3549 SMILES Strings for Serine/threonine-protein kinase B-raf [V600E]

Compound Name
SMILES String
COc1cc(Nc2cncc(n2)-c2cccc(NC(C)=O)c2)cc(OC)c1OC
COc1cc(Nc2cncc(n2)-c2ccncc2)cc(OC)c1OC
COc1cc(Nc2cncc(n2)-c2cccnc2)cc(OC)c1OC
COc1cc(Nc2cncc(n2)-c2cccc(O)c2)cc(OC)c1OC
COc1cc(Nc2cncc(n2)-c2ccc(O)cc2)cc(OC)c1OC
COc1cc(Nc2cncc(n2)-c2ccc(CO)cc2)cc(OC)c1OC
CCOC(=O)c1cccc(c1)-c1cncc(Nc2cc(OC)c(OC)c(OC)c2)n1
COc1cc(Nc2cncc(n2)-c2ccc(C=O)cc2)cc(OC)c1OC
COc1cc(Nc2cncc(n2)-c2ccc(NC(=O)Nc3ccccc3)cc2)cc(OC)c1OC
COc1cc(Nc2cncc(n2)-c2ccc(cc2)C(N)=O)cc(OC)c1OC
COc1cc(Nc2nc(cnc2NC(C)=O)-c2cccc(NC(C)=O)c2)cc(OC)c1OC
COc1cc(Nc2cncc(c2)-c2cccc(NC(C)=O)c2)cc(OC)c1OC
COc1cc(Nc2cncc(Nc3ccc(NC(C)=O)cc3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Nc3ccccc3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Nc3ccncc3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Nc3cccc(NC(C)=O)c3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Nc3ccc(O)cc3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Nc3cccc(F)c3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Nc3ccc(F)cc3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3cccc4ccccc34)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3ccc4ccccc4c3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3ccccc3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3ccncc3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3cccnc3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Sc3cccc4ccccc34)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3cccc4CCCCc34)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3cccc4[nH]ccc34)n2)cc(OC)c1OC
COc1cc(Nc2cncc(n2)-c2cccc(c2)C#N)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3ccc4CCC(=O)Oc4c3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3ccnc4ccccc34)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3cccc4ncccc34)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3ccc4ncccc4c3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3cccc4cnccc34)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3cccc4C(=O)CCCc34)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3ccc4C(=O)CCCc4c3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3cccc4C(=O)CCc34)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3ccc4C(=O)CCc4c3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3ccc4CCC(=O)c4c3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3ccccc3-c3ccccc3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3ccccc3F)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3cccc(F)c3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3cccc(Cl)c3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3cccc(NC(C)=O)c3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3ccc(NC(C)=O)cc3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3cccc(c3)C(C)=O)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3ccc(cc3)C(C)=O)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3cccc(c3)C(C)N=O)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3ccc(cc3)C(C)N=O)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3cccc4C(CCc34)N=O)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3ccc4CCC(N=O)c4c3)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3ccc4C(CCCc4c3)N=O)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3cccc4c(NC(C)=O)cccc34)n2)cc(OC)c1OC
COc1cc(Nc2cncc(Oc3ccc(NC(C)=O)c4ccccc34)n2)cc(OC)c1OC
CC(=O)Nc1cccc2c(Oc3cncc(Nc4cccc(c4)-c4cnco4)n3)cccc12
CC(=O)Nc1cccc2c(Oc3cncc(Nc4ccc5COC(=O)c5c4)n3)cccc12
CC(=O)Nc1ccc(Oc2cncc(Nc3cccc(c3)-c3cnco3)n2)c2ccccc12
CNC(=O)c1cc(ccn1)Oc2ccc(cc2)NC(=O)Nc3ccc(c(c3)C(F)(F)F)Cl
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(Cl)cc23)c1F
CNC(=O)c1cc(Oc2ccc(Nc3nc4ccc(Cl)cc4[nH]3)cc2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccc(Cl)c(c4)C(F)(F)F)[nH]c3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccc(Br)cc4)n(C)c3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccccc4)[nH]c3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccccc4Br)[nH]c3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4cccc(Br)c4)[nH]c3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccc(Br)cc4)[nH]c3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccccc4C(F)(F)F)[nH]c3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4cccc(c4)C(F)(F)F)[nH]c3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccc(cc4)C(F)(F)F)[nH]c3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4cccc(c4)C(C)(C)C)[nH]c3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccc(cc4)C(C)(C)C)[nH]c3c2)ccn1
CNC(=O)c1cc(Oc2ccc3n(C)c(Nc4ccccc4)nc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3n(C)c(Nc4ccc(Cl)c(c4)C(F)(F)F)nc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3n(C)c(Nc4ccccc4Br)nc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3n(C)c(Nc4cccc(Br)c4)nc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3n(C)c(Nc4ccc(Br)cc4)nc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3n(C)c(Nc4ccccc4C(F)(F)F)nc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3n(C)c(Nc4cccc(c4)C(F)(F)F)nc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3n(C)c(Nc4ccc(cc4)C(F)(F)F)nc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3n(C)c(Nc4cccc(c4)C(C)(C)C)nc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3n(C)c(Nc4ccc(cc4)C(C)(C)C)nc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3n(C)c(NC4CCCCC4)nc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3n(C)c(NCC4CCCCC4)nc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3n(C)c(Nc4cccc(c4)-c4ccncc4)nc3c2)ccn1
CCn1c(Nc2ccc(Br)cc2)nc2cc(Oc3ccnc(c3)C(=O)NC)ccc12
CCNC(=O)c1cc(Oc2ccc3n(C)c(Nc4ccc(Br)cc4)nc3c2)ccn1
Cn1c(Nc2ccc(Br)cc2)nc2cc(Oc3ccnc(c3)C(=O)NCCN3CCOCC3)ccc12
Cn1c(Nc2ccc(Br)cc2)nc2cc(Oc3ccnc(c3)C(=O)NCCO)ccc12
CCCC1CCCCN1NC(=O)c1cc(Oc2ccc3n(C)c(Nc4ccc(Br)cc4)nc3c2)ccn1
CN(C)C(=O)c1cc(Oc2ccc3n(C)c(Nc4ccc(Br)cc4)nc3c2)ccn1
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)ccc1Cl
O=C(Nc1ccccc1)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1
Clc1ccc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)cc1
FC(F)(F)c1cc(Cl)cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)c1
FC(F)(F)c1cccc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)c1
FC(F)(F)c1ccccc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1
FC(F)(F)c1ccc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)cc1
FC(F)(F)Oc1cccc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)c1
COc1ccc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1)C(F)(F)F
COc1cc(Cl)c(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1)C(F)(F)F
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1)C(F)(F)F
Fc1cccc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)c1
Fc1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)cc(c1)N1CCOCC1
FC(F)(F)c1ccc(N2CCOCC2)c(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)c1
Cn1c2c(Oc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)cc3)ccnc2[nH]c1=O
Cn1c2c(Oc3ccc(NC(=O)Nc4cccc(c4)C(C)(C)C)cc3)ccnc2[nH]c1=O
Cn1c2nccc(Oc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)cc3)c2[nH]c1=O
Cn1c2nccc(Oc3ccc(NC(=O)Nc4cccc(c4)C(C)(C)C)cc3)c2[nH]c1=O
Cn1c2nccc(Oc3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)cc3)c2[nH]c1=O
Cn1c2nccc(Oc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)cc3)c2n(C)c1=O
CCn1c2nccc(Oc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)cc3)c2n(CC)c1=O
Fc1ccc(cc1NC(=O)Nc1ccc(Sc2ccnc3[nH]c(=O)[nH]c23)cc1)C(F)(F)F
FC(F)(F)c1cccc(NC(=O)Nc2ccc(Sc3ccnc4[nH]c(=O)[nH]c34)cc2)c1
FC(F)(F)c1cc(NC(=O)Nc2ccc(Sc3ccnc4[nH]c(=O)[nH]c34)cc2)ccc1Cl
FC(F)(F)c1cc(NC(=S)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)ccc1Cl
O=C(Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1)c1ccccc1
FC(F)(F)c1cc(ccc1Cl)C(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1
FC(F)(F)c1cccc(c1)C(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1
Brc1cccc(c1)C(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1
COc1cccc(c1)C(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1
Fc1cc(cc(c1)C(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1)N1CCOCC1
O=C(Cc1ccccc1)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1
COc1cccc(CC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)c1
Fc1cc(F)cc(CC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)c1
FC(F)(F)Oc1cccc(CC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)c1
FC(F)(F)c1cccc(CC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)c1
FC(F)(F)c1cc(ccc1Cl)S(=O)(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1
O=c1[nH]c2nccc(Oc3ccc(NS(=O)(=O)c4ccccc4)cc3)c2[nH]1
Clc1ccc(cc1)S(=O)(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1
FC(F)(F)c1ccc(cc1)S(=O)(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1
Fc1ccc(cc1)S(=O)(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1
O=c1[nH]c2nccc(Oc3ccc(NS(=O)(=O)c4cccs4)cc3)c2[nH]1
Fc1ccccc1S(=O)(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1
Cc1ccc(cc1Nc1ncccc1-c1ccncn1)C(=O)Nc1cccc(c1)C(F)(F)F
CNc1ncc2cc(ccc2n1)-c1cc(ccc1C)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc2c(Nc3cccc(c3)C(F)(F)F)nccc2c1Nc1ncccc1-c1ccncn1
Cc1ccc2c(Nc3ccc(Cl)cc3)nccc2c1Nc1ncccc1-c1ccncn1
CNc1cc(ncn1)-c1cccnc1Nc1c(C)ccc2c(Nc3ccc(Cl)cc3)nccc12
CNc1cc(ncn1)-c1cccnc1Nc1c(C)ccc2c(Nc3ccc(cc3)C#N)nccc12
CNc1cc(ncn1)-c1cccnc1Nc1c(C)ccc2c(Nc3cccc(c3)C#C)nccc12
CNc1cc(ncn1)-c1cccnc1Nc1c(C)ccc2c(Nc3ccc4sc(C)nc4c3)nccc12
CNc1ncc2cc(ccc2n1)-c1c(C)ccc2c(Nc3ccc(Cl)cc3)nccc12
CNc1ncc2cc(ccc2n1)-c1c(C)ccc2c(Nc3cc(nn3C)C(C)(C)C)nccc12
CNc1ncc2cc(ccc2n1)-c1c(C)ccc2c(Nc3ccc4c(NC(=O)C4(C)C)c3)nccc12
Cc1ccc2c(Nc3ccc(Cl)cc3)nccc2c1Nc1ncccc1-c1ncnc2nc[nH]c12
CCCS(=O)(=O)Nc1cc(F)cc(-c2[nH]c(nc2-c2ccnc(NCC)n2)C2CC2)c1Cl
CC(C)Nc1nccc(n1)-c1nc([nH]c1-c1cc(F)cc(NS(C)(=O)=O)c1Cl)C1CC1
CCCS(=O)(=O)Nc1cc(F)cc(-c2[nH]c(nc2-c2ccnc(NC(C)C)n2)C2CC2)c1Cl
COC(=O)N[C@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(F)cc(NS(C)(=O)=O)c1Cl)C1CC1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(=O)(=O)c2ccc(F)cc2)c1F)C1CC1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(=O)(=O)c2cccc(F)c2)c1F)C1CC1 |r|
CC1(CC1)c1nc(c([nH]1)-c1cc(F)cc(NS(C)(=O)=O)c1Cl)-c1ccnc(NCCC#N)n1
Cc1cc(NS(C)(=O)=O)c(Cl)c(c1)-c1[nH]c(nc1-c1ccnc(NCCC#N)n1)C1(C)CC1
Cc1cc(NS(C)(=O)=O)c(F)c(c1)-c1[nH]c(nc1-c1ccnc(NCCC#N)n1)C1(C)CC1
CC1(CC1)c1nc(c([nH]1)-c1cc(Cl)cc(NS(C)(=O)=O)c1F)-c1ccnc(NCCC#N)n1
CC1(CC1)c1nc(c([nH]1)-c1cccc(NS(C)(=O)=O)c1Cl)-c1ccnc(NCCC#N)n1
CC(C)(C)c1nc(c([nH]1)-c1cc(Cl)cc(NS(C)(=O)=O)c1F)-c1ccnc(N)n1
CC(C)(C)c1nc(c([nH]1)-c1cc(Cl)cc(NS(=O)(=O)c2c(F)cccc2F)c1F)-c1ccnc(N)n1
Nc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(=O)(=O)c2c(F)cccc2F)c1F)C1CC1
CS(=O)(=O)Nc1cc(Cl)cc(-c2[nH]c(nc2-c2ccnc(N)n2)C2CC2)c1F
CCCS(=O)(=O)Nc1cc(Cl)cc(-c2[nH]c(nc2-c2ccnc(N)n2)C(C)(C)C)c1F
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(F)cc(NS(=O)(=O)c2c(F)cccc2F)c1Cl)C1CC1 |r|
CC(C)(C)c1nc(c([nH]1)-c1cc(F)cc(NS(C)(=O)=O)c1Cl)-c1ccnc(N)n1
CC(C)(C)c1nc(c([nH]1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1Cl)-c1ccnc(N)n1
CC(C)(C)c1nc(c([nH]1)-c1cccc(NS(C)(=O)=O)c1Cl)-c1ccnc(N)n1
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(=O)(=O)c2cc(F)cc(F)c2)c1F)C1CC1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c1F)C1CC1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(C)cc(NS(=O)(=O)CC(F)(F)F)c1F)C1CC1 |r|
CC(C)(C)c1nc(c([nH]1)-c1cc(F)cc(NS(=O)(=O)c2c(F)cccc2F)c1Cl)-c1ccnc(N)n1
CS(=O)(=O)Nc1cc(F)cc(-c2[nH]c(nc2-c2ccnc(N)n2)C2CC2)c1Cl
Nc1nccc(n1)-c1nc([nH]c1-c1cc(F)cc(NS(=O)(=O)c2c(F)cccc2F)c1Cl)C1CC1
CCCS(=O)(=O)Nc1cc(F)cc(-c2[nH]c(nc2-c2ccnc(N)n2)C2CC2)c1Cl
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(C)(=O)=O)c1F)C1CCC1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(F)cc(NS(C)(=O)=O)c1Cl)C1CCC1 |r|
CNc1nccc(n1)-c1nc([nH]c1-c1cc(F)cc(NS(=O)(=O)c2c(F)cccc2F)c1Cl)C1CC1
CNc1nccc(n1)-c1nc([nH]c1-c1cc(F)cc(NS(C)(=O)=O)c1Cl)C1CC1
CCCS(=O)(=O)Nc1cc(F)cc(-c2[nH]c(nc2-c2ccnc(NC)n2)C2CC2)c1Cl
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(F)cc(NS(C)(=O)=O)c1Cl)-c1ccc(F)cc1F |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(F)cc(NS(C)(=O)=O)c1Cl)-c1ccc(cc1)C(F)(F)F |r|
CS(=O)(=O)Nc1cc(Cl)cc(-c2[nH]c(nc2-c2ccnc(NCCC#N)n2)C2CC2)c1F
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cccc(NS(=O)(=O)C2CC2)c1F)C(C)(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cccc(NS(C)(=O)=O)c1F)C(C)(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cccc(NS(=O)(=O)C(C)C)c1F)C(C)(C)C |r|
CS(=O)(=O)Nc1cccc(-c2[nH]c(nc2-c2ccnc(NCCC#N)n2)C2CC2)c1F
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1c(F)ccc(NS(C)(=O)=O)c1Cl)C1CC1 |r,wD:5.5,(9.34,-1.06,;8.01,-1.83,;6.67,-1.06,;6.67,.48,;5.34,-1.83,;4.01,-1.06,;4.01,.48,;2.67,-1.83,;1.34,-1.06,;.01,-1.83,;.01,-3.37,;-1.33,-4.14,;-2.66,-3.37,;-2.66,-1.83,;-1.33,-1.06,;-4,-1.06,;-5.46,-1.54,;-6.37,-.29,;-5.46,.95,;-4,.48,;-2.91,1.57,;-3.31,3.05,;-4.79,3.45,;-2.22,4.14,;-.73,3.74,;-.33,2.26,;1.16,1.86,;2.25,2.95,;3.33,4.04,;1.16,4.04,;3.33,1.86,;-1.42,1.17,;-1.02,-.32,;-7.85,-.69,;-9.34,-.29,;-8.94,-1.78,)|
CS(=O)(=O)Nc1cccc(-c2[nH]c(nc2-c2ccnc(NCC3(CC3)C#N)n2)C2CC2)c1Cl
Nc1nccc(n1)-c1nc([nH]c1-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1Cl)C1CC1
Fc1cc(NS(=O)(=O)c2c(F)cccc2F)c(Cl)c(c1)-c1[nH]c(nc1-c1ccncn1)C1CC1
CS(=O)(=O)Nc1cc(F)cc(-c2[nH]c(nc2-c2ccncn2)C2CC2)c1Cl
CCCS(=O)(=O)Nc1cc(F)cc(-c2[nH]c(nc2-c2ccncn2)C2CC2)c1Cl
CNc1nccc(n1)-c1nc([nH]c1-c1cccc(NS(C)(=O)=O)c1F)C1CC1
C[C@H](O)CNc1nccc(n1)-c1nc([nH]c1-c1cccc(NS(C)(=O)=O)c1F)C1CC1 |r|
CCCS(=O)(=O)Nc1cccc(-c2[nH]c(nc2-c2ccnc(NC[C@H](C)NC(=O)OC)n2)C2CC2)c1Cl |r|
CCCS(=O)(=O)Nc1cccc(-c2[nH]c(nc2-c2ccnc(NC[C@H](C)NC(=O)OC)n2)C(C)(C)C)c1F |r|
CCCS(=O)(=O)Nc1cccc(-c2[nH]c(nc2-c2ccnc(NC[C@H](C)NC(=O)OC)n2)C2CC2)c1F |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(C)cc(NS(=O)(=O)C(C)C)c1)C1CC1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cccc(NS(=O)(=O)CCC(F)(F)F)c1F)C(C)(C)C |r|
CCCS(=O)(=O)Nc1cc(Cl)cc(-c2[nH]c(nc2-c2ccnc(NC[C@H](C)NC(=O)OC)n2)C(C)(C)C)c1F |r|
CCCS(=O)(=O)Nc1cccc(-c2[nH]c(nc2-c2ccnc(NCCC#N)n2)C2CC2)c1F
CCCS(=O)(=O)Nc1cccc(-c2[nH]c(nc2-c2ccnc(NCCC(N)=O)n2)C2CC2)c1F
CCCS(=O)(=O)Nc1c(F)ccc(-c2[nH]c(nc2-c2ccnc(NC[C@H](C)NC(=O)OC)n2)C(C)(C)C)c1F |r|
CCCS(=O)(=O)Nc1cccc(c1)-c1[nH]c(nc1-c1ccnc(NC[C@H](C)NC(=O)OC)n1)C1CC1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cccc(NS(C)(=O)=O)c1)C1CC1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(F)cc(NS(C)(=O)=O)c1Cl)C1CC1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1[nH]c(nc1-c1cc(Cl)cc(NS(C)(=O)=O)c1F)C1CC1
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(C)cc(NS(C)(=O)=O)c1F)C1CC1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(C)(=O)=O)c1)C(C)(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(=O)(=O)C(F)(F)F)c1)C(C)(C)C |r|
CCCS(=O)(=O)Nc1cc(Cl)cc(c1)-c1[nH]c(nc1-c1ccnc(NC[C@H](C)NC(=O)OC)n1)C(C)(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(=O)(=O)C2CC2)c1)C(C)(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(=O)(=O)CC(C)C)c1)C(C)(C)C |r|
CCC(C)S(=O)(=O)Nc1cc(Cl)cc(c1)-c1[nH]c(nc1-c1ccnc(NC[C@H](C)NC(=O)OC)n1)C(C)(C)C |r|
CCS(=O)(=O)Nc1cc(Cl)cc(c1)-c1[nH]c(nc1-c1ccnc(NC[C@H](C)NC(=O)OC)n1)C(C)(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(=O)(=O)C(C)C)c1)C(C)(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(NS(=O)(=O)C(C)C)c(C)c(OC)c1)C(C)(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(NS(=O)(=O)C2CC2)c(C)c(OC)c1)C(C)(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(=O)(=O)C(C)C)c1)C1CC1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(=O)(=O)C2CC2)c1C)C(C)(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(=O)(=O)C(C)C)c1C)C(C)(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(NS(=O)(=O)C(C)C)cc(OC(F)F)c1)C(C)(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(C)cc(NS(=O)(=O)C(C)C)c1)C(C)(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cccc(NS(C)(=O)=O)c1)C(C)(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(C)(=O)=O)c1)C1CC1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cccc(NS(C)(=O)=O)c1Cl)C1CC1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cccc(NS(C)(=O)=O)c1F)C1CC1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(F)cc(NS(C)(=O)=O)c1F)C1CC1 |r|
CCCS(=O)(=O)Nc1cc(Cl)cc(-c2[nH]c(nc2-c2ccnc(NC[C@H](C)NC(=O)OC)n2)C2CC2)c1F |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(C)(=O)=O)c1Cl)C1CC1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(=O)(=O)C2CC2)c1F)C1CC1 |r|
CCS(=O)(=O)Nc1cc(Cl)cc(-c2[nH]c(nc2-c2ccnc(NC[C@H](C)NC(=O)OC)n2)C2CC2)c1F |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(=O)(=O)CCC(F)(F)F)c1F)C1CC1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(C)cc(NS(C)(=O)=O)c1Cl)C1CC1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(=O)(=O)CC2CC2)c1F)C1CC1 |r|
CCS(=O)(=O)Nc1cc(F)cc(-c2[nH]c(nc2-c2ccnc(NC[C@H](C)NC(=O)OC)n2)C2CC2)c1Cl |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(F)cc(NS(=O)(=O)C2CC2)c1Cl)C1CC1 |r|
CCCS(=O)(=O)Nc1ccc(F)c(-c2[nH]c(nc2-c2ccnc(NC[C@H](C)NC(=O)OC)n2)C2CC2)c1Cl |r,wU:25.26,(-5.86,4.43,;-4.77,3.35,;-3.28,3.74,;-2.2,2.66,;-1.11,3.74,;-3.28,1.57,;-1.11,1.57,;.38,1.96,;.78,3.45,;2.27,3.85,;3.36,2.76,;4.84,3.16,;2.96,1.27,;4.05,.19,;5.51,.66,;6.42,-.58,;5.51,-1.83,;4.05,-1.35,;2.71,-2.12,;2.71,-3.66,;1.38,-4.43,;.05,-3.66,;.05,-2.12,;-1.29,-1.35,;-2.62,-2.12,;-3.96,-1.35,;-3.96,.19,;-5.29,-2.12,;-6.62,-1.35,;-6.62,.19,;-7.96,-2.12,;-9.29,-1.35,;1.38,-1.35,;7.96,-.58,;9.29,-1.35,;9.29,.19,;1.47,.88,;1.07,-.61,)|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(F)cc(NS(C)(=O)=O)c1Cl)C(C)(C)C |r|
CCCS(=O)(=O)Nc1cc(F)cc(-c2[nH]c(nc2-c2ccnc(NC[C@H](C)NC(=O)OC)n2)C(C)(C)C)c1Cl |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(C)(=O)=O)c1F)C(C)(C)C |r|
CCS(=O)(=O)Nc1cc(Cl)cc(-c2[nH]c(nc2-c2ccnc(NC[C@H](C)NC(=O)OC)n2)C(C)(C)C)c1F |r|
CC(CNc1nccc(n1)-c1nc([nH]c1-c1cccc(NS(C)(=O)=O)c1Cl)C1CC1)C#N
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(Cl)cc(NS(C)(=O)=O)c1F)C1(C)CC1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(C)cc(NS(C)(=O)=O)c1F)C1(C)CC1 |r|
CCCNc1nccc(n1)-c1nc([nH]c1-c1cc(F)cc(NS(=O)(=O)CCC)c1Cl)C1CC1
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1nc([nH]c1-c1cccc(NS(C)(=O)=O)c1Cl)C1(C)CC1 |r|
CCCNc1nccc(n1)-c1nc([nH]c1-c1cc(F)cc(NS(C)(=O)=O)c1Cl)C1CC1
CCNc1nccc(n1)-c1nc([nH]c1-c1cc(F)cc(NS(C)(=O)=O)c1Cl)C1CC1
CC(C)CNc1nccc(n1)-c1nc([nH]c1-c1cc(F)cc(NS(C)(=O)=O)c1Cl)C1CC1
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(cc34)N3CCOCC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(cc34)N3CCN(C)CC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(cc34)N3CCCC3)c2)cc1C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(cc12)N1CCOCC1)C(=O)N1CCOCC1
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)N3CCOCC3)c2)cc1C(F)(F)F
Cc1ccc(cc1Nc1ncnc2ccc(nc12)N1CCOCC1)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2ccc(nc12)N1CCOCC1)C(=O)Nc1cccc(c1)C(C)(C)[N+]#[C-]
Cc1ccc(cc1Nc1ncnc2ccc(nc12)N1CCOCC1)C(=O)n1nc(cc1N)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2ccc(nc12)N1CCOCC1)C(=O)Nc1cc(n[nH]1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2ccc(nc12)N1CCOCC1)C(=O)Nc1cc(nn1C)C(C)(C)C
CN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)N3CCOCC3)c2)cc(c1)C(F)(F)F
CN1CCCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)N3CCOCC3)c2)cc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2ccc(nc12)N1CCOCC1)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F
CN1CCN(CC1)c1ccc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
COCCN1CCN(CC1)c1ccc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN1CCC(CN2CCN(CC2)c2ccc3ncnc(Nc4cc(ccc4C)C(=O)Nc4cc(on4)C(C)(C)C)c3n2)CC1
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)N3CCN(C)CC3)c2)cc1C(F)(F)F
COCCN1CCN(CC1)c1ccc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(OC)c(c3)C(F)(F)F)c2n1
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)N3CCN(CC4CCN(C)CC4)CC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)N(C)C)c2)cc1C(F)(F)F
CN(C)c1ccc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)N3CCN(C)CC3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
COCCN1CCN(CC1)c1ccc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(cc(NS(C)(=O)=O)c3OC)C(C)(C)C)c2n1
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)N(C)C3CCOC3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(NC5CCOC5)nc34)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)N3CC[C@@H](F)C3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C |r|
CCN1CCN(CC1)c1ccc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(cc(NS(C)(=O)=O)c3OC)C(C)(C)C)c2n1
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)N3CCOCC3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)N3CCN(CCN4CCOCC4)CC3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)N3CCC(C3)N3CCOCC3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)C3=CCNCC3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C |t:26|
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(C)nc34)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)C3=CCN(CC3)C(C)C)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C |t:26|
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)C3=CCN(C)CC3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C |t:26|
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)C3CCNCC3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)C3CCN(C)CC3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
CCN1CCC(CC1)c1ccc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(cc(NS(C)(=O)=O)c3OC)C(C)(C)C)c2n1
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)C3CCN(CC3)C(C)C)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)C3CCN(CC4CC4)CC3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
COCCN1CCC(CC1)c1ccc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(cc(NS(C)(=O)=O)c3OC)C(C)(C)C)c2n1
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(CC5CCNCC5)nc34)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)C3=CCNC3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C |t:26|
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)C3CCNC3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)C3CCN(C)C3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
COCCN1CCC(C1)c1ccc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(cc(NS(C)(=O)=O)c3OC)C(C)(C)C)c2n1
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(nc34)C3CCCNC3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(CC5CNCCOC5)nc34)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(CC5CCN(C)CC5)nc34)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
CCN1CCC(Cc2ccc3ncnc(Nc4cc(ccc4C)C(=O)Nc4cc(cc(NS(C)(=O)=O)c4OC)C(C)(C)C)c3n2)CC1
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(CC5CCN(CC5)C(C)C)nc34)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4ccc(CC5CCN(CC6CC6)CC5)nc34)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
CCCN1CCC(Cc2ccc3ncnc(Nc4cc(ccc4C)C(=O)Nc4cc(cc(NS(C)(=O)=O)c4OC)C(C)(C)C)c3n2)CC1
COCCN1CCC(Cc2ccc3ncnc(Nc4cc(ccc4C)C(=O)Nc4cc(cc(NS(C)(=O)=O)c4OC)C(C)(C)C)c3n2)CC1
CCOCCN1CCC(Cc2ccc3ncnc(Nc4cc(ccc4C)C(=O)Nc4cc(cc(NS(C)(=O)=O)c4OC)C(C)(C)C)c3n2)CC1
Cc1ccc(cc1Nc1ncnc2ccc(nc12)C1=CCNCC1)C(=O)Nc1cc(on1)C(C)(C)C |t:21|
COCCN1CCN(CC1)c1ccc2ncnc(Sc3cc(ccc3C)C(=O)Nc3cccc(c3)C(C)(C)C#N)c2n1
COCCN1CCN(CC1)c1ccc2ncnc(Sc3cc(ccc3C)C(=O)Nc3cc(cc(c3)C(F)(F)F)N3CCN(C)CC3)c2n1
COCCN1CCN(CC1)c1ccc2ncnc(Sc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
COCCN1CCN(CC1)c1ccc2ncnc(Sc3cc(ccc3C)C(=O)Nc3cc(cc(NS(C)(=O)=O)c3OC)C(C)(C)C)c2n1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1Nc1ncnc2ccc(nc12)N1CCOCC1
CN1CCN(CC1)c1ccc2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(C)(C)C#N)ccc3C)c2n1
COCCN1CCN(CC1)c1ccc2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(C)(C)C#N)ccc3C)c2n1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1Nc1ncnc2ccc(nc12)N1CC[C@H](F)C1 |r|
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1Nc1ncnc2ccc(N[C@H]3CCOC3)nc12 |r|
Cc1nc(Cl)cc(Nc2cccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)c2)n1
Cc1nc(Nc2cccc(NC(=O)Nc3ccc(F)c(Cl)c3)c2)cc(n1)N1CCOCC1
Cc1nc(Nc2cccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)c2)cc(n1)N1CCOCC1
CN1CCN(CC1)c1cc(Nc2cccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)c2)nc(C)n1
CN(c1cccc(NC(=O)Nc2ccc(F)c(Cl)c2)c1)c1cc(nc(C)n1)N1CCOCC1
CN(c1cccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c1)c1cc(nc(C)n1)N1CCOCC1
CN(c1cccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c1)c1cc(nc(C)n1)N1CCN(C)CC1
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4c(N)nc(nc34)N3CCN(C)CC3)c2)cc1C(F)(F)F
CN1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(Br)cc(c3)C(F)(F)F)c2n1
CN1CCCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(cc3)C(F)(F)F)c2n1
Cc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1CCNCC1)C(=O)Nc1ccc(cc1)C(F)(F)F
CN1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(cc3)C(F)(F)F)c2n1
CN(C)CCNc1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(cc3)C(F)(F)F)c2n1
CN1CCC(CC1)N1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(cc3)C(F)(F)F)c2n1
CN1CCC(CN2CCN(CC2)c2nc(N)c3ncnc(Nc4cc(ccc4C)C(=O)Nc4ccc(cc4)C(F)(F)F)c3n2)CC1
CN1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN1CCC(CC1)N1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN1CCCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN1CCC(CC1)N1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(n[nH]3)C(C)(C)C)c2n1
CN1CCC(CN2CCN(CC2)c2nc(N)c3ncnc(Nc4cc(ccc4C)C(=O)Nc4cc(n[nH]4)C(C)(C)C)c3n2)CC1
CN1CCCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(n[nH]3)C(C)(C)C)c2n1
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4c(N)nc(nc34)N3CCN(CC3)C3CCN(C)CC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4c(N)nc(nc34)N3CCN(CC4CCN(C)CC4)CC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4c(N)nc(nc34)N3CCCN(C)CC3)c2)cc1C(F)(F)F
CN1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(n[nH]3)C(C)(C)C)c2n1
CN1CCN(CC1)c1nc(N)c2ncnc(Nc3cccc(c3)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
CN1CCCN(CC1)c1nc(N)c2ncnc(Nc3cccc(c3)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
CN1CCC(CC1)N1CCN(CC1)c1nc(N)c2ncnc(Nc3cccc(c3)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
CN1CCC(CN2CCN(CC2)c2nc(N)c3ncnc(Nc4cccc(c4)C(=O)Nc4cccc(c4)C(F)(F)F)c3n2)CC1
CN1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3Cl)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
CN1CCCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3Cl)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
CN1CCC(CC1)N1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3Cl)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
CN1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3Br)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
CN1CCCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3Br)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
CN1CCC(CC1)N1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3Br)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
CN1CCC(CN2CCN(CC2)c2nc(N)c3ncnc(Nc4cc(ccc4Br)C(=O)Nc4cccc(c4)C(F)(F)F)c3n2)CC1
COc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1CCN(C)CC1)C(=O)Nc1cccc(c1)C(F)(F)F
COc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1CCCN(C)CC1)C(=O)Nc1cccc(c1)C(F)(F)F
COc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1CCN(CC1)C1CCN(C)CC1)C(=O)Nc1cccc(c1)C(F)(F)F
COc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1CCN(CC2CCN(C)CC2)CC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1CCN2CCCC2C1)C(=O)Nc1cc(n[nH]1)C(C)(C)C
C[C@H]1CN(C[C@@H](C)N1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(n[nH]3)C(C)(C)C)c2n1 |r|
CN1C[C@H]2C[C@@H]1CN2c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(n[nH]3)C(C)(C)C)c2n1 |r|
CC(C)CN1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(n[nH]3)C(C)(C)C)c2n1
Cc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1CCN(CC2CCCO2)CC1)C(=O)Nc1cc(n[nH]1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1CCN(CC1)C1CCCC1)C(=O)Nc1cc(n[nH]1)C(C)(C)C
CN1CCCC(CN2CCN(CC2)c2nc(N)c3ncnc(Nc4cc(ccc4C)C(=O)Nc4cc(n[nH]4)C(C)(C)C)c3n2)C1
COCCN1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(n[nH]3)C(C)(C)C)c2n1
Cc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1CCN(CC1)C1CC1)C(=O)Nc1cc(n[nH]1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1CCN2CCCCC2C1)C(=O)Nc1cc(n[nH]1)C(C)(C)C
CN1CCN(CC1)C1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(n[nH]3)C(C)(C)C)c2n1
COc1ccc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3c(N)nc(nc23)N2CCN(C)CC2)c1)C(C)(C)C
COc1cc(NC(=O)c2ccc(C)c(Nc3ncnc4c(N)nc(nc34)N3CCN(C)CC3)c2)cc(c1)C(F)(F)F
CN1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
CN1CCC(CC1)N1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
Cc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1CCN(CC1)C1CCCC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1CCCN(CC1)C1CC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1CCCNCC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1CCCN(CC1)c1ccncc1)C(=O)Nc1cccc(c1)C(F)(F)F
CN1CCC(CN2CCN(CC2)c2nc(N)c3ncnc(Nc4cc(ccc4C)C(=O)Nc4cccc(c4)C(F)(F)F)c3n2)CC1
CC1CN(CC(C)N1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
Cc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1CCCN(CC1)c1ncccn1)C(=O)Nc1cccc(c1)C(F)(F)F
CC(C)N1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
CN1C[C@H]2C[C@@H]1CN2c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1 |r|
Cc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1CCNCC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1CCCN(CC1)c1ccccn1)C(=O)Nc1cccc(c1)C(F)(F)F
CN1CCCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
Cc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1C[C@@H]2C[C@H]1CN2)C(=O)Nc1cc(n[nH]1)C(C)(C)C |r|
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4c(N)nc(nc34)N3CCCOCC3)c2)cc(c1)C(F)(F)F
CN1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(C#N)c(c3)C(F)(F)F)c2n1
CN1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(nn3C)C(C)(C)C)c2n1
CN1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(ccn3)C(F)(F)F)c2n1
CN1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)c2n1
CN1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(cc(c3)C(F)(F)F)-n3cnc(C)c3)c2n1
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4c(N)nc(nc34)N3CCOCC3)c2)cc(c1)C(F)(F)F
CCN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4c(N)nc(nc34)N3CCOCC3)c2)cc(c1)C(F)(F)F
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4c(N)nc(nc34)N(C)C)c2)cc(c1)C(F)(F)F
CCN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4c(N)nc(nc34)N(C)C)c2)cc(c1)C(F)(F)F
CN1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(C)(C)C)c2n1
CCN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4c(N)nc(nc34)N3CCCOCC3)c2)cc(c1)C(F)(F)F
CN1CCN(CC1)c1nc(N)c2ncnc(Nc3ccc(F)c(c3)C(=O)Nc3cc(n[nH]3)C(C)(C)C)c2n1
CC(C)CN1CCN(CC1)c1nc(N)c2ncnc(Nc3ccc(F)c(c3)C(=O)Nc3cc(n[nH]3)C(C)(C)C)c2n1
CC(C)CN1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(nn3C)C(C)(C)C)c2n1
Cc1ccc(cc1Nc1ncnc2c(N)nc(nc12)N1CCN2CCCC2C1)C(=O)Nc1cc(nn1C)C(C)(C)C
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4c(N)nc(nc34)N3CC[C@H](F)C3)c2)cc(c1)C(F)(F)F |r|
CCN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4c(N)nc(nc34)N3CCCC3)c2)cc(c1)C(F)(F)F
CCN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4c(N)nc(nc34)N3CC[C@H](F)C3)c2)cc(c1)C(F)(F)F |r|
CN1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(F)(F)F)ccc3C)c2n1
CN1CCCN(CC1)c1nc(N)c2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(F)(F)F)ccc3C)c2n1
CN1CCN(CC1)Nc1nc(N)c2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(F)(F)F)ccc3C)c2n1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1Nc1ncnc2c(N)nc(NCc3ccncc3)nc12
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1Nc1ncnc2c(N)nc(NCc3cccnc3)nc12
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1Nc1ncnc2c(N)nc(NCc3ccccn3)nc12
CN(C)c1nc(N)c2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(F)(F)F)ccc3C)c2n1
CN1CCC(CC1)N1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(F)(F)F)ccc3C)c2n1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1Nc1ncnc2c(N)nc(nc12)N1CCN(CC1)C1CCCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1Nc1ncnc2c(N)nc(nc12)N1CCCN(CC1)C1CC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1Nc1ncnc2c(N)nc(nc12)N1CCCNCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1Nc1ncnc2c(N)nc(nc12)N1CCCN(CC1)c1ccncc1
C[C@H]1CN([C@H](C)CN1)c1nc(N)c2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(F)(F)F)ccc3C)c2n1 |r|
CN1CCC(CN2CCN(CC2)c2nc(N)c3ncnc(Nc4cc(NC(=O)c5cccc(c5)C(F)(F)F)ccc4C)c3n2)CC1
CC1CN(CC(C)N1)c1nc(N)c2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(F)(F)F)ccc3C)c2n1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1Nc1ncnc2c(N)nc(nc12)N1CCCN(CC1)c1ncccn1
CC(C)N1CCN(CC1)c1nc(N)c2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(F)(F)F)ccc3C)c2n1
CN1CC2CC1CN2c1nc(N)c2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(F)(F)F)ccc3C)c2n1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1Nc1ncnc2c(N)nc(nc12)N1CCNCC1
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCN(C)CC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)cc1C(F)(F)F
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NCc3cccc(c3)C(C)(C)C)c2n1
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3Cl)C(=O)Nc3ccc(OC)c(c3)C(F)(F)F)c2n1
COc1ccc(NC(=O)c2ccc(Cl)c(Nc3ncnc4cnc(nc34)N(C)CCN(C)C)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(Cl)c(Nc3ncnc4cnc(nc34)N3CCCCCC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(Cl)c(Nc3ncnc4cnc(nc34)N3CCCN(C)CC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(Cl)c(Nc3ncnc4cnc(nc34)N(C)CCN3CCCC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(Cl)c(Nc3ncnc4cnc(nc34)N3CCN(C)CC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(Cl)c(Nc3ncnc4cnc(nc34)N3CCCCC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(Cl)c(Nc3ncnc4cnc(NCCCN5CCOCC5)nc34)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(Cl)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(Cl)c(Nc3ncnc4cnc(nc34)N3CCCC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(Cl)c(Nc3ncnc4cnc(NCCN(C)C)nc34)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(Cl)c(Nc3ncnc4cnc(NCCN5CCOCC5)nc34)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(Cl)c(Nc3ncnc4cnc(nc34)N(C)C)c2)cc1C(F)(F)F
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3OC)C(=O)Nc3ccc(OC)c(c3)C(F)(F)F)c2n1
COc1ccc(cc1Nc1ncnc2cnc(nc12)N(C)CCN(C)C)C(=O)Nc1ccc(OC)c(c1)C(F)(F)F
COc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCCC1)C(=O)Nc1ccc(OC)c(c1)C(F)(F)F
COc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCN(C)CC1)C(=O)Nc1ccc(OC)c(c1)C(F)(F)F
COc1ccc(cc1Nc1ncnc2cnc(nc12)N(C)CCN1CCCC1)C(=O)Nc1ccc(OC)c(c1)C(F)(F)F
COc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCN(C)CC1)C(=O)Nc1ccc(OC)c(c1)C(F)(F)F
COc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)Nc1ccc(OC)c(c1)C(F)(F)F
COc1ccc(cc1Nc1ncnc2cnc(NCCCN3CCOCC3)nc12)C(=O)Nc1ccc(OC)c(c1)C(F)(F)F
COc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1ccc(OC)c(c1)C(F)(F)F
COc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)Nc1ccc(OC)c(c1)C(F)(F)F
COc1ccc(cc1Nc1ncnc2cnc(NCCN(C)C)nc12)C(=O)Nc1ccc(OC)c(c1)C(F)(F)F
COc1ccc(cc1Nc1ncnc2cnc(NCCN3CCOCC3)nc12)C(=O)Nc1ccc(OC)c(c1)C(F)(F)F
COc1ccc(cc1Nc1ncnc2cnc(nc12)N(C)C)C(=O)Nc1ccc(OC)c(c1)C(F)(F)F
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3F)C(=O)Nc3ccc(OC)c(c3)C(F)(F)F)c2n1
COc1ccc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N(C)CCN(C)C)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N3CCCCCC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N(C)CCN3CCCC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N3CCN(C)CC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N3CCCCC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(NCCCN5CCOCC5)nc34)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N3CCCC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(NCCN(C)C)nc34)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(NCCN5CCOCC5)nc34)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N(C)C)c2)cc1C(F)(F)F
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3C(F)(F)F)C(=O)Nc3ccc(OC)c(c3)C(F)(F)F)c2n1
COc1ccc(NC(=O)c2ccc(c(Nc3ncnc4cnc(nc34)N(C)CCN(C)C)c2)C(F)(F)F)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(c(Nc3ncnc4cnc(nc34)N3CCCCCC3)c2)C(F)(F)F)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(c(Nc3ncnc4cnc(nc34)N3CCCN(C)CC3)c2)C(F)(F)F)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(c(Nc3ncnc4cnc(nc34)N(C)CCN3CCCC3)c2)C(F)(F)F)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(c(Nc3ncnc4cnc(nc34)N3CCN(C)CC3)c2)C(F)(F)F)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(c(Nc3ncnc4cnc(nc34)N3CCCCC3)c2)C(F)(F)F)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(c(Nc3ncnc4cnc(NCCCN5CCOCC5)nc34)c2)C(F)(F)F)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)C(F)(F)F)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(c(Nc3ncnc4cnc(nc34)N3CCCC3)c2)C(F)(F)F)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(c(Nc3ncnc4cnc(NCCN(C)C)nc34)c2)C(F)(F)F)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(c(Nc3ncnc4cnc(NCCN5CCOCC5)nc34)c2)C(F)(F)F)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(c(Nc3ncnc4cnc(nc34)N(C)C)c2)C(F)(F)F)cc1C(F)(F)F
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3C(F)(F)F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C(F)(F)F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CC(C)(C)c1cc(NC(=O)c2ccc(c(Nc3ncnc4cnc(nc34)N3CCCCCC3)c2)C(F)(F)F)no1
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C(F)(F)F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN(CCN1CCCC1)c1ncc2ncnc(Nc3cc(ccc3C(F)(F)F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C(F)(F)F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CC(C)(C)c1cc(NC(=O)c2ccc(c(Nc3ncnc4cnc(nc34)N3CCCCC3)c2)C(F)(F)F)no1
CC(C)(C)c1cc(NC(=O)c2ccc(c(Nc3ncnc4cnc(NCCCN5CCOCC5)nc34)c2)C(F)(F)F)no1
CC(C)(C)c1cc(NC(=O)c2ccc(c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)C(F)(F)F)no1
CC(C)(C)c1cc(NC(=O)c2ccc(c(Nc3ncnc4cnc(nc34)N3CCCC3)c2)C(F)(F)F)no1
CN(C)CCNc1ncc2ncnc(Nc3cc(ccc3C(F)(F)F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CC(C)(C)c1cc(NC(=O)c2ccc(c(Nc3ncnc4cnc(NCCN5CCOCC5)nc34)c2)C(F)(F)F)no1
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3Cl)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CC(C)(C)c1cc(NC(=O)c2ccc(Cl)c(Nc3ncnc4cnc(nc34)N3CCCCCC3)c2)no1
CN(C)c1ncc2ncnc(Nc3cc(ccc3Cl)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3Cl)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN(CCN1CCCC1)c1ncc2ncnc(Nc3cc(ccc3Cl)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3Cl)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CC(C)(C)c1cc(NC(=O)c2ccc(Cl)c(Nc3ncnc4cnc(nc34)N3CCCCC3)c2)no1
CC(C)(C)c1cc(NC(=O)c2ccc(Cl)c(Nc3ncnc4cnc(NCCCN5CCOCC5)nc34)c2)no1
CC(C)(C)c1cc(NC(=O)c2ccc(Cl)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)no1
CC(C)(C)c1cc(NC(=O)c2ccc(Cl)c(Nc3ncnc4cnc(nc34)N3CCCC3)c2)no1
CN(C)CCNc1ncc2ncnc(Nc3cc(ccc3Cl)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CC(C)(C)c1cc(NC(=O)c2ccc(Cl)c(Nc3ncnc4cnc(NCCN5CCOCC5)nc34)c2)no1
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3Cl)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3OC)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
COc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1cc(on1)C(C)(C)C
COc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)Nc1cc(on1)C(C)(C)C
COc1ccc(cc1Nc1ncnc2cnc(nc12)N(C)C)C(=O)Nc1cc(on1)C(C)(C)C
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CC(C)(C)c1cc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N3CCCCCC3)c2)no1
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
COc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCCC1)C(=O)Nc1cc(on1)C(C)(C)C
CC(C)(C)c1cc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N3CCCCC3)c2)no1
CC(C)(C)c1cc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)no1
CC(C)(C)c1cc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N3CCCC3)c2)no1
CN(C)CCNc1ncc2ncnc(Nc3cc(ccc3F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CC(C)(C)c1cc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(NCCN5CCOCC5)nc34)c2)no1
CN(C)c1ncc2ncnc(Nc3cc(ccc3F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CNc1ncc2ncnc(Nc3cc(ccc3F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
COc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCN(C)CC1)C(=O)Nc1cc(on1)C(C)(C)C
COc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCN(C)CC1)C(=O)Nc1cc(on1)C(C)(C)C
COc1ccc(cc1Nc1ncnc2cnc(nc12)N(C)CCN1CCCC1)C(=O)Nc1cc(on1)C(C)(C)C
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(CN4CCCC4)cc(c3)C(F)(F)F)c2n1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCSCC1)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCC1)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(NCCF)nc12)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCC(F)(F)CC1)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCC(F)CC1)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(NCC3CCOC3)nc12)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(NCc3ccccc3)nc12)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(NCc3cccnc3)nc12)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F
COCCNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(CN4CCCC4)cc(c3)C(F)(F)F)c2n1
Cc1ccc(cc1Nc1ncnc2cnc(NC3CC3)nc12)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F
CC(C)CNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(CN4CCCC4)cc(c3)C(F)(F)F)c2n1
Cc1ccc(cc1Nc1ncnc2cnc(NCc3ccccn3)nc12)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(NCc3ccncc3)nc12)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F
CN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(CN4CCCC4)cc(c3)C(F)(F)F)c2n1
CNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(CN4CCCC4)cc(c3)C(F)(F)F)c2n1
CCN(CC)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(CN4CCCC4)cc(c3)C(F)(F)F)c2n1
Cc1ccc(cc1Nc1ncnc2cnc(NCCc3ccccc3)nc12)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(N(C)CCN(C)C)c(c3)C(F)(F)F)c2n1
CN(C)CCN(C)c1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCCCC3)c2)cc1C(F)(F)F
CN(C)CCN(C)c1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCSCC3)c2)cc1C(F)(F)F
CN(C)CCN(C)c1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCC3)c2)cc1C(F)(F)F
CN(C)CCN(C)c1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCCF)nc34)c2)cc1C(F)(F)F
CN(C)CCN(C)c1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCC(F)(F)CC3)c2)cc1C(F)(F)F
CN(C)CCN(C)c1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCC(F)CC3)c2)cc1C(F)(F)F
CN(C)CCN(C)c1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCC5CCOC5)nc34)c2)cc1C(F)(F)F
CN(C)CCN(C)c1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCc5ccccc5)nc34)c2)cc1C(F)(F)F
CN(C)CCN(C)c1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCCC3)c2)cc1C(F)(F)F
CN(C)CCN(C)c1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCc5cccnc5)nc34)c2)cc1C(F)(F)F
CN(C)CCN(C)c1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)cc1C(F)(F)F
CN(C)CCN(C)c1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCC3)c2)cc1C(F)(F)F
COCCNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(N(C)CCN(C)C)c(c3)C(F)(F)F)c2n1
CN(C)CCN(C)c1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NC5CC5)nc34)c2)cc1C(F)(F)F
CC(C)CNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(N(C)CCN(C)C)c(c3)C(F)(F)F)c2n1
CN(C)CCN(C)c1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCc5ccccn5)nc34)c2)cc1C(F)(F)F
CN(C)CCN(C)c1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCc5ccncc5)nc34)c2)cc1C(F)(F)F
CN(C)CCN(C)c1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N(C)C)c2)cc1C(F)(F)F
CNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(N(C)CCN(C)C)c(c3)C(F)(F)F)c2n1
CCN(CC)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(N(C)CCN(C)C)c(c3)C(F)(F)F)c2n1
CN(C)CCN(C)c1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCCc5ccccc5)nc34)c2)cc1C(F)(F)F
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(OCCN(C)C)cc(c3)C(F)(F)F)c2n1
CN(C)CCOc1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCSCC3)c2)cc(c1)C(F)(F)F
CN(C)CCOc1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCC3)c2)cc(c1)C(F)(F)F
CN(C)CCOc1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCCF)nc34)c2)cc(c1)C(F)(F)F
CN(C)CCOc1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCC(F)CC3)c2)cc(c1)C(F)(F)F
CN(C)CCOc1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCC5CCOC5)nc34)c2)cc(c1)C(F)(F)F
CN(C)CCOc1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCc5ccccc5)nc34)c2)cc(c1)C(F)(F)F
CN(C)CCOc1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCc5cccnc5)nc34)c2)cc(c1)C(F)(F)F
CN(C)CCOc1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)cc(c1)C(F)(F)F
CN(C)CCOc1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCC3)c2)cc(c1)C(F)(F)F
COCCNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(OCCN(C)C)cc(c3)C(F)(F)F)c2n1
CN(C)CCOc1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NC5CC5)nc34)c2)cc(c1)C(F)(F)F
CC(C)CNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(OCCN(C)C)cc(c3)C(F)(F)F)c2n1
CN(C)CCOc1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCc5ccccn5)nc34)c2)cc(c1)C(F)(F)F
CN(C)CCOc1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N(C)C)c2)cc(c1)C(F)(F)F
CNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(OCCN(C)C)cc(c3)C(F)(F)F)c2n1
CCN(CC)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(OCCN(C)C)cc(c3)C(F)(F)F)c2n1
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCCCC3)c2)cc(c1)C(F)(F)F
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCSCC3)c2)cc(c1)C(F)(F)F
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCC3)c2)cc(c1)C(F)(F)F
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCS(=O)CC3)c2)cc(c1)C(F)(F)F
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCCF)nc34)c2)cc(c1)C(F)(F)F
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCC(F)(F)CC3)c2)cc(c1)C(F)(F)F
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCC(F)CC3)c2)cc(c1)C(F)(F)F
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCC5CCOC5)nc34)c2)cc(c1)C(F)(F)F
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCc5ccccc5)nc34)c2)cc(c1)C(F)(F)F
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCCC3)c2)cc(c1)C(F)(F)F
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCc5cccnc5)nc34)c2)cc(c1)C(F)(F)F
COCCNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(cc(c3)C(F)(F)F)N(C)CCN(C)C)c2n1
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NC5CC5)nc34)c2)cc(c1)C(F)(F)F
CC(C)CNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(cc(c3)C(F)(F)F)N(C)CCN(C)C)c2n1
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCc5ccccn5)nc34)c2)cc(c1)C(F)(F)F
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCc5ccncc5)nc34)c2)cc(c1)C(F)(F)F
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N(C)C)c2)cc(c1)C(F)(F)F
CNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(cc(c3)C(F)(F)F)N(C)CCN(C)C)c2n1
CCN(CC)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(cc(c3)C(F)(F)F)N(C)CCN(C)C)c2n1
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCCc5ccccc5)nc34)c2)cc(c1)C(F)(F)F
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCC(F)(F)F)nc34)c2)cc(c1)C(F)(F)F
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NCC3CCOC3)c2n1
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(C)(C)C#N)c2n1
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCN(C)CC3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NCc3cccc(c3)C(F)(F)F)c2n1
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NC3CCCCC3)c2n1
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccccc3)c2n1
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NC3CC3)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc4N(CCN5CCCC5)C(=O)C(C)(C)c4c3)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NCC3CCOC3)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NCc3cccc(c3)C(F)(F)F)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NC3CCCCC3)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccccc3)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NC3CC3)c2n1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1ccc2N(CCN3CCCC3)C(=O)C(C)(C)c2c1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)NCC1CCOC1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)NC1CC1
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)S(=O)(=O)N(C)C)c2n1
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc4N(CCN5CCCC5)C(=O)C(C)(C)c4c3)c2n1
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NCC3CCOC3)c2n1
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(C)(C)C#N)c2n1
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N(C)CCN(C)C)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NCc3cccc(c3)C(F)(F)F)c2n1
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NC3CCCCC3)c2n1
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccccc3)c2n1
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NC3CC3)c2n1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@@H](F)C1)C(=O)Nc1ccc2N(CCN3CCCC3)C(=O)C(C)(C)c2c1 |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@@H](F)C1)C(=O)NCC1CCOC1 |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@@H](F)C1)C(=O)Nc1cccc(c1)C(C)(C)C#N |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@@H](F)C1)C(=O)NCc1cccc(c1)C(F)(F)F |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@@H](F)C1)C(=O)NC1CCCCC1 |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@@H](F)C1)C(=O)Nc1ccccc1 |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@@H](F)C1)C(=O)NC1CC1 |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)Nc1ccc2N(CCN3CCCC3)C(=O)C(C)(C)c2c1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)NCC1CCOC1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)Nc1cccc(c1)C(C)(C)C#N
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)NCc1cccc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)NC1CCCCC1
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(F)c(c3)C(F)(F)F)c2n1
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NCc3ccc(cc3)C(C)(C)C)c2n1
COc1ccc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCCN(C)CC2)c1)C(F)(F)F
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)c2n1
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NCc3ccc(cc3)C(F)(F)F)c2n1
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(OC(F)(F)F)c3)c2n1
CN(C)c1cccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCN(C)CC3)c2)c1
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(C)(C)C)c2n1
COc1ccc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCCN(C)CC2)c1)C(C)(C)C
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NCc3ccc(cc3)C(C)(C)C)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NCc3ccc(cc3)C(F)(F)F)c2n1
CN(C)c1cccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCN(C)CC3)c2)c1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(C)(C)C)c2n1
COc1ccc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCN(C)CC2)c1)C(C)(C)C
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(F)c(c3)C(F)(F)F)c2n1
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NCc3ccc(cc3)C(C)(C)C)c2n1
COc1ccc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N(C)CCN(C)C)c1)C(F)(F)F
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)c2n1
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NCc3ccc(cc3)C(F)(F)F)c2n1
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(OC(F)(F)F)c3)c2n1
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)N(C)C)c2n1
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(C)(C)C)c2n1
COc1ccc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N(C)CCN(C)C)c1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@@H](F)C1)C(=O)NCc1ccc(cc1)C(C)(C)C |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@@H](F)C1)C(=O)NCc1ccc(cc1)C(F)(F)F |r|
CN(C)c1cccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CC[C@@H](F)C3)c2)c1 |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@@H](F)C1)C(=O)Nc1cccc(c1)C(C)(C)C |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)NCc1ccc(cc1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)NCc1ccc(cc1)C(F)(F)F
CN(C)c1cccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCCC3)c2)c1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)Nc1cccc(c1)C(C)(C)C
COc1ccc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCCCC2)c1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)NCc1ccc(cc1)C(F)(F)F
CN(C)S(=O)(=O)c1cccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCN(C)CC3)c2)c1
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc4N(CCN5CCCC5)C(=O)C(C)(C)c4c3)c2n1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)Nc1ccccc1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)NC1CC1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)Nc1ccc2N(CCN3CCCC3)C(=O)C(C)(C)c2c1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)NCC1CCOC1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)NCc1cccc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)NC1CCCCC1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)Nc1ccccc1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)NC1CC1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(ccn3)C(F)(F)F)c2n1
COc1ccc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCCCC2)c1)C(F)(F)F
CN(C)c1cccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCNCC3)c2)c1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)Nc1nnc(s1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)Nc1ccc(F)c(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)NCc1ccc(cc1)C(C)(C)C
COc1ccc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCCC2)c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)Nc1cccc(OC(F)(F)F)c1
CN(C)c1cccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCC3)c2)c1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)Nc1cccc(c1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)Nc1ccc(C#N)c(c1)C(F)(F)F
CN(C)S(=O)(=O)c1cccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCC3)c2)c1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)Nc1cc(ccn1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)Nc1cccc(c1)C(C)(C)C#N
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCC3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCC1)C(=O)NCc1cccc(c1)C(C)(C)C
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(ccn3)C(F)(F)F)c2n1
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3nnc(s3)C(F)(F)F)c2n1
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(C#N)c(c3)C(F)(F)F)c2n1
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3nnc(s3)C(F)(F)F)c2n1
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(ccn3)C(F)(F)F)c2n1
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(C#N)c(c3)C(F)(F)F)c2n1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@H](F)C1)C(=O)Nc1nnc(s1)C(F)(F)F |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@H](F)C1)C(=O)Nc1ccc(F)c(c1)C(F)(F)F |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@H](F)C1)C(=O)Nc1cccc(c1)C(F)(F)F |r|
COc1ccc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N2CC[C@H](F)C2)c1)C(F)(F)F |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@H](F)C1)C(=O)Nc1ccc(Cl)c(c1)C(F)(F)F |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@H](F)C1)C(=O)Nc1cccc(OC(F)(F)F)c1 |r|
COc1ccc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N2CC[C@H](F)C2)c1)C(C)(C)C |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@H](F)C1)C(=O)Nc1ccc(C#N)c(c1)C(F)(F)F |r|
CN(C)S(=O)(=O)c1cccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CC[C@H](F)C3)c2)c1 |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1cccc(c1)C(C)(C)C
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CC[C@H](F)C3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C |r|
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3nnc(s3)C(F)(F)F)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(F)c(c3)C(F)(F)F)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
COc1ccc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCN(C)CC2)c1)C(F)(F)F
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(OC(F)(F)F)c3)c2n1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)NCc1ccc(cc1)C(C)(C)C
CN(C)S(=O)(=O)c1cccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCN(C)CC3)c2)c1
COc1ccc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCOCC2)c1)C(F)(F)F
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(C)(C)C#N)c2n1
COc1ccc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCOCC2)c1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)NCc1ccc(cc1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)NCc1cccc(c1)C(C)(C)C
CN(C)c1cccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)c1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NCc3cccc(c3)C(C)(C)C)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(C#N)c(c3)C(F)(F)F)c2n1
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCN(C)CC3)c2)cc(cc1NS(C)(=O)=O)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1nnc(s1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1ccc(F)c(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(ccc3F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN(CCN1CCCC1)c1ncc2ncnc(Nc3cc(ccc3F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN(C)S(=O)(=O)c1cccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)c1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1cc(ccn1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1cccc(c1)C(C)(C)C#N
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)NCc1cccc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)NC1CCCCC1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1ccccc1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)NCc1cccc(c1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)Nc1nnc(s1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)Nc1ccc(F)c(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)Nc1cccc(OC(F)(F)F)c1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)Nc1ccc(C#N)c(c1)C(F)(F)F
CN(C)S(=O)(=O)c1cccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCCC3)c2)c1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCCC1)C(=O)Nc1cc(ccn1)C(F)(F)F
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)NCc3cccc(c3)C(C)(C)C)c2n1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
COc1c(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCCC3)c2)cc(cc1NS(C)(=O)=O)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCNCC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1ccc(C#N)c(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCNCC1)C(=O)Nc1cccc(c1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCNCC1)C(=O)Nc1nnc(s1)C(F)(F)F
COc1ccc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCNCC2)c1)C(C)(C)C
CN(C)S(=O)(=O)c1cccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCNCC3)c2)c1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@H](F)C1)C(=O)Nc1cc(ccn1)C(F)(F)F |r|
CN(C)C(=O)c1ccc(C)c(Nc2ncnc3cnc(NC4CC[C@H](O)CC4)nc23)c1 |r,wD:24.24,(-7.34,,;-6,-.77,;-6,-2.31,;-4.67,,;-4.67,1.54,;-3.33,-.77,;-3.33,-2.31,;-2,-3.08,;-.67,-2.31,;.67,-3.08,;-.67,-.77,;.67,,;.67,1.54,;-.67,2.31,;-.67,3.85,;.67,4.62,;2,3.85,;3.33,4.62,;4.67,3.85,;4.67,2.31,;6,1.54,;6,,;7.34,-.77,;7.34,-2.31,;6,-3.08,;6,-4.62,;4.67,-2.31,;4.67,-.77,;3.33,1.54,;2,2.31,;-2,,)|
COc1ccc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(NC4CCOC4)nc23)c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(NC3CCOC3)nc12)C(=O)Nc1cc(nn1C)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(NC3CCOC3)nc12)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(NC3CCOC3)nc12)C(=O)Nc1cccc(c1)C(C)(C)C
CCN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NC5CCOC5)nc34)c2)cc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(NC3CCOC3)nc12)C(=O)Nc1cc(n[nH]1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(NC3CCOC3)nc12)C(=O)n1nc(cc1N)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(NC3CCOC3)nc12)C(=O)Nc1cc(ccn1)C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NC5CCOC5)nc34)c2)cc1C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(NC3CCOC3)nc12)C(=O)Nc1cc(on1)C(C)(C)C
COCCNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
Cc1ccc(cc1Nc1ncnc2cnc(NCC3CCOC3)nc12)C(=O)Nc1cc(on1)C(C)(C)C
CN(CC1CCOC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
Cc1ccc(cc1Nc1ncnc2cnc(NCC3CCCCO3)nc12)C(=O)Nc1cc(on1)C(C)(C)C
COC[C@@H]1CCCN1c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1 |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCC[C@H]1CO)C(=O)Nc1cc(on1)C(C)(C)C |r|
CN(C1CCOC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC(F)(F)C1)C(=O)Nc1cc(on1)C(C)(C)C
Cc1cn(cn1)-c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
C[C@H]1CN(C[C@@H](C)O1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1 |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCCOCC1)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCN(CCN2CCOCC2)CC1)C(=O)Nc1cc(on1)C(C)(C)C
Cc1cc(cc(Nc2ncnc3cnc(nc23)N2CCOCC2)c1C)C(=O)Nc1cc(nn1C)C(C)(C)C
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(cc(C)c3C)C(=O)Nc3cc(nn3C)C(C)(C)C)c2n1
Cn1nc(cc1NC(=O)c1cc(Cl)cc(Nc2ncnc3cnc(nc23)N2CCCC2)c1Cl)C(C)(C)C
Cn1nc(cc1NC(=O)c1cc(Cl)cc(Nc2ncnc3cnc(nc23)N2CCOCC2)c1Cl)C(C)(C)C
Cn1nc(cc1NC(=O)c1cc(Cl)cc(Nc2ncnc3cnc(nc23)N2CCOCC2)c1)C(C)(C)C
Cn1nc(cc1NC(=O)c1cc(Cl)cc(Nc2ncnc3cnc(nc23)N2CCCC2)c1)C(C)(C)C
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(Cl)cc(c3)C(=O)Nc3cc(nn3C)C(C)(C)C)c2n1
CN(C)C1CCN(C1)c1ncc2ncnc(Nc3cc(Cl)cc(c3)C(=O)Nc3cc(nn3C)C(C)(C)C)c2n1
Fc1ccc(cc1Nc1ncnc2cnc(NC3CCOC3)nc12)C(=O)NC1CCOC1
CC(C)(C)c1cc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(NC5CCOC5)nc34)c2)no1
CN1CCN(CC1)c1cc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)cc(c1)C(F)(F)F
CC(C)(C#N)c1cccc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)c1
Cn1nc(cc1NC(=O)c1ccc(F)c(Nc2ncnc3cnc(nc23)N2CCOCC2)c1)C(C)(C)C
CN1CCN(CC1)c1cc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)cc(c1F)C(F)(F)F
CC(C)(C#N)c1cccc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(NC5CCOC5)nc34)c2)c1
Cn1nc(cc1NC(=O)c1ccc(F)c(Nc2ncnc3cnc(NC4CCOC4)nc23)c1)C(C)(C)C
CN1CCN(CC1)c1cc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(NC5CCOC5)nc34)c2)cc(c1)C(F)(F)F
CN1CCN(CC1)c1cc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(NC5CCOC5)nc34)c2)cc(c1F)C(F)(F)F
COc1ccc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(NC5CCOC5)nc34)c2)cc1C(F)(F)F
CC(C)(C)c1cc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)[nH]n1
CC(C)(C)c1cc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(NC5CCOC5)nc34)c2)[nH]n1
Fc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1cc(ccn1)C(F)(F)F
CN1CCC(CN2CCN(CC2)c2ncc3ncnc(Nc4cc(ccc4F)C(=O)Nc4cc(on4)C(C)(C)C)c3n2)CC1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CC(C)N1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CC(C)(C)c1cc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N3CCN(CC4CC4)CC3)c2)no1
CCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN(C)C1CCN(C1)c1ncc2ncnc(Nc3cc(ccc3F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN(C1CCN(C)C1)c1ncc2ncnc(Nc3cc(ccc3F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN(C)C1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3F)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3F)C(=O)Nc3ccc(OC)c(c3)C(F)(F)F)c2n1
COc1ccc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N3CCN(CC3)C(C)C)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N3CCN(CC4CC4)CC3)c2)cc1C(F)(F)F
CCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3F)C(=O)Nc3ccc(OC)c(c3)C(F)(F)F)c2n1
COc1ccc(NC(=O)c2ccc(F)c(Nc3ncnc4cnc(nc34)N3CCC(CC3)N(C)C)c2)cc1C(F)(F)F
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N(C)CC3CCCCO3)c2)cc(c1)C(F)(F)F
CCN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N(C)CC3CCCCO3)c2)cc(c1)C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N(C)CC3CCCCO3)c2)cc1C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1cccc(OC(F)(F)F)c1
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CC[C@H](F)C3)c2)cc1C(F)(F)F |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@H](F)C1)C(=O)Nc1cc(on1)C(C)(C)C |r|
COc1ccc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCN(CC3CCN(C)CC3)CC2)c1)C(F)(F)F
CN1CCC(CN2CCN(CC2)c2ncc3ncnc(Nc4cc(ccc4C)C(=O)Nc4cc(nn4C)C(C)(C)C)c3n2)CC1
COc1ccc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCN(CC3CCN(C)CC3)CC2)c1)C(C)(C)C
CN1CCC(CN2CCN(CC2)c2ncc3ncnc(Nc4cc(ccc4C)C(=O)Nc4cccc(c4)C(C)(C)C)c3n2)CC1
CN1CCC(CN2CCN(CC2)c2ncc3ncnc(Nc4cc(ccc4C)C(=O)Nc4cccc(c4)C(F)(F)F)c3n2)CC1
CN1CCC(CN2CCN(CC2)c2ncc3ncnc(Nc4cc(ccc4C)C(=O)Nc4cc(n[nH]4)C(C)(C)C)c3n2)CC1
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCN(CC4CCN(C)CC4)CC3)c2)cc1C(F)(F)F
CN1CCC(CN2CCN(CC2)c2ncc3ncnc(Nc4cc(ccc4C)C(=O)Nc4cc(on4)C(C)(C)C)c3n2)CC1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(nn3C)C(C)(C)C)c2n1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(ccc3OC)C(C)(C)C)c2n1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
CCN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCN(CCOC)CC3)c2)cc(c1)C(F)(F)F
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(n[nH]3)C(C)(C)C)c2n1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(ccn3)C(F)(F)F)c2n1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(OC)c(c3)C(F)(F)F)c2n1
Cc1ccc(cc1Nc1ncnc2cnc(NCc3ccccc3)nc12)C(=O)Nc1cccc(c1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(NCc3ccccc3)nc12)C(=O)Nc1cc(nn1C)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(NCc3ccccc3)nc12)C(=O)Nc1cccc(c1)C(C)(C)C#N
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3C[C@H]4C[C@@H]3CN4C)c2)cc1C(F)(F)F |r|
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCN(CC4CCOC4)CC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCN(CC3)C3CC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCC(CC3)N(C)C)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3C[C@H](C)N[C@H](C)C3)c2)cc1C(F)(F)F |r|
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCN(CC3)C(C)C)c2)cc1C(F)(F)F
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CC[C@H](F)C3)c2)cc(c1)C(F)(F)F |r|
CCN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CC[C@H](F)C3)c2)cc(c1)C(F)(F)F |r|
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCC3)c2)cc(c1)C(F)(F)F
CCN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)cc(c1)C(F)(F)F
CN(C)CCN(C)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)cc(c1)C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCN(C)CC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCN(CC(C)C)CC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCC3)c2)cc1C(F)(F)F
CN1CCCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(n[nH]3)C(C)(C)C)c2n1
CC(C)CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(n[nH]3)C(C)(C)C)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(n[nH]3)C(C)(C)C)c2n1
CC(C)CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(ccn3)C(F)(F)F)c2n1
Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCC(F)(F)C3)c2)cc(c1)C(F)(F)F
Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CC[C@H](F)C3)c2)cc(c1)C(F)(F)F |r|
CC(C)CN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CC[C@H](F)C3)c2)cc(c1)C(F)(F)F |r|
CC(C)N1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CC[C@H](F)C3)c2)cc(c1)C(F)(F)F |r|
CN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CC[C@H](F)C3)c2)cc(c1)C(F)(F)F |r|
CN1CCCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CC[C@H](F)C3)c2)cc(c1)C(F)(F)F |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@H](F)C1)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F |r|
CC(C)CN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)cc(c1)C(F)(F)F
CC(C)N1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)cc(c1)C(F)(F)F
CN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)cc(c1)C(F)(F)F
CN1CCCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)cc(c1)C(F)(F)F
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(nn3C)C(C)(C)C)c2n1
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(C)(C)C)c2n1
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(cc(c3)C(F)(F)F)N(C)CCN(C)C)c2n1
CCN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N(C)CCOC)c2)cc(c1)C(F)(F)F
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(n[nH]3)C(C)(C)C)c2n1
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(ccn3)C(F)(F)F)c2n1
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(OC)c(c3)C(F)(F)F)c2n1
COCCN(C)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN(CC1CCCCO1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(nn3C)C(C)(C)C)c2n1
CN(CC1CCCCO1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCN(CCCN2CCCC2)CC1)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCN(CC2CCOC2)CC1)C(=O)Nc1cc(on1)C(C)(C)C
CN1CCCC(CN2CCN(CC2)c2ncc3ncnc(Nc4cc(ccc4C)C(=O)Nc4cc(on4)C(C)(C)C)c3n2)C1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCN2CCCC2C1)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCC(CC1)N1CCCCC1)C(=O)Nc1cc(on1)C(C)(C)C
CN1CCC(CC1)N1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CC(C)CNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
C[C@H]1CN(C[C@@H](C)O1)C1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1 |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCC(CC1)N1CCOCC1)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCC(CC1)N1CCCC1)C(=O)Nc1cc(on1)C(C)(C)C
CCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CC(C)N1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCN(CC1)C1CC1)C(=O)Nc1cc(on1)C(C)(C)C
CC(C)CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN(C)C1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
C[C@H]1CN(C[C@@H](C)N1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1 |r|
CN1C[C@H]2C[C@@H]1CN2c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1 |r|
CC(C)CNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(nn3C)C(C)(C)C)c2n1
CC(C)CNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(C)(C)C)c2n1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(N4CCN(C)CC4)c(F)c(c3)C(F)(F)F)c2n1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(cc(c3)C(F)(F)F)-n3cnc(C)c3)c2n1
CN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)cc(c1F)C(F)(F)F
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(cc(NS(C)(=O)=O)c3OC)C(C)(C)C)c2n1
CN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NC5CCOC5)nc34)c2)cc(c1F)C(F)(F)F
Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NC5CCOC5)nc34)c2)cc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CC[C@H](F)C1)C(=O)Nc1cc(n[nH]1)C(C)(C)C |r|
CN1CCC(CN2CCN(CC2)c2ncc3ncnc(Nc4cc(ccc4C)C(=O)Nc4cc(N5CCN(C)CC5)c(F)c(c4)C(F)(F)F)c3n2)CC1
CN1CCC(CN2CCN(CC2)c2ncc3ncnc(Nc4cc(ccc4C)C(=O)Nc4cc(ccn4)C(F)(F)F)c3n2)CC1
CN1CCN(CC1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CC[C@H](F)C3)c2)cc(c1F)C(F)(F)F |r|
Cc1ccc(cc1Nc1ncnc2cnc(NCc3ccccc3)nc12)C(=O)Nc1cc(n[nH]1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1cc(nn1C)C(C)(C)C
CN(CCF)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(cc(c3)C(F)(F)F)N3CCCN(C)CC3)c2n1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1cc(n[nH]1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1cc(on1)C(C)(C)C
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN(CCF)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(cc(c3)C(F)(F)F)N3CCN(C)CC3)c2n1
CC(C)CNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(ccn3)C(F)(F)F)c2n1
CC(C)CNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(C)(C)C#N)c2n1
Cc1ccc(cc1Nc1ncnc2cnc(NCc3ccccc3)nc12)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cnc(NCc3ccccc3)nc12)C(=O)Nc1cc(ccn1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1cc(OCCN2CCCC2)cc(c1)C(F)(F)F
C[C@H]1CN(C[C@@H](C)N1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)cc(c1)C(F)(F)F |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1cc(cc(c1)C(F)(F)F)N1CCOCC1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1cc(cc(c1)C(F)(F)F)N1CCN(CCO)CC1
C[C@@H]1CN(CCN1)c1cc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCOCC3)c2)cc(c1)C(F)(F)F |r|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1cc(CN2CCCC2)c(Cl)c(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1cc(OCCN2CCOCC2)cc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1ccnc1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(ccc3C#N)C(F)(F)F)c2n1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(C#N)c(c3)C(F)(F)F)c2n1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(ccc3Cl)C(F)(F)F)c2n1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(ccc3N3CCOCC3)C(F)(F)F)c2n1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(OC)cc(c3)C(F)(F)F)c2n1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(F)c(c3)C(F)(F)F)c2n1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(ccc3-n3ccnn3)C(F)(F)F)c2n1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(ccc3-n3cccn3)C(F)(F)F)c2n1
COc1c(CN2CCCC2)cc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCOCC2)c1)C(F)(F)F
COc1c(CNC(C)C)cc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCOCC2)c1)C(F)(F)F
COc1c(CN2CCCC2)cc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N2CC[C@H](F)C2)c1)C(F)(F)F |r|
COc1c(CNC(C)C)cc(cc1NC(=O)c1ccc(C)c(Nc2ncnc3cnc(nc23)N2CC[C@H](F)C2)c1)C(F)(F)F |r|
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N(C)CC3CCCO3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCC5CCCCO5)nc34)c2)cc1C(F)(F)F
COC[C@@H]1CCCN1c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(OC)c(c3)C(F)(F)F)c2n1 |r|
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCC[C@H]3CO)c2)cc1C(F)(F)F |r|
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NCC(C)C)nc34)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N(C)C3CCOC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)-n3cnc(C)c3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3C[C@H](C)O[C@H](C)C3)c2)cc1C(F)(F)F |r|
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCCOCC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCN(CCN4CCOCC4)CC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCN(CCCN4CCCC4)CC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCN(CC4CCCN(C)C4)CC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCN4CCCCC4C3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCC(CC3)N3CCCCC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCN(CC3)C3CCN(C)CC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCC(CC3)N3CCOCC3)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCC(CC3)N3C[C@H](C)O[C@H](C)C3)c2)cc1C(F)(F)F |r|
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCC(CC3)N3CCCC3)c2)cc1C(F)(F)F
CCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(OC)c(c3)C(F)(F)F)c2n1
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCC(C3)N(C)C)c2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N(C)C3CCN(C)C3)c2)cc1C(F)(F)F
COc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(nn3C)C(C)(C)C)c2n1
COc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(cc(c3)C(F)(F)F)N3CCN(CC3)C(C)C)c2n1
COc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(F)(F)F)c2n1
COc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc(OC)c(c3)C(F)(F)F)c2n1
COc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cccc(c3)C(C)(C)C)c2n1
COc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(cc(c3)C(F)(F)F)N(C)CCN(C)C)c2n1
COc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(CN4CCCC4)cc(c3)C(F)(F)F)c2n1
COc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(n[nH]3)C(C)(C)C)c2n1
COc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN(c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C)c1ncnc2cnc(nc12)N1CCOCC1
CN(c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C)c1ncnc2cnc(NC3CCOC3)nc12
COCCN1CCN(CC1)c1ncc2ncnc(N(C)c3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN(c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C)c1ncnc2cnc(nc12)N1CC[C@H](F)C1 |r|
COc1ccc(NC(=O)c2ccc(C)c(c2)N(C)c2ncnc3cnc(nc23)N2CCOCC2)cc1C(F)(F)F
COc1ccc(NC(=O)c2ccc(C)c(c2)N(C)c2ncnc3cnc(NC4CCOC4)nc23)cc1C(F)(F)F
COCCN1CCN(CC1)c1ncc2ncnc(N(C)c3cc(ccc3C)C(=O)Nc3ccc(OC)c(c3)C(F)(F)F)c2n1
COc1ccc(NC(=O)c2ccc(C)c(c2)N(C)c2ncnc3cnc(nc23)N2CC[C@H](F)C2)cc1C(F)(F)F |r|
Cc1ccc(cc1Oc1ncnc2cnc(nc12)N1CCOCC1)C(=O)Nc1cc(nn1C)C(C)(C)C
CN1CCN(CC1)C1CC(C1)Nc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1 |(13.11,4.78,;11.77,4.01,;11.77,2.47,;10.44,1.7,;9.11,2.47,;9.11,4.01,;10.44,4.78,;7.77,1.7,;7.38,.21,;5.89,.61,;6.29,2.1,;4.55,-.16,;3.22,.61,;3.22,2.15,;1.89,2.92,;.55,2.15,;-.78,2.92,;-2.11,2.15,;-2.11,.61,;-.78,-.16,;-.78,-1.7,;-2.11,-2.47,;-3.45,-1.7,;-4.78,-2.47,;-4.78,-4.01,;-3.45,-4.78,;-2.11,-4.01,;-.78,-4.78,;-6.11,-1.7,;-6.11,-.16,;-7.45,-2.47,;-8.78,-1.7,;-9.26,-.24,;-10.8,-.24,;-11.27,-1.7,;-10.03,-2.61,;-11.57,1.1,;-10.8,2.43,;-13.11,1.1,;-10.23,1.87,;.55,.61,;1.89,-.16,)|
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(NC5CC(C5)N5CCN(C)CC5)nc34)c2)cc1C(F)(F)F |(-12.95,2.15,;-12.95,.61,;-11.61,-.16,;-11.61,-1.7,;-10.28,-2.47,;-8.94,-1.7,;-7.61,-2.47,;-6.28,-1.7,;-6.28,-.16,;-4.94,-2.47,;-4.94,-4.01,;-3.61,-4.78,;-2.28,-4.01,;-.94,-4.78,;-2.28,-2.47,;-.94,-1.7,;-.94,-.16,;-2.28,.61,;-2.28,2.15,;-.94,2.92,;.39,2.15,;1.72,2.92,;3.06,2.15,;3.06,.61,;4.39,-.16,;5.73,.61,;7.21,.21,;7.61,1.7,;6.12,2.1,;8.94,2.47,;10.28,1.7,;11.61,2.47,;11.61,4.01,;12.95,4.78,;10.28,4.78,;8.94,4.01,;1.72,-.16,;.39,.61,;-3.61,-1.7,;-8.94,-.16,;-10.28,.61,;-10.28,2.15,;-11.61,2.92,;-8.94,2.92,;-8.94,1.38,)|
COCCN1CCC(CC1)Nc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
CN1CCC(CC1)Nc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccnc(c3)C(C)(C)C)c2n1
CN(C1CC(C1)N1CCN(C)CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1 |(4.55,-1.7,;4.55,-.16,;5.89,.61,;7.38,.21,;7.77,1.7,;6.29,2.1,;9.11,2.47,;10.44,1.7,;11.77,2.47,;11.77,4.01,;13.11,4.78,;10.44,4.78,;9.11,4.01,;3.22,.61,;3.22,2.15,;1.89,2.92,;.55,2.15,;-.78,2.92,;-2.11,2.15,;-2.11,.61,;-.78,-.16,;-.78,-1.7,;-2.11,-2.47,;-3.45,-1.7,;-4.78,-2.47,;-4.78,-4.01,;-3.45,-4.78,;-2.11,-4.01,;-.78,-4.78,;-6.11,-1.7,;-6.11,-.16,;-7.45,-2.47,;-8.78,-1.7,;-9.26,-.24,;-10.8,-.24,;-11.27,-1.7,;-10.03,-2.61,;-11.57,1.1,;-10.8,2.43,;-13.11,1.1,;-10.23,1.87,;.55,.61,;1.89,-.16,)|
CN(C1CC(C1)N1CCN(C)CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccnc(c3)C(C)(C)C)c2n1 |(3.73,-1.7,;3.73,-.16,;5.06,.61,;6.55,.21,;6.94,1.7,;5.46,2.1,;8.28,2.47,;9.61,1.7,;10.95,2.47,;10.95,4.01,;12.28,4.78,;9.61,4.78,;8.28,4.01,;2.39,.61,;2.39,2.15,;1.06,2.92,;-.28,2.15,;-1.61,2.92,;-2.94,2.15,;-2.94,.61,;-1.61,-.16,;-1.61,-1.7,;-2.94,-2.47,;-4.28,-1.7,;-5.61,-2.47,;-5.61,-4.01,;-4.28,-4.78,;-2.94,-4.01,;-1.61,-4.78,;-6.94,-1.7,;-6.94,-.16,;-8.28,-2.47,;-9.61,-1.7,;-10.95,-2.47,;-12.28,-1.7,;-12.28,-.16,;-10.95,.61,;-9.61,-.16,;-10.95,2.15,;-12.28,2.92,;-9.61,2.92,;-9.61,1.38,;-.28,.61,;1.06,-.16,)|
CN(C)CCCNc1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)c2n1
COc1ccc(NC(=O)c2ccc(C)c(Nc3ncnc4cnc(nc34)N3CCC(CN(C)C)CC3)c2)cc1C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCC(CN2CCCC2)CC1)C(=O)Nc1cc(n[nH]1)C(C)(C)C
CC1=Nc2ccc(NC(=O)c3ccc(C)c(Nc4ncnc5cnc(nc45)N4CCC(CN5CCCC5)CC4)c3)cc2C1(C)C |t:1|
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCN(CC2CCOC2)CC1)C(=O)Nc1cc(n[nH]1)C(C)(C)C
CN1CCC2(CCN(C2)c2ncc3ncnc(Nc4cc(ccc4C)C(=O)Nc4cc(on4)C(C)(C)C)c3n2)C1
Cc1ccc(cc1Nc1ncnc2cnc(nc12)N1CCC(CN2CCCC2)CC1)C(=O)Nc1ccnc(c1)C(C)(C)C
Cc1cn(cn1)-c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3cc(n[nH]3)C(C)(C)C)c2n1
CN(C)CCC1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccnc(c3)C(C)(C)C)c2n1
CN(C)CCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc4OC(F)(F)C(F)(F)Oc4c3)c2n1
COCCN1CCN(CC1)c1ncc2ncnc(Nc3cc(ccc3C)C(=O)Nc3ccc4c(OC(F)(F)OC4(F)F)c3)c2n1
COc1ccc(cc1C(F)(F)F)C(=O)Nc1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCN(C)CC2)c1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1Nc1ncnc2cnc(nc12)N1CCOCC1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(F)(F)F)ccc3C)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(NC(=O)c4cc(n[nH]4)C(C)(C)C)ccc3C)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(NC(=O)c4cc(on4)C(C)(C)C)ccc3C)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(C)(C)C#N)ccc3C)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(NC(=O)c4cc(nn4C)C(C)(C)C)ccc3C)c2n1
CN(C)c1ncc2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(C)(C)C#N)ccc3C)c2n1
CN(C)c1ncc2ncnc(Nc3cc(NC(=O)c4cc(cc(c4)C(F)(F)F)N4CCN(C)CC4)ccc3C)c2n1
COc1ccc(cc1C(F)(F)F)C(=O)Nc1ccc(C)c(Nc2ncnc3cnc(nc23)N(C)C)c1
CN(C)CCN(C)c1ncc2ncnc(Nc3cc(NC(=O)c4cc(cc(c4)C(F)(F)F)N4CCN(C)CC4)ccc3C)c2n1
CN(C)CCCN(C)c1ncc2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(C)(C)C#N)ccc3C)c2n1
CN(C)CCCN(C)c1ncc2ncnc(Nc3cc(NC(=O)c4cc(cc(c4)C(F)(F)F)N4CCN(C)CC4)ccc3C)c2n1
CN(C)CCCN(C)c1ncc2ncnc(Nc3cc(NC(=O)c4cc(nn4C)C(C)(C)C)ccc3C)c2n1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1Nc1ncnc2cnc(nc12)N1CCN(CC1)C1CC1
CCN1CCN(CC1)c1ncc2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(C)(C)C#N)ccc3C)c2n1
CN1CCC(CC1)Nc1ncc2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(C)(C)C#N)ccc3C)c2n1
CN(C1CCN(C)CC1)c1ncc2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(C)(C)C#N)ccc3C)c2n1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1Nc1ncnc2cnc(NC3CCOC3)nc12
CN(C1CCOCC1)c1ncc2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(C)(C)C#N)ccc3C)c2n1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1Nc1ncnc2cnc(nc12)N1CCC(F)(F)C1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1Nc1ncnc2cnc(nc12)N1CC[C@@H](F)C1 |r|
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1Nc1ncnc2cnc(nc12)N1CC[C@H](F)C1 |r|
CC(=O)N1CCN(CC1)c1ncc2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(C)(C)C#N)ccc3C)c2n1
CN(C1CCOC1)c1ncc2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(C)(C)C#N)ccc3C)c2n1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1Nc1ncnc2cnc(NC3CCOCC3)nc12
CN(CC1CCOCC1)c1ncc2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(C)(C)C#N)ccc3C)c2n1
COc1ncc2ncnc(Nc3cc(NC(=O)c4cccc(c4)C(C)(C)C#N)ccc3C)c2n1
COc1ncc2ncnc(Nc3cc(NC(=O)c4ccc(OC)c(c4)C(F)(F)F)ccc3C)c2n1
COc1ncc2ncnc(Nc3cc(NC(=O)c4cc(cc(c4)C(F)(F)F)N4CCN(C)CC4)ccc3C)c2n1
COc1ncc2ncnc(Nc3cc(NC(=O)c4ccc(Cl)c(c4)C(F)(F)F)ccc3C)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(NS(=O)(=O)CC(F)(F)F)ccc3C)c2n1
CC(C)CCS(=O)(=O)Nc1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCN(C)CC2)c1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(NS(=O)(=O)C4CCCCC4)ccc3C)c2n1
CCC(C)S(=O)(=O)Nc1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCN(C)CC2)c1
CC(C)CS(=O)(=O)Nc1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCN(C)CC2)c1
CC(C)S(=O)(=O)Nc1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCN(C)CC2)c1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(NS(=O)(=O)CCC(F)(F)F)ccc3C)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(NS(=O)(=O)CC4CC4)ccc3C)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(NS(=O)(=O)c4cccc(c4)C(F)(F)F)ccc3C)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(NS(=O)(=O)CC4CCCO4)ccc3C)c2n1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(NS(=O)(=O)C4CC4)ccc3C)c2n1
CCS(=O)(=O)Nc1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCN(C)CC2)c1
CCCS(=O)(=O)Nc1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCN(C)CC2)c1
CN1CCN(CC1)c1ncc2ncnc(Nc3cc(NS(C)(=O)=O)ccc3C)c2n1
CCN1CCN(CC1)c1cc(cc(c1)C(C)(C)C#N)C(=O)Nc1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCOCC2)c1
CN1CCN(CC1)c1cc(cc(c1)C(C)(C)C#N)C(=O)Nc1ccc(C)c(Nc2ncnc3cnc(nc23)N2CCOCC2)c1
Cc1ccc(cc1Nc1ncnc2cncnc12)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cncnc12)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncnc2cncnc12)C(=O)Nc1cc(n[nH]1)C(C)(C)C
Cc1ccc(cc1Nc1ncnc2cncnc12)C(=O)Nc1cc(nn1C)C(C)(C)C
CNc1ncnc2c(Nc3cc(ccc3C)C(=O)Nc3cc(on3)C(C)(C)C)ncnc12
CNc1ncnc2c(Nc3cc(NC(=O)c4cccc(c4)C(C)(C)C#N)ccc3C)ncnc12
CC(C)(C#N)c1cccc(c1)C(=O)Nc1cccc(Nc2ncnc3c(N)ncnc23)c1
CNc1ncnc2c(Nc3cccc(NC(=O)c4cccc(c4)C(C)(C)C#N)c3)ncnc12
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccccc3)c2c1
COc1cccc(c1)-c1ccc2ncnc(Nc3ccccc3)c2c1
Oc1ccc(cc1)-c1ccc2ncnc(Nc3ccccc3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(O)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(F)c(Cl)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(F)cc3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(Cl)cc3F)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(C)cc3F)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(c3)C(F)(F)F)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(O)cc3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(F)cc3F)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(Cl)cc3O)c2c1
COc1cccc(Nc2ncnc3ccc(cc23)-c2ccc(O)c(OC)c2)c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccccc3O)c2c1
CCS(=O)(=O)Nc1ccc(cc1)-c1ccc2ncnc(Nc3ccccc3)c2c1
COc1ccc(Nc2ncnc3ccc(cc23)-c2ccc(O)c(OC)c2)cc1O
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(c3)S(N)(=O)=O)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(C)c(O)c3)c2c1
COc1cc(ccc1O)-c1cc2c(Nc3cccc(O)c3)ncnc2cc1OC
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccccc3C(N)=O)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(cc3O)C(O)=O)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(c3)C(N)=O)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(c3)[N+]([O-])=O)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(N)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc4OCOc4c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc4cn[nH]c4c3)c2c1
COc1cc(ccc1O)-c1cc2c(Nc3ccc(C)c(O)c3)ncnc2cc1OC
COc1cc(ccc1O)-c1cc2c(Nc3cc(O)ccc3Cl)ncnc2cc1OC
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(NC(C)=O)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(NC(=O)C(F)(F)F)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(cc3)S(N)(=O)=O)c2c1
COc1cc2ncnc(Nc3cccc(O)c3)c2cc1-c1ccc(O)cc1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(F)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(O)c3C)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc4nc[nH]c4c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(NS(C)(=O)=O)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cc(O)ccc3F)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cc(O)ccc3Cl)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(O)c3Cl)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cc(O)c(Cl)cc3Cl)c2c1
Oc1ccc(cc1)-c1ccc2ncnc(Nc3cccc(O)c3)c2c1
Oc1cccc(Nc2ncnc3ccc(cc23)-c2cccc(O)c2)c1
COc1ccc(cc1)-c1ccc2ncnc(Nc3cccc(O)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc4nn[nH]c4c3)c2c1
COc1cccc(c1)-c1ccc2ncnc(Nc3cccc(O)c3)c2c1
COc1cc2ncnc(Nc3cccc(O)c3)c2cc1-c1ccc(N)cc1
Nc1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
CC(=O)Nc1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
CS(=O)(=O)Nc1cccc(c1)-c1ccc2ncnc(Nc3cccc(O)c3)c2c1
CS(=O)(=O)Nc1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1cccc(-c2ccc3ncnc(Nc4cccc5[nH]ncc45)c3c2)c1F
COc1ccc(cc1F)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(cc1Cl)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(c(C)c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(cc1C)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
Fc1ccc(cc1Cl)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
Clc1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
Fc1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc4nn[nH]c34)c2c1
COc1cc(ccc1F)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
Fc1ccc(cc1F)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
N(c1cccc2[nH]ncc12)c1ncnc2ccc(cc12)-c1ccccc1
FC(F)(F)c1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
[C-]#[N+]c1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(cc1OC)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
CN(C)c1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
Fc1ccccc1-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
[O-][N+](=O)c1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
CCOc1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
OCc1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
CS(=O)(=O)Nc1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
C1Oc2ccc(cc2O1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
NC(=O)c1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(cc1C=O)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc4n(C)ncc34)c2c1
COc1cc(ccc1O)-c1ccc2nccc(Nc3cccc(O)c3)c2c1
COc1cc(ccc1O)-c1ccc2nccc(Nc3cc(O)ccc3F)c2c1
N#Cc1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1cc(ccc1O)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
Cc1ccc(F)cc1-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1cccc(-c2ccc3ncnc(Nc4cccc5[nH]ncc45)c3c2)c1OC
CN(C)c1ccc(cc1)-c1ccc2ncnc(Nc3cccc(O)c3)c2c1
O=S(=O)Nc1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
CCS(=O)(=O)Nc1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
CCCS(=O)(=O)Nc1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
CS(=O)(=O)c1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1cccc(-c2ccc3nccc(Nc4cccc5[nH]ncc45)c3c2)c1F
COc1ccc(cc1F)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(cc1OC)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
N#Cc1cccc(c1)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(cc1Cl)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(cc1C=O)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
NC(=O)c1cccc(c1)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(OC(F)F)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccccc3F)c2c1
CS(=O)(=O)c1ccc(cc1)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
Nc1ccc(cc1)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
CCCS(=O)(=O)Nc1cccc(c1)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
COc1cccc(c1)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
Oc1ccc(cc1)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
Fc1ccccc1-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc4[nH]nc(Cl)c34)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc4[nH]c(=O)[nH]c34)c2c1
COc1cc(ccc1O)-c1ccc2nccc(Nc3cc(NS(C)(=O)=O)ccc3F)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cc(NS(C)(=O)=O)ccc3F)c2c1
Oc1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
Oc1cccc(Nc2ncnc3ccc(cc23)-c2ccccc2)c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3c(F)cccc3F)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3c(F)ccc4[nH]ncc34)c2c1
Nc1ccc(F)c(c1)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
Nc1ccc(F)c(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
Oc1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
Oc1cccc(c1)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(cc1)-c1ccc2ncnc(Oc3cccc(O)c3)c2c1
N(c1cccc2[nH]ncc12)c1ncnc2ccc(cc12)-c1ccc2[nH]ncc2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cc(O)ccc3C)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cc(O)c(C)cc3F)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(Cl)c(O)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cc(O)c(F)cc3F)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cc(O)c(Cl)cc3F)c2c1
Oc1cc(Nc2ncnc3ccc(cc23)-c2ccc(Cl)cc2)c(F)cc1F
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(F)c(O)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(F)c(O)c3F)c2c1
Oc1c(F)ccc(Nc2ncnc3ccc(cc23)-c2ccc3[nH]ncc3c2)c1F
Oc1c(F)ccc(Nc2ncnc3ccc(cc23)-c2ccc(Cl)cc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-n1cc(-c2cncc(OC)c2)c2nc(ccc12)N1CCN(C)CC1 |(-9.1,-3.71,;-7.76,-4.48,;-6.43,-3.71,;-5.1,-4.48,;-5.1,-6.02,;-6.43,-5.25,;-3.76,-3.71,;-2.43,-4.48,;-2.43,-6.02,;-1.09,-6.79,;.24,-6.02,;1.57,-6.79,;.24,-4.48,;-1.09,-3.71,;-1.09,-2.17,;1.57,-3.71,;3.04,-4.19,;3.94,-2.94,;5.43,-3.34,;5.83,-4.83,;7.32,-5.23,;8.41,-4.14,;8.01,-2.65,;9.1,-1.56,;8.7,-.07,;6.52,-2.25,;3.04,-1.7,;3.36,-.19,;2.21,.84,;.75,.37,;.43,-1.14,;1.57,-2.17,;2.61,2.33,;1.52,3.42,;1.92,4.91,;3.41,5.3,;3.81,6.79,;4.5,4.21,;4.1,2.73,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-n1cc(-c2cncc(OC)c2)c2nc(ccc12)N1CCN(CCOC)CC1 |(-9.1,-5.54,;-7.76,-6.31,;-6.43,-5.54,;-5.1,-6.31,;-5.1,-7.85,;-6.43,-7.08,;-3.76,-5.54,;-2.43,-6.31,;-2.43,-7.85,;-1.09,-8.62,;.24,-7.85,;1.57,-8.62,;.24,-6.31,;-1.09,-5.54,;-1.09,-4,;1.57,-5.54,;3.04,-6.02,;3.94,-4.77,;5.43,-5.17,;5.83,-6.66,;7.32,-7.06,;8.41,-5.97,;8.01,-4.48,;9.1,-3.39,;8.7,-1.91,;6.52,-4.08,;3.04,-3.53,;3.36,-2.02,;2.21,-.99,;.75,-1.47,;.43,-2.97,;1.57,-4,;2.61,.5,;1.52,1.58,;1.92,3.07,;3.41,3.47,;3.81,4.96,;2.72,6.05,;3.12,7.54,;2.03,8.62,;4.5,2.38,;4.1,.89,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-n1cc(-c2cncc(OC)c2)c2nc(cnc12)N(C)C1CCN(C)CC1 |(-9.1,-3.66,;-7.76,-4.43,;-6.43,-3.66,;-5.1,-4.43,;-5.1,-5.97,;-6.43,-5.2,;-3.76,-3.66,;-2.43,-4.43,;-2.43,-5.97,;-1.09,-6.74,;.24,-5.97,;1.57,-6.74,;.24,-4.43,;-1.09,-3.66,;-1.09,-2.12,;1.57,-3.66,;3.04,-4.13,;3.94,-2.89,;5.43,-3.29,;5.83,-4.77,;7.32,-5.17,;8.41,-4.08,;8.01,-2.6,;9.1,-1.51,;8.7,-.02,;6.52,-2.2,;3.04,-1.64,;3.36,-.14,;2.21,.89,;.75,.42,;.43,-1.09,;1.57,-2.12,;2.61,2.38,;4.1,2.78,;1.52,3.47,;1.92,4.96,;.83,6.05,;-.65,5.65,;-1.74,6.74,;-1.05,4.16,;.04,3.07,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-n1cc(-c2cncc(OC)c2)c2nc(ncc12)N1CCN(C)CC1 |(-9.1,-3.71,;-7.76,-4.48,;-6.43,-3.71,;-5.1,-4.48,;-5.1,-6.02,;-6.43,-5.25,;-3.76,-3.71,;-2.43,-4.48,;-2.43,-6.02,;-1.09,-6.79,;.24,-6.02,;1.57,-6.79,;.24,-4.48,;-1.09,-3.71,;-1.09,-2.17,;1.57,-3.71,;3.04,-4.19,;3.94,-2.94,;5.43,-3.34,;5.83,-4.83,;7.32,-5.23,;8.41,-4.14,;8.01,-2.65,;9.1,-1.56,;8.7,-.07,;6.52,-2.25,;3.04,-1.7,;3.36,-.19,;2.21,.84,;.75,.37,;.43,-1.14,;1.57,-2.17,;2.61,2.33,;1.52,3.42,;1.92,4.91,;3.41,5.3,;3.81,6.79,;4.5,4.21,;4.1,2.73,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-n1cc(-c2cncc(OC)c2)c2nc(ncc12)N(C)C1CCN(C)CC1 |(-9.1,-3.66,;-7.76,-4.43,;-6.43,-3.66,;-5.1,-4.43,;-5.1,-5.97,;-6.43,-5.2,;-3.76,-3.66,;-2.43,-4.43,;-2.43,-5.97,;-1.09,-6.74,;.24,-5.97,;1.57,-6.74,;.24,-4.43,;-1.09,-3.66,;-1.09,-2.12,;1.57,-3.66,;3.04,-4.13,;3.94,-2.89,;5.43,-3.29,;5.83,-4.77,;7.32,-5.17,;8.41,-4.08,;8.01,-2.6,;9.1,-1.51,;8.7,-.02,;6.52,-2.2,;3.04,-1.64,;3.36,-.14,;2.21,.89,;.75,.42,;.43,-1.09,;1.57,-2.12,;2.61,2.38,;4.1,2.78,;1.52,3.47,;1.92,4.96,;.83,6.05,;-.65,5.65,;-1.74,6.74,;-1.05,4.16,;.04,3.07,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-n1cc(-c2cncnc2)c2nc(ncc12)N(C)C1CCN(C)CC1 |(-8.75,-3.66,;-7.42,-4.43,;-6.08,-3.66,;-4.75,-4.43,;-4.75,-5.97,;-6.08,-5.2,;-3.42,-3.66,;-2.08,-4.43,;-2.08,-5.97,;-.75,-6.74,;.58,-5.97,;1.92,-6.74,;.58,-4.43,;-.75,-3.66,;-.75,-2.12,;1.92,-3.66,;3.38,-4.13,;4.29,-2.89,;5.78,-3.29,;6.17,-4.77,;7.66,-5.17,;8.75,-4.08,;8.35,-2.6,;6.86,-2.2,;3.38,-1.64,;3.7,-.14,;2.56,.89,;1.09,.42,;.77,-1.09,;1.92,-2.12,;2.96,2.38,;4.44,2.78,;1.87,3.47,;2.27,4.96,;1.18,6.05,;-.31,5.65,;-1.4,6.74,;-.71,4.16,;.38,3.07,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-n1cc(-c2cncnc2)c2nc(ncc12)N(C)C1CCN(CC)CC1 |(-8.75,-4.4,;-7.42,-5.17,;-6.08,-4.4,;-4.75,-5.17,;-4.75,-6.71,;-6.08,-5.94,;-3.42,-4.4,;-2.08,-5.17,;-2.08,-6.71,;-.75,-7.48,;.58,-6.71,;1.92,-7.48,;.58,-5.17,;-.75,-4.4,;-.75,-2.86,;1.92,-4.4,;3.38,-4.88,;4.29,-3.63,;5.78,-4.03,;6.17,-5.52,;7.66,-5.92,;8.75,-4.83,;8.35,-3.34,;6.86,-2.94,;3.38,-2.39,;3.7,-.88,;2.56,.15,;1.09,-.32,;.77,-1.83,;1.92,-2.86,;2.96,1.64,;4.44,2.04,;1.87,2.73,;2.27,4.21,;1.18,5.3,;-.31,4.91,;-1.4,5.99,;-1,7.48,;-.71,3.42,;.38,2.33,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-n1cc(-c2cncnc2)c2nc(ncc12)N(C)C1CCN(CC1)C1CC1 |(-8.75,-4.4,;-7.42,-5.17,;-6.08,-4.4,;-4.75,-5.17,;-4.75,-6.71,;-6.08,-5.94,;-3.42,-4.4,;-2.08,-5.17,;-2.08,-6.71,;-.75,-7.48,;.58,-6.71,;1.92,-7.48,;.58,-5.17,;-.75,-4.4,;-.75,-2.86,;1.92,-4.4,;3.38,-4.88,;4.29,-3.63,;5.78,-4.03,;6.17,-5.52,;7.66,-5.92,;8.75,-4.83,;8.35,-3.34,;6.86,-2.94,;3.38,-2.39,;3.7,-.88,;2.56,.15,;1.09,-.32,;.77,-1.83,;1.92,-2.86,;2.96,1.64,;4.44,2.04,;1.87,2.73,;2.27,4.21,;1.18,5.3,;-.31,4.91,;-.71,3.42,;.38,2.33,;-1.4,5.99,;-1.8,7.48,;-2.89,6.39,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-n1cc(-c2cncnc2)c2nc(ncc12)N(C)C1CCN(CCOC)CC1 |(-8.75,-5.69,;-7.42,-6.46,;-6.08,-5.69,;-4.75,-6.46,;-4.75,-8,;-6.08,-7.23,;-3.42,-5.69,;-2.08,-6.46,;-2.08,-8,;-.75,-8.77,;.58,-8,;1.92,-8.77,;.58,-6.46,;-.75,-5.69,;-.75,-4.15,;1.92,-5.69,;3.38,-6.17,;4.29,-4.92,;5.78,-5.32,;6.17,-6.81,;7.66,-7.2,;8.75,-6.12,;8.35,-4.63,;6.86,-4.23,;3.38,-3.67,;3.7,-2.17,;2.56,-1.14,;1.09,-1.61,;.77,-3.12,;1.92,-4.15,;2.96,.35,;4.44,.75,;1.87,1.44,;2.27,2.93,;1.18,4.02,;-.31,3.62,;-1.4,4.71,;-1,6.19,;-2.09,7.28,;-1.69,8.77,;-.71,2.13,;.38,1.04,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-n1cc(-c2cncnc2)c2nc(ncc12)N(C)C1CCNCC1 |(-8.75,-3.31,;-7.42,-4.08,;-6.08,-3.31,;-4.75,-4.08,;-4.75,-5.62,;-6.08,-4.85,;-3.42,-3.31,;-2.08,-4.08,;-2.08,-5.62,;-.75,-6.39,;.58,-5.62,;1.92,-6.39,;.58,-4.08,;-.75,-3.31,;-.75,-1.77,;1.92,-3.31,;3.38,-3.79,;4.29,-2.54,;5.78,-2.94,;6.17,-4.43,;7.66,-4.83,;8.75,-3.74,;8.35,-2.25,;6.86,-1.85,;3.38,-1.3,;3.7,.21,;2.56,1.24,;1.09,.76,;.77,-.74,;1.92,-1.77,;2.96,2.73,;4.44,3.13,;1.87,3.82,;2.27,5.3,;1.18,6.39,;-.31,5.99,;-.71,4.51,;.38,3.42,)|
OC(=O)c1ccc(O[C@H]2CCC(CC2)NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)cc1 |r,wU:8.7,(10.67,,;9.34,-.77,;9.34,-2.31,;8,,;6.67,-.77,;5.33,,;5.33,1.54,;4,2.31,;2.67,1.54,;2.67,,;1.33,-.77,;;,1.54,;1.33,2.31,;-1.33,-.77,;-2.67,,;-2.67,1.54,;-4,-.77,;-5.33,,;-5.33,1.54,;-6.67,2.31,;-8,1.54,;-9.34,2.31,;-8,,;-6.67,-.77,;-9.34,-.77,;-10.67,,;-9.34,-2.31,;-10.67,-1.54,;6.67,2.31,;8,1.54,)|
CNC(=O)c1ccc(O[C@H]2CCC(CC2)NC(=O)Nc2ccc(OC(F)(F)F)cc2)cc1 |r,wU:9.8,(10.67,-.77,;9.34,,;8,-.77,;8,-2.31,;6.67,,;5.33,-.77,;4,,;4,1.54,;2.67,2.31,;1.33,1.54,;1.33,,;,-.77,;-1.33,,;-1.33,1.54,;,2.31,;-2.67,-.77,;-4,,;-4,1.54,;-5.33,-.77,;-6.67,,;-6.67,1.54,;-8,2.31,;-9.34,1.54,;-10.67,2.31,;-10.67,3.85,;-10.67,5.39,;-9.34,4.62,;-12,4.62,;-9.34,,;-8,-.77,;5.33,2.31,;6.67,1.54,)|
CNC(=O)c1cc(O[C@H]2CCC(CC2)NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)ccn1 |r,wU:8.7,(11.34,1.54,;10,.77,;8.67,1.54,;8.67,3.08,;7.34,.77,;6,1.54,;4.67,.77,;3.33,1.54,;2,.77,;2,-.77,;.67,-1.54,;-.67,-.77,;-.67,.77,;.67,1.54,;-2,-1.54,;-3.33,-.77,;-3.33,.77,;-4.67,-1.54,;-6,-.77,;-6,.77,;-7.34,1.54,;-8.67,.77,;-10,1.54,;-8.67,-.77,;-7.34,-1.54,;-10,-1.54,;-11.34,-.77,;-10,-3.08,;-11.34,-2.31,;4.67,-.77,;6,-1.54,;7.34,-.77,)|
CC(C)(C)OC(=O)c1cc(O[C@H]2CCC(CC2)NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)ccn1 |r,wU:11.10,(12.21,.77,;10.67,.77,;10.67,2.31,;10.67,-.77,;9.13,.77,;7.8,1.54,;7.8,3.08,;6.46,.77,;5.13,1.54,;3.79,.77,;2.46,1.54,;1.13,.77,;1.13,-.77,;-.21,-1.54,;-1.54,-.77,;-1.54,.77,;-.21,1.54,;-2.87,-1.54,;-4.21,-.77,;-4.21,.77,;-5.54,-1.54,;-6.87,-.77,;-6.87,.77,;-8.21,1.54,;-9.54,.77,;-10.88,1.54,;-9.54,-.77,;-8.21,-1.54,;-10.88,-1.54,;-12.21,-.77,;-10.88,-3.08,;-12.21,-2.31,;3.79,-.77,;5.13,-1.54,;6.46,-.77,)|
CNC(=O)c1cc(Oc2ccc(NC(=O)NC34CC5CC(CC(C5)C3)C4)cc2)ccn1 |TLB:15:16:19:23.22.21,THB:17:18:21:25.16.24,17:16:19.18.23:21,24:16:19:23.22.21,24:22:19:25.17.16|
FC(F)(F)c1ccc(O[C@H]2CC[C@@H](CC2)NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)nc1 |r,wU:9.8,wD:12.15,(10.71,-1.64,;9.39,-.86,;8.6,-2.18,;10.17,.47,;8.06,-.07,;6.67,-.77,;5.33,,;5.33,1.54,;4,2.31,;2.67,1.54,;2.67,,;1.33,-.77,;;,1.54,;1.33,2.31,;-1.33,-.77,;-2.67,,;-2.67,1.54,;-4,-.77,;-5.33,,;-5.33,1.54,;-6.67,2.31,;-8,1.54,;-9.34,2.31,;-8,,;-6.67,-.77,;-9.34,-.77,;-10.67,,;-9.34,-2.31,;-10.67,-1.54,;6.67,2.31,;8,1.54,)|
CNC(=O)c1ccc(O[C@H]2CC[C@@H](CC2)NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)cn1 |r,wU:9.8,wD:12.15,(21.22,-29.7,;19.89,-28.92,;18.55,-29.69,;18.55,-31.23,;17.22,-28.92,;15.88,-29.69,;14.55,-28.91,;14.56,-27.37,;13.23,-26.6,;11.89,-27.36,;11.89,-28.9,;10.56,-29.66,;9.23,-28.9,;9.23,-27.36,;10.56,-26.58,;7.9,-29.67,;6.56,-28.91,;6.56,-27.37,;5.23,-29.68,;3.9,-28.91,;2.58,-29.68,;1.24,-28.92,;1.23,-27.37,;-.12,-26.61,;2.57,-26.6,;3.9,-27.37,;2.57,-25.06,;3.9,-24.29,;1.23,-24.29,;2.55,-23.51,;15.89,-26.61,;17.22,-27.37,)|
CNC(=O)c1cc(O[C@H]2CCC(CC2)NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)ccn1 |r,wD:8.7,(11.34,1.54,;10,.77,;8.67,1.54,;8.67,3.08,;7.34,.77,;6,1.54,;4.67,.77,;3.33,1.54,;2,.77,;.67,1.54,;-.67,.77,;-.67,-.77,;.67,-1.54,;2,-.77,;-2,-1.54,;-3.33,-.77,;-3.33,.77,;-4.67,-1.54,;-6,-.77,;-6,.77,;-7.34,1.54,;-8.67,.77,;-10,1.54,;-8.67,-.77,;-7.34,-1.54,;-10,-1.54,;-11.34,-.77,;-10,-3.08,;-11.34,-2.31,;4.67,-.77,;6,-1.54,;7.34,-.77,)|
Cc1ccc2c(Nc3ccc(Cl)cc3)nccc2c1NC(=O)c1csc2c(N)ncnc12
COc1ccc(Nc2nccc3c(NC(=O)c4csc5c(N)ncnc45)c(C)ccc23)cc1
Cc1ccc2c(Nc3cccc(Cl)c3)nccc2c1NC(=O)c1csc2c(N)ncnc12
Cc1ccc2c(Nc3ccc(OC(F)F)cc3)nccc2c1NC(=O)c1csc2c(N)ncnc12
CN(C)Cc1cc(Nc2nccc3c(NC(=O)c4csc5c(N)ncnc45)c(C)ccc23)ccc1Cl
CC(=O)c1ccc(Nc2nccc3c(NC(=O)c4csc5c(N)ncnc45)c(C)ccc23)cc1
Cc1ccc2c(Nc3ccc(F)c(Cl)c3)nccc2c1NC(=O)c1csc2c(N)ncnc12
Cc1ccc2c(c1NC(=O)c3csc4c3ncnc4N)ccnc2Nc5cccc(c5F)Cl
CNc1cc2nc(C)c(cc2cn1)-c1cc(NC(=O)NCCC(C)(C)C)ccc1F
CNc1cc2nc(C)c(cc2cn1)-c1cc(NC(=O)NCCC(C)(C)F)c(F)cc1C
CNC(=O)c1cc(Oc2cccc3nc(Nc4cccc(c4)C(C)(C)C)ccc23)ccn1
CNC(=O)c1cc(Oc2cccc3nc(Nc4ccc(Cl)c(c4)C(F)(F)F)ccc23)ccn1
Nc1ccc(cn1)-c1ccc2ncc3c(n(-c4cccc(c4)C(F)(F)F)c(=O)[nH]c3=O)c2n1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1NC(=O)c1cccc2c(N)nccc12
Nc1c(c(nn1-c1c(Cl)cc(Cl)cc1Cl)-c1ccncc1)-c1ccc(F)cc1 |(-1,-2.52,;-1.47,-1.05,;-2.94,-.58,;-2.94,.96,;-1.47,1.44,;-.56,.19,;.98,.19,;1.74,1.52,;.97,2.85,;3.28,1.52,;4.06,.18,;5.6,.18,;3.29,-1.15,;1.75,-1.15,;.97,-2.48,;-4.18,1.87,;-4.2,3.41,;-5.54,4.16,;-6.87,3.37,;-6.84,1.82,;-5.5,1.08,;-4.18,-1.48,;-5.52,-.72,;-6.85,-1.5,;-6.84,-3.04,;-8.17,-3.82,;-5.49,-3.8,;-4.17,-3.02,)|
Nc1c(c(nn1-c1ccccc1)-c1ccncc1)-c1ccc(F)cc1
Nc1c(c(nn1-c1ccc(Cl)cc1)-c1ccncc1)-c1ccc(F)cc1
COc1ccc(cc1)-n1nc(c(c1N)-c1ccc(F)cc1)-c1ccncc1
Nc1c(c(nn1-c1ccc(cc1)[N+]([O-])=O)-c1ccncc1)-c1ccc(F)cc1
Cc1ccc(cc1)-n1nc(c(c1N)-c1ccc(F)cc1)-c1ccncc1
Nc1c(c(nn1-c1ccc(cc1)C#N)-c1ccncc1)-c1ccc(F)cc1
Nc1c(c(nn1-c1ccc(cc1)C(F)(F)F)-c1ccncc1)-c1ccc(F)cc1
NC(=O)c1c(N)n(nc1-c1ccncc1)-c1c(Cl)cc(Cl)cc1Cl |(-5.26,-51.04,;-3.93,-51.81,;-3.93,-53.35,;-2.59,-51.04,;-1.13,-51.51,;-.66,-52.98,;-.22,-50.28,;-1.13,-49.02,;-2.59,-49.5,;-3.84,-48.59,;-3.86,-47.06,;-5.2,-46.3,;-6.52,-47.09,;-6.5,-48.64,;-5.16,-49.39,;1.32,-50.28,;2.08,-48.95,;1.31,-47.62,;3.62,-48.94,;4.4,-50.28,;5.94,-50.28,;3.63,-51.61,;2.09,-51.61,;1.32,-52.95,)|
CCOC(=O)c1c(N)n(nc1-c1ccncc1)-c1c(Cl)cc(Cl)cc1Cl |(15.66,-51.66,;16.99,-52.43,;18.32,-51.66,;19.66,-52.43,;19.66,-53.97,;20.99,-51.66,;22.46,-52.13,;22.93,-53.6,;23.37,-50.89,;22.46,-49.64,;20.99,-50.12,;19.75,-49.21,;19.73,-47.68,;18.38,-46.92,;17.06,-47.71,;17.08,-49.26,;18.43,-50,;24.91,-50.89,;25.67,-49.57,;24.89,-48.23,;27.2,-49.56,;27.98,-50.9,;29.52,-50.9,;27.21,-52.23,;25.67,-52.23,;24.9,-53.56,)|
NC(=O)c1c(N)n(nc1-c1ccncc1)-c1ccccc1
Nc1c(C(O)=O)c(nn1-c1c(Cl)cc(Cl)cc1Cl)-c1ccncc1 |(13.17,-1.44,;12.69,.03,;11.23,.5,;9.89,-.27,;8.56,.5,;9.89,-1.81,;11.23,2.04,;12.69,2.52,;13.6,1.27,;15.14,1.27,;15.91,2.6,;15.13,3.93,;17.44,2.6,;18.22,1.26,;19.76,1.27,;17.45,-.07,;15.91,-.07,;15.14,-1.4,;9.98,2.95,;9.97,4.49,;8.62,5.24,;7.3,4.45,;7.32,2.9,;8.67,2.16,)|
Nc1cc(nn1-c1c(Cl)cc(Cl)cc1Cl)-c1ccncc1 |(26.44,-.46,;25.97,1,;24.5,1.48,;24.5,3.02,;25.97,3.49,;26.88,2.24,;28.42,2.24,;29.18,3.57,;28.41,4.9,;30.72,3.57,;31.5,2.24,;33.04,2.24,;30.72,.9,;29.18,.9,;28.41,-.43,;23.26,3.92,;23.24,5.46,;21.9,6.21,;20.57,5.42,;20.6,3.88,;21.94,3.13,)|
Clc1cc(Cl)c(N\N=C\c2ccncc2)c(Cl)c1
Fc1ccc(cc1)-c1cn(nc1-c1ccncc1)-c1ccc(cc1)C(F)(F)F
COc1cc2c(cc1OCCCN3CCOCC3)c(ncn2)Nc4ccc(c(c4)Cl)F
CC1(C)OC(=C(C1=O)c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F)c1ccnc(S)n1 |c:4|
COC(=O)N[C@@H](C)CNc1nccc(n1)C1=C(C(=O)C(C)(C)O1)c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F |r,t:16|
CC1(C)OC(=C(C1=O)c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F)c1ccnc(NCCC#N)n1 |c:4|
Nc1nccc(n1)C1=C(C(=O)C2(CCCC2)O1)c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F |t:8|
CC(C)CC1(C)OC(=C(C1=O)c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F)c1ccnc(N)n1 |c:7|
CC(C)CC1(C)OC(=C(C1=O)c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F)c1ccnc(NCCC#N)n1 |c:7|
COC(=O)N[C@@H](C)CNc1nccc(n1)C1=C(C(=O)C(C)(CC(C)C)O1)c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F |r,t:16|
CC(C)CC1(C)OC(=C(C1=O)c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F)c1ccnc(NCc2nccs2)n1 |c:7|
CC(C)CC1(C)OC(=C(C1=O)c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F)c1ccnc(NC[C@H]2CCCN2)n1 |r,c:7|
CC(C)CC1(C)OC(=C(C1=O)c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F)c1ccnc(NCC2CCCO2)n1 |c:7|
CC1(C)OC(=C(C1=O)c1cc(Cl)cc(NS(=O)(=O)c2c(F)cccc2F)c1F)c1ccnc(N)n1 |c:4|
CC1(C)OC(=C(C1=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(F)ccc2F)c1F)c1ccnc(N)n1 |c:4|
CC1(C)OC(=C(C1=O)c1cc(Cl)cc(NS(=O)(=O)c2ccc(F)cc2F)c1F)c1ccnc(N)n1 |c:4|
CC1(C)OC(=C(C1=O)c1cc(Cl)cc(NS(=O)(=O)c2cccc(F)c2)c1F)c1ccnc(N)n1 |c:4|
CC1(C)OC(=C(C1=O)c1cc(Cl)cc(NS(=O)(=O)c2ccccc2F)c1F)c1ccnc(N)n1 |c:4|
CCCS(=O)(=O)Nc1cc(Cl)cc(C2=C(OC(C)(CC(C)C)C2=O)c2ccnc(N)n2)c1F |t:13|
Nc1nccc(n1)C1=C(C(=O)C2(CCCC2)O1)c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1Cl |t:8|
Nc1nccc(n1)C1=C(C(=O)C2(CCCC2)O1)c1cc(Cl)cc(NS(=O)(=O)c2c(F)cccc2F)c1Cl |t:8|
CC(C)CC1(C)OC(=C(C1=O)c1cc(Cl)cc(NS(=O)(=O)c2c(F)cccc2F)c1F)c1ccnc(N)n1 |c:7|
CC(C)CC1(C)OC(=C(C1=O)c1cc(Cl)cc(NS(=O)(=O)c2c(F)cccc2F)c1F)c1ccnc(NCCC#N)n1 |c:7|
CC1(C)OC(=C(C1=O)c1cc(Cl)cc(NS(=O)(=O)c2c(F)cccc2F)c1F)c1ccnc(NCCC#N)n1 |c:4|
COC(=O)N[C@@H](C)CNc1nccc(n1)C1=C(C(=O)C(C)(C)O1)c1cc(Cl)cc(NS(=O)(=O)c2cc(F)ccc2F)c1F |r,t:16|
CC1(C)OC(=C(C1=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(F)ccc2F)c1F)c1ccnc(NCCC#N)n1 |c:4|
C[C@H](O)CNc1nccc(n1)C1=C(C(=O)C(C)(C)O1)c1cc(Cl)cc(NS(=O)(=O)c2cc(F)ccc2F)c1F |r,t:12|
CC1(C)OC(=C(C1=O)c1cc(Cl)cc(NS(=O)(=O)c2cc(F)ccc2F)c1F)c1ccnc(NCCO)n1 |c:4|
COCCNc1nccc(n1)C1=C(C(=O)C(C)(C)O1)c1cc(Cl)cc(NS(=O)(=O)c2cc(F)ccc2F)c1F |t:12|
CCNc1nccc(n1)C1=C(C(=O)C(C)(C)O1)c1cc(Cl)cc(NS(=O)(=O)c2cc(F)ccc2F)c1F |t:10|
Nc1nccc(n1)C1=C(C(=O)C2(CCCC2)O1)c1cc(Cl)cc(NS(=O)(=O)c2cc(F)ccc2F)c1F |t:8|
Nc1nccc(n1)C1=C(C(=O)C2(CCCC2)O1)c1cc(Cl)cc(NS(=O)(=O)c2c(F)cccc2F)c1F |t:8|
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1=O
Cc1ccc(cc1-c1cc(nc(n1)N1CCOCC1)N1CCS(=O)(=O)CC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCS(=O)(=O)CC1)N1CCOCC1
Cc1ccc(cc1-c1cc(nc(n1)N1CCS(=O)(=O)CC1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F |$;;;;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1nc(cc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(cc1-c1nc(cc(n1)N1CCOCC1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2Cl)C2(CC2)C#N)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
CN(C)c1cncc(c1)C(=O)Nc1ccc(C)c(c1)-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
CN(C)Cc1cc(cc(c1)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
CCN1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)S(C)(=O)=O)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cc(no2)C(C)(C)C)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cc(on2)C(C)(C)C)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2csc(n2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)S(C)(=O)=O)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CC2(COC2)C1)N1CCOCC1
CNc1nc(cc(n1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(NCCO)n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCC(O)C1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)-n1ccnc1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(OCCO)n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(NS(C)(=O)=O)n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCCC1=O)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)-n1cc(nn1)C(C)(C)O)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(N)n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(NC(CO)CO)n1)N1CCOCC1
CC(=C)c1cc(nc(n1)N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
CC(C)c1cc(nc(n1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C)N1CCOCC1
CC(C)c1cc(nc(n1)N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOC(C)(C)C1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CC2(COC2)C1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOC[C@H]1CO |r|
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1C2CCC1COC2
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CCCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CC2CC1CO2
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CC2CCC(C1)O2
C[C@@H]1CN(CCO1)c1cc(nc(n1)N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C |r|
C[C@H]1CN(CCO1)c1cc(nc(n1)N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C |r|
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(OC2CCOCC2)nc(n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1nc(nc(N2CCOCC2)c1C)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(cnn1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(cnn1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)C(F)(F)F
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(cc1-c1ccnc(c1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccnn2)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)S(C)(=O)=O)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cnccn2)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cncnc2)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnnc2)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)F)cc1-c1ccnc(c1)N1CCOCC1
CN(C)c1cc(cc(n1)N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1ccnc(c1)N1CCO[C@H](CO)C1 |r|
C[C@@H]1CO[C@H](CN(C)C)CN1c1cc(ccn1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C |r|
C[C@H]1CO[C@@H](CN(C)C)CN1c1cc(ccn1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C |r|
CN(C)c1cncc(c1)C(=O)Nc1cnc(C)c(c1)-c1ccnc(c1)N1CCOCC1
C[C@@H]1COCCN1c1cc(ccn1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C |r|
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1ccnc(c1)N1CCO[C@H](CO)C1 |r|
CNC[C@@H]1CN(CCO1)c1cc(ccn1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C |r|
CC(=O)NC[C@@H]1CN(CCO1)c1cc(ccn1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C |r|
COC(=O)NC[C@@H]1CN(CCO1)c1cc(ccn1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C |r|
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1ccnc(c1)N1CCO[C@H](CNC(=O)CO)C1 |r|
COc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1ccnc(c1)N1CCOCC1
CC(F)(F)c1cc(ccn1)C(=O)Nc1c[nH]c(=O)c(c1)-c1ccnc(c1)N1CCOCC1
FC(F)(F)c1cc(ccn1)C(=O)Nc1c[nH]c(=O)c(c1)-c1ccnc(c1)N1CCOCC1
CC(C)(C#N)c1cc(ccn1)C(=O)Nc1c[nH]c(=O)c(c1)-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N)nc(c1)N1CCOCC1
CCn1cc(cc(c1=O)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1ccnc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1ccnc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1ccnc(c1)N1CCOCC1
COc1ccc(cc1C(F)(F)F)C(=O)Nc1cnc(C)c(c1)-c1ccnc(c1)N1CCOCC1
COc1cc(ccc1F)C(=O)Nc1cnc(C)c(c1)-c1ccnc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)F)cc1-c1ccnc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1ccnc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(C)(F)F)cc1-c1ccnc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1ccnc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)S(C)(=O)=O)cc1-c1ccnc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(c1)N1CCOCC1)C1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)C1CCOCC1
OCc1ccc(cc1-c1ccnc(c1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F
FC(F)c1ccc(cc1-c1ccnc(c1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F
FCc1ccc(cc1-c1ccnc(c1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(cc1-c1cc(nc(c1)N1CCOCC1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(c1)-c1cnn(C)c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1-c1cc(nc(c1)N1CCOCC1)C1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
CCn1cc(cc(c1=O)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cncc(n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1c[nH]c(=O)c(n1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1c[nH]c(=O)c(n1)N1CCOCC1
COc1ncc(cc1-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(cn(C)c1=O)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(cn(C)c1=O)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(c[nH]c1=O)N1CCOCC1
COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C
COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C
COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cnc1C
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(c1)C1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
CC(C)n1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C
CC(C)n1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
Cc1ccc(cc1-c1cc(N2CCOCC2)c(=O)n(C)c1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(CCO)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(CCO)c1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(CCO)c1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(OCCO)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1c[nH]c(=O)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(CC#N)c1
C[C@H](C#N)n1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C |r|
C[C@@H](C#N)n1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C |r|
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(CCS(C)(=O)=O)c1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(CCS(C)(=O)=O)c1
C[C@H](Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C)C#N |r|
C[C@@H](Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C)C#N |r|
Cc1ccc(cc1-c1cc(N2CCOCC2)c(=O)n(CCS(C)(=O)=O)c1)C(=O)Nc1cccc(c1)C(F)(F)F
CCn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
CCn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C
CCn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)ccc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)ccc1C
CCn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(cc1-c1cc(N2CCOCC2)c(=O)n(C)n1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
CCn1cc(nc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cn(CC(F)F)c(=O)c(n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
CN(C)Cc1cc(cc(c1)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
CCN1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
CN(C)c1cncc(c1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cc(cc(c2)S(C)(=O)=O)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
COc1ccc(cc1C(F)(F)F)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
COc1cc(ccc1F)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)S(C)(=O)=O)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(ccc1C(F)F)C(=O)Nc1cccc(c1)C(F)(F)F
COC(=O)NCCn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C
COC(=O)NCCn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
COc1cc(nc(c1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(OCc2ccccc2)cc(n1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(ncn1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(ncn1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1=O
Cc1ccc(cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1=O)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CCS(=O)(=O)CC1
Cc1ccc(cc1-c1cc(ccn1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F
CCN1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(cc(N)n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(ccn1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cn(C)c(=O)c(n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(s1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1csc(n1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(C#N)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cnc(OC(F)F)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(OC(F)F)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cnc(OC(F)F)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cnc(OC(F)F)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(OCC(F)F)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cnc(OCC(F)F)c(c1)N1CCOCC1
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)S(C)(=O)=O)ccc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)-c2nnco2)ccc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)F)ccc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)S(C)(=O)=O)ccc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cc(c(=O)n(CC)c2)C(F)(F)F)ccc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)O)ccc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)F)ccc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(ccc1C)C(=O)Nc1cccc(c1)S(C)(=O)=O
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cnc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)O)cnc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cc(c(=O)n(CC)c2)C(F)(F)F)cnc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)S(C)(=O)=O)cnc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cnc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)-c2nnco2)cnc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cc(on2)C2CC2)cnc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)cnc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)F)cnc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C
CN(C)Cc1cc(cc(c1)C(F)(F)F)C(=O)Nc1cnc(C)c(c1)-c1cnc(C#N)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cnc(C#N)c(c1)N1CCOCC1
CC(C)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1cnc(C#N)c(c1)N1CCOCC1
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)C)cnc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)cnc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C2CC2)cnc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C2COC2)cnc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(ccc1C)C(=O)Nc1cc(ccc1F)C(C)=C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cc(cc(c2)C(F)(F)F)N2CCN(CC)CC2)cnc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cc(CN(C)C)cc(c2)C(F)(F)F)cnc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cnnc(c2)C(F)(F)F)cnc1C
COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C2(CC2)C#N)cnc1Cl
COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)cnc1Cl
COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)cnc1Cl
COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cnnc(c2)C(F)(F)F)cnc1Cl
COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cnc1Cl
CN(C)c1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cnc1C
CN(C)c1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C2(CC2)C#N)cnc1C
CN(C)c1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)cnc1C
CN(C)c1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)cnc1C
CN(C)Cc1cc(cc(c1)C(F)(F)F)C(=O)Nc1cnc(C)c(c1)-c1cnc(N(C)C)c(c1)N1CCOCC1
CN(C)c1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cnnc(c2)C(F)(F)F)cnc1C
CN(C)c1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cnnc(c2)C2CC2)cnc1C
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cnnc(c2)C2CC2)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cnc(OC2CCOCC2)c(c1)N1C2CCC1COC2
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cnc(OC2CCOCC2)c(c1)N1C2CCC1COC2
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cnnc(c2)C(F)(F)F)ccc1C
COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)cnc1C
CCOc1ncc(cc1N1C2CCC1COC2)-c1cc(NC(=O)c2cnnc(c2)C(F)(F)F)cnc1C
COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C2(CC2)C#N)cnc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cnnc(c2)C(C)(C)C#N)ccc1C
CCOc1ncc(cc1N1CCOC[C@H]1C)-c1cc(NC(=O)c2cnnc(c2)C(F)(F)F)cnc1C |r|
CCOc1ncc(cc1N1CCOC[C@@H]1C)-c1cc(NC(=O)c2cnnc(c2)C(F)(F)F)cnc1C |r|
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cnnc(c2)C(C)(C)C#N)cnc1C
Cc1ncc(NC(=O)c2ccnc(c2)C2(CC2)C#N)cc1-c1cnc(Cl)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cnc(Cl)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cnc(Cl)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cnc(Cl)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cnc(Cl)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cnnc(c2)C(C)(C)C#N)cc1-c1cnc(Cl)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cncc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cncc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cnnc(c2)C(C)(C)C#N)cc1-c1cncc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cncc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cnc(F)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cnc(OCCO)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cnc(OCCO)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cc(ccn2)C(F)(F)F)cc1-c1cnc(OCCO)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cnnc(c2)C2(CC2)C#N)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
CCOc1ncc(cc1N1CCOC[C@H]1C)-c1cc(NC(=O)c2cnnc(c2)C(C)(C)C#N)cnc1C |r|
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cnnc(c2)C(C)(C)F)ccc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(ccc1C)C(=O)Nc1ccnc(c1)C(F)(F)F
CN(C)c1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C
CC(C)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1cnc(N(C)C)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1=O
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(O[C@H]2CCOC2)c(c1)N1CCOCC1 |r|
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(O[C@@H]2CCOC2)c(c1)N1CCOCC1 |r|
COCCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C
CC(C)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(OC2COC2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(OC2CCCC(O)C2)c(c1)N1CCOCC1
CN1CC(C1)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(OC2CC3(COC3)C2)c(c1)N1CCOCC1
COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)C)cnc1C
COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)cnc1C
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(OC2CNC2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(c(c1)N1CCOCC1)C(C)(C)C#N
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(CS(C)(=O)=O)c(c1)N1CCOCC1
CN(C(=O)c1cccc(c1)C(F)(F)F)c1cnc(C)c(c1)-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
CCN(C(=O)c1cccc(c1)C(F)(F)F)c1cnc(C)c(c1)-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
CCCN(C(=O)c1cccc(c1)C(F)(F)F)c1cnc(C)c(c1)-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
CCn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cnc1C
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(CCC#N)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(CCC#N)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(CCC#N)c1
Cc1ccc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(CCC#N)c1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(CC2(C)COC2)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(CC2(C)COC2)c1
COc1ccc(cc1C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
CCC(F)(F)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
CCOc1cc(ccc1F)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
CC(C)Oc1cccc(c1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2Cl)C2(CC2)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccccc2)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
CC(C)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)-c2nnco2)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)S(C)(=O)=O)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)C2COC2)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
CCc1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)C2CC2)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)C2COC2)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)C2(CC2)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(CC#N)c2)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cnnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cnnc(c2)C2CC2)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cnnc(c2)C(C)(C)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cc(ccn2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
CCn1cc(C(=O)Nc2ccc(C)c(c2)-c2cc(N3CCOCC3)c(=O)n(C)c2)c(C)n1
Cc1nn(C)cc1C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
CC(C)n1cc(C(=O)Nc2ccc(C)c(c2)-c2cc(N3CCOCC3)c(=O)n(C)c2)c(C)n1
Cc1ccc(NC(=O)c2cc(nn2C)C2CC2)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cc(nn2C)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
CC(C)c1cc(no1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cc(on2)C2CC2)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
CCn1cc(C(=O)Nc2cnc(C)c(c2)-c2cc(N3CCOCC3)c(=O)n(C)c2)c(C)n1
Cc1nn(C)cc1C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
CC(C)n1cc(C(=O)Nc2cnc(C)c(c2)-c2cc(N3CCOCC3)c(=O)n(C)c2)c(C)n1
Cc1cc(C(=O)Nc2cnc(C)c(c2)-c2cc(N3CCOCC3)c(=O)n(C)c2)n(C)n1
Cc1ncc(NC(=O)c2cc(nn2C)C2CC2)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
CC(C)c1cc(no1)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ncc(NC(=O)c2cc(on2)C2CC2)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1cc(C(=O)Nc2ccc(C)c(c2)-c2cc(N3CCOCC3)c(=O)n(C)c2)n(C)n1
Cc1ncc(NC(=O)c2cc(nn2C)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1nc(C(=O)Nc2cnc(C)c(c2)-c2cc(N3CCOCC3)c(=O)n(C)c2)c(C)o1
Cc1ncc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ncc(NC(=O)c2cccc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ncc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
CCOc1cc(ccc1F)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
CC(C)Oc1cc(ccc1F)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
CCOc1cccc(c1)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
CC(C)Oc1cccc(c1)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
CC(C)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
CN(C)Cc1cc(cc(c1)C(F)(F)F)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
CCN1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ncc(NC(=O)c2cccc(c2Cl)C2(CC2)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)cnc1Cl
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)cnc1Cl
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)F)cnc1Cl
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1Cl
COc1ccc(cc1C(F)(F)F)C(=O)Nc1cnc(Cl)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1Cl
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1F
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C#N
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)F)ccc1Cl
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)ccc1Cl
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1Cl
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)ccc1C#N
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1C#N
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)F)ccc1F
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)ccc1F
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1F
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)F)ccc1C#N
CC(C)c1cc(ccn1)C(=O)Nc1ccc(Cl)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
CC(C)c1cc(ccn1)C(=O)Nc1cnc(Cl)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(cnc1Cl)C(=O)Nc1cccc(c1)C(F)(F)F |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(cnc1Cl)C(=O)Nc1cccc(c1)C(C)(C)O |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(ccc1Cl)C(=O)Nc1cccc(c1)C(F)(F)F |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(ccc1Cl)C(=O)Nc1cccc(c1)C(F)F |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;$|
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(ccc1Cl)C(=O)Nc1cccc(c1)C(C)(C)C#N |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;$|
Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(c2)-c2cc(N3CCOCC3)c(=O)n(C)c2)cc(c1)C(F)(F)F |$;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;$|
Cc1ccc(cc1-c1cc(N2CCOCC2)c(=O)n(C)c1)C(=O)Nc1ccccc1 |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;$|
Cc1ccc(cc1-c1cc(N2CCOCC2)c(=O)n(C)c1)C(=O)Nc1cccc(c1)C(F)F |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;$|
Cc1ccc(cc1-c1cc(N2CCOCC2)c(=O)n(C)c1)C(=O)Nc1cccc(c1)C(C)(C)C#N |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;$|
Cc1ccc(cc1-c1cc(N2CCOCC2)c(=O)n(C)c1)C(=O)Nc1ccccn1 |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;$|
Cc1ccc(cc1-c1cc(N2CCOCC2)c(=O)n(C)c1)C(=O)Nc1cccnc1 |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;$|
CCc1cccc(NC(=O)c2ccc(C)c(c2)-c2cc(N3CCOCC3)c(=O)n(C)c2)c1 |$;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;;$|
CC(C)c1cccc(NC(=O)c2ccc(C)c(c2)-c2cc(N3CCOCC3)c(=O)n(C)c2)c1 |$;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;;$|
Cc1ccc(cc1-c1cc(N2CCOCC2)c(=O)n(C)c1)C(=O)Nc1cccc(c1)-c1nnco1 |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;$|
Cc1nc(no1)-c1cccc(NC(=O)c2ccc(C)c(c2)-c2cc(N3CCOCC3)c(=O)n(C)c2)c1 |$;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;;$|
Cc1ccc(cc1-c1cc(N2CCOCC2)c(=O)n(C)c1)C(=O)Nc1cccc(c1)C(C)(C)O |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
COc1cccc(NC(=O)c2ccc(C)c(c2)-c2cc(N3CCOCC3)c(=O)n(C)c2)c1 |$;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;;$|
Cc1ccc(cc1-c1cc(N2CCOCC2)c(=O)n(C)c1)C(=O)Nc1cccc(OC(F)(F)F)c1 |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;$|
COc1cncc(NC(=O)c2ccc(C)c(c2)-c2cc(N3CCOCC3)c(=O)n(C)c2)c1 |$;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;;$|
Cc1ncc(cc1-c1cc(N2CCOCC2)c(=O)n(C)c1)C(=O)Nc1cccc(c1)C(F)(F)F |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
Cc1ncc(cc1-c1cc(N2CCOCC2)c(=O)n(C)c1)C(=O)Nc1cccc(c1)C(C)(C)C#N |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;$|
Cc1ncc(cc1-c1cc(N2CCOCC2)c(=O)n(C)c1)C(=O)Nc1cccc(c1)C(F)F |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;$|
Cc1ncc(cc1-c1cc(N2CCOCC2)c(=O)n(C)c1)C(=O)Nc1cccc(c1)C(C)(C)O |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2=O)c(=O)n(C)c1
CN(C)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
CCN(C)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)N2CCC2)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
COCCN(C)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
CN(CCO)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
CNCCN(C)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccc(C(O)CO)c(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccc(CCl)c(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CC3CC(C2)O3)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CC3CC(C2)O3)c(=O)n(C)c1
Cc1ccc(cc1-c1cc(N2CCOCC2)c(=O)n(C)c1)C(=O)Nc1ccc(CNC(=O)OC(C)(C)C)c(c1)C(F)(F)F |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;HN;;;;;;;;;;;;;$|
Cc1ccc(NC(=O)c2cc(CN)cc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2ccccc2)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
CCC(F)(F)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)n(C)c(=O)c1
CCc1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2ccnc(c2)C2CC2)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2ccnc(c2)C2COC2)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2ccnc(c2)C2(CC2)C#N)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
CCn1cc(cc(c1=O)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)n(C)c(=O)c1
CC(C)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2cccc(c2)S(C)(=O)=O)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2cnnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
CCN1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2cc(F)cc(c2)N2CCOCC2)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2cccc(c2)C2COC2)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2cccc(c2)-c2nnco2)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)S(C)(=O)=O)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2cnnc(c2)C2CC2)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
CN(C)Cc1cc(cc(c1)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
CCn1cc(cc(c1=O)C(F)(F)F)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ncc(NC(=O)c2ccccc2)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ncc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
CC(C)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ncc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ncc(NC(=O)c2cccc(c2)S(C)(=O)=O)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ncc(NC(=O)c2ccnc(c2)C2CC2)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ncc(NC(=O)c2cccc(c2)C(C)(C)S(C)(=O)=O)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cn1c(cc(cc1=O)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)cnc1Cl)N1CCOCC1
Cc1ccc(cc1-c1cc(N2CCOCC2)n(C)c(=O)c1)C(=O)Nc1cccc(c1)C(F)F |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;$|
Cc1ccc(cc1-c1cc(N2CCOCC2)n(C)c(=O)c1)C(=O)Nc1cccc(c1)C(C)(C)C#N |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;$|
Cc1ccc(cc1-c1cc(N2CCOCC2)n(C)c(=O)c1)C(=O)Nc1cccc(c1)C(C)(C)O |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
Cc1ccc(cc1-c1cc(N2CCOCC2)n(C)c(=O)c1)C(=O)Nc1cccc(c1)C(F)(F)F |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
Cc1ccc(cc1-c1cc(N2CCOCC2)n(C)c(=O)c1)C(=O)Nc1ccccc1 |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;$|
CCn1c(cc(cc1=O)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1C)N1CCOCC1
CCn1c(cc(cc1=O)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)CC)ccc1C)N1CCOCC1
CCn1c(cc(cc1=O)-c1cc(NC(=O)c2ccnc(c2)C(C)C)ccc1C)N1CCOCC1
C[C@@H]1COCCN1c1cc(cc(=O)n1C)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1C |r|
C[C@@H]1COCCN1c1cc(cc(=O)n1C)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)cnc1C |r|
C[C@H]1COCCN1c1cc(cc(=O)n1C)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1C |r|
C[C@H]1COCCN1c1cc(cc(=O)n1C)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)cnc1C |r|
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2C3CCC2COC3)n(C)c(=O)c1
Cn1c(cc(cc1=O)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)cnc1Cl)N1C2CCC1COC2
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCO[C@@H](CO)C2)n(C)c(=O)c1 |r|
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCO[C@H](CO)C2)n(C)c(=O)c1 |r|
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cncc(n1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cncc(n1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cncc(n1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cncc(n1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cncc(n1)N1CCOCC1
CCC(F)(F)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1cncc(n1)N1CCOCC1
CCOc1ncc(nc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
CCOc1ncc(nc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C
CCOc1ncc(nc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cnc1C
CCOc1ncc(nc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)cnc1C
CCOc1ncc(nc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)cnc1C
CCOc1ncc(nc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)cnc1C
CCOc1ncc(nc1N1CCOCC1)-c1cc(NC(=O)c2cc(ccn2)C(F)(F)F)cnc1C
CCOc1ncc(nc1N1CCOCC1)-c1cc(NC(=O)c2cc(CN(C)C)cc(c2)C(F)(F)F)cnc1C
COc1ncc(nc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)S(C)(=O)=O)ccc1C
COc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)ccc1C
COc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1C
CCC(F)(F)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(OC)nn1
COc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C2CC2)ccc1C
COc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2cnnc(c2)C(F)(F)F)ccc1C
COc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)ccc1C
COc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)S(C)(=O)=O)ccc1C
COc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)O)ccc1C
COc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2cnnc(c2)C(C)(C)C#N)ccc1C
COc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(N)ccc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)CC)ccc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)F)ccc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)F)ccc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C2CC2)ccc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)ccc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)ccc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2cnnc(c2)C(C)(C)C#N)ccc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C2(CC2)C#N)ccc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)O)ccc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2cnnc(c2)C(F)(F)F)ccc1C
CCOc1nnc(cc1N1CCOC[C@@H]1C)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C |r|
CCOc1nnc(cc1N1CCOC[C@@H]1C)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C |r|
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccc(CNC)c(c2)C(F)(F)F)ccc1C
CCNCc1ccc(cc1C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(OCC)nn1 |$;;HN;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;$|
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccc(CN(C)C)c(c2)C(F)(F)F)ccc1C
Cc1ccc(N)cc1-c1cc(N2CCOCC2)c(OC2CCOCC2)nn1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cc(N2CCOCC2)c(OC2CCOCC2)nn1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c(OC2CCOCC2)nn1
Cc1ccc(NC(=O)c2cc(ccn2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(OC2CCOCC2)nn1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cc(N2CCOCC2)c(OC2CCOCC2)nn1
Cc1ccc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1cc(N2CCOCC2)c(OC2CCOCC2)nn1
Cc1ccc(NC(=O)c2cnnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(OC2CCOCC2)nn1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(OC2CCOCC2)nn1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(OCCO)nn1
Cc1ccc(NC(=O)c2cc(ccn2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(OCCO)nn1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c(OCCO)nn1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cc(N2CCOCC2)c(OCCO)nn1
CCC(F)(F)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(OCCO)nn1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(OCCO)nn1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(OCCO)nn1
CC(C)Oc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1C
CC(C)Oc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)F)ccc1C
CC(C)Oc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2cc(ccn2)C(F)(F)F)ccc1C
CC(C)Oc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)ccc1C
CC(C)Oc1nnc(nc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C
COCCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1C
COCCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)F)ccc1C
COCCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2cc(ccn2)C(F)(F)F)ccc1C
COCCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)ccc1C
COCCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(nn1)S(C)(=O)=O
COc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)cnc1C
COc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)F)cnc1C
COc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)cnc1C
COc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C2CC2)cnc1C
CCC(F)(F)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c(OC)nn1
COc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)cnc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)cnc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2cc(ccn2)C(F)(F)F)cnc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C2CC2)cnc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cnc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2cnnc(c2)C(F)(F)F)cnc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cnc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)cnc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)CC)cnc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)S(C)(=O)=O)cnc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)F)cnc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)cnc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)C)cnc1C
CCOc1nnc(cc1N1CCOC[C@H]1C)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C |r|
CCOc1nnc(cc1N1CCOC[C@H]1C)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cnc1C |r|
CCOc1nnc(cc1N1CCOC[C@H]1C)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C |r|
CCOc1nnc(cc1N1CCOC(C1)c1ncc[nH]1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C |$;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;$|
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccc(CNC)c(c2)C(F)(F)F)cnc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccc(CO)c(c2)C(F)(F)F)cnc1C
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c(OC2CCOCC2)nn1
Cc1ncc(NC(=O)c2cc(ccn2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(OC2CCOCC2)nn1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cc(N2CCOCC2)c(OC2CCOCC2)nn1
Cc1ncc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(OC2CCOCC2)nn1
Cc1ncc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1cc(N2CCOCC2)c(OC2CCOCC2)nn1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(OC2CCOCC2)nn1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cc(N2CCOCC2)c(OC2CCOCC2)nn1
Cc1ncc(NC(=O)c2cnnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(OC2CCOCC2)nn1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(OC2CCOCC2)nn1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)S(C)(=O)=O)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2cccc(c2)-c2nnco2)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
CCn1cc(cc(c1=O)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)n1
CCc1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)n1
CCC(F)(F)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2cnnc(c2)C2CC2)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2cnnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2ccnc(c2)C2COC2)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
CCN1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2cccc(CC#N)c2)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2ccnc(c2)C2CC2)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2ccnc(c2)C2(CC2)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
CN(C)Cc1cc(cc(c1)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)n1
C[C@H]1COCCN1c1cc(nn(C)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)ccc1C |r|
C[C@H]1COCCN1c1cc(nn(C)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C |r|
C[C@H]1COCCN1c1cc(nn(C)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1C |r|
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cc(N2CCOC(C)(C)C2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOC(C)(C)C2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCOC(C)(C)C2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cc(N2C3CCC2COC3)c(=O)n(C)n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2C3CCC2COC3)c(=O)n(C)n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2C3CCC2COC3)c(=O)n(C)n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2(C)C)c(=O)n(C)n1
C[C@@H]1COCCN1c1cc(nn(C)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C |r|
C[C@@H]1COCCN1c1cc(nn(C)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)ccc1C |r|
C[C@@H]1COCCN1c1cc(nn(C)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1C |r|
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(C2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cc(C2CCOCC2)c(=O)n(C)n1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
CCC(F)(F)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ncc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ncc(NC(=O)c2ccnc(c2)C2CC2)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ncc(NC(=O)c2ccnc(c2)C2(CC2)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1ccc(C#N)c(c1)N1CCOCC1
CN(C)Cc1cc(cc(c1)C(F)(F)F)C(=O)Nc1cnc(C)c(c1)-c1ccc(C#N)c(c1)N1CCOCC1
CC(C)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1ccc(C#N)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1ccc(c(c1)N1CCOCC1)S(C)(=O)=O
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(cc(=O)n1C)N1C2CCC1COC2
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)ccc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccccc2)ccc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C)ccc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2cccc(c2)C(F)F)ccc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2cccc(c2)-c2nnco2)ccc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)C)ccc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2cccc(c2)C(C)(F)F)ccc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)S(C)(=O)=O)ccc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2cc(c(=O)n(CC)c2)C(F)(F)F)ccc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2cccc(c2)S(C)(=O)=O)ccc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)O)ccc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)CC)ccc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C2COC2)ccc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C2(CC2)C#N)ccc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2cnnc(c2)C(C)(C)C#N)ccc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C)N1CCOC[C@H]1C |r|
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)O)ccc1C)N1CCOC[C@H]1C |r|
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)O)ccc1C)N1CCOC[C@@H]1C |r|
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C)N1CCOC[C@@H]1C |r|
CCNc1nc(cc(n1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cnc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)cnc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2cc(c(=O)n(CC)c2)C(F)(F)F)cnc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(F)F)cnc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2cccc(c2)C(F)F)cnc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)O)cnc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C)cnc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)cnc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2cccc(c2)C(C)(C)C#N)cnc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2cnnc(c2)C2CC2)cnc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C2(CC2)C#N)cnc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C2COC2)cnc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2cnnc(c2)C(C)(C)C#N)cnc1C)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(ccc1C)C(=O)Nc1ccccc1)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(ccc1C)C(=O)Nc1cccc(c1)C(C)(C)C#N)N1CCOCC1 |$;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;$|
CCNc1nc(cc(n1)-c1cc(ccc1C)C(=O)Nc1cccc(c1)C(F)F)N1CCOCC1 |$;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;$|
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(NCCO)n1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(NCCO)n1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(NCCO)n1)N1CCOCC1
Cc1ccc(NC(=O)c2cnnc(c2)C(C)(C)C#N)cc1-c1cc(nc(NCCO)n1)N1CCOCC1
C[C@H](O)CNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cnc1C)N1CCOCC1 |r|
C[C@H](O)CNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C)N1CCOCC1 |r|
C[C@H](O)CNc1nc(cc(n1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C)N1CCOCC1 |r|
C[C@@H](O)CNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C)N1CCOCC1 |r|
C[C@@H](O)CNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cnc1C)N1CCOCC1 |r|
C[C@@H](O)CNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)cnc1C)N1CCOCC1 |r|
C[C@@H](CO)Nc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cnc1C)N1CCOCC1 |r|
C[C@@H](CO)Nc1nc(cc(n1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C)N1CCOCC1 |r|
C[C@@H](CO)Nc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C)N1CCOCC1 |r|
C[C@H](CO)Nc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cnc1C)N1CCOCC1 |r|
C[C@H](CO)Nc1nc(cc(n1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C)N1CCOCC1 |r|
C[C@H](CO)Nc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C)N1CCOCC1 |r|
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(NC(C)(C)CO)n1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(NC(C)(C)CO)n1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(NC(C)(C)CO)n1)N1CCOCC1
OCC1(CCOCC1)Nc1nc(Cl)cc(n1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(NC2(CO)CCOCC2)n1)N1CCOCC1
CN(C)c1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C)N1CCOCC1
CN(C)c1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1C)N1CCOCC1
CC(C)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(nc(n1)N(C)C)N1CCOCC1
CN(C)c1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)ccc1C)N1CCOCC1
CN(C)c1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)S(C)(=O)=O)ccc1C)N1CCOCC1
CN(C)c1nc(cc(n1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C)N1CCOCC1
CCOc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1C)N1CCOCC1
CCOc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)ccc1C)N1CCOCC1
CCOc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)C)ccc1C)N1CCOCC1
CCOc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CC(O)C1)N1CCOCC1
Cc1ccc(cc1-c1cc(nc(n1)N1CC(O)C1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F |$;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(n1)N1CC(O)C1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CC(O)C1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(n1)N1CC(O)C1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(nc(n1)N1CC(O)C1)N1CCOCC1
CC(C)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(nc(n1)N1CC(O)C1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(nc(n1)N1CC(O)C1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CC(O)C1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCNCC1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(OC2CNC2)n1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(OC2CNC2)n1)N1CCOCC1
CC(C)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(nc(OC2CNC2)n1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(nc(OC2CNC2)n1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(nc(OC2CNC2)n1)N1CCOCC1
C[C@H]1COC(=O)N1c1nc(cc(n1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C)N1CCOCC1 |r|
C[C@H]1COC(=O)N1c1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C)N1CCOCC1 |r|
C[C@H]1COC(=O)N1c1nc(cc(n1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C)N1CCOCC1 |r|
C[C@H]1COC(=O)N1c1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cnc1C)N1CCOCC1 |r|
C[C@H]1COC(=O)N1c1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(F)F)ccc1C)N1CCOCC1 |r|
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(NC2CNC2)n1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(NC2CNC2)n1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)C(C)(C)O)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cc(N2CCOCC2)n2nccc2n1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)n2nccc2n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)n2nccc2n1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)n2nccc2n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cc(N2CCOCC2)n2nccc2n1
Cc1ccc(NC(=O)c2cnnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)n2nccc2n1
Cc1ccc(NC(=O)c2ccnc(c2)C2(CC2)C#N)cc1-c1cc(N2CCOCC2)n2nccc2n1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cc(N2CCOCC2)n2nccc2n1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)n2nccc2n1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)n2nccc2n1
CCC(F)(F)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)n2nccc2n1
Cc1ncc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)n2nccc2n1
Cc1ncc(NC(=O)c2ccnc(c2)C2(CC2)C#N)cc1-c1cc(N2CCOCC2)n2nccc2n1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(N2CCOCC2)n2nccc2n1
Cc1ncc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(N2CCOCC2)n2nccc2n1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(N2CCOCC2)n2nccc2n1
Cc1ccc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1cc(N2CCOCC2)n2nccc2n1
Cc1ncc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1cc(N2CCOCC2)n2nccc2n1
Cc1ncc(NC(=O)c2cc(ccn2)C(F)(F)F)cc1-c1cc(N2CCOCC2)n2nccc2n1
C[C@@H]1COCCN1c1nc(cc2[nH]cnc12)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C |r|
Cc1ncc(NC(=O)c2cccc(c2)S(C)(=O)=O)cc1-c1cc(N2CCOCC2)c2nc[nH]c2c1
CCn1cc(C(=O)Nc2cnc(C)c(c2)-c2cc3[nH]cnc3c(n2)N2CCOCC2)c(C)n1
Cc1nn(C)cc1C(=O)Nc1cnc(C)c(c1)-c1cc2[nH]cnc2c(n1)N1CCOCC1
CC(C)n1cc(C(=O)Nc2cnc(C)c(c2)-c2cc3[nH]cnc3c(n2)N2CCOCC2)c(C)n1
Cc1cc(C(=O)Nc2cnc(C)c(c2)-c2cc3[nH]cnc3c(n2)N2CCOCC2)n(C)n1
Cc1ncc(NC(=O)c2cc(nn2C)C2CC2)cc1-c1cc2[nH]cnc2c(n1)N1CCOCC1
Cc1ncc(NC(=O)c2cc(on2)C2CC2)cc1-c1cc2[nH]cnc2c(n1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1cc2[nH]cnc2c(n1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)-c2nnco2)cc1-c1cc2[nH]cnc2c(n1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cc2[nH]cnc2c(n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cn2ccnc2c(n1)N1CCOCC1
C[C@@H]1COCCN1c1nc(cn2ccnc12)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C |r|
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(cc2[nH]c(=O)oc12)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc2nccn2c(n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1nc(N2CCOCC2)c2sccc2n1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1nc(N2CCOCC2)c2[nH]ccc2n1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2n1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOC(C2)c2ncc[nH]2)c2nccn2n1 |$;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;$|
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1nc(N2CCOCC2)c2cccnc2n1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1nc2CN(CCc2c(n1)N1CCOCC1)C(=O)OC(C)(C)C
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1nc2CCNCc2c(n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1nc2CNCc2c(n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1nc(N2CCOCC2)c2n(C)ncc2n1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1nc(N2CCOCC2)c2occc2n1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1nc(N2CCOCC2)c2ncsc2n1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1nc(N2CCOCC2)c2cnn(C)c2n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cc(N2CCOCC2)c2nccn2n1
CC(C)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c2nccn2n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c2nccn2n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2n1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c2nccn2n1
Cc1ccc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(N2CCOCC2)c2nccn2n1
Cc1ccc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ccc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ccc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ccc(NC(=O)c2ccc(CBr)c(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ccc(NC(=O)c2cccc(c2)C(F)F)cc1-c1nc2CCS(=O)(=O)c2c(n1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1nc2CCS(=O)(=O)c2c(n1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1nc2CCS(=O)(=O)c2c(n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1nc2CCS(=O)(=O)c2c(n1)N1CCOCC1
C[C@@H]1COCCN1c1nc(cc2[nH]cnc12)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C |r|
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cn2ccnc2c(n1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1nc(N2CCOCC2)c2n(C)ncc2n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1nc(N2CCOCC2)c2sccc2n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1nc(N2CCOCC2)c2[nH]ccc2n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1nc2CCN(Cc2c(n1)N1CCOCC1)C(=O)OC(C)(C)C
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1nc2CNCCc2c(n1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1nc2CNCc2c(n1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2n1
Cc1ncc(NC(=O)c2cc(ccn2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2n1
CC(C)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c2nccn2n1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cc(N2CCOCC2)c2nccn2n1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2n1
Cc1ncc(NC(=O)c2ccc(C(O)CO)c(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2n1
CNC(=O)C1CN(CCO1)c1cc(nn2ccnc12)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C
Cc1ncc(NC(=O)c2ccc(CBr)c(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2n1
Cc1ncc(NC(=O)c2cc(ccn2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ncc(NC(=O)c2ccc(C#N)c(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ncc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c2nccn2c1
CC(C)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c2nccn2c1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ncc(NC(=O)c2ccc(CBr)c(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1nc2CS(=O)(=O)Cc2c(n1)N1CCOCC1
Cc1c(cc(NC(=O)c2cccc(c2)C(F)(F)F)c[n+]1[O-])-c1nc2CS(=O)(=O)Cc2c(n1)N1CCOCC1
Cc1ccc(cc1-c1cc(N2CCOCC2)c2nccn2n1)C(=O)Nc1cccc(c1)C(F)(F)F |$;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
Cc1ccc(cc1-c1nc2CNCc2c(n1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F |$;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
Cc1ccc(NC(=O)c2cnnc(c2)C2(CC2)C#N)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2cc(ccn2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2cncc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2cnnc(c2)C2(CC2)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cc(ccn2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cncc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cc(ccn2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cc(ccn2)C(C)(C)O)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cc(ccn2)C(C)(C)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cc(cc(c2)C(F)(F)F)C(C)(C)NC(=O)OC(C)(C)C)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cncc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2cc(ccn2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
CC(C)Oc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)cnc1C
CC(C)Oc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)cnc1C
CC(C)Oc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)F)cnc1C
CCC(F)(F)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c(OCC(F)F)nn1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c(OCC(F)F)nn1
Cc1ncc(NC(=O)c2cc(ccn2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(OCC(F)F)nn1
Cc1ncc(NC(=O)c2cncc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(OCC(F)F)nn1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(OCC(F)F)nn1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(nn1)S(C)(=O)=O
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c(nn1)S(C)(=O)=O
Cc1ncc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(nn1)S(C)(=O)=O
Cc1ncc(NC(=O)c2cc(ccn2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(nn1)S(C)(=O)=O
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(nn1)S(C)(=O)=O
CCC(F)(F)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c(nn1)S(C)(=O)=O
CCC(F)(F)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(nn1)S(C)(=O)=O
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cc(N2CCOCC2)c(nn1)S(C)(=O)=O
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cc(N2CCOCC2)c(nn1)S(C)(=O)=O
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c(nn1)S(C)(=O)=O
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(nn1)S(C)(=O)=O
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(nn1)S(C)(=O)=O
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cc(N2CCOCC2)c(nn1)S(C)(=O)=O
Cc1ccc(NC(=O)c2cc(ccn2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(nn1)S(C)(=O)=O
COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)nnc1C
Cc1ncc(NC(=O)c2cncc(c2)C(F)(F)F)cc1-c1cnc(OCC(F)F)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cnnc(c2)C2(CC2)C#N)cc1-c1cnc(OCC(F)F)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)S(C)(=O)=O)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C2(CC2)C#N)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C2CC2)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cc(ccn2)C(F)(F)F)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cc(ccn2)C(C)(C)C#N)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cnnc(c2)C2(CC2)C#N)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)ccc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)O)ccc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cc(ccn2)C(C)(C)C#N)ccc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cc(ccn2)C(C)(C)O)ccc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)S(C)(=O)=O)ccc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cncc(c2)C(F)(F)F)ccc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)cnc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)cnc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cnc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)O)cnc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cc(ccn2)C(C)(F)F)cnc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cc(ccn2)C(C)(C)F)cnc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cc(ccn2)C(C)(C)C#N)cnc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cc(ccn2)C(C)(C)O)cnc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cncc(c2)C(F)(F)F)cnc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(ccc1C)C(=O)Nc1cc(ncc1F)C(F)(F)F |$;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;$|
Cc1ncc(NC(=O)c2cnnc(c2)C(C)(C)C#N)cc1-c1cnc(OCC(F)F)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cnc(OC2CC3(COC3)C2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cnc(OC2CC3(COC3)C2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cnc(OC2CC3(COC3)C2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C2CC2)cc1-c1cnc(OC2CC3(COC3)C2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cnc(OC2CC3(COC3)C2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cc(ccn2)C(C)(C)F)cc1-c1cnc(OC2CC3(COC3)C2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cc(ccn2)C(C)(C)O)cc1-c1cnc(OC2CC3(COC3)C2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cc(ccn2)C(C)(C)C#N)cc1-c1cnc(OC2CC3(COC3)C2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cc(ccn2)C(C)(C)F)cc1-c1cnc(OCCO)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cc(ccn2)C(C)(C)O)cc1-c1cnc(OCCO)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cc(ccn2)C(C)(C)C#N)cc1-c1cnc(OCCO)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cc(ccn2)C(C)(F)F)cc1-c1cnc(OCCO)c(c1)N1CCOCC1
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)S(C)(=N)=O)ccc1C
Cc1ncc(NC(=O)c2cccc(c2)C(O)C(F)(F)F)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cnc(OC(F)F)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cnc(OC(F)F)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cnc(OC(F)F)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cc(ccn2)C(C)(C)C#N)cc1-c1cnc(OC(F)F)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cnc(OC(F)F)c(c1)N1CCOCC1
CCC(F)(F)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1cnc(OC(F)F)c(c1)N1CCOCC1
C[C@@H](O)COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C |r|
C[C@@H](CO)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C |r|
CN(CCO)c1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C
CNC(=O)c1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1C
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1c[nH]c(=O)c(c1)N1CCOCC1
C[C@H](O)COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)S(C)(=O)=O)ccc1C |r|
C[C@H](O)COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)cnc1C |r|
C[C@@H](O)CNc1cc(cc(n1)N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)ccc1C |r|
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(OCC2COCCO2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(CC2(O)CCOCC2)c(c1)N1CCOCC1
[#6]-c1ncc(-[#7]-[#6](=O)-c2cccc(c2)C(F)(F)F)cc1-c1cnc(\[#6]=[#6]-2\[#6]-[#6]-[#8]-[#6]-[#6]-2)c(c1)-[#7]-1-[#6]-[#6]-[#8]-[#6]-[#6]-1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cnc(OCCO)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cnc(OCCO)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C2CC2)cc1-c1cnc(OCCO)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cnc(OCCO)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cncc(c2)C(F)(F)F)cc1-c1cnc(OCCO)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cnc(OCCO)c(c1)N1CCOCC1
COC(=O)NC[C@@H](C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C |r|
Cc1ncc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cc(NCCO)nc(N2CCOCC2)c1F
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(nc(NCCO)c1F)N1CCOCC1
Cc1ccc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cc(nc(NCCO)c1F)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(NCCO)nc(N2CCOCC2)c1F
Cc1ccc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(NCCO)nc(N2CCOCC2)c1F
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cc(NCCO)nc(N2CCOCC2)c1F
Cc1ccc(NC(=O)c2ccnc(c2)C2(CC2)C#N)cc1-c1cc(NCCO)nc(N2CCOCC2)c1F
Cc1ccc(NC(=O)c2cnnc(c2)C(C)(C)C#N)cc1-c1cc(NCCO)nc(N2CCOCC2)c1F
Cc1ccc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cc(NCCO)nc(N2CCOCC2)c1F
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1c(F)c(NCCO)nc(N2CCOCC2)c1F |(-2,5,;-.67,4.23,;.67,5,;2,4.23,;2,2.69,;3.33,1.93,;4.67,2.69,;4.67,4.23,;6,1.93,;7.34,2.69,;8.67,1.93,;8.67,.38,;7.34,-.38,;6,.38,;7.34,-1.93,;8.67,-2.69,;6,-2.69,;8.67,-1.15,;.67,1.93,;-.67,2.69,;-2,1.93,;-2,.38,;-.67,-.38,;-3.33,-.38,;-3.33,-1.93,;-2,-2.69,;-2,-4.23,;-.67,-5,;-4.67,.38,;-4.67,1.93,;-6,2.69,;-7.34,1.93,;-8.67,2.69,;-8.67,4.23,;-7.34,5,;-6,4.23,;-3.33,2.69,;-3.33,4.23,)|
Cc1ccc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1c(F)c(NCCO)nc(N2CCOCC2)c1F |(-2,5,;-.67,4.23,;.67,5,;2,4.23,;2,2.69,;3.33,1.93,;4.67,2.69,;4.67,4.23,;6,1.93,;7.34,2.69,;8.67,1.93,;8.67,.38,;7.34,-.38,;6,.38,;7.34,-1.93,;8.67,-2.69,;6,-2.69,;8.67,-1.15,;.67,1.93,;-.67,2.69,;-2,1.93,;-2,.38,;-.67,-.38,;-3.33,-.38,;-3.33,-1.93,;-2,-2.69,;-2,-4.23,;-.67,-5,;-4.67,.38,;-4.67,1.93,;-6,2.69,;-7.34,1.93,;-8.67,2.69,;-8.67,4.23,;-7.34,5,;-6,4.23,;-3.33,2.69,;-3.33,4.23,)|
Cc1ccc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(nc(NCCO)c1F)N1CCOCC1
COc1nnc(cc1N1CCOCC1)-c1cc(ccc1C)C(=O)Nc1ccnc(c1)C(F)(F)F |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
COc1nnc(cc1N1CCOCC1)-c1cc(ccc1C)C(=O)Nc1ccnc(c1)C(C)(F)F |$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
CCOc1nnc(cc1N1CCOCC1)-c1cc(ccc1C)C(=O)Nc1ccnc(c1)C(C)(F)F |$;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
COC[C@@H](C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C |r|
CO[C@@H](C)COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C |r|
C[C@@H](O)CNc1cc(nc(n1)N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)ccc1C |r|
C[C@@H](O)CNc1cc(nc(n1)N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)ccc1C |r|
C[C@@H](O)CNc1cc(nc(n1)N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)ccc1C |r|
C[C@@H](O)CNc1cc(nc(n1)N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C |r|
CCOc1ccc(nc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)cnc1C
CCOc1ccc(nc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)cnc1C
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(O[C@H]2CCOC[C@H]2F)c(c1)N1CCOCC1 |r|
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(OC2CCOCC2F)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(OCCOCCO)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(OC2CCS(=O)(=O)CC2)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
CCn1cc(cc(c1=O)C(F)(F)F)C(=O)Nc1cnc(C)c(c1)-c1cc(NCCO)nc(c1)N1CCOCC1
CCN1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1cnc(C)c(c1)-c1cc(NCCO)nc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cnnc(c2)C2CC2)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cnnc(c2)C(C)(C)C#N)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C2(CC2)C#N)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cnnc(c2)C2CC2)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(NC2CCOC2)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(NCC2CCOC2)nc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C2CC2)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
CCC(F)(F)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1cc(NCCO)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
CCn1cc(cc(c1=O)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(NCC(C)(C)O)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(NCC(O)C(F)(F)F)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1C[C@H](O)CC1=O |r|
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CC[C@@H](O)C1=O |r|
CC(O)C(=O)Nc1cc(cc(n1)N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
Cc1ccc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ccc(NC(=O)c2ccnc(c2)C2CC2)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
CC(C)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ccc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ccc(NC(=O)c2ccnc(c2)C2(CC2)C#N)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(C)(O)C1
Cc1ccc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(C)(O)C1
Cc1ccc(NC(=O)c2cccc(c2)S(C)(=O)=O)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(C)(O)C1
Cc1ccc(NC(=O)c2cnncc2C(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ccc(NC(=O)c2cnnc(c2)C2CC2)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(C)(O)C1
Cc1ccc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ncc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
CC(C)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ncc(NC(=O)c2cccc(c2)S(C)(=O)=O)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
CN(C)Cc1cc(cc(c1)C(F)(F)F)C(=O)Nc1cnc(C)c(c1)-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
CCn1cc(cc(c1=O)C(F)(F)F)C(=O)Nc1cnc(C)c(c1)-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
CCN1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1cnc(C)c(c1)-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ncc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ncc(NC(=O)c2cccc(c2)C(C)(C)S(C)(=O)=O)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ncc(NC(=O)c2cccc(c2)-c2nnco2)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ncc(NC(=O)c2cc(on2)C2CC2)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ccc(NC(=O)c2cc(on2)C2CC2)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ccc(NC(=O)c2cccc(c2)S(C)(=O)=O)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ccc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)S(C)(=O)=O)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ccc(NC(=O)c2cccc(c2)-c2nnco2)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
Cc1ncc(NC(=O)c2cnnc(c2)C2CC2)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(C)(O)C1
Cc1ncc(NC(=O)c2ccnc(c2)C2CC2)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(C)(O)C1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(C)(O)C1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(C)(O)C1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(C)(O)C1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(C)(O)C1
Cc1ncc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(C)(O)C1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(C)(O)C1
Cc1ncc(NC(=O)c2ccnc(c2)C2(CC2)C#N)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(C)(O)C1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(C)(O)C1
Cc1ccc(NC(=O)c2ccnc(c2)C2(CC2)C#N)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(C)(O)C1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(c1)N1CCOCC1)N1CCOCC1
CCn1cc(cc(c1=O)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(nc(c1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CCOCC1
CC(C)c1cc(ccn1)C(=O)Nc1ccc(C)c(c1)-c1cc(nc(c1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1cc(nc(c1)N1CCOCC1)N1CCOCC1
CC(C)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1cc(nc(c1)N1CCOCC1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(c1)N1CCOCC1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1cc(nc(c1)N1CCOCC1)N1CCOCC1
CCn1cc(cc(c1=O)C(F)(F)F)C(=O)Nc1cnc(C)c(c1)-c1cc(nc(c1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cncc(c2)C(F)(F)F)cc1-c1cc(nc(c1)-c1cnn(C)c1)N1CCOCC1
Cc1n[nH]c(C)c1-c1cc(cc(n1)N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)ccc1C
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CCNCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CCNCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CCC(O)C1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CCC(O)C1
Cc1ccc(NC(=O)[C@@H]2CCN[C@@H](C2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)C1COCCO1 |r|
CCOc1cc(cc(n1)N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)ccc1C
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1ccnc(c1)N1CCOCC1=O
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1ccnc(c1)N1CCOCC1=O
CC(C)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1ccnc(c1)N1CCOCC1
C[C@@H]1COCCN1c1cc(cc(NCCO)n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)cnc1C |r|
C[C@@H]1COCCN1c1cc(cc(NCCO)n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)cnc1C |r|
C[C@@H]1COCCN1c1cc(cc(NCCO)n1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)cnc1C |r|
C[C@@H]1COCCN1c1cc(cc(NCCO)n1)-c1cc(NC(=O)c2ccnc(c2)C(F)F)cnc1C |r|
CCOc1cc(cc(n1)N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)cnc1C
CCOc1cc(cc(n1)N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)cnc1C
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cc(nc(c1)N1CCOCC1)C1COCCO1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)C1COCCO1
CCOc1cc(cc(n1)N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)F)cnc1C
CCOc1cc(cc(n1)N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cnc1C
CCOc1cc(cc(n1)N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)O)cnc1C
CCOc1cc(cc(n1)N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C2CC2)cnc1C
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)O)cc1-c1cc(OC2CCOCC2)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(OC2CCOCC2)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(OC2CCOCC2)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cnnc(c2)C(C)(C)C#N)cc1-c1cc(OC2CCOCC2)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cnnc(c2)C2CC2)cc1-c1cc(OC2CCOCC2)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cc(OC2CCOCC2)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(OCCO)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C2CC2)cc1-c1cc(OCCO)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cc(OCCO)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(OCCO)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(OCCO)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(OCCO)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cnnc(c2)C2CC2)cc1-c1cc(OCCO)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cc(ccn2)C(F)(F)F)cc1-c1cc(OCCO)nc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cc(OCCO)nc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)C1COCCO1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)C1COCCO1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)F)cc1-c1cc(nc(c1)N1CCOCC1)C1COCCO1
CCC(F)(F)c1cc(ccn1)C(=O)Nc1cnc(C)c(c1)-c1cc(nc(c1)N1CCOCC1)C1COCCO1
Cc1ncc(NC(=O)c2ccnc(c2)C2CC2)cc1-c1cc(nc(c1)N1CCOCC1)C1COCCO1
FC(F)c1cccc(c1)C(=O)Nc1c[nH]c(=O)c(c1)-c1ccnc(c1)N1CCOCC1 |$;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;$|
Cc1cc(=O)c(cn1-c1ccnc(c1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F |$;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
CCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
FC(F)(F)CN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CCN1CCN(Cc2ccc(cc2F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CCN1CCN(Cc2cc(cc(c2)C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CCN1CCN(Cc2cc(F)cc(c2)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
FC(F)(F)c1cc(ccc1CN1CCOCC1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1cc(ccc1CN1CCCCC1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CN(C)[C@H]1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)C1 |r|
CN(C)[C@@H]1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)C1 |r|
CN1CCN(Cc2ccc(cc2)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
FC(F)(F)c1cc(ccc1CN1CCN2CCC[C@@H]2C1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
C[C@H]1CN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)C[C@@H](C)O1 |r|
FC(F)(F)c1nnc2CN(Cc3ccc(cc3C(F)(F)F)C(=O)N[C@@H]3[C@H]4Oc5ccc(Oc6ccnc7NC(=O)CCc67)cc5[C@@H]34)CCn12 |r|
O[C@H]1CCCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)C1 |r|
O[C@@H]1CCCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)C1 |r|
OCCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CCN1CCN(Cc2ccc(cc2Cl)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CCN1CCN(Cc2ccc(cc2Br)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CN(C)C1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CN1CCN(Cc2ccc(cc2F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CN1CCN(Cc2ccc(cc2Cl)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CN1CCN(Cc2ccc(cc2Br)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CN(C)Cc1ccc(cc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CC(C)(N)c1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
NC1(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1cc(ccc1CN1CCNCC1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
C[C@H]1CN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CCN1 |r|
CN(C)[C@@H]1CCCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)C1 |r|
CN(C)[C@@H]1CN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CCN1 |r|
CCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@H]2[C@@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@H]23)CC1 |r|
FC(F)(F)c1cccc(c1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
Fc1ccc(cc1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
Cc1cccc(F)c1C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
Fc1ccccc1C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
Fc1cccc(c1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1ccc(cc1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
Fc1ccc(cc1F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
Fc1cc(ccc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CC(C)(C#N)c1cccc(c1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1ccccc1C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1ccnc(c1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
O=C(N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12)c1cccc(c1)C1(CC1)C#N |r|
CN(C)[C@H]1CCCN(C1)c1ccc(cc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CN(C)[C@@H]1CCCN(C1)c1ccc(cc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CN1CCN(CC1)c1ccc(cc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CCN1CCN(CC1)c1ccc(cc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CN1CCC(CC1)Oc1ccc(cc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CN1CCN(CCOc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
FC(F)(F)c1cccc(\C=C\C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)c1 |r|
O=C(N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12)c1ccc(o1)-c1ccccc1 |r|
CCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)NC2C3Oc4c(cc(Oc5ccnc6NC(=O)CCc56)cc4C)C23)CC1
CN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)NC2C3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4C23)CC1
CCN1CCN(Cc2ccc(cc2C)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CN1CCN(Cc2ccc(cc2C)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
Cc1cc(ccc1CO)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1cccc(CC(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)c1 |r|
FC(F)(F)c1cc(ccn1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1cncc(c1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1cccc(n1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CC1CN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC(C)N1C(=O)OC(C)(C)C |r|
CN(C)Cc1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CCCCCC(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CCCCCCC(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CCCCCCCC(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CCCCCCCCCC(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CN(C)C1CCN(CC1)c1ccc(cc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
COc1cc(ccc1CN1CCN(C)CC1)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CCN1CCN(Cc2ccc(cc2OC)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CCN1CCC(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
[#6]-[#6]-[#7]-1-[#6]-[#6]\[#6](-[#6]-[#6]-1)=[#6]/c1ccc(cc1C(F)(F)F)-[#6](=O)-[#7]-[#6@@H]-1-[#6@H]-2-[#8]-c3ccc(-[#8]-c4ccnc5-[#7]-[#6](=O)-[#6]-[#6]-c45)cc3-[#6@@H]-1-2 |r|
OCc1ccc(cc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CN1C(C)(C)CC(CC1(C)C)Oc1ccc(cc1C(F)(F)F)C(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CCN1CCN(Cc2ccc(cc2OC(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)CCc56)cc4[C@@H]23)CC1 |r|
CCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)OCc56)cc4[C@@H]23)CC1 |r|
CN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)OCc56)cc4[C@@H]23)CC1 |r|
CCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc(c5)C(=O)NC)cc4[C@@H]23)CC1 |r|
CNC(=O)c1cc(Oc2ccc3O[C@@H]4[C@@H](NC(=O)c5ccc(CN6CCN(C)CC6)c(c5)C(F)(F)F)[C@@H]4c3c2)ccn1 |r|
CCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc(N)c5)cc4[C@@H]23)CC1 |r|
CCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)NCc56)cc4[C@@H]23)CC1 |r|
CN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)N[C@@H]2[C@H]3Oc4ccc(Oc5ccnc6NC(=O)NCc56)cc4[C@@H]23)CC1 |r|
N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)NCc45)cc3[C@@H]12 |r|
O=c1[nH]nc2CCCc3[nH]c4cccc1c4c23
CC1(C)Cc2[nH]c3cc(F)cc4c3c2c(C1)n[nH]c4=O
CC1(C)Cc2n(CCN3CCCCC3)c3cccc4c3c2c(C1)n[nH]c4=O
CCN(CC)CCn1c2CC(C)(C)Cc3n[nH]c(=O)c4cccc1c4c23
CC1(C)Cc2n(CC3CO3)c3cccc4c3c2c(C1)n[nH]c4=O
CC(C)N1Cc2[nH]c3cccc4c3c2c(C1)n[nH]c4=O
O=C(C1CC1)N1Cc2[nH]c3cccc4c3c2c(C1)n[nH]c4=O
CC(C)(C)C(=O)N1Cc2[nH]c3cccc4c3c2c(C1)n[nH]c4=O
CC(C)(N)C(=O)N1Cc2[nH]c3cccc4c3c2c(C1)n[nH]c4=O
C[C@]12CCCN1Cc1n[nH]c(=O)c3cc(F)cc4[nH]c2c1c34 |r|
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(Cl)cc23)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(Cl)cc2)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(OC)nc2)c1F
Fc1ccc(NS(=O)(=O)N2CCCC2)c(F)c1C(=O)c1c[nH]c2ncc(F)c(I)c12
Fc1cnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)N4CCCC4)c3F)c2c1NCC1CC1
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)C#N)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(Cl)cc23)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(Cl)cc2)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(OC)nc2)c1F
Fc1ccc(NS(=O)(=O)N2CCCC2)c(F)c1C(=O)c1c[nH]c2ncc(cc12)-c1ccc(Cl)cc1
CN(C)c1ncc(cn1)-c1cnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
Cc1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
Fc1ccc(NS(=O)(=O)N2CCCC2)c(F)c1C(=O)c1c[nH]c2ncc(I)cc12
COc1ncc(cn1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N(C)C4CC4)c3F)c2c1
CNS(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(OC)nc2)c1F
CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C#N)c1F
CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cccnc2)c1F
CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(C)nc2)c1F
CN(C)c1ccc(cn1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N(C)C)c3F)c2c1
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C#N)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cccnc2)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(C)nc2)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(F)cc2)c1F
CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(F)cc2)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccccc2)c1F
CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccccc2)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(Br)cc23)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)C#N)c1F
CCCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(OC)nc2)c1F
COc1ncc(cn1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCC(C4)OCc4ccccc4)c3F)c2c1
CC1C=C(C=N1)c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)CC4CC4)c3F)c2c1 |c:2,4|
Fc1c(NS(=O)(=O)N2CCCC2)cccc1C(=O)c1c[nH]c2ncc(cc12)-c1cccnc1
COc1ncc(c(OC)n1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
Cc1ccc(cn1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
CN(C)c1ccc(cn1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
CC(C)c1ncc(cn1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
Fc1c(NS(=O)(=O)N2CCCC2)cccc1C(=O)c1c[nH]c2ncc(cc12)-c1cnc(nc1)C1CC1
COc1cc(ccc1C#N)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
Fc1c(NS(=O)(=O)N2CCCC2)cccc1C(=O)c1c[nH]c2ncc(cc12)-c1ccc(cc1)C1(CC1)C#N
CC(C)c1ncc(cn1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N(C)C)c3F)c2c1
CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(nc2)C(F)(F)F)c1F
COc1cc(ccc1C#N)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N(C)C)c3F)c2c1
CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C2(CC2)C#N)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(C)nc2)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C(C)C)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(nc2)C(F)(F)F)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(C#N)c(OC)c2)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C2(CC2)C#N)c1F
Fc1ccc(cc1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
Fc1c(NS(=O)(=O)N2CCCC2)cccc1C(=O)c1c[nH]c2ncc(cc12)-c1ccccc1
CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(NC3CC3)nc2)c1F
COCCS(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(OC)nc2)c1F
COC(=O)CCS(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(OC)nc2)c1F
COc1ncc(cn1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)C4CC4)c3F)c2c1
CCNS(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(OC)nc2)c1F
CCNS(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(I)cc23)c1F
CC(C)CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(I)cc23)c1F
CC(C)NS(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(I)cc23)c1F
COc1ncc(cn1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N(C)CC(C)C)c3F)c2c1
COCCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(OC)nc2)c1F
COc1ncc(cn1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCCC4C)c3F)c2c1
COc1ncc(cn1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N(C)C(C)C)c3F)c2c1
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(nc2)N(C)C)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(NC3CC3)nc2)c1F
CCCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
CCCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C2(CC2)C#N)c1F
COCCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C2(CC2)C#N)c1F
COCCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(NC3CC3)nc2)c1F
CCCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(NC3CC3)nc2)c1F
COc1ncc(cn1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N(C)CC4CC4)c3F)c2c1
CN(CC1CC1)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
COCCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
CCCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(nc2)C2CC2)c1F
COc1ncc(cn1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CC(F)(F)C4)c3F)c2c1
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncnc(N[C@@H](C)C4CC4)c23)c1F |r|
Fc1c(NS(=O)(=O)N2CCCC2)cccc1C(=O)c1c[nH]c2ncc(cc12)-c1ccc(cc1)C#N
Fc1c(NS(=O)(=O)N2CCCC2)cccc1C(=O)c1c[nH]c2ncc(cc12)-c1cnc(nc1)C#N
Cc1ncc(cn1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
Fc1c(NS(=O)(=O)N2CCCC2)cccc1C(=O)c1c[nH]c2ncc(cc12)-c1cncc(c1)C#N
Fc1c(NS(=O)(=O)N2CCCC2)cccc1C(=O)c1c[nH]c2ncc(cc12)-c1ccc(nc1)C#N
Fc1c(NS(=O)(=O)N2CCCC2)cccc1C(=O)c1c[nH]c2ncc(cc12)-c1ccc(nc1)C(F)(F)F
CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C#N)c1F
CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(C)nc2)c1F
CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cncc(c2)C#N)c1F
CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(nc2)C#N)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C#N)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cncc(c2)C#N)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(nc2)C#N)c1F
CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C(C)(C)O)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C(C)(C)O)c1F
CC(C)(O)c1ccc(cc1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
CN(C)c1ncc(cn1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N(C)C)c3F)c2c1
CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)N2CCCC2)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)N2CCCC2)c1F
Fc1c(NS(=O)(=O)N2CCCC2)cccc1C(=O)c1c[nH]c2ncc(cc12)-c1cnc(nc1)N1CCCC1
Fc1c(NS(=O)(=O)N2CCCC2)cccc1C(=O)c1c[nH]c2ncc(cc12)-c1cnc(nc1)N1CCOCC1
CCC(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)N2CCOCC2)c1F
CN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C2(CC2)[N+]#[C-])c1F
CN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C2(CC2)[N+]#[C-])c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
Fc1ccc(NS(=O)(=O)N2CCCC2)c(F)c1C(=O)c1c[nH]c2ncc(cc12)-c1cnc(nc1)C1CC1
CCCNS(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnn(C)c2)c1F
OC(=O)C1(CC1)c1ccc(cc1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
CCOc1cnc(cn1)-c1cnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)N(C)C)c3F)c2c1
CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C(C)(C)C#N)c1F
CC1(C)CCN(C1)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
CC1CCN(C1)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
Fc1ccc(NS(=O)(=O)N2CCCC2)c(F)c1C(=O)c1c[nH]c2ncc(cc12)-c1ccc(cc1)C1(CC1)[N+]#[C-]
CN(C1CC1)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
CCCNS(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
CN(C1CC1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
NC(=O)C1(CC1)c1ccc(cc1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
COC(=O)C1(CC1)c1ccc(cc1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
CN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C(C)(C)C#N)c1F
CCOc1ncc(cn1)-c1cnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)N(C)CC)c3F)c2c1
CCOC(=O)C1CCCN1S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(OC)nc2)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)N2CCOCC2)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cccc(c2)N2CCOCC2)c1F
CN1CCN(CC1)c1ncc(cn1)-c1cnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
Fc1ccc(NS(=O)(=O)N2CCCC2)c(F)c1C(=O)c1c[nH]c2ncc(cc12)-c1cnc(nc1)N1CCNCC1
OC1CCN(CC1)c1ncc(cn1)-c1cnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)N2CCN(C)CC2)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)N2CCN(CC2)C(=O)OC(C)(C)C)c1F
CC(C)(O)c1nc(cs1)-c1cnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
Fc1ccc(NS(=O)(=O)N2CCCC2)c(F)c1C(=O)c1c[nH]c2ncc(cc12)-c1cnc(nc1)N1CCOCC1
CN(C1CCN(C1)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F)C(C)=O
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)N2CCNCC2)c1F
Fc1ccc(NS(=O)(=O)N2CCCC2)c(F)c1C(=O)c1c[nH]c2ncc(cc12)-c1cnc(nc1)N1CCC1
COc1ncc(s1)-c1cnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
C[C@@H]1CCN(C1)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F |r|
CNC1CCN(C1)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
Fc1c(NS(=O)(=O)N2CCCC2)cccc1C(=O)c1c[nH]c2ncc(cc12)C1CC1
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)N2CCC(O)CC2)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cccc(c2)C2(CC2)C#N)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)N2CCC2)c1F
Nc1ncc(cn1)-c1cnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
Fc1c(NS(=O)(=O)N2CCCC2)cccc1C(=O)c1c[nH]c2ncc(cc12)-c1ccncc1
Fc1ccc(NS(=O)(=O)N2CCCC2)c(F)c1C(=O)c1c[nH]c2ncc(cc12)-c1ccnc(n1)N1CCOCC1
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccnc(F)c2)c1F
CN1CCN(CC1)c1cc(ccn1)-c1cnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
Fc1ccc(NS(=O)(=O)N2CCCC2)c(F)c1C(=O)c1c[nH]c2ncc(cc12)-c1ccnc(OC2CCC2)c1
Fc1ccc(NS(=O)(=O)N2CCC(F)(F)C2)c(F)c1C(=O)c1c[nH]c2ncc(cc12)-c1cnc(nc1)C1CC1
F[C@H]1CCN(C1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F |r|
COC(=O)C(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)N2CCCC2)c1F
Fc1ccc(NS(=O)(=O)N2CCCC2)c(F)c1C(=O)c1c[nH]c2ncc(cc12)-c1cc(ncn1)C(F)(F)F
Fc1ccc(NS(=O)(=O)N2CCCC2)c(F)c1C(=O)c1c[nH]c2ncc(cc12)-c1ccnc(c1)C1CC1
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)C2CCC2)c1F
CCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)C2CC2)c1F
Nc1cc(ncn1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C#N)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C(F)(F)F)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cccc(c2)N(C)C)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)N2CCCC2)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)-c2nnc(C)o2)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)-c2nnc(NC)s2)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cncc(c2)C(C)(C)O)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(nc2)C(C)(C)O)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)N(CC)CC)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc3CC(=O)Nc3c2)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(s2)-c2noc(C)n2)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc3nc(N)ncc3c2)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(nc2)C(=O)NC2CC2)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc3nc(ncc3c2)N(C)C)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C2(O)CC2)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cncs2)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2csc(n2)C(C)(C)O)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(OC)nn2)c1F
Fc1ccc(NS(=O)(=O)N2CCCC2)c(F)c1C(=O)c1c[nH]c2ncc(cc12)-c1cc(ncn1)N1CCOCC1
CN1CCN(CC1)c1cc(ncn1)-c1cnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
C[C@H]1CCN(C1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F |r|
Fc1c(NS(=O)(=O)N2CCCC2)cccc1C(=O)c1c[nH]c2ncc(cc12)-c1cc(ncn1)N1CCOCC1
CN1CCN(CC1)c1cc(ncn1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
CN1CCN(CC1)c1cccc(n1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
COc1ccnc(n1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
Cc1ccnc(n1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)N4CCCC4)c3F)c2c1
F[C@@H]1CCN(C1)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F |r|
CNS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
CCNS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
NS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
CCC(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(Cl)cc2)c1F
F[C@@H]1CCN(C1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F |r|
FC1CCN(C1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
CN(CC(F)(F)F)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
CCCNS(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(C)cc23)c1F
CCC(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(OC)nc2)c1F
CCC(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)N2CCCC2)c1F
CCC(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(NC3CC3)nc2)c1F
CCC(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C2(CC2)C#N)c1F
CCC(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
CCC(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C(C)C)c1F
CCC(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(nc2)N(C)C)c1F
CCC(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(C)nc2)c1F
Fc1c(NS(=O)(=O)N2CCCC2)cccc1C(=O)c1c[nH]c2ncc(cc12)-c1cnc(NC2CC2)nc1
CC(C)N(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
CCCNS(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(I)cc23)c1F
CCCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(OC)nc2)c1F
CN(CC1CC1)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(nc2)C2CC2)c1F
CCCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(nc2)C2CC2)c1F
CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(nc2)C2CC2)c1F
CN(CC1CC1)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(C)nc2)c1F
CCCN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(C)nc2)c1F
CN(C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(I)cc23)c1F
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
CCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(on4)C(C)(C)C)ccc3F)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(on4)C(C)(C)C)ccc3Cl)c2cc1OC
CCOc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCOC
CCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCC
CC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3ncnc4cc5OCCOc5cc34)c2)no1
COCCOc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCCCC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCC(CO)CC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCN(C)CC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCN(CCO)CC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCOCC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCN(C)CC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCOCC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCCCC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCC(CO)CC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCN(CC1)S(C)(=O)=O
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCS(=O)(=O)CC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCOCC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCN(C)CC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCC(CO)CC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCN(CCO)CC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCC(O)C1 |w:39.43|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCN(CC1)S(C)(=O)=O
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CC[C@H](O)C1 |r|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CC[C@@H](O)C1 |r|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCOCC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCN(C)CC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCC(CO)CC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCN(CCO)CC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCS(=O)(=O)CC1
COCCOc1ccc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2c1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCS(C)(=O)=O
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)F)c3)c2cc1OCCCS(C)(=O)=O
COCCOc1ccc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2c1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCS(C)(=O)=O
COCCOc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
CC(C)(C)c1cc(NC(=O)Nc2cccc(Sc3ncnc4cc(F)c(F)cc34)c2)no1
COc1ccc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2c1
COc1ccc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2c1
CCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
CCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCOC
CC(C)(C)c1cc(NC(=O)Nc2cccc(Sc3ncnc4cc5OCCOc5cc34)c2)no1
COc1cc(OC2CCOCC2)c2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2c1
CCOc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCCCC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCC(CO)CC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCN(C)CC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCN(CC1)S(C)(=O)=O
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCN(CCO)CC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCS(=O)(=O)CC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCOCC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCCCC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCC(CO)CC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCN(C)CC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCN(CCO)CC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCN(CC1)S(C)(=O)=O
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCOCC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCS(=O)(=O)CC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCOCC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCN(C)CC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCC(CO)CC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCN(CCO)CC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCCCC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCN(CC1)S(C)(=O)=O
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCOCC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCCCC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCN(CC1)S(C)(=O)=O
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCN(C)CC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCC(CCO)CC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCC(CO)CC1
COCCOc1ccc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2c1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCS(C)(=O)=O
COc1cc2nc(Cl)nc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
CC(C)(C)c1cc(NC(=O)Nc2cccc(Sc3ncnc4ccc(OCCCN5CCS(=O)(=O)CC5)cc34)c2)no1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCS(=O)(=O)CC1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3ncnc4ccc(cc34)-c3ccc(CNCCS(C)(=O)=O)o3)c2)no1
COc1cc(OC2CCOCC2)c2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2c1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1O
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1O[C@H]1CCNC1 |r|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1O[C@H]1CCN(C)C1 |r|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1O[C@@H]1CCNC1 |r|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1O[C@@H]1CCN(C)C1 |r|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OC[C@H](O)CN1CCN(C)CC1 |r|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCC1CCNCC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCC1CCN(C)CC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1O[C@H]1CCN(CC(F)F)C1 |r|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1O[C@H]1CCN(CC(F)(F)F)C1 |r|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OC1CCN(CC(F)F)CC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1O
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1O[C@H]1CCN(C1)C(=O)OC(C)(C)C |r|
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC1CCN(C)C1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1O[C@H]1CCN(CC(F)F)C1 |r|
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC[C@@H](O)CN1CCN(C)CC1 |r|
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC[C@H](O)CN1CCN(C)CC1 |r|
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)-c4ccccc4)c3)c2cc1OC
COc1cc(NC(=O)Nc2cccc(Sc3ncnc4cc(OC)c(OC)cc34)c2)cc(c1)C(F)(F)F
COc1cc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)cc(c1)C(F)(F)F
COCCOc1cc(NC(=O)Nc2cccc(Oc3ncnc4cc(OCCOC)c(OC)cc34)c2)cc(c1)C(F)(F)F
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cccc(c4)C(C)(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cccc(c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cccc(c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C4CCOCC4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C4CC4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C#N)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C4(C)CC4)c3)c2cc1OC
COCC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)on1
COCCOc1cc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)cc(c1)C(F)(F)F
COCC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)no1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)CO)c3)c2cc1OC
COc1cc2cccc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C4CCCC4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(CC(F)(F)F)nn4-c4ccccc4)c3)c2cc1OC
COc1ccc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)cc1C(F)(F)F
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccc(OC)c(c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(Cl)cc(c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(ccn4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(ccc4Cl)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4nccc(n4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cccc(c4)C(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(ncn4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)ccc1C(F)(F)F
COCCOc1cc(NC(=O)Nc2cccc(Sc3ncnc4cc(OC)c(OC)cc34)c2)ccc1C(F)(F)F
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(cc(c4)C(F)(F)F)C(=O)N4CCOCC4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccc(c(F)c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(CN5CCOCC5)cc(c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C4(CCC4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C4(CCC4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(CF)CF)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(CF)CF)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(CF)CF)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C4CCCC4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4C)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(n(C)n4)C(F)(F)F)c3)c2cc1OC
CCOC(=O)Cn1nc(cc1NC(=O)Nc1cccc(Oc2ncnc3cc(OC)c(OC)cc23)c1)C(C)(C)C
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(CF)CF)c3)c2cc1OC
CCOC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)n(n1)-c1ccccc1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(n(n4)-c4ccccc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(n(n4)-c4ccccc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(F)cc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccc(cc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4ccc(cc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccc(Cl)cc4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccc(OC(F)(F)F)cc4)c3)c2cc1OC
COc1cccc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)c1
CCOc1cccc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)c1
COc1ccc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)cc1Cl
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cccc(c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccccc4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cccc(c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4ccc(c(F)c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(CN5CCOCC5)cc(c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4ccc(c(OC)c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(CF)CF)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4C)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(n(C)n4)C(F)(F)F)c3)c2cc1OC
CCOC(=O)Cn1nc(cc1NC(=O)Nc1cccc(Sc2ncnc3cc(OC)c(OC)cc23)c1)C(C)(C)C
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(CF)CF)c3)c2cc1OC
CCCOC(C)(C)c1cc(NC(=O)Nc2cccc(Sc3ncnc4cc(OC)c(OC)cc34)c2)n(n1)-c1ccccc1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(F)cc4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc(NC(=O)Nc2cccc(Sc3ncnc4cc(OC)c(OC)cc34)c2)cc(c1)C(F)(F)F
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C4CCCC4)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)-c4ccccc4)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(cc(c4)C(F)(F)F)C(=O)N4CCOCC4)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C4CCCC4)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(n(C)n4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4C)C(C)(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(F)F)c3)c2cc1OC
CCOC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3ncnc4cc(OCCOC)c(OC)cc34)c2)n(n1)-c1ccccc1
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(CF)CF)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C4CC4)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C4CCOCC4)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)COC)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C4CCCC4)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4C)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccc(c(F)c4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccc(c(OC)c4)C(F)(F)F)c3)c2cc1OC
CCOC(=O)Cn1nc(cc1NC(=O)Nc1cccc(Oc2ncnc3cc(OCCOC)c(OC)cc23)c1)C(C)(C)C
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(n(n4)-c4ccccc4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(F)cc4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(CF)CF)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(CF)CF)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4ccc(c(F)c4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4ccc(c(OC)c4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C4CCCC4)c3)c2cc1OC
CCOC(=O)Cn1nc(cc1NC(=O)Nc1cccc(Sc2ncnc3cc(OCCOC)c(OC)cc23)c1)C(C)(C)C
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(CF)CF)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4C)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(n(C)n4)C(F)(F)F)c3)c2cc1OC
CCOC(C)(C)c1cc(NC(=O)Nc2cccc(Sc3ncnc4cc(OCCOC)c(OC)cc34)c2)n(n1)-c1ccccc1
COCCOc1cc2ncnc(Sc3cccc(NC(=O)NC4=CC(=NC4c4ccc(F)cc4)C(F)(F)F)c3)c2cc1OC |c:24,t:22|
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(n(n4)-c4ccccc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)c2cc1OCCCN1CCS(=O)(=O)CC1
COc1ccc(NC(=O)Nc2cccc(Sc3ncnc4cc(OC)c(OCCCN5CCS(=O)(=O)CC5)cc34)c2)cc1C(F)(F)F
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(C)C)c3)c2cc1OCCOC
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)ncnc2cc1OCCN1CCOCC1
COc1ccc(NC(=O)Nc2cccc(Sc3ncnc4cc(OCCN5CCOCC5)c(OC)cc34)c2)cc1C(F)(F)F
COc1ccc(NC(=O)Nc2cccc(Oc3ncnc4cc(OCCN5CCOCC5)c(OC)cc34)c2)cc1C(F)(F)F
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)ncnc2cc1OCCN1CCOCC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cnn(c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(S(=O)c3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)NC4=CC(=CC4)C(C)(C)CO)c3)c2cc1OC |c:21,t:19|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCS(=O)(=O)CC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)ncnc2cc1O
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)c2cc1O
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C(F)(F)F)c3)c2cc1OC
CCOc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C(F)(F)F)c3)ncnc2cc1OC
CCOc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C(F)(F)F)c3)ncnc2cc1OC
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C(F)(F)F)c3)ncnc2cc1O
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C(F)(F)F)c3)c2cc1O
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C(F)(F)F)c3F)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(on4)C(C)(C)C(F)(F)F)ccc3F)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(C)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(no4)C(C)(C)F)c(F)cc3F)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(on4)C(C)(C)C)c(F)cc3F)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)F)c(F)cc3F)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C(C)(C)C)c(F)cc3F)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c(F)cc3F)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C(C)(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cccc(c4)C(C)(C)C#N)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cccc(c4)C(C)(C)C#N)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cccc(c4)C(C)(C)C#N)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4C)C(C)(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cccc(C)c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4cccc(C)c4)C(C)(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4cccc(C)c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C(C)(C)C)c3C)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c3C)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3C)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)F)c3C)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3C)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(no4)C(C)(C)F)ccc3F)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(on4)C(C)(CF)CF)ccc3F)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c3F)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3F)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(CF)CF)c3F)c2cc1OC
COc1cc2ncnc(Oc3ccc(Cl)c(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3ccc(Cl)c(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3ccc(Cl)c(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3ccc(Cl)c(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)CN4CCOCC4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cnccc4C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cccnc4C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)CF)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C#N)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C#N)c3)c2cc1OC
COc1cc2nc(Cl)nc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cccnc4)C(C)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)nc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cc[nH]c(=O)c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cncc(F)c4)C(C)C)c3)c2cc1OC
COc1ccc(cc1)-n1nc(cc1NC(=O)Nc1cccc(Oc2ncnc3cc(OC)c(OC)cc23)c1)C(C)(F)F
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cncc(F)c4)C(C)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(=O)[nH]c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccnc(C)c4)C(C)(C)C)c3)c2cc1OC
CCn1nc(cc1NC(=O)Nc1cccc(Sc2ncnc3cc(OC)c(OC)cc23)c1)C(C)(C)C
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cccnc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4cccnc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cncc(F)c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4cncc(F)c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(cc4)C#N)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(cc4)C#N)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4C4CCCCC4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4C4CCCCC4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4CC(C)C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4CC(C)C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4C(C)C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4C(C)C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccncc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccncc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cccc(C)c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4Cl)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4Cl)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccn4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccn4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C4(CC4)C(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C4(CC4)C(F)(F)F)c3)c2cc1OC
COc1ccc(cc1)-n1nc(cc1NC(=O)Nc1cccc(Oc2ncnc3cc(OC)c(OC)cc23)c1)C(C)C
COc1ccc(cc1)-n1nc(cc1NC(=O)Nc1cccc(Sc2ncnc3cc(OC)c(OC)cc23)c1)C(C)C
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cccnc4)C(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4cccnc4)C(C)C)c3)c2cc1OC
CCc1cc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)n(n1)-c1ccccc1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C4CC4)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C4CC4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C4CCC4)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C4CCC4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4Cc4ccccc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4Cc4ccccc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cccc(F)c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4cccc(F)c4)C(C)(C)C)c3)c2cc1OC
COc1ccc(cc1)-n1nc(cc1NC(=O)Nc1cccc(Oc2ncnc3cc(OC)c(OC)cc23)c1)C(C)(C)C
COc1ccc(cc1)-n1nc(cc1NC(=O)Nc1cccc(Sc2ncnc3cc(OC)c(OC)cc23)c1)C(C)(C)C
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cccc(Cl)c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4cccc(Cl)c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(Cl)cc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(Cl)cc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3ccc(F)c(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3ccc(F)c(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(cc4)C(C)(C)C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(cc4)C(C)(C)C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4F)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4F)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(cc4)C(F)(F)F)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(cc4)C(F)(F)F)C(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4C(F)(F)F)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4C(F)(F)F)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C4(CC4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C4(CC4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cccc(c4)C(F)(F)F)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4cccc(c4)C(F)(F)F)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(C)C#N)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C4(CC4)C(F)(F)F)c3)c2cc1OC
CCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)F)c3)c2cc1OC
CCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)c2cc1OC
CCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(CF)CF)c3)c2cc1OC
CCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c3)c2cc1OC
CCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(CF)CF)c3)c2cc1OC
CCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)c2cc1OC
CCOc1cc2c(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c3)ncnc2cc1OC
CCOc1cc2c(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)F)c3)ncnc2cc1OC
CCOc1cc2c(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)ncnc2cc1OC
CCOc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(CF)CF)c3)ncnc2cc1OC
CCOc1cc2c(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)ncnc2cc1OC
CCOc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(CF)CF)c3)ncnc2cc1OC
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)F)c3)ncnc2cc1OCCN1CCOCC1
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)F)ccc3F)c2cc1OC
COc1ccc(cn1)-n1nc(cc1NC(=O)Nc1cccc(Oc2ncnc3cc(OC)c(OC)cc23)c1)C(C)(C)C
CCc1cc(NC(=O)Nc2cccc(Sc3ncnc4cc(OC)c(OC)cc34)c2)n(n1)-c1ccccc1
Cc1ncc(cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1=O)C(=O)Nc1cccc(c1)C(F)(F)F
CC(=C)c1cc(nc(n1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C)N1CCOCC1
Cc1ccc(cc1-c1cc(OCc2ccccc2)cc(n1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(ncn1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(O[C@@H]2CC[C@H](O)CC2)c(c1)N1CCOCC1 |r,wD:25.26,28.30,(-2.15,-1.94,;-.82,-2.71,;.52,-1.94,;1.85,-2.71,;1.85,-4.25,;3.19,-5.02,;4.52,-4.25,;4.52,-2.71,;5.85,-5.02,;7.19,-4.25,;8.52,-5.02,;8.52,-6.56,;7.15,-7.43,;5.85,-6.56,;7.13,-8.97,;7.11,-10.51,;5.59,-8.96,;8.67,-8.99,;.52,-5.02,;-.82,-4.25,;-2.15,-5.02,;-2.15,-6.56,;-3.48,-7.33,;-4.82,-6.56,;-6.15,-7.33,;-6.15,-8.87,;-4.82,-9.64,;-4.82,-11.18,;-6.15,-11.95,;-6.15,-13.49,;-7.48,-11.18,;-7.48,-9.64,;-4.82,-5.02,;-3.48,-4.25,;-6.15,-4.25,;-5.75,-2.76,;-6.84,-1.67,;-8.33,-2.07,;-8.73,-3.56,;-7.64,-4.65,)|
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(O[C@H]2CC[C@H](O)C2)c(c1)N1CCOCC1 |r|
Cc1ncc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cnc(OC2CNC2)c(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cnc(c(c1)N1CCOCC1)C(C)(C)C#N
Cc1ncc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cnc(CS(C)(=O)=O)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cc(Br)cc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
COc1ncc(nc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cnc1C
COc1ncc(nc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C2(CC2)C#N)cnc1C
COc1ncc(nc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(F)F)cnc1C
COc1ncc(nc1N1CCOCC1)-c1cc(NC(=O)c2cc(CN(C)C)cc(c2)C(F)(F)F)cnc1C
COc1ncc(nc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)F)cnc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)S(C)(=O)=O)ccc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccc(CCl)c(c2)C(F)(F)F)ccc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccc(CN(C)CC)c(c2)C(F)(F)F)ccc1C
Cc1ccc(NC(=O)c2cnnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(OC2CCOCC2)nn1
CC(C)Oc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C
CCOc1nnc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccc(CCl)c(c2)C(F)(F)F)cnc1C
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2oc(=O)[nH]c2c1
C[C@@H]1COCCN1c1nc(cc2CCSc12)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C |r|
Cc1ncc(NC(=O)c2ccc(C#N)c(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2n1
Cc1ncc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(N2CCOCC2)c2nccn2n1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c2nccn2n1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(nc(c1)-c1cnn(C)c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1ccnc(c1)N1CCOCC1
O=C1CCc2c(Oc3ccc4CC5C(C5c4c3)c3nc4ccccc4[nH]3)ccnc2N1
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Cc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Sc1ccccc1NC(=O)C1C2Cc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
O=C1CCc2c(Oc3ccc4OC5C(C5c4c3)c3nc4ccccc4[nH]3)ccnc2N1
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
FC(F)(F)c1ccc2nc([nH]c2c1)[C@H]1[C@@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@H]12 |r|
FC(F)(F)c1ccc2nc([nH]c2c1)[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
Clc1cc2nc([nH]c2cc1Cl)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Clc1cc2nc([nH]c2cc1Cl)[C@H]1[C@@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@H]12 |r|
Clc1cc2nc([nH]c2cc1Cl)[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
Cc1cc2[nH]c(nc2cc1F)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Cc1cc2[nH]c(nc2cc1F)[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
Cc1cc2[nH]c(nc2cc1F)[C@H]1[C@@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@H]12 |r|
FC(F)(F)c1cc2[nH]c(nc2cc1Cl)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
FC(F)(F)c1cc2[nH]c(nc2cc1Cl)[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1cc2[nH]c(nc2cc1Cl)[C@H]1[C@@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@H]12 |r|
O=C1CCc2c(Oc3ccc4OC5C(C5c4c3)c3nc4ccc(cc4[nH]3)C#N)ccnc2N1
Fc1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Cc1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
O=C1CCc2c(Oc3ccc4OC5C(C5c4c3)c3nc4ccncc4[nH]3)ccnc2N1
FC(F)(F)c1cc(Cl)c2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Fc1cc2nc([nH]c2cc1F)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Clc1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Brc1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
FC(F)(F)Oc1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Cn1c(nc2ccccc12)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
COc1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Fc1cc2[nH]c(nc2cc1Cl)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
FC(F)(F)c1cccc2nc([nH]c12)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Fc1cccc2nc([nH]c12)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
CC(C)(C)c1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
O=C1CCc2c(Oc3ccc4OC5C(C5c4c3)c3nc4cc5CCCc5cc4[nH]3)ccnc2N1
NC(=O)c1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Cn1c(nc2ccc(cc12)C(F)(F)F)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Cn1c(nc2cc(ccc12)C(F)(F)F)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Oc3c(cccc3Oc3ccnc4NC(=O)CCc34)C12
Clc1cccc2nc([nH]c12)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Oc1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
O=C1CCc2c(Oc3ccc4OC5C(C5c4c3)c3nc(no3)-c3ccccc3)ccnc2N1
O=C(COC(=O)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12)c1ccccc1
O=C1CCc2c(Oc3ccc4OC5C(C5c4c3)c3nc(c[nH]3)-c3ccncc3)ccnc2N1
Clc1ccccc1-c1c[nH]c(n1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
FC(F)(F)c1c[nH]c(n1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
OCCn1c(nc2cc(ccc12)C(F)(F)F)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Cc1cc(Oc2ccnc3NC(=O)CCc23)cc2C3C(Oc12)C3c1nc2ccc(cc2[nH]1)C(F)(F)F
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Oc3cc(Cl)c(Oc4ccnc5NC(=O)CCc45)cc3C12
Cc1cc2nc([nH]c2cc1F)C1C2Oc3cc(Cl)c(Oc4ccnc5NC(=O)CCc45)cc3C12
CNC(=O)Nc1cc(Oc2ccc3OC4C(C4c3c2)c2nc3ccc(cc3[nH]2)C(F)(F)F)ccn1
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccncn4)cc3C12
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5[nH]ccc45)cc3C12
FC(F)(F)c1c[nH]c(n1)-c1cc(Oc2ccc3OC4C(C4c3c2)c2nc3ccc(cc3[nH]2)C(F)(F)F)ccn1
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ncnc5[nH]cnc45)cc3C12
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccncc4)cc3C12
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)OCc45)cc3C12
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4c(Cl)cnc5NC(=O)CCc45)cc3C12
OC(=O)C1C2Cc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
OC(=O)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
CCn1nc(C#Cc2cc(ccc2C)C(=O)Nc2ccc(CN3CCN(C)CC3)c(c2)C(F)(F)F)c2c(N)ncnc12
CN1CCC(CC1)n1nc(C#Cc2cc(NC(=O)c3cccc(c3)C(F)(F)F)ccc2C)c2c(N)ncnc12
Cc1ccc(NC(=O)c2ccc(C)c(c2)C(F)(F)F)cc1C#Cc1nn([C@H]2CC[C@H](O)CC2)c2ncnc(N)c12 |r,wU:26.27,wD:29.31,(-5.46,5.4,;-3.98,5.8,;-3.58,7.29,;-2.09,7.69,;-1,6.6,;.49,7,;1.57,5.91,;1.18,4.42,;3.06,6.31,;3.46,7.79,;4.95,8.19,;6.04,7.1,;7.53,7.5,;5.64,5.62,;4.15,5.22,;6.73,4.53,;8.22,4.93,;6.33,3.04,;7.82,3.44,;-1.4,5.11,;-2.89,4.71,;-3.29,3.22,;-3.68,1.74,;-4.08,.25,;-3.18,-1,;-4.08,-2.24,;-3.68,-3.73,;-2.2,-4.13,;-1.8,-5.62,;-2.89,-6.7,;-2.49,-8.19,;-4.38,-6.31,;-4.77,-4.82,;-5.55,-1.77,;-6.88,-2.54,;-8.22,-1.77,;-8.22,-.23,;-6.88,.54,;-6.88,2.08,;-5.55,-.23,)|
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(Cl)cc2)c1F
O=C1CCc2c(Oc3ccc4CC5C(C5c4c3)c3nc4ccccc4s3)ccnc2N1
O=C1CCc2c(Oc3ccc4OC5C(C5c4c3)c3nc4ccc(cc4[nH]3)-c3ccccc3)ccnc2N1
O=C1CCc2c(Oc3ccc4OC5C(C5c4c3)c3nc(c[nH]3)-c3ccccc3)ccnc2N1
CNC(=O)c1cc(Oc2ccc3OC4C(C4c3c2)c2nc3ccc(cc3[nH]2)C(F)(F)F)ccn1
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1cc(Cl)cc(NS(C)(=O)=O)c1)C(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1cccc(NS(C)(=O)=O)c1F)C(C)C |r|
CCCS(=O)(=O)Nc1cc(Cl)cc(c1)-c1nn(cc1-c1ccnc(NC[C@H](C)NC(=O)OC)n1)C(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1c(F)ccc(NS(C)(=O)=O)c1F)C(C)C |r,wD:5.5,(-7.74,6.48,;-6.41,5.71,;-5.08,6.48,;-5.08,8.02,;-3.74,5.71,;-3.74,4.17,;-5.08,3.4,;-2.41,3.4,;-2.41,1.86,;-1.08,1.09,;.26,1.86,;1.59,1.09,;1.59,-.45,;.26,-1.22,;-1.08,-.45,;.26,-2.76,;-.99,-3.66,;-.51,-5.13,;1.03,-5.13,;1.5,-3.66,;2.99,-3.27,;3.39,-1.78,;2.3,-.69,;4.88,-1.38,;5.97,-2.47,;5.57,-3.96,;6.66,-5.05,;6.26,-6.53,;5.86,-8.02,;4.77,-6.13,;7.74,-6.93,;4.08,-4.36,;3.68,-5.84,;-1.28,-6.46,;-.51,-7.8,;-2.82,-6.46,)|
CCCS(=O)(=O)Nc1ccc(F)c(-c2nn(cc2-c2ccnc(NC[C@H](C)NC(=O)OC)n2)C(C)C)c1F |r,wD:25.26,(6.55,-9.31,;6.95,-7.82,;5.86,-6.73,;6.26,-5.24,;4.77,-4.85,;7.74,-5.64,;6.66,-3.76,;5.57,-2.67,;5.97,-1.18,;4.88,-.09,;3.39,-.49,;2.3,.6,;2.99,-1.98,;1.5,-2.38,;1.03,-3.84,;-.51,-3.84,;-.99,-2.38,;.26,-1.47,;.26,.07,;1.59,.84,;1.59,2.38,;.26,3.15,;-1.08,2.38,;-2.41,3.15,;-2.41,4.69,;-3.74,5.46,;-5.08,4.69,;-3.74,7,;-5.08,7.77,;-5.08,9.31,;-6.41,7,;-7.74,7.77,;-1.08,.84,;-1.28,-5.17,;-.51,-6.51,;-2.82,-5.17,;4.08,-3.07,;3.68,-4.55,)|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1cc(Cl)cc(NS(C)(=O)=O)c1F)C(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1cc(F)cc(NS(C)(=O)=O)c1F)C(C)C |r|
CCn1cc(c(n1)-c1cc(Cl)cc(NS(C)(=O)=O)c1F)-c1ccnc(NC[C@H](C)NC(=O)OC)n1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1cc(C)cc(NS(C)(=O)=O)c1F)C(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1cc(C)cc(NS(C)(=O)=O)c1Cl)C(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1cc(F)cc(NS(C)(=O)=O)c1Cl)C(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1ccnc(NS(C)(=O)=O)c1F)C(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1ccc(F)c(NS(C)(=O)=O)c1F)C(C)C |r|
COC(=O)N[C@H](C)CNc1nccc(n1)-c1cn(nc1-c1cc(Cl)cc(NS(C)(=O)=O)c1F)C(C)C |r|
CCS(=O)(=O)Nc1c(F)ccc(-c2nn(cc2-c2ccnc(NC[C@H](C)NC(=O)OC)n2)C(C)C)c1F |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1cc(NS(C)(=O)=O)c(C)c(OC)c1)C(C)C |r|
CC(C)n1cc(c(n1)-c1cc(Cl)cc(NS(C)(=O)=O)c1F)-c1ccnc(NCCN(C)C)n1
CNc1nccc(n1)-c1cn(nc1-c1cc(Cl)cc(NS(C)(=O)=O)c1F)C(C)C
CC(C)n1cc(c(n1)-c1cc(Cl)cc(NS(C)(=O)=O)c1F)-c1ccnc(N)n1
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1c[nH]nc1-c1cc(Cl)cc(NS(C)(=O)=O)c1F |r|
COC(=O)NC[C@H](C)Nc1nccc(n1)-c1cn(nc1-c1cc(Cl)cc(NS(C)(=O)=O)c1F)C(C)C |r|
CCCS(=O)(=O)Nc1c(F)ccc(-c2nn(cc2-c2ccnc(NC[C@H](C)NC(=O)OC)n2)C(C)C)c1F |r|
CN1CCN(CCNc2nccc(n2)-c2c(nc3occn23)-c2cccc(O)c2)S1(=O)=O
CCN1CCN(CCNc2nccc(n2)-c2c(nc3occn23)-c2cccc(O)c2)S1(=O)=O
COc1ccc(cc1)S(=O)(=O)NCCNc1nccc(n1)-c1c(nc2sccn12)-c1ccccc1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(cc2)C(F)(F)F)n1
Oc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(F)cc2)n1
Oc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccc(F)cc2)n1
Oc1c(Br)cc(C=C2C(=O)Nc3ccc(I)cc23)cc1Br
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(Oc2ccc3nccnc3c2)c1
COc1ccc(NC(=O)Nc2cccc(Oc3ccc4nccnc4c3)c2)cc1
FC(F)(F)c1cc(NC(=O)Nc2cccc(Oc3ccc4nccnc4c3)c2)ccc1Cl
FC(F)(F)c1cccc(NC(=O)Nc2cccc(Oc3ccc4nccnc4c3)c2)c1
Fc1ccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)cc1Oc1ccc2ncc(nc2c1)N1CCOCC1
FC(F)(F)c1cccc(NC(=O)Nc2ccc(Oc3ccc4nccnc4c3)cc2)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc2[nH]cnc2c(n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc2[nH]cnc2c(n1)N1CCOCC1
Cc1ncc(NC(=O)c2cc(cc(c2)S(C)(=O)=O)C(F)(F)F)cc1-c1ccnc(c1)N1CCOCC1
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cc(CF)cc(c2)N2CCN(CC)CC2)cnc1C
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(O[C@H]2CCOC2)c(c1)N1CCOCC1=O |r|
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(O[C@H]2CC[C@H](O)CC2)c(c1)N1CCOCC1 |r,wU:28.30,wD:25.26,(-2.15,13.29,;-.82,12.52,;.52,13.29,;1.85,12.52,;1.85,10.98,;3.19,10.21,;4.52,10.98,;4.52,12.52,;5.85,10.21,;7.19,10.98,;8.52,10.21,;8.52,8.67,;7.19,7.84,;5.85,8.67,;7.19,6.3,;7.19,4.76,;5.65,6.3,;8.73,6.3,;.52,10.21,;-.82,10.98,;-2.15,10.21,;-2.15,8.67,;-3.48,7.9,;-4.82,8.67,;-6.15,7.9,;-6.15,6.36,;-7.48,5.59,;-7.48,4.05,;-6.15,3.28,;-6.15,1.74,;-4.82,4.05,;-4.82,5.59,;-4.82,10.21,;-3.48,10.98,;-6.15,10.98,;-5.75,12.46,;-6.84,13.55,;-8.33,13.15,;-8.73,11.67,;-7.64,10.58,)|
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(O[C@H]2CC[C@@H](O)C2)c(c1)N1CCOCC1 |r|
Cc1ccc(NC(=O)c2ccc(CCN)c(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
CNCc1cc(cc(c1)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(N)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ncc(N)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
CCN1C=C(C=C(C1O)C(F)(F)F)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)n(C)c(=O)c1 |c:3,5|
CNc1nc(cc(n1)-c1cc(ccc1C)C(=O)Nc1cccc(c1)C(C)(C)C#N)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(cc2oc(=O)[nH]c12)N1CCOCC1
Cc1ccc(NC(=O)c2cnnc(c2)C2(CC2)C#N)cc1-c1cc(nc(c1)N1CCOCC1)N1CC(O)C1
FC(F)(F)c1cc(NC(=O)Nc2cccc(c2)C(=O)c2ccc3nccnc3c2)ccc1Cl
FC(F)(F)c1cccc(NC(=O)Nc2cccc(c2)C(=O)c2ccc3nccnc3c2)c1
Fc1ccc(NC(=O)Nc2cccc(c2)C(F)(F)F)cc1C(=O)c1ccc2nccnc2c1
Fc1ccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)cc1C(=O)c1ccc2nccnc2c1
Fc1cccc(NC(=O)Nc2cccc(c2)C(=O)c2ccc3ncc(nc3c2)N2CCOCC2)c1
FC(F)(F)c1cccc(NC(=O)Nc2cccc(c2)C(=O)c2ccc3ncc(nc3c2)N2CCOCC2)c1
FC(F)(F)c1cc(NC(=O)Nc2cccc(c2)C(=O)c2ccc3ncc(nc3c2)N2CCOCC2)ccc1Cl
Fc1cccc(NC(=O)Nc2cccc(c2)C(=O)c2ccc3ncc(nc3c2)N2CCCC2)c1
FC(F)(F)c1cc(NC(=O)Nc2cccc(c2)C(=O)c2ccc3ncc(nc3c2)-c2cccnc2)ccc1Cl
Cn1cc(cn1)-c1cnc2ccc(cc2n1)C(=O)c1cccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c1
FC(F)(F)c1cc(NC(=O)Nc2cccc(c2)C(=O)c2ccc3ncc(nc3c2)-c2cn[nH]c2)ccc1Cl
Fc1cccc(NC(=O)Nc2ccc(F)c(c2)C(=O)c2ccc3ncc(nc3c2)N2CCOCC2)c1
Fc1ccc(NC(=O)Nc2cccc(c2)C(F)(F)F)cc1C(=O)c1ccc2ncc(nc2c1)N1CCOCC1
Fc1cc(NC(=O)Nc2cccc(c2)C(F)(F)F)cc(c1)C(=O)c1ccc2ncc(nc2c1)N1CCOCC1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)C(=O)c1ccc2ncc(nc2c1)N1CCOCC1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)C(=O)c1ccc2ncc(nc2c1)N1CCCC1
FC(F)(F)c1ccc(cc1Cl)C(=O)Nc1cccc(c1)C(=O)c1ccc2ncc(nc2c1)-c1cccnc1
Fc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1C(=O)c1ccc2ncc(nc2c1)N1CCOCC1
Fc1cc(NC(=O)c2cccc(c2)C(F)(F)F)cc(c1)C(=O)c1ccc2ncc(nc2c1)N1CCOCC1
Fc1cc(NC(=O)c2cccc(c2)C(F)(F)F)cc(C(=O)c2ccc3ncc(nc3c2)N2CCOCC2)c1F
Fc1ccc(NC(=O)c2ccc(Cl)c(c2)C(F)(F)F)cc1C(=O)c1ccc2ncc(nc2c1)N1CCOCC1
Fc1cc(NC(=O)Nc2cccc(c2)C(F)(F)F)cc(C(=O)c2ccc3ncc(nc3c2)N2CCOCC2)c1F
Fc1ccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)cc1C(=O)c1ccc2ncc(nc2c1)N1CCOCC1
Fc1ccc(NC(=O)c2ccc(Cl)c(c2)C(F)(F)F)c(Cl)c1C(=O)c1ccc2nccnc2c1
Fc1cc(NC(=O)c2cccc(c2)C(F)(F)F)c(F)c(C(=O)c2ccc3nccnc3c2)c1F
Fc1cccc(c1)C(=O)Nc1cccc(c1)C(=O)c1ccc2ncc(nc2c1)N1CCCC1
Nc1ncnc2n(C[C@H]3SSC[C@H]3O)nc(-c3ccc(Oc4ccccc4)cc3)c12 |r|
CCN1CCN(CCNc2nccc(n2)-c2c(nc3sccn23)-c2ccc(F)c(O)c2)S1(=O)=O
COc1cc(ccc1F)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccc(F)cc2)n1
COc1cc(ccc1F)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccc(Cl)cc2)n1
Oc1cc(ccc1F)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(F)cc2)n1
Oc1cc(ccc1F)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(Cl)cc2)n1
Oc1cc(ccc1F)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccccc2)n1
Oc1cc(ccc1F)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccc(Cl)cc2)n1
COc1ccc(cc1)S(=O)(=O)NCCCNc1nccc(n1)-c1c(nc2sccn12)-c1ccc(F)c(O)c1
Nc1cc(ccc1F)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccc(F)cc2)n1
COc1cc(ccc1F)-c1nc2occn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccc(Cl)cc2)n1
Oc1cc(ccc1F)-c1nc2occn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(F)cc2)n1
Oc1cc(ccc1F)-c1nc2occn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(Cl)cc2)n1
Oc1cc(ccc1F)-c1nc2occn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccc(Cl)cc2)n1
COc1ccc(cc1)S(=O)(=O)NCCCNc1nccc(n1)-c1c(nc2occn12)-c1ccc(F)c(O)c1
Oc1cc(ccc1F)-c1nc2occn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccccc2)n1
Cn1cc(cn1)-c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)CC4CC4)c3F)c2c1
CN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C2(CC2)C#N)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C2(CC2)C#N)c1F
Fc1ccc(NS(=O)(=O)N2CCCC2)c(F)c1C(=O)c1c[nH]c2ncc(cc12)-c1ccc(cc1)C1(CC1)C#N
CC(N(C)C)S(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1F
Cc1c(Nc2c(F)ccc(NS(=O)(=O)CCCF)c2F)ccc2ncn(C)c(=O)c12
CCCS(=O)(=O)Nc1cccc(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
Cc1c(Nc2cccc(NS(=O)(=O)CCCF)c2Cl)ccc2ncn(C)c(=O)c12
CCCS(=O)(=O)Nc1cc(F)c(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1F
Cc1c(Nc2c(F)c(F)cc(NS(=O)(=O)CCCF)c2F)ccc2ncn(C)c(=O)c12
CCCS(=O)(=O)Nc1cc(F)c(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
Cc1c(Nc2c(F)c(F)cc(NS(=O)(=O)CCCF)c2Cl)ccc2ncn(C)c(=O)c12
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
Cc1c(ccc2c1C(=O)N(C=N2)C)Nc3c(ccc(c3Cl)NS(=O)(=O)CCCF)F
CCCS(=O)(=O)Nc1cc(F)cc(Nc2ccc3ncn(C)c(=O)c3c2C)c1F
CCCS(=O)(=O)Nc1cc(F)cc(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1cc(Cl)cc(Nc2ccc3ncn(C)c(=O)c3c2C)c1F
CCCS(=O)(=O)Nc1ccc(Cl)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ncc(Cl)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ncc(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1F
Cc1c(Nc2c(F)cnc(NS(=O)(=O)CCCF)c2F)ccc2ncn(C)c(=O)c12
CCCS(=O)(=O)Nc1ncc(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
Cc1c(Nc2c(F)cnc(NS(=O)(=O)CCCF)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)c3ccco3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CCCC3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC[C@@H](F)C3)c2Cl)ccc2ncn(C)c(=O)c12 |r|
Cc1c(Nc2c(F)ccc(NS(=O)(=O)c3cc(F)ccc3F)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)c3ccccn3)c2Cl)ccc2ncn(C)c(=O)c12
COCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1C#N
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(Cc4ccccc4)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(CCOC)c(=O)c3c2C)c1Cl |$;;;;;;;;;;;;;;;;;;;;;;;O;;;;;;;;$|
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C4CC4)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(-c4ccccc4)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C4CCC4)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn([C@@H]4CCOC4)c(=O)c3c2C)c1Cl |r|
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn([C@H]4CCOC4)c(=O)c3c2C)c1Cl |r|
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C(C)C)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(CC)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(CC4CC4)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C4CCCC4)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ccc(Cl)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1F
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1C
Cc1c(Nc2c(F)cnc(NS(=O)(=O)CC3CC3)c2F)ccc2ncn(C)c(=O)c12
CCS(=O)(=O)Nc1ncc(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1F
Cc1c(Nc2cc(F)cc(NS(=O)(=O)CCCF)c2Cl)ccc2ncn(C)c(=O)c12
CCS(=O)(=O)Nc1ncc(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1cc(C)cc(Nc2ccc3ncn(C)c(=O)c3c2C)c1F
Cc1c(Nc2c(F)cnc(NS(=O)(=O)CC3CC3)c2Cl)ccc2ncn(C)c(=O)c12
CCCS(=O)(=O)Nc1cc(Cl)cc(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
Cc1c(Nc2c(F)ccc(NS(=O)(=O)c3ccccc3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)CC3CC3)c2Cl)ccc2ncn(C)c(=O)c12
CC(C)CS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
CCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1cccc(Nc2ccc3ncn(C)c(=O)c3c2C)c1C#N
CCN(C)S(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Oc2ccc3ncn(C)c(=O)c3c2C)c1Cl
Cc1c(Oc2c(F)ccc(NS(=O)(=O)CCCF)c2F)ccc2ncn(C)c(=O)c12
CCCS(=O)(=O)Nc1nccc(Oc2ccc3ncn(C)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(-c4cccnc4)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(CC(F)(F)F)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2C#C)c1Cl
CCC(C)S(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ncc(F)c(Oc2ccc3ncn(C)c(=O)c3c2C)c1F
CCCS(=O)(=O)Nc1ncc(F)c(Oc2ccc3ncn(C)c(=O)c3c2C)c1Cl
Cc1c(Oc2c(F)cnc(NS(=O)(=O)CCCF)c2F)ccc2ncn(C)c(=O)c12
CCCS(=O)(=O)Nc1ccc(F)c(Sc2ccc3ncn(C)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1cccc(Oc2ccc3ncn(C)c(=O)c3c2C)c1C#N
Cc1c(Oc2c(F)ccc(NS(=O)(=O)CCCF)c2Cl)ccc2ncn(C)c(=O)c12
CCCS(=O)(=O)Nc1cccc(Oc2ccc3ncn(C)c(=O)c3c2C)c1F
CCCS(=O)(=O)Nc1ccc(F)c(Oc2ccc3ncn(C)c(=O)c3c2C)c1C#N
CCCS(=O)(=O)Nc1cc(Cl)cc(Oc2ccc3ncn(C)c(=O)c3c2C)c1F
CCCS(=O)(=O)Nc1ccc(F)c(Oc2ccc3ncn(C)c(=O)c3c2C)c1F
CCCS(=O)(=O)Nc1cc(F)c(F)c(Oc2ccc3ncn(C)c(=O)c3c2C)c1F
CCCS(=O)(=O)Nc1cc(F)c(F)c(Oc2ccc3ncn(C)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1cc(F)cc(Oc2ccc3ncn(C)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1cc(C)cc(Oc2ccc3ncn(C)c(=O)c3c2C)c1F
CCCS(=O)(=O)Nc1cc(F)cc(Oc2ccc3ncn(C)c(=O)c3c2C)c1F
Cc1c(Oc2cc(F)cc(NS(=O)(=O)CCCF)c2F)ccc2ncn(C)c(=O)c12
CCCS(=O)(=O)Nc1cccc(Oc2ccc3ncn(C)c(=O)c3c2C)c1Cl
Cc1c(Oc2cccc(NS(=O)(=O)CCCF)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Oc2cccc(NS(=O)(=O)CCCF)c2F)ccc2ncn(C)c(=O)c12
Cc1ccc2c(Nc3ccc(O)c(Cl)c3F)nccc2c1NC(=O)c1csc2c(N)ncnc12 |$;;;;;;N;;;;;;;;;;;;;;;;;;;;;;;;;;;$|
O=C1CCc2c(Oc3ccc4OCC(Cc4c3)c3nc4ccccc4[nH]3)ccnc2N1
Clc1cccc2nc([nH]c12)C1COc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1
O=C1CCc2c(Oc3ccc4OCC(Cc4c3)c3nc(c[nH]3)-c3ccccc3)ccnc2N1
O=C1CCc2c(Oc3ccc4OCC(Cc4c3)c3nc(c[nH]3)-c3ccncc3)ccnc2N1
CC(C)(C)c1c[nH]c(n1)C1COc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1
O=C1CCc2c(Oc3ccc4OCC(Cc4c3)c3nc(c[nH]3)-c3ccsc3)ccnc2N1
O=C1CCc2c(Oc3ccc4OCC(Cc4c3)c3nc(c[nH]3)-c3cccs3)ccnc2N1
Clc1ccccc1-c1cnc([nH]1)C1COc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1
Clc1cccc(c1)-c1cnc([nH]1)C1COc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1
O=C1CCc2c(Oc3ccc4OCC(Cc4c3)c3nc(c[nH]3)-c3coc4ccccc34)ccnc2N1
O=C1CCc2c(Oc3ccc4OCC(Cc4c3)c3ncc([nH]3)-c3cccnc3)ccnc2N1
CS(=O)(=O)c1ccc(cc1)-c1cnc([nH]1)C1COc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1
Fc1ccc(cc1)-c1cnc([nH]1)C1COc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1
O=C1CCc2c(Oc3ccc4OCC(Cc4c3)c3ncc([nH]3)-c3ccc4OCOc4c3)ccnc2N1
O=C1CCc2c(Oc3ccc4OCC(Cc4c3)c3ncc([nH]3)-c3ccc4OCCOc4c3)ccnc2N1
O=C1CCc2c(Oc3ccc4OCC(=Cc4c3)c3nc(c[nH]3)-c3ccccc3)ccnc2N1 |c:13|
O=C1CCc2c(Oc3ccc4OCC(Cc4c3)c3nc(no3)-c3ccccc3)ccnc2N1
O=C1CCc2c(Oc3ccc4OCC(Cc4c3)c3cc([nH]n3)-c3ccccc3)ccnc2N1
O=C1CCc2c(Oc3ccc4OC[C@@H](Oc4c3)c3nc(c[nH]3)-c3ccccc3)ccnc2N1 |r|
O=C1CCc2c(Oc3ccc4OC[C@H](Oc4c3)c3nc(c[nH]3)-c3ccccc3)ccnc2N1 |r|
Cc1cc(Oc2ccc3OCC(Cc3c2)c2ncc([nH]2)-c2ccccc2)ccn1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4cccc(Cl)c4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(Br)csc23)c(OC)c1
Cc1ccc2c(nccc2c1NC(=O)c1csc2c(N)ncnc12)C(O)c1ccccc1F
COc1ccc(Cc2nccc3c(NC(=O)c4csc5c(NCc6ccc(OC)cc6OC)ncnc45)c(C)ccc23)cc1
COc1ccc(cc1)C(O)c1nccc2c(NC(=O)c3csc4c(N)ncnc34)c(C)ccc12
COc1ccc(cc1)C(=O)c1nccc2c(NC(=O)c3csc4c(N)ncnc34)c(C)ccc12
COc1ccc(CNc2ncnc3c(csc23)C(=O)Nc2c(C)ccc3c(Cc4cccc(Cl)c4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(csc23)C(=O)Nc2c(C)ccc3c(Cc4ccccc4Cl)nccc23)c(OC)c1
Cc1ccc2c(nccc2c1NC(=O)c1csc2c(N)ncnc12)C(=O)c1ccccc1Cl
Cc1ccc2c(Nc3cccc(Cl)c3)nccc2c1NC(=O)c1cnc2c(N)ncnn12
COc1ccc(CNc2ncnc3c(csc23)C(=O)Nc2c(C)ccc3c(Cc4ccc(F)cc4)nccc23)c(OC)c1
Cc1ccc2c(nccc2c1NC(=O)c1csc2c(N)ncnc12)C(O)c1ccccc1Cl
Cc1ccc2c(nccc2c1NC(=O)c1csc2c(N)ncnc12)C(O)c1ccc(F)cc1
COc1ccc(CNc2ncnc3c(csc23)C(=O)Nc2c(C)ccc3c(Cc4cccc(Cl)c4)nccc23)c(OC)c1
Cc1ccc2c(nccc2c1NC(=O)c1csc2c(N)ncnc12)C(O)c1cccc(Cl)c1
COc1ccc(CNc2ncnc3c(csc23)C(=O)Nc2c(C)ccc3c(Cc4ccc(Cl)cc4)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(csc23)C(=O)Nc2c(C)ccc3c(Cc4cccc(c4)C(F)(F)F)nccc23)c(OC)c1
Cc1ccc2c(nccc2c1NC(=O)c1csc2c(N)ncnc12)C(O)c1ccc(Cl)cc1
Cc1ccc2c(nccc2c1NC(=O)c1csc2c(N)ncnc12)C(=O)c1cccc(c1)C(F)(F)F
Cc1ccc2c(nccc2c1NC(=O)c1csc2c(N)ncnc12)C(O)c1cccc(c1)C(F)(F)F
Cc1ccc2c(nccc2c1NC(=O)c1cccc2c(N)ncnc12)C(O)c1ccccc1Cl
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Cc4ccccc4Cl)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(csc23)C(=O)Nc2c(C)ccc3c(Cc4ccc(Cl)cc4F)nccc23)c(OC)c1
Cc1ccc2c(nccc2c1NC(=O)c1csc2c(N)ncnc12)C(=O)c1ccc(Cl)cc1F
Cc1ccc2c(nccc2c1NC(=O)c1csc2c(N)ncnc12)C(O)c1ccc(Cl)cc1F
Cc1ccc2c(Nc3cccc(Cl)c3F)nccc2c1NC(=O)c1cnc2c(N)ncnn12
Cc1ccc2c(nccc2c1NC(=O)c1csc2c(N)ncnc12)C(O)c1ccc(cc1)C(F)(F)F
COc1ccc(CNc2ncnc3c(csc23)C(=O)Nc2c(C)ccc3c(Cc4ccc(cc4)C(F)(F)F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(csc23)C(=O)Nc2c(C)ccc3c(nccc23)C(C)Oc2ccccc2)c(OC)c1
COc1ccc(CNc2ncnc3c(csc23)C(=O)Nc2c(C)ccc3c(Cc4ccc(nc4)N(C)C)nccc23)c(OC)c1
CN(C)c1ccc(cn1)C(O)c1nccc2c(NC(=O)c3csc4c(N)ncnc34)c(C)ccc12
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4cccc(Cl)c4)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4ccccc4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4ccc(CN(C)C)cc4)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4ccc(Cl)cc4F)nccc23)c(OC)c1
Cc1ccc2c(Cc3ccc(Cl)c(c3)C3OCCO3)nccc2c1NC(=O)c1csc2c(N)ncnc12
Cc1ccc2c(Nc3cccc(c3)C(F)(F)F)nccc2c1NC(=O)c1cnc2c(N)ncnn12
Cc1ccc2c(Nc3ccccc3F)nccc2c1NC(=O)c1cnc2c(N)ncnn12
COc1ccc(CNc2ncnc3c(cc(C)cc23)C(=O)Nc2c(C)ccc3c(Nc4cccc(Cl)c4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cc(F)cc23)C(=O)Nc2c(C)ccc3c(Nc4cccc(Cl)c4F)nccc23)c(OC)c1
COC(=O)c1cc(I)cc2c(NCc3ccc(OC)cc3OC)ncnc12
COc1ccc(CNc2ncnc3c(cc(cc23)N2CCN(C)CC2)C(=O)Nc2c(C)ccc3c(Nc4cccc(Cl)c4F)nccc23)c(OC)c1
Cc1ccc2c(Nc3ccc(Cl)cc3F)nccc2c1NC(=O)c1cnc2c(N)ncnn12
COc1ccc(Nc2nccc3c(NC(=O)c4cnc5c(N)ncnn45)c(C)ccc23)cc1Cl
COc1ccc(Nc2nccc3c(NC(=O)c4cccc5c(NCc6ccc(OC)cc6OC)ncnc45)c(C)ccc23)cc1
Cc1ccc2c(Nc3ccc(F)c(Cl)c3)nccc2c1NC(=O)c1cnc2c(N)ncnn12
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4ccc(nc4)N(C)C)nccc23)c(OC)c1
COc1ccc(Nc2nccc3c(NC(=O)c4cccc5c(NCc6ccc(OC)cc6OC)ncnc45)c(C)ccc23)c(F)c1
COc1ccc(Nc2nccc3c(NC(=O)c4cnc5c(N)ncnn45)c(C)ccc23)c(F)c1
CN(C)Cc1ccc(Nc2nccc3c(c(C)ccc23)[N+]([O-])=O)cc1C(F)(F)F
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4ccc(cc4)C(C)=O)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4ccc(Cl)c(CN(C)C)c4)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4ccc(C)cc4)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(nccc23)C(=O)Nc2c(C)ccc3c(Nc4cccc(Cl)c4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4ccc(F)cc4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4ccc(OC)c(OC)c4)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cncc23)C(=O)Nc2c(C)ccc3c(Nc4cccc(Cl)c4F)nccc23)c(OC)c1
Cc1ccc2c(Nc3ccc(Cl)c(F)c3F)nccc2c1NC(=O)c1cnc2c(N)ncnn12
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4ccnc(c4)C(F)(F)F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4cc(F)ccc4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4cc(Cl)ccc4F)nccc23)c(OC)c1
CCOc1ccc(Nc2nccc3c(NC(=O)c4cccc5c(NCc6ccc(OC)cc6OC)ncnc45)c(C)ccc23)c(F)c1
COc1ccc(CNc2ncnc3c(cc(OC)cc23)C(=O)Nc2c(C)ccc3c(Nc4cccc(Cl)c4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4ccc5OCCOc5c4)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4ccc(cc4F)C#N)nccc23)c(OC)c1
Cc1ccc2c(Nc3cccc(Cl)c3F)nccc2c1NC(=O)c1cc(OCCN2CCOCC2)cc2c(N)ncnc12
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4cc(ccc4F)C#N)nccc23)c(OC)c1
Cc1ccc2c(Nc3cccc(Cl)c3F)nccc2c1NC(=O)c1cccc2c(N)ncnc12
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4ccc5CCN(C)Cc5c4)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4cccc(C#N)c4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cc(F)cc23)C(=O)Nc2c(C)ccc3c(Nc4cc(Cl)ccc4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cc(F)cc23)C(=O)Nc2c(C)ccc3c(Nc4ccc(F)cc4F)nccc23)c(OC)c1
Cc1ccc2c(Nc3cccc(Cl)c3F)nccc2c1NC(=O)c1cc(OCCO[Si](C)(C)C(C)(C)C)cc2c(N)ncnc12
COc1ccc(F)c(Nc2nccc3c(NC(=O)c4cccc5c(NCc6ccc(OC)cc6OC)ncnc45)c(C)ccc23)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4ccc(C)cc4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4cc(ccc4F)S(C)(=O)=O)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4cc(F)c(F)cc4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4cc(Br)ccc4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(F)ccc3c(Nc4cccc(Cl)c4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(ccc(F)c23)C(=O)Nc2c(C)ccc3c(Nc4cccc(Cl)c4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4c(F)cc(F)cc4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4c(F)c(F)c(F)c(F)c4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4cccc(OCCN5CCOCC5)c4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cn(C)c23)C(=O)Nc2c(C)ccc3c(Nc4cccc(Cl)c4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4cccc(Cl)c4F)ncnc23)c(OC)c1
Cc1ccc2c(Nc3cccc(Cl)c3F)nccc2c1NC(=O)c1cccc2c(N)nccc12
Cc1ccc2c(Nc3cccc(c3)C(F)(F)F)nccc2c1NC(=O)c1cccc2c(N)nccc12
Cn1cnc2ccc(Oc3c(F)ccc(NS(=O)(=O)N4CC[C@@H](F)C4)c3C#N)cc2c1=O
Cn1cnc2ccc(Oc3c(F)ccc(NS(=O)(=O)N4CC[C@H](F)C4)c3C#N)cc2c1=O
CCCS(=O)(=O)Nc1ccc(F)c(Oc2ccc3ncn(C)c(=O)c3c2)c1C#N
CN(C)S(=O)(=O)Nc1ccc(Cl)c(Oc2ccc3ncn(C)c(=O)c3c2)c1C#N
Cn1cnc2ccc(Oc3c(Cl)ccc(NS(=O)(=O)N4CCCC4)c3C#N)cc2c1=O
CN(C)S(=O)(=O)Nc1ccc(Cl)c(Oc2ccc3ncn(C)c(=O)c3c2)c1F
Cn1cnc2ccc(Oc3c(Cl)ccc(NS(=O)(=O)N4CCCC4)c3F)cc2c1=O
CO[C@@H]1CCN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3C)c2Cl)C1
CCN(C)S(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2Cl)c1Cl
CN(C)S(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2Cl)c1Cl
CCN(C)S(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2F)c1Cl
CO[C@@H]1CCN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3F)c2Cl)C1
CO[C@@H]1CCN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3Cl)c2Cl)C1
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CCCC4)c3Cl)c(F)c2c1=O
CO[C@@H]1CCN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3Br)c2Cl)C1
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC5CC4C5)c3Cl)c(Cl)c2c1=O
CO[C@@H]1CCN(S(=O)(=O)Nc2ccc(F)c(Oc3ccc4ncn(C)c(=O)c4c3C)c2Cl)C1
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CCCC4)c3Cl)c(Br)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CCCC4)c3Cl)c(Cl)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC5CC4C5)c3Cl)c(F)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC[C@@H](F)C4)c3Cl)c(F)c2c1=O
CO[C@@H]1CN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3F)c2Cl)C[C@@H]1F
CO[C@H]1CN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3Br)c2Cl)C[C@H]1F
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC5CC5C4)c3Cl)c(Cl)c2c1=O
CO[C@@H]1CN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3Cl)c2Cl)C[C@@H]1F
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC[C@@H](F)C4)c3Cl)c(Cl)c2c1=O
Cn1cnc2ccc(Oc3c(F)ccc(NS(=O)(=O)N4CC[C@@H](F)C4)c3Cl)c(F)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4C[C@@H](F)[C@@H](F)C4)c3Cl)c(F)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4C[C@@H](F)[C@@H](F)C4)c3Cl)c(Cl)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CCC(F)(F)C4)c3Cl)c(F)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC[C@@H](F)C4)c3Cl)c(Br)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CCC(F)(F)C4)c3Cl)c(Cl)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC[C@@H](OC(F)F)C4)c3Cl)c(F)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC[C@H](F)C4)c3Cl)c(F)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC[C@H](F)C4)c3Cl)c(Cl)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC[C@@H](OC(F)F)C4)c3Cl)c(Cl)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC5CC5C4)c3Cl)c(F)c2c1=O
Cn1cnc2ccc(Nc3c(F)c(F)cc(NS(=O)(=O)N4CCCC4)c3Cl)c(Cl)c2c1=O
CO[C@@H]1CCN(S(=O)(=O)Nc2cc(F)c(F)c(Nc3ccc4ncn(C)c(=O)c4c3Cl)c2Cl)C1
Cn1cnc2ccc(Nc3c(F)c(F)cc(NS(=O)(=O)N4CC[C@@H](F)C4)c3Cl)c(Cl)c2c1=O
CO[C@@H]1CCN(S(=O)(=O)Nc2cc(F)c(F)c(Nc3ccc4ncn(C)c(=O)c4c3Cl)c2F)C1
Cc1c(Nc2c(F)c(F)cc(NS(=O)(=O)N3CC[C@@H](F)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cn1cnc2ccc(Nc3c(F)c(F)cc(NS(=O)(=O)N4CC[C@@H](F)C4)c3F)c(Cl)c2c1=O
CO[C@@H]1CCN(S(=O)(=O)Nc2ccc(F)c(Oc3ccc4ncn(C)c(=O)c4c3Cl)c2Cl)C1
Cn1cnc2ccc(Oc3c(F)ccc(NS(=O)(=O)N4CC[C@@H](F)C4)c3Cl)c(Cl)c2c1=O
Cn1cnc2ccc(Oc3c(F)ccc(NS(=O)(=O)N4CCCC4)c3Cl)c(Cl)c2c1=O
Cn1cnc2ccc(Nc3c(F)c(F)cc(NS(=O)(=O)N4CCCC4)c3Cl)c(F)c2c1=O
Cn1cnc2ccc(Nc3c(F)c(F)cc(NS(=O)(=O)N4CC5CC4C5)c3Cl)c(F)c2c1=O
O=c1c2c(F)c(Nc3c(F)ccc(NS(=O)(=O)N4CCCC4)c3Cl)ccc2ncn1CF
Cn1cnc2ccc(Nc3c(F)c(F)cc(NS(=O)(=O)N4CCCC4)c3F)c(Cl)c2c1=O
Cn1cnc2ccc(Oc3c(F)ccc(NS(=O)(=O)N4CCCC4)c3Cl)c(F)c2c1=O
CCN(C)S(=O)(=O)Nc1cc(F)c(F)c(Nc2ccc3ncn(C)c(=O)c3c2F)c1Cl
Cn1cnc2ccc(Nc3c(F)c(F)cc(NS(=O)(=O)N4CC[C@@H](F)C4)c3Cl)c(F)c2c1=O
CO[C@@H]1CCN(S(=O)(=O)Nc2cc(F)c(F)c(Nc3ccc4ncn(C)c(=O)c4c3F)c2Cl)C1
CO[C@@H]1CCN(S(=O)(=O)Nc2ccc(F)c(Oc3ccc4ncn(C)c(=O)c4c3F)c2Cl)C1
Cn1cnc2ccc(Oc3c(F)ccc(NS(=O)(=O)N4CC5CC4C5)c3Cl)c(F)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CCCC4)c3Cl)c(C#N)c2c1=O
C=Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CCCC3)c2Cl)ccc2ncn(C)c(=O)c12
CCc1c(Nc2c(F)ccc(NS(=O)(=O)N3CCCC3)c2Cl)ccc2ncn(C)c(=O)c12
[2H]C([2H])([2H])O[C@@H]1CCN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3Cl)c2Cl)C1
[2H]C([2H])([2H])O[C@@H]1CCN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3F)c2Cl)C1
[2H]C([2H])([2H])O[C@@H]1CCN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3C)c2Cl)C1
Cn1cnc2ccc(Nc3cc(Cl)cc(NS(=O)(=O)N4CC[C@@H](F)C4)c3F)c(Cl)c2c1=O
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC[C@@H](OC(F)F)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cn1cnc2ccc(Nc3cc(Cl)cc(NS(=O)(=O)N4CC[C@@H](F)C4)c3F)c(F)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4C[C@@H](F)[C@@H](F)C4)c3Cl)c(Cl)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC[C@@H](OC(F)F)C4)c3Cl)c(Cl)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CCC(F)(F)C4)c3Cl)c(Cl)c2c1=O
CC[C@@H]1CCN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3F)c2Cl)C1
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CCC(F)(F)C4)c3Cl)c(F)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4C[C@@H](F)[C@@H](F)C4)c3Cl)c(F)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC5CC5C4)c3Cl)c(F)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC[C@@H](OC(F)F)C4)c3Cl)c(F)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC5CC4C5)c3Cl)c(Cl)c2c1=O
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N(C)C)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N(C)C3CCOC3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N(C)C3CC3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N(C)C3CCC3)c2Cl)ccc2ncn(C)c(=O)c12
COC1CCN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3C)c2Cl)CC1
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CCC(C(F)(F)F)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CCC(O)CC3)c2Cl)ccc2ncn(C)c(=O)c12
CO[C@H]1CN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3C)c2Cl)C[C@@H]1F
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CCOCC3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CCC4CC4C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC4CCC3C4)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CCC4(CC4)C3)c2Cl)ccc2ncn(C)c(=O)c12
CN(C)S(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2F)c1Cl
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CCCCC3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3C[C@H](F)[C@@H](F)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC[C@H](F)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC4CC3C4)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC4CC4(C)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC[C@@H](OC(F)F)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3C[C@@H](F)[C@@H](F)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Oc2c(F)ccc(NS(=O)(=O)N3CC4CC4C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC4CC4C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CCC(F)(F)C3)c2Cl)ccc2ncn(C)c(=O)c12
CCC1CCN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3Cl)c2Cl)C1
Cc1c(Nc2c(F)c(F)cc(NS(=O)(=O)N3C[C@@H](F)[C@@H](F)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)c(F)cc(NS(=O)(=O)N3CCCC3)c2Cl)ccc2ncn(C)c(=O)c12
CCN(C)S(=O)(=O)Nc1cc(F)c(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
Cc1c(Nc2c(F)c(F)cc(NS(=O)(=O)N(C)C)c2Cl)ccc2ncn(C)c(=O)c12
CO[C@@H]1CCN(S(=O)(=O)Nc2cc(F)c(F)c(Nc3ccc4ncn(C)c(=O)c4c3C)c2Cl)C1
CO[C@H]1CN(S(=O)(=O)Nc2cc(F)c(F)c(Nc3ccc4ncn(C)c(=O)c4c3C)c2Cl)C[C@H]1F
Cc1c(Nc2c(F)c(F)cc(NS(=O)(=O)N3CC4CC3C4)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)c(F)cc(NS(=O)(=O)N3CC4CC4C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2cc(Cl)cc(NS(=O)(=O)N3CC[C@@H](F)C3)c2F)ccc2ncn(C)c(=O)c12
Cc1c(Nc2cc(Cl)cc(NS(=O)(=O)N3CCCC3)c2F)ccc2ncn(C)c(=O)c12
CO[C@@H]1CCN(S(=O)(=O)Nc2cc(Cl)cc(Nc3ccc4ncn(C)c(=O)c4c3C)c2F)C1
CC[C@@H]1CCN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3Cl)c2Cl)C1
Cn1cnc2ccc(Oc3c(F)ccc(NS(=O)(=O)N4CC[C@H](F)C4)c3Cl)c(Cl)c2c1=O
Cn1cnc2ccc(Oc3c(F)ccc(NS(=O)(=O)N4CC5CC5C4)c3Cl)c(Cl)c2c1=O
CCN(C)S(=O)(=O)Nc1ccc(F)c(Oc2ccc3ncn(C)c(=O)c3c2Cl)c1Cl
CN(C)S(=O)(=O)Nc1ccc(F)c(Oc2ccc3ncn(C)c(=O)c3c2Cl)c1Cl
CN(C)S(=O)(=O)Nc1ccc(F)c(Oc2ccc3ncn(C)c(=O)c3c2Cl)c1Cl
CCN(C)S(=O)(=O)Nc1ccc(F)c(Oc2ccc3ncn(C)c(=O)c3c2Cl)c1Cl
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CCCC3)c2F)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC[C@@H](F)C3)c2F)ccc2ncn(C)c(=O)c12
COCC1CN(S(=O)(=O)Nc2ccc(F)c(Oc3ccc4ncn(C)c(=O)c4c3C)c2Cl)C1
Cc1c(Oc2c(F)ccc(NS(=O)(=O)N3CC(F)C3)c2Cl)ccc2ncn(C)c(=O)c12
COC1CN(S(=O)(=O)Nc2ccc(F)c(Oc3ccc4ncn(C)c(=O)c4c3C)c2Cl)C1
COCC1CN(S(=O)(=O)Nc2ccc(F)c(Oc3ccc4ncn(C)c(=O)c4c3Cl)c2Cl)C1
COC1CN(S(=O)(=O)Nc2ccc(F)c(Oc3ccc4ncn(C)c(=O)c4c3Cl)c2Cl)C1
Cn1cnc2ccc(Oc3c(F)ccc(NS(=O)(=O)N4CC(F)C4)c3Cl)c(Cl)c2c1=O
COCC1CN(S(=O)(=O)Nc2ccc(F)c(Oc3ccc4ncn(C)c(=O)c4c3F)c2Cl)C1
Cn1cnc2ccc(Oc3c(F)ccc(NS(=O)(=O)N4CC(F)C4)c3Cl)c(F)c2c1=O
COC1CN(S(=O)(=O)Nc2ccc(F)c(Oc3ccc4ncn(C)c(=O)c4c3F)c2Cl)C1
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CCC3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC(F)C3)c2Cl)ccc2ncn(C)c(=O)c12
CN1C=Nc2ccc(c(c2C1=O)Cl)Nc3c(ccc(c3Cl)NS(=O)(=O)N4CC(C4)F)F
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC(F)C4)c3Cl)c(F)c2c1=O
COC1CN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3C)c2Cl)C1
COC1CN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3Cl)c2Cl)C1
COC1CN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3F)c2Cl)C1
COCC1CN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3C)c2Cl)C1
COCC1CN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3Cl)c2Cl)C1
COCC1CN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3F)c2Cl)C1
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC(F)(F)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC(F)(F)C4)c3Cl)c(Cl)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC(F)(F)C4)c3Cl)c(F)c2c1=O
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC(COC(F)F)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC(COC(F)F)C4)c3Cl)c(Cl)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC(COC(F)F)C4)c3Cl)c(F)c2c1=O
COCC1(C)CN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3C)c2Cl)C1
CCOC1CN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3Cl)c2Cl)C1
CCOC1CN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3F)c2Cl)C1
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC(OC(F)F)C4)c3Cl)c(Cl)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC(OC(F)F)C4)c3Cl)c(F)c2c1=O
COCC1(F)CN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3C)c2Cl)C1
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC(C#N)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC(C)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC4C(F)C4C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC4CC4(F)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2cc(F)cc(NS(=O)(=O)N3CCCC3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2cc(F)cc(NS(=O)(=O)N3CC[C@@H](F)C3)c2Cl)ccc2ncn(C)c(=O)c12
CO[C@@H]1CCN(S(=O)(=O)Nc2cc(F)cc(Nc3ccc4ncn(C)c(=O)c4c3C)c2Cl)C1
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CCC4CC43)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2cc(F)cc(NS(=O)(=O)N3CCCC3)c2F)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC(C)(F)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC(COC(F)(F)F)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC4(CCC4)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC5(CCC5)C4)c3Cl)c(Cl)c2c1=O
Cn1cnc2ccc(Nc3c(F)ccc(NS(=O)(=O)N4CC5(CCC5)C4)c3Cl)c(F)c2c1=O
CCOC1CN(S(=O)(=O)Nc2ccc(F)c(Nc3ccc4ncn(C)c(=O)c4c3C)c2Cl)C1
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC(OC(F)F)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC(OC(F)(F)F)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC4(CC4)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1c(Nc2c(F)ccc(NS(=O)(=O)N3CC(COCF)C3)c2Cl)ccc2ncn(C)c(=O)c12
Cn1cnc2ccc(Oc3c(F)ccc(NS(=O)(=O)N4CC5(CCC5)C4)c3C#N)cc2c1=O
N#Cc1c(NS(=O)(=O)N2CC3(CCC3)C2)ccc(F)c1Oc1ccc2ncn(CC(F)(F)F)c(=O)c2c1
N#Cc1c(NS(=O)(=O)N2CC3(CCC3)C2)ccc(F)c1Oc1ccc2ncn(CC(F)F)c(=O)c2c1
N#Cc1c(NS(=O)(=O)N2CC3(CCC3)C2)ccc(F)c1Oc1ccc2ncn(C3CC3)c(=O)c2c1
N#Cc1c(NS(=O)(=O)N2CC3(CCC3)C2)ccc(F)c1Oc1ccc2ncn(CCF)c(=O)c2c1
N#Cc1c(NS(=O)(=O)N2CC3(CCC3)C2)cc(F)c(F)c1Oc1ccc2ncn(CCF)c(=O)c2c1
N#Cc1c(NS(=O)(=O)N2CC3(CC[C@H]3F)C2)ccc(F)c1Oc1ccc2ncn(CC(F)F)c(=O)c2c1