Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 62 hits in this display
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
IC50: 4nMAssay Description:Inhibition of recombinant RET M918T (unknown origin) incubated for 120 mins by Perkin Elmer electrophoretic mobility shift platform methodMore data for this Ligand-Target Pair
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
IC50: 7nMAssay Description:Inhibition of recombinant CCDC6-RET (unknown origin) incubated for 120 mins by Perkin Elmer electrophoretic mobility shift platform methodMore data for this Ligand-Target Pair
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
IC50: 17nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) incubated for 120 mins by Perkin Elmer electrophoretic mobility shift platform methodMore data for this Ligand-Target Pair
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
IC50: 31nMAssay Description:Inhibition of wildtype RET (unknown origin) incubated for 120 mins by Perkin Elmer electrophoretic mobility shift platform methodMore data for this Ligand-Target Pair
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
IC50: 168nMAssay Description:Inhibition of recombinant RET V804L (unknown origin) incubated for 120 mins by Perkin Elmer electrophoretic mobility shift platform methodMore data for this Ligand-Target Pair
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
Kd: <250nMAssay Description:Competition binding assays used herein were developed, validated and performed as described in Fabian et al., Nature Biotechnology 2005, 23, 329-336....More data for this Ligand-Target Pair
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
Kd: <250nMAssay Description:Competition binding assays used herein were developed, validated and performed as described in Fabian et al., Nature Biotechnology 2005, 23, 329-336....More data for this Ligand-Target Pair
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
Kd: <250nMAssay Description:Competition binding assays used herein were developed, validated and performed as described in Fabian et al., Nature Biotechnology 2005, 23, 329-336....More data for this Ligand-Target Pair
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
Kd: 375nMAssay Description:Competition binding assays used herein were developed, validated and performed as described in Fabian et al., Nature Biotechnology 2005, 23, 329-336....More data for this Ligand-Target Pair
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
Kd: <250nMAssay Description:Competition binding assays used herein were developed, validated and performed as described in Fabian et al., Nature Biotechnology 2005, 23, 329-336....More data for this Ligand-Target Pair
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
BDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)
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