,.61,;7.15,-.93,;8.48,-1.7,;8.48,-3.24,;7.15,-4.01,;5.82,-3.24,;5.82,-1.7,;4.48,-.93,;2.99,-1.33,;2.6,.16,;4.08,.56,;1.26,-.61,;-.07,.16,;-.07,1.7,;1.26,2.47,;2.6,1.7,;-1.41,2.47,;-1.41,4.01,;-2.74,1.7,;-3.14,.21,;-4.63,.61,;-4.23,2.1,;-4.63,-.93,;-6.09,-1.41,;-7,-.16,;-8.48,.24,;-6.09,1.09,)|

O=C([C@H]1C[C@@]2(C1)COC(=O)N2)N1CCC2(CC(C2)c2cccc(c2)C2CC2)CC1 |r,wU:2.1,wD:4.4,(-2.84,4.01,;-2.84,2.47,;-4.18,1.7,;-4.57,.21,;-6.06,.61,;-5.66,2.1,;-6.06,-.93,;-7.53,-1.41,;-8.43,-.16,;-9.92,.24,;-7.53,1.09,;-1.51,1.7,;-1.51,.16,;-.18,-.61,;1.16,.16,;1.56,-1.33,;3.04,-.93,;2.65,.56,;4.38,-1.7,;4.38,-3.24,;5.71,-4.01,;7.05,-3.24,;7.05,-1.7,;5.71,-.93,;8.38,-.93,;9.92,-.93,;9.15,.4,;1.16,1.7,;-.18,2.47,)|

CC(C)c1cccc(c1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:20.22,wD:22.25,(9.82,-1.7,;8.48,-.93,;8.48,.61,;7.15,-1.7,;7.15,-3.24,;5.82,-4.01,;4.48,-3.24,;4.48,-1.7,;5.82,-.93,;3.15,-.93,;1.66,-1.33,;1.26,.16,;2.75,.56,;-.07,-.61,;-1.41,.16,;-1.41,1.7,;-.07,2.47,;1.26,1.7,;-2.74,2.47,;-2.74,4.01,;-4.07,1.7,;-4.47,.21,;-5.96,.61,;-5.56,2.1,;-5.96,-.93,;-7.42,-1.41,;-8.33,-.16,;-9.82,.24,;-7.42,1.09,)|

Cc1cccc(c1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.20,wD:20.23,(9.15,-.93,;7.82,-1.7,;7.82,-3.24,;6.48,-4.01,;5.15,-3.24,;5.15,-1.7,;6.48,-.93,;3.81,-.93,;2.33,-1.33,;1.93,.16,;3.42,.56,;.59,-.61,;-.74,.16,;-.74,1.7,;.59,2.47,;1.93,1.7,;-2.07,2.47,;-2.07,4.01,;-3.41,1.7,;-3.8,.21,;-5.29,.61,;-4.89,2.1,;-5.29,-.93,;-6.76,-1.41,;-7.66,-.16,;-9.15,.24,;-6.76,1.09,)|

COc1cccc(c1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:19.21,wD:21.24,(9.2,.64,;9.2,-.9,;7.86,-1.67,;7.82,-3.24,;6.48,-4.01,;5.15,-3.24,;5.15,-1.7,;6.48,-.93,;3.81,-.93,;2.33,-1.33,;1.93,.16,;3.42,.56,;.59,-.61,;-.74,.16,;-.74,1.7,;.59,2.47,;1.93,1.7,;-2.07,2.47,;-2.07,4.01,;-3.41,1.7,;-3.8,.21,;-5.29,.61,;-4.89,2.1,;-5.29,-.93,;-6.76,-1.41,;-7.66,-.16,;-9.15,.24,;-6.76,1.09,)|

FC(F)(F)Oc1cccc(c1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:22.24,wD:24.27,(8.53,2.18,;8.53,.64,;10.07,.64,;6.99,.64,;8.53,-.9,;7.2,-1.67,;7.15,-3.24,;5.82,-4.01,;4.48,-3.24,;4.48,-1.7,;5.82,-.93,;3.15,-.93,;1.66,-1.33,;1.26,.16,;2.75,.56,;-.07,-.61,;-1.41,.16,;-1.41,1.7,;-.07,2.47,;1.26,1.7,;-2.74,2.47,;-2.74,4.01,;-4.07,1.7,;-4.47,.21,;-5.96,.61,;-5.56,2.1,;-5.96,-.93,;-7.42,-1.41,;-8.33,-.16,;-9.82,.24,;-7.42,1.09,)|

Cc1cccc(C2CC3(C2)CCN(CC3)C(=O)[C@H]2C[C@@]3(C2)COC(=O)N3)c1C |r,wU:17.18,wD:19.21,(9.15,-.93,;7.82,-1.7,;7.82,-3.24,;6.48,-4.01,;5.15,-3.24,;5.15,-1.7,;3.81,-.93,;2.33,-1.33,;1.93,.16,;3.42,.56,;.59,-.61,;-.74,.16,;-.74,1.7,;.59,2.47,;1.93,1.7,;-2.07,2.47,;-2.07,4.01,;-3.41,1.7,;-3.8,.21,;-5.29,.61,;-4.89,2.1,;-5.29,-.93,;-6.76,-1.41,;-7.66,-.16,;-9.15,.24,;-6.76,1.09,;6.48,-.93,;6.48,.61,)|

CC(C)(C)c1cccc(c1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)CCC(=O)N2 |r,wU:21.23,wD:23.26,(9.82,-1.7,;8.48,-.93,;8.48,.61,;9.82,-.16,;7.15,-1.7,;7.15,-3.24,;5.82,-4.01,;4.48,-3.24,;4.48,-1.7,;5.82,-.93,;3.15,-.93,;1.66,-1.33,;1.26,.16,;2.75,.56,;-.07,-.61,;-1.41,.16,;-1.41,1.7,;-.07,2.47,;1.26,1.7,;-2.74,2.47,;-2.74,4.01,;-4.07,1.7,;-4.47,.21,;-5.96,.61,;-5.56,2.1,;-5.96,-.93,;-7.42,-1.41,;-8.33,-.16,;-9.82,.24,;-7.42,1.09,)|

Cc1ccc(C2CC3(C2)CCN(CC3)C(=O)[C@H]2C[C@@]3(C2)COC(=O)N3)c(C)c1 |r,wU:16.17,wD:18.20,(9.15,-4.01,;7.82,-3.24,;7.82,-1.7,;6.48,-.93,;5.15,-1.7,;3.81,-.93,;2.33,-1.33,;1.93,.16,;3.42,.56,;.59,-.61,;-.74,.16,;-.74,1.7,;.59,2.47,;1.93,1.7,;-2.07,2.47,;-2.07,4.01,;-3.41,1.7,;-3.8,.21,;-5.29,.61,;-4.89,2.1,;-5.29,-.93,;-6.76,-1.41,;-7.66,-.16,;-9.15,.24,;-6.76,1.09,;5.15,-3.24,;3.81,-4.01,;6.48,-4.01,)|

CC(C)(C)c1cc(ccn1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:21.23,wD:23.26,(9.82,-.16,;8.48,-.93,;8.48,.61,;9.82,-1.7,;7.15,-1.7,;5.82,-.93,;4.48,-1.7,;4.48,-3.24,;5.82,-4.01,;7.15,-3.24,;3.15,-.93,;1.66,-1.33,;1.26,.16,;2.75,.56,;-.07,-.61,;-1.41,.16,;-1.41,1.7,;-.07,2.47,;1.26,1.7,;-2.74,2.47,;-2.74,4.01,;-4.07,1.7,;-4.47,.21,;-5.96,.61,;-5.56,2.1,;-5.96,-.93,;-7.42,-1.41,;-8.33,-.16,;-9.82,.24,;-7.42,1.09,)|

Cc1ccc(cc1C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2)C(C)(C)C |r,wU:18.20,wD:20.23,(3.21,-4.01,;4.54,-3.24,;5.88,-4.01,;7.21,-3.24,;7.21,-1.7,;5.88,-.93,;4.54,-1.7,;3.21,-.93,;1.72,-1.33,;1.32,.16,;2.81,.56,;-.01,-.61,;-1.35,.16,;-1.35,1.7,;-.01,2.47,;1.32,1.7,;-2.68,2.47,;-2.68,4.01,;-4.01,1.7,;-4.41,.21,;-5.9,.61,;-5.5,2.1,;-6.06,-.92,;-7.57,-1.24,;-8.34,.09,;-9.88,.09,;-7.31,1.24,;8.54,-.93,;9.88,-.16,;8.54,.61,;9.88,-1.7,)|

FC(F)(F)c1cccc(c1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:21.23,wD:23.26,(9.92,-.13,;8.59,-.9,;9.36,-2.24,;7.82,.43,;7.26,-1.67,;7.21,-3.24,;5.88,-4.01,;4.54,-3.24,;4.54,-1.7,;5.88,-.93,;3.21,-.93,;1.72,-1.33,;1.32,.16,;2.81,.56,;-.01,-.61,;-1.35,.16,;-1.35,1.7,;-.01,2.47,;1.32,1.7,;-2.68,2.47,;-2.68,4.01,;-4.01,1.7,;-4.41,.21,;-5.9,.61,;-5.5,2.1,;-6.06,-.92,;-7.57,-1.24,;-8.34,.09,;-9.88,.09,;-7.31,1.24,)|

CC(C)(C)c1cccc(n1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:21.23,wD:23.26,(9.88,-.16,;8.54,-.93,;8.54,.61,;9.88,-1.7,;7.21,-1.7,;7.21,-3.24,;5.88,-4.01,;4.54,-3.24,;4.54,-1.7,;5.88,-.93,;3.21,-.93,;1.72,-1.33,;1.32,.16,;2.81,.56,;-.01,-.61,;-1.35,.16,;-1.35,1.7,;-.01,2.47,;1.32,1.7,;-2.68,2.47,;-2.68,4.01,;-4.01,1.7,;-4.41,.21,;-5.9,.61,;-5.5,2.1,;-6.06,-.92,;-7.57,-1.24,;-8.34,.09,;-9.88,.09,;-7.31,1.24,)|

FC(F)(F)C1(CC1)c1ccc(cc1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:26.30,wD:24.27,(-6.85,5.1,;-5.4,5.63,;-5.93,7.07,;-4.87,4.18,;-3.95,6.15,;-4.22,7.67,;-2.77,7.14,;-3.18,4.82,;-3.95,3.48,;-3.18,2.15,;-1.64,2.15,;-.87,3.48,;-1.64,4.82,;-.87,.82,;-1.27,-.67,;.21,-1.07,;.61,.42,;-.56,-2.4,;.21,-3.74,;1.75,-3.74,;2.52,-2.4,;1.75,-1.07,;2.52,-5.07,;1.75,-6.4,;4.06,-5.07,;5.15,-6.16,;6.24,-5.07,;5.15,-3.98,;7.15,-6.32,;8.61,-5.84,;8.61,-4.3,;9.86,-3.39,;7.15,-3.82,)|

FC(F)(F)c1ccc(cc1Cl)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:22.24,wD:24.27,(9.92,-4.14,;8.59,-3.37,;7.82,-4.7,;9.36,-2.04,;7.26,-2.6,;5.88,-3.34,;4.54,-2.57,;4.54,-1.03,;5.88,-.26,;7.21,-1.03,;8.54,-.26,;3.21,-.26,;1.72,-.66,;1.32,.83,;2.81,1.22,;-.01,.06,;-1.35,.83,;-1.35,2.37,;-.01,3.14,;1.32,2.37,;-2.68,3.14,;-2.68,4.68,;-4.01,2.37,;-4.41,.88,;-5.9,1.28,;-5.5,2.76,;-6.06,-.25,;-7.57,-.57,;-8.34,.76,;-9.88,.76,;-7.31,1.9,)|

Cc1ccc(C)c(c1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:19.21,wD:21.24,(9.21,-.93,;7.88,-1.7,;7.88,-3.24,;6.54,-4.01,;5.21,-3.24,;3.87,-4.01,;5.21,-1.7,;6.54,-.93,;3.87,-.93,;2.39,-1.33,;1.99,.16,;3.48,.56,;.66,-.61,;-.68,.16,;-.68,1.7,;.66,2.47,;1.99,1.7,;-2.01,2.47,;-2.01,4.01,;-3.35,1.7,;-3.74,.21,;-5.23,.61,;-4.83,2.1,;-5.39,-.92,;-6.9,-1.24,;-7.67,.09,;-9.21,.09,;-6.64,1.24,)|

COc1ccc(cc1C(F)(F)F)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:23.25,wD:25.28,(9.92,-3.28,;8.58,-4.04,;7.25,-3.25,;5.88,-4.01,;4.54,-3.24,;4.54,-1.7,;5.88,-.93,;7.25,-1.68,;8.58,-.9,;9.9,-.12,;7.79,.43,;9.36,-2.23,;3.21,-.93,;1.72,-1.33,;1.32,.16,;2.81,.56,;-.01,-.61,;-1.35,.16,;-1.35,1.7,;-.01,2.47,;1.32,1.7,;-2.68,2.47,;-2.68,4.01,;-4.01,1.7,;-4.41,.21,;-5.9,.61,;-5.5,2.1,;-6.06,-.92,;-7.57,-1.24,;-8.34,.09,;-9.88,.09,;-7.31,1.24,)|

CC(C)(C)c1ccnc(c1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:21.23,wD:23.26,(9.88,-.16,;8.54,-.93,;8.54,.61,;9.88,-1.7,;7.21,-1.7,;7.21,-3.24,;5.88,-4.01,;4.54,-3.24,;4.54,-1.7,;5.88,-.93,;3.21,-.93,;1.72,-1.33,;1.32,.16,;2.81,.56,;-.01,-.61,;-1.35,.16,;-1.35,1.7,;-.01,2.47,;1.32,1.7,;-2.68,2.47,;-2.68,4.01,;-4.01,1.7,;-4.41,.21,;-5.9,.61,;-5.5,2.1,;-6.06,-.92,;-7.57,-1.24,;-8.34,.09,;-9.88,.09,;-7.31,1.24,)|

CC(C)(C)c1ccc(F)c(c1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:22.24,wD:24.27,(9.88,-.16,;8.54,-.93,;8.54,.61,;9.88,-1.7,;7.21,-1.7,;7.21,-3.24,;5.88,-4.01,;4.54,-3.24,;3.21,-4.01,;4.54,-1.7,;5.88,-.93,;3.21,-.93,;1.72,-1.33,;1.32,.16,;2.81,.56,;-.01,-.61,;-1.35,.16,;-1.35,1.7,;-.01,2.47,;1.32,1.7,;-2.68,2.47,;-2.68,4.01,;-4.01,1.7,;-4.41,.21,;-5.9,.61,;-5.5,2.1,;-6.06,-.92,;-7.57,-1.24,;-8.34,.09,;-9.88,.09,;-7.31,1.24,)|

CCOc1ccc(cc1C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2)C(C)(C)C |r,wU:20.22,wD:22.25,$;;;;;;;;;;;;;;;;;;;;;;;;;;;;N;;;;$,(.54,-4.01,;1.87,-3.24,;3.21,-4.01,;4.54,-3.24,;5.88,-4.01,;7.21,-3.24,;7.21,-1.7,;5.88,-.93,;4.54,-1.7,;3.21,-.93,;1.72,-1.33,;1.32,.16,;2.81,.56,;-.01,-.61,;-1.35,.16,;-1.35,1.7,;-.01,2.47,;1.32,1.7,;-2.68,2.47,;-2.68,4.01,;-4.01,1.7,;-4.41,.21,;-5.9,.61,;-5.5,2.1,;-6.06,-.92,;-7.57,-1.24,;-8.34,.09,;-9.88,.09,;-7.31,1.24,;8.54,-.93,;9.88,-.16,;8.54,.61,;9.88,-1.7,)|

Cc1ccccc1C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.20,wD:20.23,(7.21,.61,;7.21,-.93,;8.54,-1.7,;8.54,-3.24,;7.21,-4.01,;5.88,-3.24,;5.88,-1.7,;4.54,-.93,;3.05,-1.33,;2.66,.16,;4.14,.56,;1.32,-.61,;-.01,.16,;-.01,1.7,;1.32,2.47,;2.66,1.7,;-1.35,2.47,;-1.35,4.01,;-2.68,1.7,;-3.08,.21,;-4.57,.61,;-4.17,2.1,;-4.73,-.92,;-6.23,-1.24,;-7,.09,;-8.54,.09,;-5.97,1.24,)|

CC(C)c1cccc(c1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:20.22,wD:22.25,(8.54,.61,;8.54,-.93,;9.88,-1.7,;7.21,-1.7,;7.21,-3.24,;5.88,-4.01,;4.54,-3.24,;4.54,-1.7,;5.88,-.93,;3.21,-.93,;1.72,-1.33,;1.32,.16,;2.81,.56,;-.01,-.61,;-1.35,.16,;-1.35,1.7,;-.01,2.47,;1.32,1.7,;-2.68,2.47,;-2.68,4.01,;-4.01,1.7,;-4.41,.21,;-5.9,.61,;-5.5,2.1,;-6.06,-.92,;-7.57,-1.24,;-8.34,.09,;-9.88,.09,;-7.31,1.24,)|

Cc1cccc(C2CC3(C2)CCN(CC3)C(=O)[C@H]2C[C@@]3(C2)COC(=O)N3)c1C |r,wU:17.18,wD:19.21,(9.21,-.93,;7.88,-1.7,;7.88,-3.24,;6.54,-4.01,;5.21,-3.24,;5.21,-1.7,;3.87,-.93,;2.39,-1.33,;1.99,.16,;3.48,.56,;.66,-.61,;-.68,.16,;-.68,1.7,;.66,2.47,;1.99,1.7,;-2.01,2.47,;-2.01,4.01,;-3.35,1.7,;-3.74,.21,;-5.23,.61,;-4.83,2.1,;-5.39,-.92,;-6.9,-1.24,;-7.67,.09,;-9.21,.09,;-6.64,1.24,;6.54,-.93,;6.54,.61,)|

COc1ccc(cc1C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2)C(C)(C)C |r,wU:19.21,wD:21.24,(1.87,-3.24,;3.21,-4.01,;4.54,-3.24,;5.88,-4.01,;7.21,-3.24,;7.21,-1.7,;5.88,-.93,;4.54,-1.7,;3.21,-.93,;1.72,-1.33,;1.32,.16,;2.81,.56,;-.01,-.61,;-1.35,.16,;-1.35,1.7,;-.01,2.47,;1.32,1.7,;-2.68,2.47,;-2.68,4.01,;-4.01,1.7,;-4.41,.21,;-5.9,.61,;-5.5,2.1,;-6.06,-.92,;-7.57,-1.24,;-8.34,.09,;-9.88,.09,;-7.31,1.24,;8.54,-.93,;9.88,-.16,;8.54,.61,;9.88,-1.7,)|

FC1(F)Oc2ccc(cc2O1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:22.25,wD:24.28,(10.39,-1.7,;9.06,-2.47,;10.39,-3.24,;8.16,-3.72,;6.69,-3.24,;5.36,-4.01,;4.02,-3.24,;4.02,-1.7,;5.36,-.93,;6.69,-1.7,;8.16,-1.22,;2.69,-.93,;1.2,-1.33,;.8,.16,;2.29,.56,;-.53,-.61,;-1.86,.16,;-1.86,1.7,;-.53,2.47,;.8,1.7,;-3.2,2.47,;-3.2,4.01,;-4.53,1.7,;-4.93,.21,;-6.42,.61,;-6.02,2.1,;-6.58,-.92,;-8.08,-1.24,;-8.85,.09,;-10.39,.09,;-7.82,1.24,)|

COc1ccccc1C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:19.21,wD:21.24,(5.88,1.44,;7.21,.67,;7.21,-.87,;8.54,-1.7,;8.54,-3.24,;7.21,-4.01,;5.88,-3.24,;5.88,-1.7,;4.54,-.93,;3.05,-1.33,;2.66,.16,;4.14,.56,;1.32,-.61,;-.01,.16,;-.01,1.7,;1.32,2.47,;2.66,1.7,;-1.35,2.47,;-1.35,4.01,;-2.68,1.7,;-3.08,.21,;-4.57,.61,;-4.17,2.1,;-4.73,-.92,;-6.23,-1.24,;-7,.09,;-8.54,.09,;-5.97,1.24,)|

COc1ccc(cc1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:19.21,wD:21.24,(9.92,-3.27,;8.59,-4.04,;7.26,-3.27,;5.88,-4.01,;4.54,-3.24,;4.54,-1.7,;5.88,-.93,;7.21,-1.7,;3.21,-.93,;1.72,-1.33,;1.32,.16,;2.81,.56,;-.01,-.61,;-1.35,.16,;-1.35,1.7,;-.01,2.47,;1.32,1.7,;-2.68,2.47,;-2.68,4.01,;-4.01,1.7,;-4.41,.21,;-5.9,.61,;-5.5,2.1,;-6.06,-.92,;-7.57,-1.24,;-8.34,.09,;-9.88,.09,;-7.31,1.24,)|

Fc1ccc(nc1C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2)C(F)(F)F |r,wU:18.20,wD:20.23,(3.21,-4.01,;4.54,-3.24,;5.88,-4.01,;7.21,-3.24,;7.26,-1.67,;5.88,-.93,;4.54,-1.7,;3.21,-.93,;1.72,-1.33,;1.32,.16,;2.81,.56,;-.01,-.61,;-1.35,.16,;-1.35,1.7,;-.01,2.47,;1.32,1.7,;-2.68,2.47,;-2.68,4.01,;-4.01,1.7,;-4.41,.21,;-5.9,.61,;-5.5,2.1,;-6.06,-.92,;-7.57,-1.24,;-8.34,.09,;-9.88,.09,;-7.31,1.24,;8.59,-.9,;9.92,-.13,;9.36,-2.24,;7.82,.43,)|

FC(F)(F)c1cccc(n1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:21.23,wD:23.26,(9.92,-.13,;8.59,-.9,;9.36,-2.24,;7.82,.43,;7.26,-1.67,;7.21,-3.24,;5.88,-4.01,;4.54,-3.24,;4.54,-1.7,;5.88,-.93,;3.21,-.93,;1.72,-1.33,;1.32,.16,;2.81,.56,;-.01,-.61,;-1.35,.16,;-1.35,1.7,;-.01,2.47,;1.32,1.7,;-2.68,2.47,;-2.68,4.01,;-4.01,1.7,;-4.41,.21,;-5.9,.61,;-5.5,2.1,;-6.06,-.92,;-7.57,-1.24,;-8.34,.09,;-9.88,.09,;-7.31,1.24,)|

Cc1nc(ccc1F)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:19.21,wD:21.24,(9.21,-.93,;7.88,-1.7,;6.54,-.93,;5.21,-1.7,;5.21,-3.24,;6.54,-4.01,;7.88,-3.24,;9.21,-4.01,;3.87,-.93,;2.39,-1.33,;1.99,.16,;3.48,.56,;.66,-.61,;-.68,.16,;-.68,1.7,;.66,2.47,;1.99,1.7,;-2.01,2.47,;-2.01,4.01,;-3.35,1.7,;-3.74,.21,;-5.23,.61,;-4.83,2.1,;-5.39,-.92,;-6.9,-1.24,;-7.67,.09,;-9.21,.09,;-6.64,1.24,)|

CC(C)(C)c1nccc(n1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:21.23,wD:23.26,(9.88,-.16,;8.54,-.93,;8.54,.61,;9.88,-1.7,;7.21,-1.7,;7.21,-3.24,;5.88,-4.01,;4.54,-3.24,;4.54,-1.7,;5.88,-.93,;3.21,-.93,;1.72,-1.33,;1.32,.16,;2.81,.56,;-.01,-.61,;-1.35,.16,;-1.35,1.7,;-.01,2.47,;1.32,1.7,;-2.68,2.47,;-2.68,4.01,;-4.01,1.7,;-4.41,.21,;-5.9,.61,;-5.5,2.1,;-6.06,-.92,;-7.57,-1.24,;-8.34,.09,;-9.88,.09,;-7.31,1.24,)|

CC(C)(C)c1coc(n1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:20.22,wD:22.25,(9.92,-1.65,;8.43,-2.05,;8.83,-.56,;9.52,-3.14,;6.94,-2.45,;6.17,-3.78,;4.66,-3.46,;4.5,-1.93,;5.91,-1.3,;3.17,-1.16,;1.68,-1.56,;1.28,-.07,;2.77,.33,;-.05,-.84,;-1.38,-.07,;-1.38,1.47,;-.05,2.24,;1.28,1.47,;-2.72,2.24,;-2.72,3.78,;-4.05,1.47,;-4.45,-.02,;-5.94,.38,;-5.54,1.87,;-6.1,-1.15,;-7.61,-1.47,;-8.38,-.14,;-9.92,-.14,;-7.34,1.01,)|

CC(C)(C)c1ncc(o1)C1CC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:20.22,wD:22.25,(9.92,-1.65,;8.43,-2.05,;8.83,-.56,;9.52,-3.14,;6.94,-2.45,;6.17,-3.78,;4.66,-3.46,;4.5,-1.93,;5.91,-1.3,;3.17,-1.16,;1.68,-1.56,;1.28,-.07,;2.77,.33,;-.05,-.84,;-1.38,-.07,;-1.38,1.47,;-.05,2.24,;1.28,1.47,;-2.72,2.24,;-2.72,3.78,;-4.05,1.47,;-4.45,-.02,;-5.94,.38,;-5.54,1.87,;-6.1,-1.15,;-7.61,-1.47,;-8.38,-.14,;-9.92,-.14,;-7.34,1.01,)|

Fc1cnc(C2CC3(C2)CCN(CC3)C(=O)[C@H]2C[C@@]3(C2)COC(=O)N3)c(F)c1 |r,wU:16.17,wD:18.20,(9.21,-4.01,;7.88,-3.24,;7.88,-1.7,;6.54,-.93,;5.21,-1.7,;3.87,-.93,;2.39,-1.33,;1.99,.16,;3.48,.56,;.66,-.61,;-.68,.16,;-.68,1.7,;.66,2.47,;1.99,1.7,;-2.01,2.47,;-2.01,4.01,;-3.35,1.7,;-3.74,.21,;-5.23,.61,;-4.83,2.1,;-5.39,-.92,;-6.9,-1.24,;-7.67,.09,;-9.21,.09,;-6.64,1.24,;5.21,-3.24,;3.87,-4.01,;6.54,-4.01,)|

FC(F)(F)c1ccc(cc1)C1CCC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:22.24,wD:24.27,(10.43,.68,;9.09,-.09,;9.49,1.39,;10.43,-.86,;7.6,-.49,;7.21,-1.98,;5.72,-2.38,;4.63,-1.29,;5.03,.2,;6.52,.6,;3.14,-1.69,;2.24,-2.93,;.77,-2.46,;.77,-.92,;2.24,-.44,;-.56,-1.69,;-1.9,-.92,;-1.9,.62,;-.56,1.39,;.77,.62,;-3.23,1.39,;-3.23,2.93,;-4.56,.62,;-4.96,-.86,;-6.45,-.47,;-6.05,1.02,;-6.61,-2,;-8.12,-2.32,;-8.89,-.98,;-10.43,-.98,;-7.86,.16,)|

CC1OC(=O)N[C@@]11C[C@@H](C1)C(=O)N1CCC2(CCC(C2)c2ccc(cc2)C(F)(F)F)CC1 |r,wU:8.11,wD:6.10,(-5.45,-3.04,;-6.61,-1.89,;-8.12,-2.21,;-8.89,-.87,;-10.43,-.87,;-7.86,.27,;-6.45,-.35,;-4.96,-.75,;-4.56,.73,;-6.05,1.13,;-3.23,1.5,;-3.23,3.04,;-1.9,.73,;-1.9,-.81,;-.56,-1.58,;.77,-.81,;.77,-2.35,;2.24,-2.82,;3.14,-1.58,;2.24,-.33,;4.63,-1.18,;5.72,-2.27,;7.21,-1.87,;7.6,-.38,;6.52,.71,;5.03,.31,;9.09,.02,;10.43,.79,;9.49,1.51,;10.43,-.75,;.77,.73,;-.56,1.5,)|

O=C([C@H]1C[C@@]2(C1)COC(=O)N2)N1CC2(C1)CCC(C2)c1ccccc1 |r,wU:2.1,wD:4.4,(-1.43,2.71,;-1.43,1.17,;-2.76,.4,;-3.16,-1.09,;-4.65,-.69,;-4.25,.8,;-4.81,-2.22,;-6.31,-2.54,;-7.08,-1.21,;-8.62,-1.21,;-6.05,-.07,;-.09,.4,;.3,-1.09,;1.79,-.69,;1.39,.8,;1.79,-2.23,;3.26,-2.71,;4.16,-1.46,;3.26,-.22,;5.65,-1.06,;6.74,-2.15,;8.23,-1.75,;8.62,-.27,;7.54,.82,;6.05,.42,)|

O=C([C@H]1C[C@@]2(C1)COC(=O)N2)N1CC2(C1)CC[C@H](C2)c1ccccc1 |r,wU:2.1,wD:4.4,17.22,(-1.45,2.71,;-1.45,1.17,;-2.78,.4,;-3.18,-1.09,;-4.67,-.69,;-4.27,.8,;-4.83,-2.22,;-6.33,-2.54,;-7.1,-1.21,;-8.64,-1.21,;-6.07,-.07,;-.11,.4,;.28,-1.09,;1.77,-.69,;1.37,.8,;1.77,-2.23,;3.24,-2.71,;4.14,-1.46,;3.24,-.22,;5.67,-1.35,;6.76,-2.44,;8.25,-2.04,;8.64,-.55,;7.56,.54,;6.07,.14,)|

FC(F)(F)c1ccc(cc1)C1CCC2(CN(C2)C(=O)[C@H]2C[C@@]3(C2)COC(=O)N3)C1 |r,wU:19.20,wD:21.23,(9.23,.19,;8.55,-1.19,;9.4,-2.47,;10.09,-1.09,;7.01,-1.29,;6.33,-2.67,;4.79,-2.77,;3.94,-1.49,;4.62,-.11,;6.16,-.01,;2.4,-1.62,;1.49,-2.87,;.03,-2.39,;.03,-.85,;-.21,.67,;-1.73,.43,;-1.49,-1.1,;-2.98,1.33,;-2.98,2.87,;-4.39,.7,;-4.78,-.78,;-6.27,-.38,;-5.87,1.1,;-6.19,-1.92,;-7.63,-2.47,;-8.6,-1.28,;-10.09,-.88,;-7.76,.01,;1.49,-.38,)|

FC(F)(F)c1ccc(cc1)[C@@H]1CCC2(CN(C2)C(=O)[C@H]2C[C@@]3(C2)COC(=O)N3)C1 |r,wU:19.20,wD:10.10,21.23,(9.22,.19,;8.57,-1.21,;9.46,-2.47,;10.11,-1.08,;7.04,-1.35,;6.39,-2.74,;4.85,-2.88,;3.97,-1.62,;4.62,-.22,;6.15,-.09,;2.43,-1.62,;1.52,-2.86,;.06,-2.39,;.06,-.85,;-.18,.67,;-1.7,.43,;-1.46,-1.09,;-2.95,1.34,;-2.95,2.88,;-4.36,.71,;-4.75,-.78,;-6.24,-.38,;-5.84,1.11,;-6.16,-1.92,;-7.6,-2.47,;-8.57,-1.27,;-10.11,-1.15,;-7.73,.02,;1.52,-.37,)|

FC(F)(F)c1ccc(cc1)[C@H]1CCC2(CN(C2)C(=O)[C@H]2C[C@@]3(C2)COC(=O)N3)C1 |r,wU:10.10,19.20,wD:21.23,(9.12,.44,;8.54,-.99,;9.48,-2.2,;10.06,-.77,;7.01,-1.2,;6.43,-2.63,;4.91,-2.84,;3.96,-1.62,;4.54,-.2,;6.07,.02,;2.42,-1.62,;1.52,-2.87,;.05,-2.39,;.05,-.85,;-.19,.67,;-1.71,.43,;-1.47,-1.1,;-2.96,1.33,;-2.96,2.87,;-4.36,.7,;-4.76,-.78,;-6.25,-.38,;-5.85,1.1,;-6.17,-1.92,;-7.61,-2.47,;-8.57,-1.28,;-10.06,-1.08,;-7.74,.01,;1.52,-.38,)|

FC(F)(F)c1ccc(cc1)[C@@H]1CCC2(CN(C2)C(=O)[C@H]2C[C@@]3(C2)COC(=O)N3)C1 |r,wU:19.20,wD:10.10,21.23,(9.2,.19,;8.55,-1.21,;9.43,-2.47,;10.08,-1.07,;7.01,-1.35,;6.36,-2.74,;4.83,-2.88,;3.94,-1.62,;4.59,-.22,;6.13,-.09,;2.4,-1.62,;1.5,-2.86,;.03,-2.39,;.03,-.85,;-.21,.67,;-1.73,.43,;-1.49,-1.09,;-2.97,1.34,;-2.97,2.88,;-4.38,.71,;-4.78,-.78,;-6.27,-.38,;-5.87,1.11,;-6.19,-1.92,;-7.62,-2.47,;-8.59,-1.27,;-10.08,-1.07,;-7.75,.02,;1.5,-.37,)|

FC(F)(F)c1ccc(cc1)[C@H]1CCC2(CN(C2)C(=O)[C@H]2C[C@@]3(C2)COC(=O)N3)C1 |r,wU:10.10,19.20,wD:21.23,(9.18,.23,;8.54,-1.17,;9.44,-2.42,;10.08,-1.02,;7.01,-1.32,;6.38,-2.72,;4.84,-2.87,;3.95,-1.62,;4.58,-.22,;6.12,-.07,;2.41,-1.62,;1.5,-2.87,;.04,-2.39,;.04,-.85,;-.2,.67,;-1.72,.43,;-1.48,-1.09,;-2.97,1.33,;-2.97,2.87,;-4.38,.71,;-4.78,-.78,;-6.26,-.38,;-5.87,1.11,;-6.18,-1.92,;-7.62,-2.47,;-8.59,-1.27,;-10.08,-1.08,;-7.75,.02,;1.5,-.38,)|

CC(C)(C)c1ccc(cc1)C1CCC2(CN(C2)C(=O)[C@H]2C[C@@]3(C2)COC(=O)N3)C1 |r,wU:19.20,wD:21.23,(9.17,.26,;8.54,-1.14,;9.45,-2.39,;10.08,-.98,;7.01,-1.3,;6.39,-2.71,;4.85,-2.87,;3.95,-1.62,;4.58,-.22,;6.11,-.06,;2.41,-1.62,;1.5,-2.87,;.04,-2.39,;.04,-.85,;-.2,.67,;-1.72,.43,;-1.48,-1.1,;-2.97,1.33,;-2.97,2.87,;-4.38,.7,;-4.77,-.78,;-6.26,-.38,;-5.86,1.1,;-6.18,-1.92,;-7.62,-2.47,;-8.59,-1.28,;-10.08,-1.15,;-7.75,.01,;1.5,-.38,)|

CC(C)(C)c1cccc(c1)C1CCC2(CN(C2)C(=O)[C@H]2C[C@@]3(C2)COC(=O)N3)C1 |r,wU:19.20,wD:21.23,(9.51,-2.32,;8,-2.58,;7.46,-4.03,;8.98,-3.77,;7.01,-1.4,;7.55,.05,;6.56,1.23,;5.04,.97,;4.51,-.47,;5.49,-1.66,;2.97,-.47,;2.07,-1.72,;.6,-1.24,;.6,.3,;.36,1.82,;-1.16,1.58,;-.92,.06,;-2.41,2.49,;-2.41,4.03,;-3.81,1.86,;-4.21,.37,;-5.7,.77,;-5.3,2.26,;-5.62,-.77,;-7.06,-1.32,;-8.03,-.12,;-9.51,.08,;-7.19,1.17,;2.07,.78,)|

CC1OC(=O)N[C@@]11C[C@@H](C1)C(=O)N1CC2(C1)CCC(C2)c1cccc(c1)C(C)(C)C |r,wU:8.11,wD:6.10,(-4.3,-1.56,;-5.59,-.72,;-7.03,-1.27,;-8,-.08,;-9.48,.13,;-7.16,1.22,;-5.67,.82,;-4.18,.42,;-3.78,1.91,;-5.27,2.3,;-2.38,2.53,;-2.38,4.07,;-1.13,1.63,;.39,1.87,;.63,.35,;-.89,.11,;.63,-1.19,;2.1,-1.67,;3,-.42,;2.1,.82,;4.54,-.42,;5.12,1,;6.65,1.21,;7.59,-0,;7.01,-1.43,;5.49,-1.64,;7.96,-2.65,;9.48,-2.44,;7.38,-4.07,;8.9,-3.86,)|

O=C([C@H]1C[C@@]2(C1)COC(=O)N2)N1CC2(C1)CCC(C2)C1CC1 |r,wU:2.1,wD:4.4,(-.57,2.87,;-.57,1.33,;-1.98,.7,;-2.38,-.78,;-3.87,-.38,;-3.47,1.1,;-3.78,-1.92,;-5.22,-2.47,;-6.19,-1.28,;-7.68,-1.01,;-5.35,.01,;.67,.43,;2.19,.67,;2.44,-.85,;.91,-1.1,;2.44,-2.39,;3.9,-2.87,;4.81,-1.62,;3.9,-.38,;6.35,-1.62,;7.68,-2.39,;7.68,-.85,)|

O=C([C@H]1C[C@@]2(C1)COC(=O)N2)N1CC2(C1)CCC(C2)C1CCCCC1 |r,wU:2.1,wD:4.4,(-1.44,2.88,;-1.44,1.34,;-2.85,.71,;-3.25,-.77,;-4.73,-.37,;-4.33,1.11,;-4.65,-1.91,;-6.09,-2.46,;-7.06,-1.27,;-8.55,-1.06,;-6.22,.02,;-.19,.44,;1.33,.68,;1.57,-.84,;.05,-1.09,;1.57,-2.38,;3.03,-2.86,;3.94,-1.61,;3.03,-.37,;5.48,-1.61,;6.35,-2.88,;7.89,-2.76,;8.55,-1.37,;7.67,-.1,;6.14,-.22,)|

O=C([C@H]1C[C@@]2(C1)COC(=O)N2)N1CC2(C1)CCC(C2)C1CCCC1 |r,wU:2.1,wD:4.4,(-1.14,2.87,;-1.14,1.33,;-2.54,.7,;-2.94,-.78,;-4.43,-.38,;-4.03,1.1,;-4.35,-1.92,;-5.79,-2.47,;-6.76,-1.28,;-8.24,-1.07,;-5.92,.01,;.11,.43,;1.63,.67,;1.87,-.85,;.35,-1.1,;1.87,-2.39,;3.34,-2.87,;4.24,-1.62,;3.34,-.38,;5.78,-1.62,;6.87,-2.71,;8.24,-2.01,;8,-.49,;6.48,-.25,)|

O=C([C@H]1C[C@@]2(C1)COC(=O)N2)N1CC2(C1)CCC(C2)C1CCC1 |r,wU:2.1,wD:4.4,(-.99,2.87,;-.99,1.33,;-2.4,.7,;-2.8,-.78,;-4.29,-.38,;-3.89,1.1,;-4.21,-1.92,;-5.64,-2.47,;-6.61,-1.28,;-8.1,-1.07,;-5.77,.01,;.25,.43,;1.77,.67,;2.01,-.85,;.49,-1.1,;2.01,-2.39,;3.48,-2.87,;4.38,-1.62,;3.48,-.38,;5.92,-1.62,;7.01,-2.71,;8.1,-1.62,;7.01,-.54,)|

CC(C)(C)c1cccc(c1)C1CCC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:22.24,wD:24.27,(7.66,-4.22,;8.36,-2.84,;9.9,-2.76,;9.2,-4.13,;7.52,-1.55,;8.1,-.13,;7.16,1.09,;5.63,.88,;5.05,-.54,;5.99,-1.76,;3.51,-.54,;2.6,-1.79,;1.14,-1.31,;1.14,.23,;2.6,.71,;-.19,-.54,;-1.53,.23,;-1.54,1.77,;-.19,2.54,;1.14,1.77,;-2.79,2.68,;-2.79,4.22,;-4.2,2.05,;-4.6,.56,;-6.08,.96,;-5.68,2.45,;-6,-.58,;-7.44,-1.13,;-8.41,.07,;-9.9,.21,;-7.57,1.36,)|

CC(C)(C)c1ccc(cc1)C1CCC2(C1)CCN(CC2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:22.24,wD:24.27,(9.63,-2.96,;8.76,-1.69,;9.41,-.3,;10.29,-1.57,;7.22,-1.81,;6.56,-3.21,;5.03,-3.33,;4.15,-2.06,;4.81,-.67,;6.34,-.55,;2.61,-2.06,;1.71,-3.31,;.24,-2.83,;.24,-1.29,;1.71,-.82,;-1.25,-1.69,;-2.34,-.6,;-1.94,.88,;-.45,1.28,;.64,.19,;-3.18,1.79,;-3.18,3.33,;-4.59,1.16,;-4.99,-.32,;-6.48,.07,;-6.08,1.56,;-6.4,-1.46,;-7.83,-2.01,;-8.8,-.82,;-10.29,-.69,;-7.96,.47,)|

CC(C)c1cccc(c1)C1CC2(C1)CCN(C2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:19.21,wD:21.24,(7.56,-3.25,;8.17,-1.84,;9.7,-1.66,;7.25,-.6,;7.86,.81,;6.94,2.05,;5.41,1.87,;4.8,.45,;5.72,-.78,;3.26,.38,;2.23,-.76,;1.09,.28,;2.12,1.42,;.24,-1.01,;-1.24,-.6,;-1.33,.94,;.12,1.48,;-2.67,1.71,;-2.67,3.25,;-4,.94,;-4.4,-.55,;-5.89,-.15,;-5.49,1.34,;-5.81,-1.69,;-7.24,-2.24,;-8.21,-1.04,;-9.7,-.99,;-7.37,.25,)|

CC(C)(C)c1cccc(c1)C1CC2(C1)CCN(C2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:20.22,wD:22.25,(9.63,-1.89,;8.09,-2.01,;7.42,-3.39,;8.86,-3.34,;7.23,-.73,;7.89,.65,;7.03,1.93,;5.49,1.81,;4.82,.43,;5.69,-.85,;3.29,.31,;2.2,-.78,;1.11,.31,;2.2,1.4,;.2,-.93,;-1.26,-.46,;-1.26,1.08,;.2,1.56,;-2.59,1.85,;-2.59,3.39,;-3.93,1.08,;-4.33,-.4,;-5.81,-.01,;-5.42,1.48,;-5.73,-1.54,;-7.17,-2.1,;-8.14,-.9,;-9.63,-.83,;-7.3,.39,)|

CC(C)c1cccc(c1)C1CCC2(CN(C2)C(=O)[C@H]2C[C@@]3(C2)COC(=O)N3)C1 |r,wU:18.19,wD:20.22,(9.48,-2.44,;7.95,-2.55,;7.28,-3.94,;7.08,-1.28,;7.75,.11,;6.88,1.38,;5.35,1.27,;4.68,-.12,;5.54,-1.39,;3.14,-.23,;2.24,-1.48,;.77,-1,;.77,.54,;-.72,.14,;-1.11,1.63,;.37,2.03,;-2.45,2.4,;-2.45,3.94,;-3.78,1.63,;-4.18,.14,;-5.67,.54,;-5.27,2.03,;-5.59,-1,;-7.03,-1.55,;-7.99,-.35,;-9.48,-.22,;-7.16,.94,;2.24,1.01,)|

CC(C)c1cccc(c1)C1CCC2(CN(C2)C(=O)[C@H]2C[C@@]3(C2)CCC(=O)N3)C1 |r,wU:18.19,wD:20.22,(9.48,-2.44,;7.95,-2.55,;7.28,-3.94,;7.08,-1.28,;7.75,.11,;6.88,1.38,;5.35,1.27,;4.68,-.12,;5.54,-1.39,;3.14,-.23,;2.24,-1.48,;.77,-1,;.77,.54,;-.72,.14,;-1.11,1.63,;.37,2.03,;-2.45,2.4,;-2.45,3.94,;-3.78,1.63,;-4.18,.14,;-5.67,.54,;-5.27,2.03,;-5.59,-1,;-7.03,-1.55,;-7.99,-.35,;-9.48,-.22,;-7.16,.94,;2.24,1.01,)|

CC(C)c1ccc(cc1)C1CCC2(CN(C2)C(=O)[C@H]2C[C@@]3(C2)COC(=O)N3)C1 |r,wU:18.19,wD:20.22,(9.62,.42,;8.95,-.97,;9.82,-2.24,;7.41,-1.08,;6.74,-2.47,;5.21,-2.58,;4.34,-1.31,;5.01,.08,;6.55,.19,;2.81,-1.42,;1.9,-2.67,;.44,-2.19,;.44,-.65,;-1.05,-1.05,;-1.45,.43,;.04,.83,;-2.78,1.2,;-2.78,2.74,;-4.12,.43,;-4.52,-1.05,;-6,-.65,;-5.6,.83,;-5.92,-2.19,;-7.36,-2.74,;-8.33,-1.55,;-9.82,-1.41,;-7.49,-.26,;1.9,-.18,)|

O=C([C@H]1C[C@@]2(C1)COC(=O)N2)N1CCC2(CC(C2)c2ccccc2)C1 |r,wU:2.1,wD:4.4,(-1.73,2.74,;-1.73,1.2,;-3.06,.43,;-3.46,-1.05,;-4.95,-.65,;-4.55,.83,;-4.87,-2.19,;-6.3,-2.74,;-7.27,-1.55,;-8.76,-1.47,;-6.43,-.26,;-.39,.43,;-.39,-1.11,;1.07,-1.58,;1.98,-.34,;3.06,-1.42,;4.15,-.34,;3.06,.75,;5.69,-.22,;6.56,-1.49,;8.09,-1.38,;8.76,.01,;7.89,1.28,;6.36,1.17,;1.07,.91,)|

CC(C)(C)c1cccc(c1)C1CC2(C1)CN(C2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:19.21,wD:21.24,(8.07,.84,;8.07,-.7,;9.4,-1.47,;9.4,.07,;6.74,-1.47,;6.74,-3.01,;5.4,-3.78,;4.07,-3.01,;4.07,-1.47,;5.4,-.7,;2.74,-.7,;1.25,-1.1,;.85,.38,;2.34,.78,;-.64,-.01,;-1.04,1.47,;.45,1.87,;-2.37,2.24,;-2.37,3.78,;-3.7,1.47,;-4.1,-.01,;-5.59,.39,;-5.19,1.87,;-5.51,-1.15,;-6.95,-1.7,;-7.92,-.51,;-9.4,-.43,;-7.08,.78,)|

Cc1cccc(c1)C1CC2(C1)CN(C2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:16.18,wD:18.21,(8.74,-.7,;7.4,-1.47,;7.4,-3.01,;6.07,-3.78,;4.74,-3.01,;4.74,-1.47,;6.07,-.7,;3.4,-.7,;1.91,-1.1,;1.52,.38,;3,.78,;.03,-.01,;-.37,1.47,;1.12,1.87,;-1.7,2.24,;-1.7,3.78,;-3.04,1.47,;-3.44,-.01,;-4.92,.39,;-4.52,1.87,;-4.84,-1.15,;-6.28,-1.7,;-7.25,-.51,;-8.74,-.37,;-6.41,.78,)|

CC(C)c1cccc(c1)C1CC2(C1)CN(C2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.20,wD:20.23,(9.4,-1.47,;8.07,-.7,;8.07,.84,;6.74,-1.47,;6.74,-3.01,;5.4,-3.78,;4.07,-3.01,;4.07,-1.47,;5.4,-.7,;2.74,-.7,;1.25,-1.1,;.85,.38,;2.34,.78,;-.64,-.01,;-1.04,1.47,;.45,1.87,;-2.37,2.24,;-2.37,3.78,;-3.7,1.47,;-4.1,-.01,;-5.59,.39,;-5.19,1.87,;-5.51,-1.15,;-6.95,-1.7,;-7.92,-.51,;-9.4,-.3,;-7.08,.78,)|

Cc1ccc(cc1C)C1CC2(C1)CN(C2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:17.19,wD:19.22,(8.74,-3.78,;7.4,-3.01,;6.07,-3.78,;4.74,-3.01,;4.74,-1.47,;6.07,-.7,;7.4,-1.47,;8.74,-.7,;3.4,-.7,;1.91,-1.1,;1.52,.38,;3,.78,;.03,-.01,;-.37,1.47,;1.12,1.87,;-1.7,2.24,;-1.7,3.78,;-3.04,1.47,;-3.44,-.01,;-4.92,.39,;-4.52,1.87,;-4.84,-1.15,;-6.28,-1.7,;-7.25,-.51,;-8.74,-.37,;-6.41,.78,)|

O=C([C@H]1C[C@@]2(C1)COC(=O)N2)N1CC2(CC(C2)C2CCCCC2)C1 |r,wU:2.1,wD:4.4,(-1.04,3.78,;-1.04,2.24,;-2.37,1.47,;-2.77,-.01,;-4.26,.39,;-3.86,1.87,;-4.18,-1.15,;-5.61,-1.7,;-6.58,-.51,;-8.07,-.3,;-5.74,.78,;.3,1.47,;.7,-.01,;2.18,.38,;2.58,-1.1,;4.07,-.7,;3.67,.78,;5.4,-1.47,;5.4,-3.01,;6.74,-3.78,;8.07,-3.01,;8.07,-1.47,;6.74,-.7,;1.78,1.87,)|

Cc1cc(C)cc(c1)C1CC2(C1)CN(C2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:17.19,wD:19.22,(8.74,.07,;7.4,-.7,;7.4,-2.24,;6.07,-3.01,;6.07,-4.55,;4.74,-2.24,;4.74,-.7,;6.07,.07,;3.4,.07,;1.91,-.33,;1.52,1.15,;3,1.55,;.03,.76,;-.37,2.24,;1.12,2.64,;-1.7,3.01,;-1.7,4.55,;-3.04,2.24,;-3.44,.76,;-4.92,1.16,;-4.52,2.64,;-4.84,-.38,;-6.28,-.93,;-7.25,.26,;-8.74,.47,;-6.41,1.55,)|

Cc1ccc(C2CC3(C2)CN(C3)C(=O)[C@H]2C[C@@]3(C2)COC(=O)N3)c(C)c1 |r,wU:14.15,wD:16.18,(8.74,-3.78,;7.4,-3.01,;6.07,-3.78,;4.74,-3.01,;4.74,-1.47,;3.4,-.7,;1.91,-1.1,;1.52,.38,;3,.78,;.03,-.01,;-.37,1.47,;1.12,1.87,;-1.7,2.24,;-1.7,3.78,;-3.04,1.47,;-3.44,-.01,;-4.92,.39,;-4.52,1.87,;-4.84,-1.15,;-6.28,-1.7,;-7.25,-.51,;-8.74,-.37,;-6.41,.78,;6.07,-.7,;6.07,.84,;7.4,-1.47,)|

O=C([C@H]1C[C@@]2(C1)COC(=O)N2)N1CC2(CC(C2)c2cccc(c2)C2CC2)C1 |r,wU:2.1,wD:4.4,(-2.45,3.78,;-2.45,2.24,;-3.78,1.47,;-4.18,-.01,;-5.67,.39,;-5.27,1.87,;-5.59,-1.15,;-7.02,-1.7,;-7.99,-.51,;-9.53,-.51,;-7.15,.78,;-1.11,1.47,;-.71,-.01,;.77,.38,;1.17,-1.1,;2.66,-.7,;2.26,.78,;3.99,-1.47,;3.99,-3.01,;5.33,-3.78,;6.66,-3.01,;6.66,-1.47,;5.33,-.7,;7.99,-.7,;9.53,-.7,;8.76,.63,;.37,1.87,)|

O=C([C@H]1C[C@@]2(C1)COC(=O)N2)N1CC2(CC(C2)c2cccc(c2)C2CCC2)C1 |r,wU:2.1,wD:4.4,(-2.62,3.78,;-2.62,2.24,;-3.95,1.47,;-4.35,-.01,;-5.84,.39,;-5.44,1.87,;-5.76,-1.15,;-7.2,-1.7,;-8.17,-.51,;-9.71,-.51,;-7.33,.78,;-1.29,1.47,;-.89,-.01,;.6,.38,;1,-1.1,;2.49,-.7,;2.09,.78,;3.82,-1.47,;3.82,-3.01,;5.15,-3.78,;6.49,-3.01,;6.49,-1.47,;5.15,-.7,;7.82,-.7,;9.31,-1.1,;9.71,.38,;8.22,.78,;.2,1.87,)|

O=C([C@H]1C[C@@]2(C1)COC(=O)N2)N1CC2(CC(C2)c2ccc3CCCc3c2)C1 |r,wU:2.1,wD:4.4,(-2.14,3.78,;-2.14,2.24,;-3.48,1.47,;-3.88,-.01,;-5.36,.39,;-4.97,1.87,;-5.52,-1.15,;-7.03,-1.47,;-7.8,-.13,;-9.33,.03,;-6.77,1.01,;-.81,1.47,;.68,1.87,;1.08,.39,;2.56,.78,;2.96,-.7,;1.47,-1.1,;4.3,-1.47,;4.3,-3.01,;5.63,-3.78,;6.96,-3.01,;8.43,-3.49,;9.33,-2.24,;8.43,-1,;6.96,-1.47,;5.63,-.7,;-.41,-.01,)|

O=C([C@H]1C[C@@]2(C1)COC(=O)N2)N1CC2(CC(C2)c2ccccc2)C1 |r,wU:2.1,wD:4.4,(-.96,3.78,;-.96,2.24,;-2.29,1.47,;-2.69,-.01,;-4.18,.39,;-3.78,1.87,;-4.34,-1.15,;-5.85,-1.47,;-6.62,-.13,;-8.15,.03,;-5.59,1.01,;.37,1.47,;1.86,1.87,;2.26,.39,;3.75,.78,;4.15,-.7,;2.66,-1.1,;5.48,-1.47,;5.48,-3.01,;6.81,-3.78,;8.15,-3.01,;8.15,-1.47,;6.81,-.7,;.77,-.01,)|

O=C([C@H]1C[C@@]2(C1)COC(=O)N2)N1CC2(C1)CCC(CC2)c1ccccc1 |r,wU:2.1,wD:4.4,(-1.35,4.01,;-1.35,2.47,;-2.68,1.7,;-3.08,.21,;-4.57,.61,;-4.17,2.1,;-4.73,-.92,;-6.24,-1.24,;-7.01,.09,;-8.54,.25,;-5.98,1.24,;-.02,1.7,;1.47,2.1,;1.87,.61,;.38,.21,;1.87,-.93,;3.2,-1.7,;4.54,-.93,;4.54,.61,;3.2,1.38,;5.87,-1.7,;5.87,-3.24,;7.2,-4.01,;8.54,-3.24,;8.54,-1.7,;7.2,-.93,)|

O=C([C@H]1C[C@@]2(C1)COC(=O)N2)N1CC2(CC(C2)C2CCCC2)C1 |r,wU:2.1,wD:4.4,(-.84,3.55,;-.84,2.01,;-2.18,1.24,;-2.58,-.24,;-4.06,.16,;-3.67,1.64,;-4.22,-1.38,;-5.73,-1.7,;-6.5,-.36,;-8.03,-.2,;-5.47,.78,;.49,1.24,;1.98,1.64,;2.38,.16,;3.86,.55,;4.26,-.93,;2.77,-1.33,;5.6,-1.7,;5.76,-3.23,;7.26,-3.55,;8.03,-2.22,;7,-1.08,;.89,-.24,)|

O=C([C@H]1C[C@@]2(C1)COC(=O)N2)N1CC2(CC(C2)C2CCC2)C1 |r,wU:2.1,wD:4.4,(-.57,3.37,;-.57,1.83,;-1.9,1.06,;-2.3,-.42,;-3.79,-.03,;-3.39,1.46,;-3.95,-1.56,;-5.46,-1.88,;-6.23,-.54,;-7.76,-.38,;-5.2,.6,;.77,1.06,;2.25,1.46,;2.65,-.03,;4.14,.37,;4.54,-1.12,;3.05,-1.51,;5.87,-1.89,;6.27,-3.37,;7.76,-2.97,;7.36,-1.49,;1.16,-.42,)|

CC1(CC1)C1CC2(C1)CN(C2)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:13.15,wD:15.18,(7.48,-1.19,;6.15,-1.96,;5.38,-3.3,;6.92,-3.3,;4.81,-1.19,;4.42,.3,;2.93,-.1,;3.33,-1.59,;2.53,1.38,;1.04,.99,;1.44,-.5,;-.29,1.76,;-.29,3.3,;-1.63,.99,;-2.02,-.5,;-3.51,-.1,;-3.11,1.38,;-3.67,-1.63,;-5.18,-1.95,;-5.95,-.62,;-7.48,-.46,;-4.92,.52,)|

CN([C@H]1C[C@H](C1)c1ccccc1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:14.15,2.1,4.6,wD:16.18,$;;;;;;;;;;;;;;;;;;;;;;HN$,(.65,-2.54,;.65,-1,;1.98,-.23,;2.38,1.26,;3.87,.86,;3.47,-.63,;5.2,1.63,;6.54,.86,;7.87,1.63,;7.87,3.17,;6.54,3.94,;5.2,3.17,;-.68,-.23,;-.68,1.31,;-2.02,-1,;-2.42,-2.49,;-3.9,-2.09,;-3.5,-.6,;-4.06,-3.62,;-5.57,-3.94,;-6.34,-2.61,;-7.87,-2.45,;-5.31,-1.46,)|

CN([C@H]1C[C@@H](C1)c1ccccc1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:14.15,2.1,wD:16.18,4.6,$;;;;;;;;;;;;;;;;;;;;;;HN$,(.65,-2.54,;.65,-1,;1.98,-.23,;2.38,1.26,;3.87,.86,;3.47,-.63,;5.2,1.63,;6.54,.86,;7.87,1.63,;7.87,3.17,;6.54,3.94,;5.2,3.17,;-.68,-.23,;-.68,1.31,;-2.02,-1,;-2.42,-2.49,;-3.9,-2.09,;-3.5,-.6,;-4.06,-3.62,;-5.57,-3.94,;-6.34,-2.61,;-7.87,-2.45,;-5.31,-1.46,)|

CN([C@H]1C[C@H](C1)c1cccc(c1)C1CCC1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.20,2.1,4.6,wD:20.23,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.96,-2.54,;-.96,-1,;.37,-.23,;.77,1.26,;2.26,.86,;1.86,-.63,;3.59,1.63,;3.59,3.17,;4.93,3.94,;6.26,3.17,;6.26,1.63,;4.93,.86,;7.6,.86,;7.99,-.63,;9.48,-.23,;9.08,1.26,;-2.29,-.23,;-2.29,1.31,;-3.63,-1,;-4.03,-2.49,;-5.51,-2.09,;-5.11,-.6,;-5.67,-3.62,;-7.18,-3.94,;-7.95,-2.61,;-9.48,-2.45,;-6.92,-1.46,)|

CN([C@H]1C[C@H](C1)c1ccc(cc1)C(C)(C)C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.19,2.1,4.6,wD:20.22,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.68,-3.31,;-.68,-1.77,;.65,-1,;1.05,.49,;2.54,.09,;2.14,-1.4,;3.87,.86,;5.2,.09,;6.54,.86,;6.54,2.4,;5.2,3.17,;3.87,2.4,;7.87,3.17,;9.21,2.4,;7.87,4.71,;9.21,3.94,;-2.02,-1,;-2.02,.54,;-3.35,-1.77,;-3.75,-3.26,;-5.24,-2.86,;-4.84,-1.37,;-5.4,-4.39,;-6.9,-4.71,;-7.67,-3.38,;-9.21,-3.22,;-6.64,-2.23,)|

CN([C@H]1C[C@@H](C1)c1ccc(cc1)C(C)(C)C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.19,2.1,wD:20.22,4.6,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.68,-3.31,;-.68,-1.77,;.65,-1,;1.05,.49,;2.54,.09,;2.14,-1.4,;3.87,.86,;5.2,.09,;6.54,.86,;6.54,2.4,;5.2,3.17,;3.87,2.4,;7.87,3.17,;9.21,2.4,;7.87,4.71,;9.21,3.94,;-2.02,-1,;-2.02,.54,;-3.35,-1.77,;-3.75,-3.26,;-5.24,-2.86,;-4.84,-1.37,;-5.4,-4.39,;-6.9,-4.71,;-7.67,-3.38,;-9.21,-3.22,;-6.64,-2.23,)|

CN([C@H]1C[C@H](C1)c1cccc(c1)C(C)(C)C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.19,2.1,4.6,wD:20.22,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.68,-2.54,;-.68,-1,;.65,-.23,;1.05,1.26,;2.54,.86,;2.14,-.63,;3.87,1.63,;3.87,3.17,;5.2,3.94,;6.54,3.17,;6.54,1.63,;5.2,.86,;7.87,.86,;9.21,1.63,;7.87,-.68,;9.21,.09,;-2.02,-.23,;-2.02,1.31,;-3.35,-1,;-3.75,-2.49,;-5.24,-2.09,;-4.84,-.6,;-5.4,-3.62,;-6.9,-3.94,;-7.67,-2.61,;-9.21,-2.45,;-6.64,-1.46,)|

CN([C@H]1C[C@H](C1)c1cccc(c1)C(C)(C)C)C(=O)[C@H]1C[C@@]2(C1)CCC(=O)N2 |r,wU:18.19,2.1,4.6,wD:20.22,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.68,-2.54,;-.68,-1,;.65,-.23,;1.05,1.26,;2.54,.86,;2.14,-.63,;3.87,1.63,;3.87,3.17,;5.2,3.94,;6.54,3.17,;6.54,1.63,;5.2,.86,;7.87,.86,;9.21,1.63,;7.87,-.68,;9.21,.09,;-2.02,-.23,;-2.02,1.31,;-3.35,-1,;-3.75,-2.49,;-5.24,-2.09,;-4.84,-.6,;-5.4,-3.62,;-6.9,-3.94,;-7.67,-2.61,;-9.21,-2.45,;-6.64,-1.46,)|

CN([C@H]1C[C@H](C1)c1cc(C)cc(C)c1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:16.17,2.1,4.6,wD:18.20,$;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.02,-3.31,;-.02,-1.77,;1.32,-1,;1.72,.49,;3.2,.09,;2.81,-1.4,;4.54,.86,;5.87,.09,;7.2,.86,;8.54,.09,;7.2,2.4,;5.87,3.17,;5.87,4.71,;4.54,2.4,;-1.35,-1,;-1.35,.54,;-2.68,-1.77,;-3.08,-3.26,;-4.57,-2.86,;-4.17,-1.37,;-4.73,-4.39,;-6.24,-4.71,;-7.01,-3.38,;-8.54,-3.22,;-5.98,-2.23,)|

CN([C@H]1C[C@@H](C1)c1cc(C)cc(C)c1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:16.17,2.1,wD:18.20,4.6,$;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.02,-3.31,;-.02,-1.77,;1.32,-1,;1.72,.49,;3.2,.09,;2.81,-1.4,;4.54,.86,;5.87,.09,;7.2,.86,;8.54,.09,;7.2,2.4,;5.87,3.17,;5.87,4.71,;4.54,2.4,;-1.35,-1,;-1.35,.54,;-2.68,-1.77,;-3.08,-3.26,;-4.57,-2.86,;-4.17,-1.37,;-4.73,-4.39,;-6.24,-4.71,;-7.01,-3.38,;-8.54,-3.22,;-5.98,-2.23,)|

CC(C)c1cccc(c1)[C@@H]1C[C@@H](C1)N(C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:17.18,11.14,9.9,wD:19.21,$;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(9.21,1.63,;7.87,.86,;7.87,-.68,;6.54,1.63,;6.54,3.17,;5.2,3.94,;3.87,3.17,;3.87,1.63,;5.2,.86,;2.54,.86,;1.05,1.26,;.65,-.23,;2.14,-.63,;-.68,-1,;-.68,-2.54,;-2.02,-.23,;-2.02,1.31,;-3.35,-1,;-3.75,-2.49,;-5.24,-2.09,;-4.84,-.6,;-5.4,-3.62,;-6.9,-3.94,;-7.67,-2.61,;-9.21,-2.45,;-6.64,-1.46,)|

COc1cccc(c1)[C@@H]1C[C@@H](C1)N(C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:16.17,10.13,8.8,wD:18.20,$;;;;;;;;;;;;;;;;;;;;;;;;HN$,(9.21,1.63,;7.87,.86,;6.54,1.63,;6.54,3.17,;5.2,3.94,;3.87,3.17,;3.87,1.63,;5.2,.86,;2.54,.86,;1.05,1.26,;.65,-.23,;2.14,-.63,;-.68,-1,;-.68,-2.54,;-2.02,-.23,;-2.02,1.31,;-3.35,-1,;-3.75,-2.49,;-5.24,-2.09,;-4.84,-.6,;-5.4,-3.62,;-6.9,-3.94,;-7.67,-2.61,;-9.21,-2.45,;-6.64,-1.46,)|

COc1cccc(c1)[C@H]1C[C@@H](C1)N(C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:16.17,10.13,wD:18.20,8.8,$;;;;;;;;;;;;;;;;;;;;;;;;HN$,(9.21,1.63,;7.87,.86,;6.54,1.63,;6.54,3.17,;5.2,3.94,;3.87,3.17,;3.87,1.63,;5.2,.86,;2.54,.86,;1.05,1.26,;.65,-.23,;2.14,-.63,;-.68,-1,;-.68,-2.54,;-2.02,-.23,;-2.02,1.31,;-3.35,-1,;-3.75,-2.49,;-5.24,-2.09,;-4.84,-.6,;-5.4,-3.62,;-6.9,-3.94,;-7.67,-2.61,;-9.21,-2.45,;-6.64,-1.46,)|

CC(C)c1ccc(cc1)[C@@H]1C[C@@H](C1)N(C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:17.18,11.14,9.9,wD:19.21,$;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(9.21,2.4,;7.87,3.17,;7.87,4.71,;6.54,2.4,;6.54,.86,;5.2,.09,;3.87,.86,;3.87,2.4,;5.2,3.17,;2.54,.09,;1.05,.49,;.65,-1,;2.14,-1.4,;-.68,-1.77,;-.68,-3.31,;-2.02,-1,;-2.02,.54,;-3.35,-1.77,;-3.75,-3.26,;-5.24,-2.86,;-4.84,-1.37,;-5.4,-4.39,;-6.9,-4.71,;-7.67,-3.38,;-9.21,-3.22,;-6.64,-2.23,)|

CN([C@H]1C[C@H](C1)c1ccc(F)c(c1)C(C)(C)C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:19.20,2.1,4.6,wD:21.23,$;;;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.68,-2.54,;-.68,-1,;.65,-.23,;1.05,1.26,;2.54,.86,;2.14,-.63,;3.87,1.63,;3.87,3.17,;5.2,3.94,;6.54,3.17,;7.87,3.94,;6.54,1.63,;5.2,.86,;7.87,.86,;9.21,1.63,;7.87,-.68,;9.21,.09,;-2.02,-.23,;-2.02,1.31,;-3.35,-1,;-3.75,-2.49,;-5.24,-2.09,;-4.84,-.6,;-5.4,-3.62,;-6.9,-3.94,;-7.67,-2.61,;-9.21,-2.45,;-6.64,-1.46,)|

CN([C@H]1C[C@H](C1)c1cccc(c1)C1(CC1)C(F)(F)F)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:23.26,wD:21.23,2.1,4.6,$;;;;;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(3.84,-1.32,;3.07,.01,;1.53,.01,;.44,1.1,;-.65,.01,;.44,-1.08,;-2.19,.01,;-2.96,1.35,;-4.5,1.35,;-5.27,.01,;-4.5,-1.32,;-2.96,-1.32,;-5.27,-2.66,;-6.45,-3.65,;-6.71,-2.13,;-4.09,-3.65,;-2.91,-4.64,;-5.08,-4.83,;-3.1,-2.47,;3.84,1.35,;3.07,2.68,;5.38,1.35,;6.47,.26,;7.56,1.35,;6.47,2.43,;8.47,.1,;9.93,.58,;9.93,2.12,;11.18,3.02,;8.47,2.59,)|

CN([C@H]1C[C@@H](C1)c1cccc(c1)C1(CC1)C(F)(F)F)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:23.26,4.6,wD:21.23,2.1,$;;;;;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(3.84,-1.32,;3.07,.01,;1.53,.01,;.44,1.1,;-.65,.01,;.44,-1.08,;-2.19,.01,;-2.96,1.35,;-4.5,1.35,;-5.27,.01,;-4.5,-1.32,;-2.96,-1.32,;-5.27,-2.66,;-6.45,-3.65,;-6.71,-2.13,;-4.09,-3.65,;-2.91,-4.64,;-5.08,-4.83,;-3.1,-2.47,;3.84,1.35,;3.07,2.68,;5.38,1.35,;6.47,.26,;7.56,1.35,;6.47,2.43,;8.47,.1,;9.93,.58,;9.93,2.12,;11.18,3.02,;8.47,2.59,)|

CN([C@H]1C[C@H](C1)c1ccccc1C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:15.16,2.1,4.6,wD:17.19,$;;;;;;;;;;;;;;;;;;;;;;;HN$,(.65,-2.54,;.65,-1,;1.98,-.23,;2.38,1.26,;3.87,.86,;3.47,-.63,;5.2,1.63,;5.2,3.17,;6.54,3.94,;7.87,3.17,;7.87,1.63,;6.54,.86,;6.54,-.68,;-.68,-.23,;-.68,1.31,;-2.02,-1,;-2.42,-2.49,;-3.9,-2.09,;-3.5,-.6,;-4.06,-3.62,;-5.57,-3.94,;-6.34,-2.61,;-7.87,-2.45,;-5.31,-1.46,)|

CN([C@H]1C[C@@H](C1)c1ccccc1C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:15.16,2.1,wD:17.19,4.6,$;;;;;;;;;;;;;;;;;;;;;;;HN$,(.65,-2.54,;.65,-1,;1.98,-.23,;2.38,1.26,;3.87,.86,;3.47,-.63,;5.2,1.63,;5.2,3.17,;6.54,3.94,;7.87,3.17,;7.87,1.63,;6.54,.86,;6.54,-.68,;-.68,-.23,;-.68,1.31,;-2.02,-1,;-2.42,-2.49,;-3.9,-2.09,;-3.5,-.6,;-4.06,-3.62,;-5.57,-3.94,;-6.34,-2.61,;-7.87,-2.45,;-5.31,-1.46,)|

CN([C@H]1C[C@H](C1)c1cccc(C)c1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:15.16,2.1,4.6,wD:17.19,$;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.02,-2.54,;-.02,-1,;1.32,-.23,;1.72,1.26,;3.2,.86,;2.81,-.63,;4.54,1.63,;4.54,3.17,;5.87,3.94,;7.2,3.17,;7.2,1.63,;8.54,.86,;5.87,.86,;-1.35,-.23,;-1.35,1.31,;-2.68,-1,;-3.08,-2.49,;-4.57,-2.09,;-4.17,-.6,;-4.73,-3.62,;-6.24,-3.94,;-7.01,-2.61,;-8.54,-2.45,;-5.98,-1.46,)|

CN([C@H]1C[C@@H](C1)c1cccc(C)c1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:15.16,2.1,wD:17.19,4.6,$;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.02,-2.54,;-.02,-1,;1.32,-.23,;1.72,1.26,;3.2,.86,;2.81,-.63,;4.54,1.63,;4.54,3.17,;5.87,3.94,;7.2,3.17,;7.2,1.63,;8.54,.86,;5.87,.86,;-1.35,-.23,;-1.35,1.31,;-2.68,-1,;-3.08,-2.49,;-4.57,-2.09,;-4.17,-.6,;-4.73,-3.62,;-6.24,-3.94,;-7.01,-2.61,;-8.54,-2.45,;-5.98,-1.46,)|

CCc1cccc(c1)[C@@H]1C[C@@H](C1)N(C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:16.17,10.13,8.8,wD:18.20,$;;;;;;;;;;;;;;;;;;;;;;;;HN$,(9.21,1.63,;7.87,.86,;6.54,1.63,;6.54,3.17,;5.2,3.94,;3.87,3.17,;3.87,1.63,;5.2,.86,;2.54,.86,;1.05,1.26,;.65,-.23,;2.14,-.63,;-.68,-1,;-.68,-2.54,;-2.02,-.23,;-2.02,1.31,;-3.35,-1,;-3.75,-2.49,;-5.24,-2.09,;-4.84,-.6,;-5.4,-3.62,;-6.9,-3.94,;-7.67,-2.61,;-9.21,-2.45,;-6.64,-1.46,)|

CN([C@H]1C[C@H](C1)c1cccc(C)c1C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:16.17,2.1,4.6,wD:18.20,$;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.02,-2.54,;-.02,-1,;1.32,-.23,;1.72,1.26,;3.2,.86,;2.81,-.63,;4.54,1.63,;4.54,3.17,;5.87,3.94,;7.2,3.17,;7.2,1.63,;8.54,.86,;5.87,.86,;5.87,-.68,;-1.35,-.23,;-1.35,1.31,;-2.68,-1,;-3.08,-2.49,;-4.57,-2.09,;-4.17,-.6,;-4.73,-3.62,;-6.24,-3.94,;-7.01,-2.61,;-8.54,-2.45,;-5.98,-1.46,)|

CN([C@H]1C[C@@H](C1)c1cccc(C)c1C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:16.17,2.1,wD:18.20,4.6,$;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.02,-2.54,;-.02,-1,;1.32,-.23,;1.72,1.26,;3.2,.86,;2.81,-.63,;4.54,1.63,;4.54,3.17,;5.87,3.94,;7.2,3.17,;7.2,1.63,;8.54,.86,;5.87,.86,;5.87,-.68,;-1.35,-.23,;-1.35,1.31,;-2.68,-1,;-3.08,-2.49,;-4.57,-2.09,;-4.17,-.6,;-4.73,-3.62,;-6.24,-3.94,;-7.01,-2.61,;-8.54,-2.45,;-5.98,-1.46,)|

CN([C@H]1C[C@H](C1)c1ccc(cc1)C1CC1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:17.19,2.1,4.6,wD:19.22,$;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.79,-3.21,;-.79,-1.67,;.55,-.9,;.95,.59,;2.43,.19,;2.04,-1.29,;3.77,.96,;5.1,.19,;6.43,.96,;6.43,2.5,;5.1,3.27,;3.77,2.5,;7.77,3.27,;9.31,3.27,;8.54,4.61,;-2.12,-.9,;-2.12,.64,;-3.45,-1.67,;-3.85,-3.15,;-5.34,-2.75,;-4.94,-1.27,;-5.5,-4.29,;-7.01,-4.61,;-7.78,-3.27,;-9.31,-3.11,;-6.75,-2.13,)|

CN([C@H]1C[C@H](C1)c1ccc(C)c(C)c1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:16.17,2.1,4.6,wD:18.20,$;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.02,-2.54,;-.02,-1,;1.32,-.23,;1.72,1.26,;3.2,.86,;2.81,-.63,;4.54,1.63,;4.54,3.17,;5.87,3.94,;7.2,3.17,;8.54,3.94,;7.2,1.63,;8.54,.86,;5.87,.86,;-1.35,-.23,;-1.35,1.31,;-2.68,-1,;-3.08,-2.49,;-4.57,-2.09,;-4.17,-.6,;-4.73,-3.62,;-6.24,-3.94,;-7.01,-2.61,;-8.54,-2.45,;-5.98,-1.46,)|

CC(C)c1ccc(cc1F)[C@@H]1C[C@@H](C1)N(C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.19,12.15,10.10,wD:20.22,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(9.21,2.4,;7.87,3.17,;7.87,4.71,;6.54,2.4,;5.2,3.17,;3.87,2.4,;3.87,.86,;5.2,.09,;6.54,.86,;7.87,.09,;2.54,.09,;1.05,.49,;.65,-1,;2.14,-1.4,;-.68,-1.77,;-.68,-3.31,;-2.02,-1,;-2.02,.54,;-3.35,-1.77,;-3.75,-3.26,;-5.24,-2.86,;-4.84,-1.37,;-5.4,-4.39,;-6.9,-4.71,;-7.67,-3.38,;-9.21,-3.22,;-6.64,-2.23,)|

CC(C)c1cc(ccc1F)[C@@H]1C[C@@H](C1)N(C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.19,12.15,10.10,wD:20.22,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(9.21,1.63,;7.87,.86,;7.87,-.68,;6.54,1.63,;5.2,.86,;3.87,1.63,;3.87,3.17,;5.2,3.94,;6.54,3.17,;7.87,3.94,;2.54,.86,;1.05,1.26,;.65,-.23,;2.14,-.63,;-.68,-1,;-.68,-2.54,;-2.02,-.23,;-2.02,1.31,;-3.35,-1,;-3.75,-2.49,;-5.24,-2.09,;-4.84,-.6,;-5.4,-3.62,;-6.9,-3.94,;-7.67,-2.61,;-9.21,-2.45,;-6.64,-1.46,)|

CN([C@H]1C[C@H](C1)c1ccc(C)cc1C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:16.17,2.1,4.6,wD:18.20,$;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.02,-2.54,;-.02,-1,;1.32,-.23,;1.72,1.26,;3.2,.86,;2.81,-.63,;4.54,1.63,;4.54,3.17,;5.87,3.94,;7.2,3.17,;8.54,3.94,;7.2,1.63,;5.87,.86,;5.87,-.68,;-1.35,-.23,;-1.35,1.31,;-2.68,-1,;-3.08,-2.49,;-4.57,-2.09,;-4.17,-.6,;-4.73,-3.62,;-6.24,-3.94,;-7.01,-2.61,;-8.54,-2.45,;-5.98,-1.46,)|

CCc1ccc(cc1)[C@@H]1C[C@@H](C1)N(C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:16.17,10.13,8.8,wD:18.20,$;;;;;;;;;;;;;;;;;;;;;;;;HN$,(9.21,3.17,;7.87,3.94,;6.54,3.17,;6.54,1.63,;5.2,.86,;3.87,1.63,;3.87,3.17,;5.2,3.94,;2.54,.86,;1.05,1.26,;.65,-.23,;2.14,-.63,;-.68,-1,;-.68,-2.54,;-2.02,-.23,;-2.02,1.31,;-3.35,-1,;-3.75,-2.49,;-5.24,-2.09,;-4.84,-.6,;-5.4,-3.62,;-6.9,-3.94,;-7.67,-2.61,;-9.21,-2.45,;-6.64,-1.46,)|

CCc1ccc(cc1C)[C@@H]1C[C@@H](C1)N(C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:17.18,11.14,9.9,wD:19.21,$;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(9.21,3.17,;7.87,3.94,;6.54,3.17,;5.2,3.94,;3.87,3.17,;3.87,1.63,;5.2,.86,;6.54,1.63,;7.87,.86,;2.54,.86,;1.05,1.26,;.65,-.23,;2.14,-.63,;-.68,-1,;-.68,-2.54,;-2.02,-.23,;-2.02,1.31,;-3.35,-1,;-3.75,-2.49,;-5.24,-2.09,;-4.84,-.6,;-5.4,-3.62,;-6.9,-3.94,;-7.67,-2.61,;-9.21,-2.45,;-6.64,-1.46,)|

CN([C@H]1C[C@H](C1)c1ccc(C2CC2)c(C)c1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.20,2.1,4.6,wD:20.23,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.79,-3.21,;-.79,-1.67,;.55,-.9,;.95,.59,;2.43,.19,;2.04,-1.29,;3.77,.96,;3.77,2.5,;5.1,3.27,;6.43,2.5,;7.77,3.27,;9.31,3.27,;8.54,4.61,;6.43,.96,;7.77,.19,;5.1,.19,;-2.12,-.9,;-2.12,.64,;-3.45,-1.67,;-3.85,-3.15,;-5.34,-2.75,;-4.94,-1.27,;-5.5,-4.29,;-7.01,-4.61,;-7.78,-3.27,;-9.31,-3.11,;-6.75,-2.13,)|

CN([C@H]1C[C@H](C1)c1ccc(C)c(c1)C1CC1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.20,2.1,4.6,wD:20.23,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.79,-2.54,;-.79,-1,;.55,-.23,;.95,1.26,;2.43,.86,;2.04,-.63,;3.77,1.63,;3.77,3.17,;5.1,3.94,;6.43,3.17,;7.77,3.94,;6.43,1.63,;5.1,.86,;7.77,.86,;8.54,-.47,;9.31,.86,;-2.12,-.23,;-2.12,1.31,;-3.45,-1,;-3.85,-2.49,;-5.34,-2.09,;-4.94,-.6,;-5.5,-3.62,;-7.01,-3.94,;-7.78,-2.61,;-9.31,-2.45,;-6.75,-1.46,)|

CN([C@H]1C[C@H](C1)c1ccc2CCCCc2c1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.20,2.1,4.6,wD:20.23,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.68,-2.54,;-.68,-1,;.65,-.23,;1.05,1.26,;2.54,.86,;2.14,-.63,;3.87,1.63,;3.87,3.17,;5.2,3.94,;6.54,3.17,;7.87,3.94,;9.21,3.17,;9.21,1.63,;7.87,.86,;6.54,1.63,;5.2,.86,;-2.02,-.23,;-2.02,1.31,;-3.35,-1,;-3.75,-2.49,;-5.24,-2.09,;-4.84,-.6,;-5.4,-3.62,;-6.9,-3.94,;-7.67,-2.61,;-9.21,-2.45,;-6.64,-1.46,)|

CN([C@@H]1C[C@H](Cc2ccccc2)C1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:15.16,2.1,4.4,wD:17.19,$;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.02,-1.38,;-.02,.16,;1.32,.93,;2.81,.53,;3.2,2.01,;4.54,2.78,;5.87,2.01,;5.87,.47,;7.2,-.3,;8.54,.47,;8.54,2.01,;7.2,2.78,;1.72,2.41,;-1.35,.93,;-1.35,2.47,;-2.68,.16,;-3.08,-1.33,;-4.57,-.93,;-4.17,.55,;-4.73,-2.46,;-6.24,-2.78,;-7.01,-1.45,;-8.54,-1.29,;-5.98,-.31,)|

CN([C@H]1C[C@H](Cc2ccccc2)C1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:15.16,2.1,wD:17.19,4.4,$;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.02,-1.38,;-.02,.16,;1.32,.93,;1.72,2.41,;3.2,2.01,;4.54,2.78,;5.87,2.01,;5.87,.47,;7.2,-.3,;8.54,.47,;8.54,2.01,;7.2,2.78,;2.81,.53,;-1.35,.93,;-1.35,2.47,;-2.68,.16,;-3.08,-1.33,;-4.57,-.93,;-4.17,.55,;-4.73,-2.46,;-6.24,-2.78,;-7.01,-1.45,;-8.54,-1.29,;-5.98,-.31,)|

CN([C@H]1C[C@H](C1)C(C)(C)C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:12.12,2.1,4.6,wD:14.15,$;;;;;;;;;;;;;;;;;;;;HN$,(1.32,-2.15,;1.32,-.61,;2.65,.16,;3.05,1.64,;4.54,1.24,;4.14,-.24,;5.87,2.01,;7.2,1.24,;5.87,3.55,;7.2,2.78,;-.02,.16,;-.02,1.7,;-1.35,-.61,;-1.75,-2.1,;-3.24,-1.7,;-2.84,-.22,;-3.4,-3.23,;-4.9,-3.55,;-5.67,-2.22,;-7.2,-2.06,;-4.64,-1.08,)|

CN([C@H]1C[C@@H](C1)C(C)(C)C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:12.12,2.1,wD:14.15,4.6,$;;;;;;;;;;;;;;;;;;;;HN$,(1.32,-2.15,;1.32,-.61,;2.65,.16,;3.05,1.64,;4.54,1.24,;4.14,-.24,;5.87,2.01,;7.2,1.24,;5.87,3.55,;7.2,2.78,;-.02,.16,;-.02,1.7,;-1.35,-.61,;-1.75,-2.1,;-3.24,-1.7,;-2.84,-.22,;-3.4,-3.23,;-4.9,-3.55,;-5.67,-2.22,;-7.2,-2.06,;-4.64,-1.08,)|

CN([C@@H]1C[C@@H](C1)C1CCCCC1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:14.15,2.1,4.6,wD:16.18,$;;;;;;;;;;;;;;;;;;;;;;HN$,(.65,-2.54,;.65,-1,;1.98,-.23,;3.47,-.63,;3.87,.86,;2.38,1.26,;5.2,1.63,;6.54,.86,;7.87,1.63,;7.87,3.17,;6.54,3.94,;5.2,3.17,;-.68,-.23,;-.68,1.31,;-2.02,-1,;-2.42,-2.49,;-3.9,-2.09,;-3.5,-.6,;-4.06,-3.62,;-5.57,-3.94,;-6.34,-2.61,;-7.87,-2.45,;-5.31,-1.46,)|

CN([C@H]1C[C@@H](C1)C1CCCCC1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:14.15,2.1,wD:16.18,4.6,$;;;;;;;;;;;;;;;;;;;;;;HN$,(.65,-2.54,;.65,-1,;1.98,-.23,;2.38,1.26,;3.87,.86,;3.47,-.63,;5.2,1.63,;6.54,.86,;7.87,1.63,;7.87,3.17,;6.54,3.94,;5.2,3.17,;-.68,-.23,;-.68,1.31,;-2.02,-1,;-2.42,-2.49,;-3.9,-2.09,;-3.5,-.6,;-4.06,-3.62,;-5.57,-3.94,;-6.34,-2.61,;-7.87,-2.45,;-5.31,-1.46,)|

CN([C@H]1C[C@H](C1)c1ccc(cc1)C1(C)CC1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.20,2.1,4.6,wD:20.23,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.68,-3.21,;-.68,-1.67,;.65,-.9,;1.05,.59,;2.54,.19,;2.14,-1.29,;3.87,.96,;5.2,.19,;6.54,.96,;6.54,2.5,;5.2,3.27,;3.87,2.5,;7.87,3.27,;9.21,2.5,;8.64,4.61,;7.1,4.61,;-2.02,-.9,;-2.02,.64,;-3.35,-1.67,;-3.75,-3.15,;-5.24,-2.75,;-4.84,-1.27,;-5.4,-4.29,;-6.9,-4.61,;-7.67,-3.27,;-9.21,-3.11,;-6.64,-2.13,)|

CCC(C)c1ccc(cc1)[C@@H]1C[C@@H](C1)N(C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.19,12.15,10.10,wD:20.22,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(9.87,3.17,;8.54,2.4,;7.2,3.17,;7.2,4.71,;5.87,2.4,;5.87,.86,;4.54,.09,;3.2,.86,;3.2,2.4,;4.54,3.17,;1.87,.09,;.38,.49,;-.02,-1,;1.47,-1.4,;-1.35,-1.77,;-1.35,-3.31,;-2.68,-1,;-2.68,.54,;-4.02,-1.77,;-4.42,-3.26,;-5.9,-2.86,;-5.5,-1.37,;-6.06,-4.39,;-7.57,-4.71,;-8.34,-3.38,;-9.87,-3.22,;-7.31,-2.23,)|

CN([C@H]1C[C@H](C1)c1cccc(c1)C1(C)CC1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.20,2.1,4.6,wD:20.23,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.68,-2.54,;-.68,-1,;.65,-.23,;1.05,1.26,;2.54,.86,;2.14,-.63,;3.87,1.63,;3.87,3.17,;5.2,3.94,;6.54,3.17,;6.54,1.63,;5.2,.86,;7.87,.86,;9.21,1.63,;7.1,-.47,;8.64,-.47,;-2.02,-.23,;-2.02,1.31,;-3.35,-1,;-3.75,-2.49,;-5.24,-2.09,;-4.84,-.6,;-5.4,-3.62,;-6.9,-3.94,;-7.67,-2.61,;-9.21,-2.45,;-6.64,-1.46,)|

CCc1cc(C)cc(c1)[C@@H]1C[C@@H](C1)N(C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:17.18,11.14,9.9,wD:19.21,$;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(9.21,.86,;7.87,.09,;6.54,.86,;6.54,2.4,;5.2,3.17,;5.2,4.71,;3.87,2.4,;3.87,.86,;5.2,.09,;2.54,.09,;1.05,.49,;.65,-1,;2.14,-1.4,;-.68,-1.77,;-.68,-3.31,;-2.02,-1,;-2.02,.54,;-3.35,-1.77,;-3.75,-3.26,;-5.24,-2.86,;-4.84,-1.37,;-5.4,-4.39,;-6.9,-4.71,;-7.67,-3.38,;-9.21,-3.22,;-6.64,-2.23,)|

CN([C@H]1C[C@H](C1)c1cc(C)cc(c1)C1CC1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.20,2.1,4.6,wD:20.23,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.79,-3.31,;-.79,-1.77,;.55,-1,;.95,.49,;2.43,.09,;2.04,-1.4,;3.77,.86,;3.77,2.4,;5.1,3.17,;5.1,4.71,;6.43,2.4,;6.43,.86,;5.1,.09,;7.77,.09,;8.54,-1.24,;9.31,.09,;-2.12,-1,;-2.12,.54,;-3.45,-1.77,;-3.85,-3.26,;-5.34,-2.86,;-4.94,-1.37,;-5.5,-4.39,;-7.01,-4.71,;-7.78,-3.38,;-9.31,-3.22,;-6.75,-2.23,)|

CC(C)c1cc(C)cc(c1)[C@@H]1C[C@@H](C1)N(C)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:18.19,12.15,10.10,wD:20.22,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(9.21,.86,;7.87,.09,;7.87,-1.45,;6.54,.86,;6.54,2.4,;5.2,3.17,;5.2,4.71,;3.87,2.4,;3.87,.86,;5.2,.09,;2.54,.09,;1.05,.49,;.65,-1,;2.14,-1.4,;-.68,-1.77,;-.68,-3.31,;-2.02,-1,;-2.02,.54,;-3.35,-1.77,;-3.75,-3.26,;-5.24,-2.86,;-4.84,-1.37,;-5.4,-4.39,;-6.9,-4.71,;-7.67,-3.38,;-9.21,-3.22,;-6.64,-2.23,)|

CN([C@H]1C[C@H](C1)c1cc(C)cc(Cl)c1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:16.17,2.1,4.6,wD:18.20,$;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.02,-3.31,;-.02,-1.77,;1.32,-1,;1.72,.49,;3.2,.09,;2.81,-1.4,;4.54,.86,;4.54,2.4,;5.87,3.17,;5.87,4.71,;7.2,2.4,;7.2,.86,;8.54,.09,;5.87,.09,;-1.35,-1,;-1.35,.54,;-2.68,-1.77,;-3.08,-3.26,;-4.57,-2.86,;-4.17,-1.37,;-4.73,-4.39,;-6.24,-4.71,;-7.01,-3.38,;-8.54,-3.22,;-5.98,-2.23,)|

CN([C@H]1C[C@H](C1)c1cccc(c1)C1CC1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:17.19,2.1,4.6,wD:19.22,$;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.79,-2.54,;-.79,-1,;.55,-.23,;.95,1.26,;2.43,.86,;2.04,-.63,;3.77,1.63,;3.77,3.17,;5.1,3.94,;6.43,3.17,;6.43,1.63,;5.1,.86,;7.77,.86,;8.54,-.47,;9.31,.86,;-2.12,-.23,;-2.12,1.31,;-3.45,-1,;-3.85,-2.49,;-5.34,-2.09,;-4.94,-.6,;-5.5,-3.62,;-7.01,-3.94,;-7.78,-2.61,;-9.31,-2.45,;-6.75,-1.46,)|

CN([C@H]1C[C@H](C1)c1ccc2CCCc2c1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:17.19,2.1,4.6,wD:19.22,$;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.53,-2.54,;-.53,-1,;.8,-.23,;1.2,1.26,;2.69,.86,;2.29,-.63,;4.02,1.63,;4.02,3.17,;5.35,3.94,;6.69,3.17,;8.15,3.65,;9.06,2.4,;8.15,1.15,;6.69,1.63,;5.35,.86,;-1.87,-.23,;-1.87,1.31,;-3.2,-1,;-3.6,-2.49,;-5.09,-2.09,;-4.69,-.6,;-5.25,-3.62,;-6.75,-3.94,;-7.52,-2.61,;-9.06,-2.45,;-6.49,-1.46,)|

CN([C@H]1C[C@H](C1)c1ccc2CCc2c1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:16.18,2.1,4.6,wD:18.21,$;;;;;;;;;;;;;;;;;;;;;;;;HN$,(-.12,-2.54,;-.12,-1,;1.21,-.23,;1.61,1.26,;3.1,.86,;2.7,-.63,;4.43,1.63,;4.43,3.17,;5.77,3.94,;7.1,3.17,;8.64,3.17,;8.64,1.63,;7.1,1.63,;5.77,.86,;-1.45,-.23,;-1.45,1.31,;-2.79,-1,;-3.19,-2.49,;-4.67,-2.09,;-4.27,-.6,;-4.83,-3.62,;-6.34,-3.94,;-7.11,-2.61,;-8.64,-2.45,;-6.08,-1.46,)|

CCN([C@H]1C[C@H](C1)c1cc(C)cc(C)c1)C(=O)[C@H]1C[C@@]2(C1)COC(=O)N2 |r,wU:17.18,3.2,5.7,wD:19.21,$;;;;;;;;;;;;;;;;;;;;;;;;;HN$,(1.32,-4.08,;-.02,-3.31,;-.02,-1.77,;1.32,-1,;1.72,.49,;3.2,.09,;2.81,-1.4,;4.54,.86,;5.87,.09,;7.2,.86,;8.54,.09,;7.2,2.4,;5.87,3.17,;5.87,4.71,;4.54,2.4,;-1.35,-1,;-1.35,.54,;-2.68,-1.77,;-3.08,-3.26,;-4.57,-2.86,;-4.17,-1.37,;-4.73,-4.39,;-6.24,-4.71,;-7.01,-3.38,;-8.54,-3.22,;-5.98,-2.23,)|

Cn1nc2C3CCCC(Cc2c1-c1ccccc1)N3C(=O)c1ccc2ncccc2c1 |TLB:19:18:3.10.9:7.6.5|

Cn1cc2[C@@H]3CCC[C@H](Cc2c1C1CC1)N3C(=O)c1ccc2ncccc2c1 |r,TLB:16:15:3.10.9:7.6.5|

COc1cccc(C(=O)N2C3CCCC2c2cn(C)c(c2C3)-c2ccccc2)c1Cl |TLB:7:9:15.20.21:11.12.13|

COc1cccc(C(=O)N(C)C2CCCCCc3c2cn(C)c3-c2ccccc2)c1Cl

COc1cccc(C(=O)N2[C@@H]3CCC[C@H]2c2cn(C)c(c2C3)-c2ccccc2)c1Cl |r,TLB:7:9:15.20.21:11.12.13|

CN(C1CCCCCc2c1cn(C)c2-c1ccccc1)C(=O)c1ccccc1-n1cncn1

CN(C1CCCCCc2c1cn(C)c2-c1ccccc1)C(=O)c1cccc(c1)-n1cnnc1

CN(C1CCCCCc2c1cn(C)c2-c1ccccc1)C(=O)c1ccc(cc1)-n1cncn1

CN(C1CCCCCc2c1cn(C)c2-c1ccccc1)C(=O)c1cccc(c1)-n1ccnc1

Cn1cnc(n1)C(=O)N1C2CCCC1c1nn(C)c(c1C2)-c1ccccc1 |TLB:6:8:14.19.20:10.11.12|

Cn1ncc(C(=O)N2C3CCCC2c2nn(C)c(c2C3)-c2ccccc2)c1Cl |TLB:5:7:13.18.19:9.10.11|

COc1c(cnn1C)C(=O)N1C2CCCC1c1nn(C)c(c1C2)-c1ccccc1 |TLB:8:10:16.21.22:12.13.14|

Cn1nc(c(Br)c1C(=O)N1C2CCCC1c1nn(C)c(c1C2)-c1ccccc1)C(F)(F)F |TLB:7:9:15.20.21:11.12.13|

Cn1ncc(C(=O)N2C3CCCC2c2nn(C)c(c2C3)-c2ccccc2)c1C1CC1 |TLB:5:7:13.18.19:9.10.11|

Cn1nc2C3CCCC(Cc2c1-c1ccccc1)N3C(=O)c1ncn(n1)-c1ccccc1 |TLB:19:18:3.10.9:7.6.5|

Cn1nc2C3CCCC(Cc2c1-c1ccccc1)N3C(=O)c1ccn(n1)-c1ccccc1 |TLB:19:18:3.10.9:7.6.5|

COc1cc(nn1-c1ccccc1)C(=O)N1C2CCCC1c1nn(C)c(c1C2)-c1ccccc1 |TLB:13:15:21.26.27:17.18.19|

Cn1nc2C3CCCC(Cc2c1-c1ccccc1)N3C(=O)c1cccc2n(C)ccc12 |TLB:19:18:3.10.9:7.6.5|

Cn1nc2C3CCCC(Cc2c1-c1ccccc1)N3C(=O)c1cc2[nH]ccc2cc1Cl |TLB:19:18:3.10.9:7.6.5|

Cc1cc(cc2cn[nH]c12)C(=O)N1C2CCCC1c1nn(C)c(c1C2)-c1ccccc1 |TLB:10:12:18.23.24:14.15.16|

Cn1ccc2c(ccnc12)C(=O)N1C2CCCC1c1nn(C)c(c1C2)-c1ccccc1 |TLB:10:12:18.23.24:14.15.16|

Cn1nc2C3CCCC(Cc2c1-c1ccccc1)N3C(=O)c1cnc2[nH]ccc2c1Cl |TLB:19:18:3.10.9:7.6.5|

Cn1nc2C3CCCC(Cc2c1-c1ccccc1)N3C(=O)c1cnc2[nH]ccc2c1F |TLB:19:18:3.10.9:7.6.5|

Cn1cc(C(=O)N2C3CCCC2c2nn(C)c(c2C3)-c2ccccc2)c2cccnc12 |TLB:4:6:12.17.18:8.9.10|

Cn1nc2C3CCCC(Cc2c1-c1ccccc1)N3C(=O)c1cccc2ncnn12 |TLB:19:18:3.10.9:7.6.5|

Cn1nc2C3CCCC(Cc2c1-c1ccccc1)N3C(=O)c1ccc2nccc(Cl)c2c1 |TLB:19:18:3.10.9:7.6.5|

Cn1nc2C3CCCC(Cc2c1-c1ccccc1)N3C(=O)c1ccc2nccc(O)c2c1 |TLB:19:18:3.10.9:7.6.5|

Cn1nc2C3CCCC(Cc2c1-c1ccccc1)N3C(=O)c1cccc2nccnc12 |TLB:19:18:3.10.9:7.6.5|

Cn1nc2C3CCCC(Cc2c1-c1ccccc1)N3C(=O)c1ccc2nccnc2c1 |TLB:19:18:3.10.9:7.6.5|

Cn1nc2C3CCCC(Cc2c1-c1ccccc1)N3C(=O)c1ccc2ncncc2c1 |TLB:19:18:3.10.9:7.6.5|

[H][C@]12CCC[C@]([H])(N1C(=O)c1cc3cccnc3nc1C(F)(F)F)c1nn(C)c(c1C2)-c1ccccc1 |THB:8:7:30.29.24:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1cccc(OC)c1Cl)c1nn(C)c(c1C2)-c1ccc(F)cc1 |THB:8:7:25.24.19:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1ccccc1-n1nccn1)c1nn(C)c(c1C2)-c1ccc(F)cc1 |THB:8:7:27.26.21:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1nn(C)cc1C)c1nn(C)c(c1C2)-c1ccc(F)cc1 |THB:8:7:23.22.17:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1nn(C)c3ncccc13)c1nn(C)c(c1C2)-c1ccc(F)cc1 |THB:8:7:26.25.20:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1ccc3ncccc3c1)c1nn(C)c(c1C2)-c1ccc(F)cc1 |THB:8:7:26.25.20:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1cccc(OC)c1Cl)c1nn(C)c(c1C2)-c1cccc(F)c1 |THB:8:7:25.24.19:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1ncn(n1)-c1ccccc1)c1nn(C)c(c1C2)-c1cccc(F)c1 |THB:8:7:27.26.21:4.3.2|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cccc(F)c1)N3C(=O)c1cnc2ccoc2c1 |r,TLB:20:19:10.3.9:7.6.5|

[H][C@]12CCC[C@]([H])(N1C(=O)c1ccc3ncccc3c1)c1nn(C)c(c1C2)-c1cccc(F)c1 |THB:8:7:26.25.20:4.3.2|

[H][C@@]12CCC[C@@]([H])(N1C(=O)c1ccc3ncccc3c1)c1nn(C)c(c1C2)-c1cccc(F)c1 |THB:8:7:26.25.20:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1ccc3ncccc3c1)c1nn(C3CC3)c(c1C2)-c1cccc(F)c1 |THB:8:7:28.27.20:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1cccc(c1)-n1cncn1)c1nn(C)c(c1C2)-c1cccc(Cl)c1 |THB:8:7:27.26.21:4.3.2|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cccc(Cl)c1)N3C(=O)c1cccc(c1)-c1cn[nH]c1 |r,TLB:20:19:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cccc(Cl)c1)N3C(=O)c1cccc(c1)-n1cccn1 |r,TLB:20:19:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cccc(Cl)c1)N3C(=O)c1cccc(c1)-n1cnnn1 |r,TLB:20:19:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cccc(Cl)c1)N3C(=O)c1cc(ccc1Cl)-n1cnnc1 |r,TLB:20:19:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cccc(Cl)c1)N3C(=O)c1ccc(cc1)-n1cnnc1 |r,TLB:20:19:3.10.9:7.6.5|

CC(C)n1cnc(n1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cccc(Cl)c1 |r,TLB:8:10:16.21.22:12.13.14|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cccc(Cl)c1)N3C(=O)c1ncn(n1)-c1ccccc1F |r,TLB:20:19:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cccc(Cl)c1)N3C(=O)c1ncn(n1)-c1ccccn1 |r,TLB:20:19:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cccc(Cl)c1)N3C(=O)c1ncn(n1)-c1cccc(F)c1 |r,TLB:20:19:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cccc(Cl)c1)N3C(=O)c1ncn(n1)-c1cccc(Cl)c1 |r,TLB:20:19:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cccc(Cl)c1)N3C(=O)c1cnn(c1C(F)(F)F)-c1ccccc1 |r,TLB:20:19:3.10.9:7.6.5|

Cc1nc(nn1-c1cccc(c1)C(F)(F)F)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cccc(Cl)c1 |r,TLB:16:18:24.29.30:20.21.22|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cccc(Cl)c1)N3C(=O)c1ncn(n1)-c1cccc(c1)C(F)(F)F |r,TLB:20:19:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cccc(Cl)c1)N3C(=O)c1ncn(Cc2ccccc2)n1 |r,TLB:20:19:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cccc(Cl)c1)N3C(=O)c1noc2ccccc12 |r,TLB:20:19:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cccc(Cl)c1)N3C(=O)c1nn(C)c2ccccc12 |r,TLB:20:19:3.10.9:7.6.5|

Cn1nc2C3CCCC(Cc2c1-c1cccc(Cl)c1)N3C(=O)c1ccc2ncccc2c1 |TLB:20:19:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cccc(Cl)c1)N3C(=O)c1ccc2nccnc2c1 |r,TLB:20:19:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccc2nccc(OCCF)c2c1 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1cccc(OCCF)c1 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2C3CCCC(Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccccc1-n1nccn1 |TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccccc1-c1ncn[nH]1 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccccc1-c1nc(Cl)n[nH]1 |r,TLB:21:20:3.10.9:7.6.5|

Cn1cc(cn1)-c1cccc(c1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |r,TLB:12:14:20.25.26:16.17.18|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1cccc(c1)-n1cnnc1 |r,TLB:21:20:3.10.9:7.6.5|

Cc1ccc(c(c1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)cc(F)c1)-n1nccn1 |r,TLB:7:9:15.20.21:11.12.13|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1cccc(F)c1-n1nccn1 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1cccc(F)c1-c1ncco1 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2C3CCCC(Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccccc1-c1ncccn1 |TLB:21:20:3.10.9:7.6.5|

[H][C@]12CCC[C@]([H])(N1C(=O)c1cnn(C)c1OC)c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |THB:8:7:24.23.18:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1cc(n(CC)n1)C(F)(F)F)c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |THB:8:7:27.26.21:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1cn[nH]c1C1CC1)c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |THB:8:7:24.23.18:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1cnn(CCO)c1C1CC1)c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |THB:8:7:27.26.21:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1cn(CC(F)(F)F)nc1C1CC1)c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |THB:8:7:29.28.23:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1cnn(c1C1CC1)-c1ccccc1)c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |THB:8:7:30.29.24:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1cnn(c1C1CC1)-c1cccc(c1)C(F)(F)F)c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |THB:8:7:34.33.28:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1nc(C)n(n1)-c1ccccc1)c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |THB:8:7:28.27.22:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1nc(C)n(n1)-c1ccc(F)cc1)c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |THB:8:7:29.28.23:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1nc(CC)n(n1)-c1ccccc1)c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |THB:8:7:29.28.23:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1ccnc(F)c1)c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |THB:8:7:23.22.17:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1cncc(OC)c1)c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |THB:8:7:24.23.18:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1ccc(N)cn1)c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |THB:8:7:23.22.17:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1cc3cc(OC)ccc3o1)c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |THB:8:7:27.26.21:4.3.2|

[H][C@]12CCC[C@]([H])(N1C(=O)c1ccc3nc(C)oc3c1)c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |THB:8:7:26.25.20:4.3.2|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccc2nc(N)oc2c1 |r,TLB:21:20:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1cc2ncccc2o1 |r,TLB:21:20:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1cc2occc2cn1 |r,TLB:21:20:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1nn(C)c2ncccc12 |r,TLB:21:20:10.3.9:7.6.5|

Cn1nc2C3CCCC(Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccc2ncccc2c1 |TLB:21:20:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccc2ncccc2c1 |r,TLB:21:20:10.3.9:7.6.5|

Cn1nc2[C@@H]3CCC[C@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccc2ncccc2c1 |r,TLB:21:20:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1cc2ccccc2cn1 |r,TLB:21:20:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccc2ccncc2c1 |r,TLB:21:20:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccc2nccc(Br)c2c1 |r,TLB:21:20:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccc2ncc(Br)cc2c1 |r,TLB:21:20:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1cc(Br)c2ncccc2c1 |r,TLB:21:20:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccc2nc(Cl)ccc2c1 |r,TLB:21:20:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccc(F)c2ncccc12 |r,TLB:21:20:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1cc(F)c2ncccc2c1 |r,TLB:21:20:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccc2nc(ccc2c1)C(F)(F)F |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1cc(O)c2ncccc2c1 |r,TLB:21:20:3.10.9:7.6.5|

COc1cccc2ncc(cc12)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |r,TLB:12:14:20.25.26:16.17.18|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1cc([N+]([O-])=O)c2ncccc2c1 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1cc(N)c2ncccc2c1 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccc2cncnc2c1 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccc2nccnc2c1 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccc2ncncc2c1 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1cc2nccnc2cc1F |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1nccc2ncccc12 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1cnc2ncccc2c1 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccnc2ncccc12 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccnc2cnccc12 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccnc2ccncc12 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccc2ncccc2n1 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccc2n(CCF)ccc(=O)c2c1 |r,TLB:21:20:3.10.9:7.6.5|

CN1C(=O)COc2ccc(cc12)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |r,TLB:12:14:20.25.26:16.17.18|

CN1CCOc2cc(cnc12)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)cc(F)c1 |r,TLB:11:13:19.24.25:15.16.17|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1ccc(F)c(F)c1)N3C(=O)c1ccccc1-n1nccn1 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2C3CCCC(Cc2c1-c1ccc(F)c(F)c1)N3C(=O)c1ccc2ncccc2c1 |TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1ccc(F)c(F)c1)N3C(=O)c1ccc2ncccc2c1 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2C3CCCC(Cc2c1-c1ccc(F)c(F)c1)N3C(=O)c1ccc2nccnc2c1 |TLB:21:20:3.10.9:7.6.5|

COc1cc(F)cc(c1)-c1c2C[C@@H]3CCC[C@@H](N3C(=O)c3ccc4nccnc4c3)c2nn1C |r,TLB:18:17:30.10.11:13.14.15|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1ccc(Cl)c(F)c1)N3C(=O)c1ccc2nccnc2c1 |r,TLB:21:20:3.10.9:7.6.5|

COc1ccc(cc1Cl)-c1c2C[C@@H]3CCC[C@@H](N3C(=O)c3ccc4nccnc4c3)c2nn1C |r,TLB:18:17:30.10.11:13.14.15|

COc1ccc(cc1Cl)-c1c2C[C@@H]3CCC[C@@H](N3C(=O)c3ccccc3-n3nccn3)c2nn1C |r,TLB:18:17:31.10.11:13.14.15|

COc1ccc(cc1Cl)-c1c2C[C@@H]3CCC[C@@H](N3C(=O)c3nn(C)c4ncccc34)c2nn1C |r,TLB:18:17:30.10.11:13.14.15|

COc1ccc(cc1Cl)-c1c2C[C@@H]3CCC[C@@H](N3C(=O)c3ccc4ncccc4c3)c2nn1C |r,TLB:18:17:30.10.11:13.14.15|

COc1cc(Cl)cc(c1)-c1c2C[C@@H]3CCC[C@@H](N3C(=O)c3ccc4nc(C)oc4c3)c2nn1C |r,TLB:18:17:30.10.11:13.14.15|

COc1cc(Cl)cc(c1)-c1c2C[C@@H]3CCC[C@@H](N3C(=O)c3ccc4ncccc4c3)c2nn1C |r,TLB:18:17:30.10.11:13.14.15|

COc1cc(Cl)cc(c1)-c1c2C[C@@H]3CCC[C@@H](N3C(=O)c3ccc4nccnc4c3)c2nn1C |r,TLB:18:17:30.10.11:13.14.15|

COc1cc(OC)cc(c1)-c1c2C[C@@H]3CCC[C@@H](N3C(=O)c3ccc4nc(C)oc4c3)c2nn1C |r,TLB:19:18:31.11.12:14.15.16|

COc1cc(OC)cc(c1)-c1c2C[C@@H]3CCC[C@@H](N3C(=O)c3ccc4nccnc4c3)c2nn1C |r,TLB:19:18:31.11.12:14.15.16|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(Cl)cc(Cl)c1)N3C(=O)c1cccc(c1)-n1cnnc1 |r,TLB:21:20:3.10.9:7.6.5|

CN1CCOc2cc(cnc12)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(Cl)cc(Cl)c1 |r,TLB:11:13:19.24.25:15.16.17|

COc1c(cnn1C)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(Cl)cc(Cl)c1 |r,TLB:8:10:16.21.22:12.13.14|

Cn1ncc(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(Cl)cc(Cl)c2)c1C1CC1 |r,TLB:5:7:13.18.19:9.10.11|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(Cl)cc(Cl)c1)N3C(=O)c1cn(nn1)-c1ccccc1 |r,TLB:21:20:3.10.9:7.6.5|

COc1cncc(c1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(Cl)cc(Cl)c1 |r,TLB:8:10:16.21.22:12.13.14|

Cc1ccc(c(n1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(Cl)cc(Cl)c1)-n1nccn1 |r,TLB:7:9:15.20.21:11.12.13|

Cc1cc2ccc(cc2o1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(Cl)cc(Cl)c1 |r,TLB:10:12:18.23.24:14.15.16|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(Cl)cc(Cl)c1)N3C(=O)c1cc2ncccc2o1 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(Cl)cc(Cl)c1)N3C(=O)c1cccn2cncc12 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(Cl)cc(Cl)c1)N3C(=O)c1cnc2ccccn12 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(Cl)cc(Cl)c1)N3C(=O)c1ccc2ncccc2c1 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(Cl)cc(Cl)c1)N3C(=O)c1ccc2nccnc2c1 |r,TLB:21:20:3.10.9:7.6.5|

Cn1nc2C3CCCC(Cc2c1-c1ccc(F)c(c1)C(F)F)N3C(=O)c1ccc2ncccc2c1 |TLB:23:22:3.10.9:7.6.5|

Cn1nc2C3CCCC(Cc2c1-c1ccc(F)c(c1)C(F)F)N3C(=O)c1ccc2nccnc2c1 |TLB:23:22:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(c1)C(F)(F)F)N3C(=O)c1ccc2nccnc2c1 |r,TLB:24:23:3.10.9:7.6.5|

COc1cc(Cl)cc(c1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:9:11:17.22.23:13.14.15|

COc1cc(NC(C)=O)cc(c1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:12:14:20.25.26:16.17.18|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cccc(c1)-n1cnnc1 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccccc1-n1cnnc1 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cccc(F)c1-n1cncn1 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccc(F)cc1-n1cncn1 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cc(F)ccc1-n1cncn1 |r,TLB:22:21:3.10.9:7.6.5|

Cc1ccc(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c(c1)-n1cncn1 |r,TLB:5:7:13.18.19:9.10.11|

Cc1ccc(c(c1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1)-n1cncn1 |r,TLB:7:9:15.20.21:11.12.13|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cc(ccc1-n1cncn1)C(F)(F)F |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccccc1-n1ncnc1C(F)(F)F |r,TLB:22:21:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccccc1-n1ccnc1 |r,TLB:22:21:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cc(F)ccc1-n1cccn1 |r,TLB:22:21:10.3.9:7.6.5|

Cn1cc(cn1)-c1cccc(c1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:12:14:25.20.26:16.17.18|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cccc(c1)-n1cc(F)cn1 |r,TLB:22:21:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cccc(c1)-n1cc(cn1)C(F)(F)F |r,TLB:22:21:10.3.9:7.6.5|

COc1cnn(c1)-c1cccc(c1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:13:15:26.21.27:17.18.19|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cccc(c1)-n1ccc(n1)C(F)(F)F |r,TLB:22:21:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cccc(c1)-n1nccn1 |r,TLB:22:21:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cc(F)ccc1-n1nccn1 |r,TLB:22:21:10.3.9:7.6.5|

Cc1cccc(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c1-n1nccn1 |r,TLB:6:8:19.14.20:10.11.12|

COc1cccc(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c1-n1nccn1 |r,TLB:7:9:20.15.21:11.12.13|

COc1ccc(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c(c1)-n1nccn1 |r,TLB:6:8:19.14.20:10.11.12|

COc1ccc(c(c1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1)-n1nccn1 |r,TLB:8:10:21.16.22:12.13.14|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cccc(c1-n1nccn1)C(F)(F)F |r,TLB:22:21:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cc(ccc1-n1nccn1)C(F)(F)F |r,TLB:22:21:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccccc1-n1ccnn1 |r,TLB:22:21:10.3.9:7.6.5|

COc1cccc(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c1-n1ccnn1 |r,TLB:7:9:20.15.21:11.12.13|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnn2CCCCc12 |r,TLB:22:21:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnc2CCCOc2c1 |r,TLB:22:21:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnn2CCCOc12 |r,TLB:22:21:10.3.9:7.6.5|

CC1COc2c(cnn2C1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:23.18.24:14.15.16|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cc2OCCCn2n1 |r,TLB:22:21:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnn(C)c1C(F)(F)F |r,TLB:22:21:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnn(c1C(F)(F)F)C(C)(C)C |r,TLB:22:21:10.3.9:7.6.5|

CCc1nc(nn1-c1ccccc1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:13:15:26.21.27:17.18.19|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cc(n(n1)-c1ccccc1)C(F)(F)F |r,TLB:22:21:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1nc(n(n1)-c1ccccc1)C(F)(F)F |r,TLB:22:21:10.3.9:7.6.5|

COc1nc(nn1-c1ccccc1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:13:15:26.21.27:17.18.19|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ncn(n1)-c1cccc(F)c1 |r,TLB:22:21:10.3.9:7.6.5|

Cc1nc(nn1-c1ccc(F)cc1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:13:15:21.26.27:17.19.18|

COc1ccccc1-n1cnc(n1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:13:15:17.18.19:27.21.26|

COc1cccc(c1)-n1cnc(n1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:13:15:17.18.19:27.21.26|

COc1ccncc1C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:8:10:16.21.22:12.14.13|

COc1cccc(n1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:8:10:16.21.22:12.14.13|

COc1ccnc(c1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:8:10:16.21.22:12.14.13|

COc1ccc(nc1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:8:10:16.21.22:12.14.13|

COc1ccc(cn1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:8:10:16.21.22:12.14.13|

CC(C)Oc1cncc(c1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:18.23.24:14.16.15|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cccc(OC(F)(F)F)n1 |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccc(OC(F)(F)F)cn1 |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cccc(n1)C#N |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnccn1 |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccncn1 |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccnnc1 |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cncnc1 |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cncc(c1)-n1cccn1 |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccc(nc1)-n1cccn1 |r,TLB:22:21:3.10.9:5.7.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccc(nc1)-n1cccc1 |r,TLB:22:21:3.10.9:5.7.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccc(nc1)-n1ccnc1 |r,TLB:22:21:3.10.9:5.7.6|

Cc1ccc(c(n1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1)-n1nccn1 |r,TLB:7:9:15.20.21:13.11.12|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cncc(c1)N1CCCC1 |r,TLB:22:21:3.10.9:5.7.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cncc(c1)N1CCCC1=O |r,TLB:22:21:3.10.9:5.7.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cncc(c1)N1CCOCC1 |r,TLB:22:21:3.10.9:5.7.6|

Cc1cc2ccc(cn2c1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:18.23.24:16.14.15|

Cc1nc2ccc(cc2o1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:18.23.24:16.14.15|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnn2ccccc12 |r,TLB:22:21:3.10.9:5.7.6|

Cc1ccn2ncc(C(=O)N3[C@H]4CCC[C@@H]3c3nn(C)c(c3C4)-c3cc(F)c(F)c(F)c3)c2c1 |r,TLB:8:10:16.21.22:14.12.13|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccn2nccc2c1 |r,TLB:22:21:3.10.9:5.7.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccc2ccnn2c1 |r,TLB:22:21:3.10.9:5.7.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cc2ccccn2n1 |r,TLB:22:21:3.10.9:5.7.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cccc2nccn12 |r,TLB:22:21:3.10.9:5.7.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cccc2cncn12 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccc2cncn2c1 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccc2nccn2c1 |r,TLB:22:21:3.10.9:7.6.5|

Cc1ccn2c(cnc2c1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:18.23.24:14.15.16|

Cn1ccc2c(ccnc12)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:18.23.24:14.15.16|

Cn1cc(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c2cccnc12 |r,TLB:4:6:12.17.18:8.9.10|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccn2ncccc12 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccn2ccncc12 |r,TLB:22:21:3.10.9:7.6.5|

COc1cccc2n(C)nc(C(=O)N3[C@H]4CCC[C@@H]3c3nn(C)c(c3C4)-c3cc(F)c(F)c(F)c3)c12 |r,TLB:11:13:19.24.25:15.16.17|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1nn(C)c2ncccc12 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnn2ncccc12 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cc2ncccn2n1 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnn2cccnc12 |r,TLB:22:21:3.10.9:7.6.5|

Cc1cnc2c(cnn2c1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:18.23.24:14.15.16|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccn2nccc2n1 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnn2ccncc12 |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccc2nccn2n1 |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnc2cccnn12 |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccn2ncnc2c1 |r,TLB:22:21:3.10.9:7.5.6|

Cn1cc(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c2nccnc12 |r,TLB:4:6:12.17.18:8.10.9|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnc2ncccn12 |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccnc2ccccc12 |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1nccc2ccccc12 |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccc2ncccc2c1 |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccc2cccnc2c1 |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ncnc2ccccc12 |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccc2nccnc2c1 |r,TLB:22:21:3.10.9:7.5.6|

Cc1cnc2cc(ccc2n1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:11:13:19.24.25:15.17.16|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnc2ccccc2n1 |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cc2ccccc2nn1 |r,TLB:22:21:3.10.9:7.5.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccc2nnccc2c1 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccc2ncccc2n1 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnc2cccnc2c1 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cncc2cccnc12 |r,TLB:22:21:3.10.9:7.6.5|

COc1c(F)cc(cc1F)-c1c2C[C@@H]3CCC[C@@H](N3C(=O)c3ccccc3-n3nccn3)c2nn1C |r,TLB:19:18:32.11.12:14.15.16|

COc1c(F)cc(cc1F)-c1c2C[C@@H]3CCC[C@@H](N3C(=O)c3nn(C)c4ncccc34)c2nn1C |r,TLB:19:18:31.11.12:14.15.16|

COc1c(F)cc(cc1F)-c1c2C[C@@H]3CCC[C@@H](N3C(=O)c3ccc4ncccc4c3)c2nn1C |r,TLB:19:18:31.11.12:14.15.16|

COc1cc(cc(F)c1F)-c1c2C[C@@H]3CCC[C@@H](N3C(=O)c3ccccc3-n3nccn3)c2nn1C |r,TLB:19:18:32.11.12:14.15.16|

COc1cc(cc(F)c1F)-c1c2C[C@@H]3CCC[C@@H](N3C(=O)c3nn(C)c4ncccc34)c2nn1C |r,TLB:19:18:31.11.12:14.15.16|

COc1cc(cc(F)c1F)-c1c2C[C@@H]3CCC[C@@H](N3C(=O)c3ccc4ncccc4c3)c2nn1C |r,TLB:19:18:31.11.12:14.15.16|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc2ccccc2n1C)N3C(=O)c1ccc2ncccc2c1 |r,wD:4.26,8.25,TLB:23:22:3.10.9:7.6.5,(-6.77,2.27,;-5.23,2.27,;-4.33,3.52,;-2.86,3.04,;-1.77,4.13,;-.23,4.13,;.86,3.04,;.86,1.5,;-.23,.41,;-1.77,.41,;-2.86,1.5,;-4.33,1.03,;-4.8,-.44,;-6.27,-.91,;-6.27,-2.45,;-7.41,-3.48,;-7.09,-4.99,;-5.63,-5.47,;-4.48,-4.44,;-4.8,-2.93,;-3.9,-1.68,;-2.36,-1.68,;-.52,2.29,;.91,2.85,;1.17,4.37,;2.08,1.84,;2.08,.3,;3.41,-.47,;4.74,.3,;6.08,-.47,;7.41,.3,;7.41,1.84,;6.08,2.61,;4.74,1.84,;3.41,2.61,)|

Cn1nc2C3CCCC(Cc2c1-c1ccc(s1)C(F)(F)F)N3C(=O)c1ccc2ncccc2c1 |TLB:22:21:3.10.9:7.6.5|

COc1ccc(cc1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:8:10:16.21.22:12.13.14|

Cc1ccc(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c(F)c1 |r,TLB:5:7:13.18.19:9.10.11|

COc1ccc(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c(F)c1 |r,TLB:6:8:14.19.20:10.11.12|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cc(F)cc(c1)-n1cccn1 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cc(F)cc(c1)-n1cnnc1 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccc(F)c(c1)-n1cnnc1 |r,TLB:22:21:3.10.9:7.6.5|

Cc1ccc(cc1-n1cnnc1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:12:14:20.25.26:16.17.18|

Cc1cc(cc(c1)-n1cnnc1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:12:14:20.25.26:16.17.18|

Cc1c(cccc1-n1cnnc1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:12:14:20.25.26:16.17.18|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccccc1-n1nccn1 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccc(F)cc1-n1nccn1 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cccc(F)c1-n1nccn1 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cc(F)ccc1-n1nccn1 |r,TLB:22:21:3.10.9:7.6.5|

Cc1ccc(c(c1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1)-n1nccn1 |r,TLB:7:9:15.20.21:11.12.13|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cccc(c1-n1nccn1)C(F)(F)F |r,TLB:22:21:3.10.9:7.6.5|

Cc1cnn(n1)-c1ccccc1C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:12:14:20.25.26:16.17.18|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccccc1-n1ncc(n1)C(F)(F)F |r,TLB:22:21:3.10.9:7.6.5|

COc1ccc(c(c1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1)-n1cncn1 |r,TLB:8:10:16.21.22:12.13.14|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccccc1-n1cc(nn1)C(F)(F)F |r,TLB:22:21:3.10.9:7.6.5|

CC(C)c1cc(ncn1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:9:11:17.22.23:13.14.15|

COc1cc(ncn1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:8:10:16.21.22:12.13.14|

CN(C)c1ccc(cn1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:9:11:17.22.23:13.14.15|

COc1cncc(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c1C |r,TLB:7:9:15.20.21:11.12.13|

COc1ncc(cc1C)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:9:11:17.22.23:13.14.15|

COc1ncc(cc1F)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:9:11:17.22.23:13.14.15|

COc1ncc(F)cc1C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:9:11:17.22.23:13.14.15|

COc1cc(cnc1OC)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:18.23.24:14.15.16|

COc1ccc(nc1OC)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:18.23.24:14.15.16|

COc1nccc(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c1Cl |r,TLB:7:9:15.20.21:11.12.13|

COc1nc(ccc1Cl)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:9:11:17.22.23:13.14.15|

Cc1nccc(Cl)c1C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:8:10:16.21.22:12.13.14|

Cc1cncc(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c1Cl |r,TLB:6:8:14.19.20:10.11.12|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1c(F)cncc1Cl |r,TLB:22:21:3.10.9:7.6.5|

Cc1nc(ccc1C(=O)CN1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1)C1CC1 |r,TLB:9:10:21.22.16:12.13.14|

Cc1nc(ccc1C(=O)CN1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1)C1(CC1)C#N |r|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3CC(=O)c1ccnc(c1)-n1cccn1 |r,TLB:22:21:10.9.3:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3CC(=O)c1cc(ccn1)-n1cccn1 |r,TLB:22:21:10.9.3:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3CC(=O)c1cnccc1-n1cccn1 |r,TLB:22:21:10.9.3:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3CC(=O)c1cccc(n1)-n1cccn1 |r,TLB:22:21:10.9.3:7.6.5|

Cc1ccc(c(n1)C(=O)CN1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1)-n1cccn1 |r,TLB:9:10:21.22.16:12.13.14|

COc1c(cncc1-n1cccn1)C(=O)CN1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:15:16:27.28.22:18.19.20|

Cc1ccc(c(n1)C(=O)CN1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1)-n1cncn1 |r,TLB:9:10:21.22.16:12.13.14|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3CC(=O)c1cncc(c1)-n1cnnc1 |r,TLB:22:21:10.9.3:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3CC(=O)c1cc(ccn1)-n1cnnc1 |r,TLB:22:21:10.9.3:7.6.5|

Cc1cc(cc(n1)C(=O)CN1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1)-n1cnnc1 |r,TLB:9:10:21.22.16:12.13.14|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3CC(=O)c1cncc(c1)-n1nccn1 |r,TLB:22:21:10.9.3:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3CC(=O)c1ncccc1-n1nccn1 |r,TLB:22:21:10.9.3:7.6.5|

Cc1cc(cc(n1)C(=O)CN1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1)-n1nccn1 |r,TLB:9:10:21.22.16:12.13.14|

Cc1c(cnn1C)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:7:9:15.20.21:11.12.13|

CCc1c(cnn1C)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:8:10:16.21.22:12.13.14|

Cc1nn(C)c(C)c1C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:8:10:16.21.22:12.13.14|

COc1c(cnn1C)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:8:10:16.21.22:12.13.14|

COc1nn(C)cc1C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:8:10:16.21.22:12.13.14|

Cc1c(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c(F)nn1C |r,TLB:3:5:11.16.17:7.8.9|

Cn1ncc(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c1C(F)F |r,TLB:5:7:13.18.19:9.10.11|

Cc1c(cnn1C1CC1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:9:11:17.22.23:13.14.15|

Cc1nn(cc1C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1)C1CC1 |r,TLB:6:8:14.19.20:10.11.12|

Cn1cc(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c(n1)C1CC1 |r,TLB:4:6:12.17.18:8.9.10|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccn2cccc2c1 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnn2cccc(F)c12 |r,TLB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnn2cc(F)ccc12 |r,TLB:22:21:3.10.9:7.6.5|

Cc1cccc2c(cnn12)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:18.23.24:14.15.16|

COc1cccn2ncc(C(=O)N3[C@H]4CCC[C@@H]3c3nn(C)c(c3C4)-c3cc(F)c(F)c(F)c3)c12 |r,TLB:10:12:18.23.24:14.15.16|

[H][C@]12CCC[C@]([H])(N1C(=O)c1cnn3cc(OC)ccc13)c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |THB:8:7:27.26.21:4.3.2|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccn2cncc2c1 |r,TLB:22:21:10.3.9:7.6.5|

Cc1c(ccc2cncn12)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:23.18.24:14.15.16|

Cc1ncc2ccc(cn12)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:23.18.24:14.15.16|

Cc1c(ccc2nccn12)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:23.18.24:14.15.16|

Cc1cc(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)n2ccnc2c1 |r,TLB:4:6:17.12.18:8.9.10|

Cc1cnc2cccc(C(=O)N3[C@H]4CCC[C@@H]3c3nn(C)c(c3C4)-c3cc(F)c(F)c(F)c3)n12 |r,TLB:9:11:22.17.23:13.14.15|

Cc1cnc2ccc(cn12)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:23.18.24:14.15.16|

Cc1cn2cc(ccc2n1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:23.18.24:14.15.16|

Cc1cn2c(cccc2n1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:23.18.24:14.15.16|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnc2ccccn12 |r,TLB:22:21:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnc2cc(F)ccn12 |r,TLB:22:21:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnc2cc(Cl)ccn12 |r,TLB:22:21:10.3.9:7.6.5|

Cc1nc2ccccn2c1C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:23.18.24:14.15.16|

Cc1nc2cc(C)ccn2c1C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:11:13:24.19.25:15.16.17|

Cc1nc2ccccn2c1C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(C)cc(F)c1 |r,TLB:10:12:23.18.24:14.15.16|

Cc1cccc2ncc(C(=O)N3[C@H]4CCC[C@@H]3c3nn(C)c(c3C4)-c3cc(F)c(F)c(F)c3)n12 |r,TLB:9:11:22.17.23:13.14.15|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnc2cc(ccn12)C(F)(F)F |r,TLB:22:21:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1c(nc2ccccn12)C(F)F |r,TLB:22:21:10.3.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1n(C)nc2ccccc12 |r,TLB:22:21:10.3.9:7.6.5|

Cc1cc2nc(cc(C)n2n1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:11:13:24.19.25:15.16.17|

Cc1c(cnc2ccnn12)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:23.18.24:14.15.16|

CC(C)c1cc(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)n2ncc(C)c2n1 |r,TLB:6:8:19.14.20:10.11.12|

Cc1nn2c(cc(C)nc2c1C)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:12:14:25.20.26:16.17.18|

Cc1cc2nc(cc(C3CC3)n2n1)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:13:15:26.21.27:17.18.19|

Cc1nn2ncccc2c1C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:23.18.24:14.15.16|

Cc1cn2ccnc(C(=O)N3[C@H]4CCC[C@@H]3c3nn(C)c(c3C4)-c3cc(F)c(F)c(F)c3)c2n1 |r,TLB:8:10:21.16.22:12.13.14|

Cc1nc2c(C)ccc(C)n2c1C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:12:14:25.20.26:16.17.18|

Cc1nc2cccnn2c1C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:23.18.24:14.15.16|

Cc1nc2cc(C)cnn2c1C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:11:13:19.24.25:17.15.16|

Cn1cnc2c(ccnc12)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:18.23.24:16.14.15|

Cn1cnc2cc(cnc12)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:18.23.24:16.14.15|

Cn1ccc2c(ncnc12)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:18.23.24:16.14.15|

Cn1nc2[C@@H]3CCC[C@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccnc2n(C)ncc12 |r,THB:22:21:3.10.9:7.6.5|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ncnc2n(C)ncc12 |r,TLB:22:21:3.10.9:5.7.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccn2cnnc2c1 |r,TLB:22:21:3.10.9:5.7.6|

Cc1nc(C(=O)N2[C@H]3CCC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c2cnccn12 |r,TLB:4:6:12.17.18:10.8.9|

Cc1cc(F)cc(c1)-c1c2C[C@@H]3CCC[C@@H](N3C(=O)c3ccc4ncccc4c3)c2nn1C |r,TLB:17:16:29.9.10:14.12.13|

Cc1ccnc2ccc(cc12)C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:11:13:19.24.25:17.15.16|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccc2nc(O)ccc2c1 |r,TLB:21:20:3.10.9:5.7.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)cc(F)c1)N3C(=O)c1ccc2[n+]([O-])cccc2c1 |r,TLB:21:20:3.10.9:5.7.6|

Cc1ccc2ncnc(C(=O)N3[C@H]4CCC[C@@H]3c3nn(C)c(c3C4)-c3cc(F)c(F)c(F)c3)c2c1 |r,TLB:9:11:17.22.23:15.13.14|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccc2nccnc2c1 |r,TLB:22:21:3.10.9:5.7.6|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1ccc2nccnc2c1 |r,TLB:22:21:3.10.9:7.6.5|

CC1CCCc2ncc(C(=O)N3[C@H]4CCC[C@@H]3c3nn(C)c(c3C4)-c3cc(F)c(F)c(F)c3)n12 |r,TLB:9:11:17.22.23:13.14.15|

Cn1nc2[C@H]3CCC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cnc2CCCCn12 |r,TLB:22:21:3.10.9:7.6.5|

Cc1nn2CC(C)(C)OCc2c1C(=O)N1[C@H]2CCC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:12:14:20.25.26:16.17.18|

Cn1nc2[C@H]3CC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cccc(Cl)c1 |r,TLB:21:20:3.9.8:6.5|

COc1cccc(c1)C(=O)N1[C@H]2CC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:8:10:15.20.21:12.13|

COc1cccc(c1)C(=O)N1[C@H]2CC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)ccc1F |r,wD:14.15,11.11,TLB:8:10:15.20.21:12.13,(6.99,3.71,;5.57,4.29,;4.35,3.35,;4.56,1.82,;3.34,.88,;1.91,1.46,;1.71,2.99,;2.92,3.93,;.06,3.53,;-.09,5.01,;-1.25,2.24,;-.09,.62,;.25,2.12,;-.7,3.32,;-2.24,3.33,;-3.21,2.13,;-4.74,2.27,;-5.35,.86,;-6.84,.48,;-4.19,-.16,;-2.87,.62,;-1.48,-.05,;-4.34,-1.69,;-3.08,-2.58,;-3.22,-4.12,;-1.96,-5.01,;-4.62,-4.76,;-5.88,-3.87,;-5.73,-2.34,;-6.99,-1.45,)|

COc1cccc(c1)C(=O)N1[C@H]2CC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)cc1F |r,wD:14.15,11.11,TLB:8:10:15.20.21:12.13,(6.98,4.39,;5.56,4.97,;4.34,4.03,;4.55,2.5,;3.33,1.56,;1.9,2.14,;1.7,3.67,;2.91,4.61,;.07,4.18,;-.08,5.65,;-1.25,2.88,;-.08,1.26,;.26,2.76,;-.69,3.97,;-2.23,3.97,;-3.2,2.77,;-4.73,2.91,;-5.34,1.5,;-6.84,1.13,;-4.18,.48,;-2.86,1.27,;-1.47,.6,;-4.33,-1.05,;-3.07,-1.94,;-3.21,-3.47,;-1.96,-4.36,;-4.61,-4.12,;-4.75,-5.65,;-5.87,-3.23,;-5.73,-1.69,;-6.98,-.8,)|

COc1cccc(c1)C(=O)N1[C@H]2CC[C@@H]1c1nn(C)c(c1C2)-c1cccc(F)c1F |r,wD:14.15,11.11,TLB:8:10:15.20.21:12.13,(6.95,3.75,;5.52,4.33,;4.3,3.39,;4.51,1.86,;3.29,.92,;1.87,1.5,;1.66,3.02,;2.88,3.97,;-.04,3.53,;-.19,5.01,;-1.36,2.24,;-.19,.62,;.15,2.12,;-.8,3.32,;-2.34,3.33,;-3.31,2.13,;-4.84,2.27,;-5.45,.86,;-6.95,.48,;-4.29,-.16,;-2.97,.62,;-1.58,-.05,;-4.44,-1.69,;-5.84,-2.34,;-5.98,-3.87,;-4.72,-4.76,;-3.32,-4.12,;-2.07,-5.01,;-3.18,-2.58,;-1.78,-1.94,)|

COc1cccc(C(=O)N2[C@H]3CC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c1OC |r,TLB:7:9:14.19.20:11.12|

COc1cccc(C(=O)N2[C@H]3CC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c1F |r,TLB:7:9:14.19.20:11.12|

COc1cccc(C(=O)N2[C@H]3CC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c1Cl |r,TLB:7:9:14.19.20:11.12|

COc1cccc(n1)C(=O)N1[C@H]2CC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:8:10:15.20.21:12.13|

Cc1c(cnn1C)C(=O)N1[C@H]2CC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:7:9:14.19.20:11.12|

Cc1cc(F)cc(c1)-c1c2C[C@@H]3CC[C@@H](N3C(=O)c3cnn(C)c3C3CC3)c2nn1C |r,TLB:16:15:27.9.10:12.13|

Cn1ncc(C(=O)N2[C@H]3CC[C@@H]2c2nn(C)c(c2C3)-c2ccccc2)c1C1CC1 |r,TLB:5:7:12.17.18:9.10|

Cn1ncc(C(=O)N2[C@H]3CC[C@@H]2c2nn(C)c(c2C3)-c2ccc(F)c(F)c2)c1C1CC1 |r,TLB:5:7:12.17.18:9.10|

Cn1ncc(C(=O)N2[C@H]3CC[C@@H]2c2nn(C)c(c2C3)-c2ccc(F)cc2F)c1C1CC1 |r,wD:11.11,8.7,TLB:5:7:12.17.18:9.10,(6.19,2.93,;4.73,2.45,;4.26,.98,;2.72,.98,;2.24,2.44,;.84,3.1,;.72,4.63,;-.4,2.24,;.57,.71,;.91,2.21,;-.05,3.41,;-1.59,3.41,;-2.55,2.2,;-4.09,2.34,;-4.69,.92,;-6.19,.57,;-3.53,-.09,;-2.21,.7,;-.82,.04,;-3.66,-1.62,;-5.06,-2.27,;-5.19,-3.81,;-3.93,-4.69,;-4.07,-6.23,;-2.54,-4.04,;-2.4,-2.51,;-1.01,-1.86,;3.48,3.35,;3.47,4.89,;4.24,6.23,;2.7,6.22,)|

Cn1ncc(C(=O)N2[C@H]3CC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)cc(F)c2)c1C1CC1 |r,TLB:5:7:12.17.18:9.10|

Cn1ncc(C(=O)N2[C@H]3CC[C@@H]2c2nn(C)c(c2C3)-c2ccc(F)c(F)c2F)c1C1CC1 |r,wD:11.11,8.7,TLB:5:7:12.17.18:9.10,(6.19,2.93,;4.73,2.45,;4.26,.98,;2.72,.98,;2.24,2.44,;.84,3.1,;.72,4.63,;-.4,2.24,;.57,.71,;.91,2.21,;-.05,3.41,;-1.59,3.41,;-2.55,2.2,;-4.09,2.34,;-4.69,.92,;-6.19,.57,;-3.53,-.09,;-2.21,.7,;-.82,.04,;-3.66,-1.62,;-5.06,-2.27,;-5.19,-3.81,;-3.93,-4.69,;-4.07,-6.23,;-2.54,-4.04,;-1.28,-4.93,;-2.4,-2.51,;-1.01,-1.86,;3.48,3.35,;3.47,4.89,;4.24,6.23,;2.7,6.22,)|

Cn1ncc(C(=O)N2[C@H]3CC[C@@H]2c2nn(C)c(c2C3)-c2cc(F)c(F)c(F)c2)c1C1CC1 |r,TLB:5:7:12.17.18:9.10|

Cc1nc(c([nH]1)C(=O)N1[C@H]2CC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1)C(F)(F)F |r,TLB:6:8:13.18.19:10.11|

Cn1nc2[C@H]3CC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cccc2cc[nH]c12 |r,TLB:21:20:3.9.8:6.5|

Cn1nc2[C@H]3CC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1c(F)ccc2cc[nH]c12 |r,TLB:21:20:3.9.8:6.5|

Cc1[nH]c2c(cccc2c1C)C(=O)N1[C@H]2CC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:11:13:18.23.24:15.16|

Cn1nc2[C@H]3CC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cccc2cn[nH]c12 |r,TLB:21:20:3.9.8:6.5|

Cn1nc2[C@H]3CC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1cccc2nc[nH]c12 |r,TLB:21:20:3.9.8:6.5|

Cc1nc2ccc(cc2o1)C(=O)N1[C@H]2CC[C@@H]1c1nn(C)c(c1C2)-c1cc(F)c(F)c(F)c1 |r,TLB:10:12:17.22.23:14.15|

Cn1nc2[C@H]3CC[C@@H](Cc2c1-c1cc(F)c(F)c(F)c1)N3C(=O)c1nccc2occc12 |r,TLB:21:20:3.9.8:6.5|