1451 SMILES Strings for Sodium channel protein type 10 subunit alpha

Compound Name
SMILES String
Fc1ccc(Oc2ccccc2C(=O)Nc2cc[nH]c(=O)c2)cc1
Fc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1
Fc1ccc(Oc2ccccc2C(=O)Nc2ccc(=O)[nH]c2)cc1
Fc1ccc(Oc2ccc(cc2C(=O)Nc2ccc(=O)[nH]c2)C(F)(F)F)cc1
Fc1ccc(Oc2cc(ccc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1
Fc1ccc(Oc2cc(ccc2C(=O)Nc2ccc(=O)[nH]c2)C(F)(F)F)cc1
Fc1ccc(Oc2cc(ccc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c(F)c1
COCCOc1ccc(Oc2cc(ccc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1
FC(F)(F)c1ccc(C(=O)Nc2cc[nH]c(=O)c2)c(Oc2ccccc2)c1
Cc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
Cc1ccccc1Oc1cc(ccc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
Cc1ccc(Oc2cc(ccc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1
Fc1ccc(Oc2cc(Cl)ccc2C(=O)Nc2cc[nH]c(=O)c2)c(F)c1
Fc1ccc(Oc2cc(Cl)ccc2C(=O)Nc2cc[nH]c(=O)c2)c(Cl)c1
Fc1ccc(Oc2cc(Cl)ccc2C(=O)Nc2cc[nH]c(=O)c2)cc1
COc1cc(F)ccc1Oc1cc(Cl)ccc1C(=O)Nc1cc[nH]c(=O)c1
Cc1cccc(F)c1Oc1cc(Cl)ccc1C(=O)Nc1cc[nH]c(=O)c1
Fc1cccc(Cl)c1Oc1cc(Cl)ccc1C(=O)Nc1cc[nH]c(=O)c1
Fc1cccc(F)c1Oc1cc(Cl)ccc1C(=O)Nc1cc[nH]c(=O)c1
Cc1cc(F)ccc1Oc1cc(Cl)ccc1C(=O)Nc1cc[nH]c(=O)c1
Fc1ccc(Oc2cc(ccc2C(=O)Nc2cc[nH]c(=O)c2)C#N)cc1
COc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1cc[nH]c(=O)c1)C#N
Cc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1cc[nH]c(=O)c1)C#N
Fc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c(F)c1
FC(F)(F)c1ccc(Oc2ccc(cc2)[N+]#[C-])c(c1)C(=O)Nc1cc[nH]c(=O)c1
Fc1cccc(F)c1Oc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
Cc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1
Cc1ccccc1Oc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
Fc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c(Cl)c1
COc1cc(F)ccc1Oc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
Cc1cc(F)ccc1Oc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
FC(F)(F)c1ccc(Oc2ccccc2)c(c1)C(=O)Nc1cc[nH]c(=O)c1
Fc1ccc(Oc2ccc(OC(F)(F)F)cc2C(=O)Nc2cc[nH]c(=O)c2)c(F)c1
Fc1cccc(F)c1Oc1ccc(OC(F)(F)F)cc1C(=O)Nc1cc[nH]c(=O)c1
Cc1ccc(Oc2ccc(OC(F)(F)F)cc2C(=O)Nc2cc[nH]c(=O)c2)cc1
Cc1ccccc1Oc1ccc(OC(F)(F)F)cc1C(=O)Nc1cc[nH]c(=O)c1
Fc1ccc(Oc2ccc(OC(F)(F)F)cc2C(=O)Nc2cc[nH]c(=O)c2)c(Cl)c1
Fc1ccc(Oc2ccc(OC(F)(F)F)cc2C(=O)Nc2cc[nH]c(=O)c2)cc1
Cc1cccc(F)c1Oc1ccc(OC(F)(F)F)cc1C(=O)Nc1cc[nH]c(=O)c1
Cc1cc(F)ccc1Oc1ccc(OC(F)(F)F)cc1C(=O)Nc1cc[nH]c(=O)c1
FC(F)(F)Oc1ccc(Oc2ccccc2)c(c1)C(=O)Nc1cc[nH]c(=O)c1
COc1cc(F)ccc1Oc1ccc(OC(F)(F)F)cc1C(=O)Nc1cc[nH]c(=O)c1
Fc1ccc(Oc2cccc(c2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1
CCOc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1
COc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1
CCOc1ccccc1Oc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
COc1cc(C)ccc1Oc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
COc1cccc(F)c1Oc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
Cc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c(Cl)c1
Cc1cc(Cl)ccc1Oc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
Fc1cc(Cl)ccc1Oc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
COc1ccc(F)cc1Oc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
CCCOc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1
COc1c(F)cccc1Oc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
COc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c(F)c1
Cc1ccc(F)cc1Oc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
COc1cc(F)cc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c1
FC(F)(F)c1ccc(Oc2ccc(Cl)cc2)c(c1)C(=O)Nc1cc[nH]c(=O)c1
COc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1F
Cc1cc(F)ccc1Oc1ccc(cc1C(=O)Nc1cc(Cl)[nH]c(=O)c1)C(F)(F)F
Cc1cc(NC(=O)c2cc(ccc2Oc2ccc(F)cc2C)C(F)(F)F)cc(=O)[nH]1
CCCOc1ccccc1Oc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
COc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c(C)c1
CC(C)Oc1ccccc1Oc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
FC(F)(F)c1ccc(Oc2ccccc2Cl)c(c1)C(=O)Nc1cc[nH]c(=O)c1
Fc1ccc(Oc2ccc(Cl)cc2C(=O)Nc2cc[nH]c(=O)c2)c(Cl)c1
Fc1ccc(Oc2ccc(Cl)cc2C(=O)Nc2cc[nH]c(=O)c2)cc1
Cc1cc(F)ccc1Oc1ccc(Cl)cc1C(=O)Nc1cc[nH]c(=O)c1
Fc1ccc(Oc2ccc(Cl)cc2C(=O)Nc2cc[nH]c(=O)c2)c(F)c1
COc1cc(C)ccc1Oc1ccc(Cl)cc1C(=O)Nc1cc[nH]c(=O)c1
COc1ccc(Oc2ccc(Cl)cc2C(=O)Nc2cc[nH]c(=O)c2)cc1F
FC(F)(F)Oc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1
FC(F)Oc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1
FC(F)(F)c1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1
FC(F)(F)Oc1ccccc1Oc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
FC(F)Oc1ccccc1Oc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
Fc1ccc(Oc2cc(ccc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c(Cl)c1
FC(F)(F)c1ccc(C(=O)Nc2cc[nH]c(=O)c2)c(Oc2ccc(Cl)cc2)c1
FC(F)(F)c1ccc(Oc2cc(ccc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1
FC(F)(F)Oc1ccccc1Oc1cc(ccc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
COc1ccc(Oc2cc(ccc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1F
FC(F)Oc1ccc(Oc2cc(ccc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1
FC(F)Oc1ccccc1Oc1cc(ccc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
COc1ccc(Oc2cc(ccc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c(F)c1
OCCn1ccc(NC(=O)c2ccc(cc2Oc2ccc(F)cc2)C(F)(F)F)cc1=O
Cc1c[nH]c(=O)cc1NC(=O)c1ccc(cc1Oc1ccc(F)cc1C)C(F)(F)F
COc1c(F)cccc1Oc1cc(ccc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
Fc1ccc(Oc2cc(ccc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)C(F)(F)F)cc1
COc1ccc(Oc2cc(ccc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)C(F)(F)F)cc1F
Fc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c(F)c1F
Cc1cc(C)c(C)c(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c1
Cc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c(F)c1F
Cc1cc(C)c(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1C
Cc1cc(C)c(C)c(Oc2ccc(F)cc2C(=O)Nc2cc[nH]c(=O)c2)c1
Fc1ccc(Oc2ccccc2)c(c1)C(=O)Nc1cc[nH]c(=O)c1
Fc1ccc(Oc2ccc(cc2)C2CC2)c(c1)C(=O)Nc1cc[nH]c(=O)c1
CC(C)(C)Oc1ccc(Oc2ccc(F)cc2C(=O)Nc2cc[nH]c(=O)c2)cc1
CCOc1ccc(Oc2ccc(F)cc2C(=O)Nc2cc[nH]c(=O)c2)cc1
CC(C)c1ccc(Oc2ccc(F)cc2C(=O)Nc2cc[nH]c(=O)c2)cc1
CCCOc1ccc(Oc2ccc(F)cc2C(=O)Nc2cc[nH]c(=O)c2)cc1
Fc1ccc(Oc2ccc(OC(F)(F)F)cc2)c(c1)C(=O)Nc1cc[nH]c(=O)c1
COCCc1ccc(Oc2ccc(F)cc2C(=O)Nc2cc[nH]c(=O)c2)cc1
COc1ccc(Oc2ccc(F)cc2C(=O)Nc2cc[nH]c(=O)c2)c(Cl)c1
COc1ccc(Oc2ccc(F)cc2C(=O)Nc2cc[nH]c(=O)c2)cc1
Cc1cc(C)c(Oc2ccc(F)cc2C(=O)Nc2cc[nH]c(=O)c2)cc1C
Fc1ccc(Oc2ccc(OCC(F)(F)F)cc2)c(c1)C(=O)Nc1cc[nH]c(=O)c1
Fc1ccc(Oc2ccc(OCC3CC3)cc2)c(c1)C(=O)Nc1cc[nH]c(=O)c1
Fc1ccc(Oc2cc(Cl)c(F)cc2C(=O)Nc2cc[nH]c(=O)c2)c(Cl)c1
COc1ccc(Oc2cc(ccc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c(Cl)c1F
COc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)C(F)(F)F
Cc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)C(F)(F)F
Fc1ccc(Oc2cc(Cl)c(Cl)cc2C(=O)Nc2cc[nH]c(=O)c2)cc1
COc1cc(F)ccc1Oc1cc(Cl)c(Cl)cc1C(=O)Nc1cc[nH]c(=O)c1
COc1ccc(Oc2cc(Cl)c(Cl)cc2C(=O)Nc2cc[nH]c(=O)c2)cc1F
CC(C)CCOc1cc(ccc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
CC(C)COc1cc(ccc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
FC(F)(F)c1ccc(C(=O)Nc2cc[nH]c(=O)c2)c(OC2C[C@H]3CCC2C3)c1 |r,TLB:19:20:26:24.23|
CC1(COc2cc(ccc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)CC1
FC(F)(F)c1ccc(C(=O)Nc2cc[nH]c(=O)c2)c(OCC2CCCC2)c1
FC(F)(F)c1ccc(C(=O)Nc2cc[nH]c(=O)c2)c(OCC2CCOC2)c1
FC(F)(F)c1ccc(C(=O)Nc2cc[nH]c(=O)c2)c(OC2CCC2)c1
FC(F)(F)CCCOc1cc(ccc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
CC1(C)CC1COc1cc(ccc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
FC(F)(F)c1ccc(C(=O)Nc2cc[nH]c(=O)c2)c(OC2C[C@@H]3C[C@@H]3C2)c1 |r|
FC(F)(F)c1ccc(C(=O)Nc2cc[nH]c(=O)c2)c(OCC2CC2(F)F)c1
FC(F)(F)c1ccc(C(=O)Nc2cc[nH]c(=O)c2)c(OC2CC3CCC2C3)c1 |TLB:19:20:26:24.23|
FC(F)(F)c1ccc(C(=O)Nc2cc[nH]c(=O)c2)c(OC2CCCCC2)c1
FC(F)(F)CCCOc1cc(Cl)ccc1C(=O)Nc1cc[nH]c(=O)c1
FC(F)(F)c1ccc(OCC2CCCC2)c(c1)C(=O)Nc1cc[nH]c(=O)c1
CC(C)COc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
FC(F)(F)CCOc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
FC(F)(F)CCCOc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
CC1(C)CC1COc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
FC(F)(F)c1ccc(OC2C[C@@H]3C[C@@H]3C2)c(c1)C(=O)Nc1cc[nH]c(=O)c1 |r|
FC(F)(F)Oc1ccc(OCC2CCCC2)c(c1)C(=O)Nc1cc[nH]c(=O)c1
FC(F)(F)Oc1ccc(OC2CCCCC2)c(c1)C(=O)Nc1cc[nH]c(=O)c1
FC(F)(F)CCOc1ccc(OC(F)(F)F)cc1C(=O)Nc1cc[nH]c(=O)c1
FC(F)(F)CCCOc1ccc(OC(F)(F)F)cc1C(=O)Nc1cc[nH]c(=O)c1
CC(C)(C)c1ccc(C(=O)Nc2cc[nH]c(=O)c2)c(Oc2ccc(nc2)C(F)(F)F)c1
CC(C)(C)c1ccc(C(=O)Nc2ccc(=O)[nH]c2)c(Oc2ccc(nc2)C(F)(F)F)c1
FC(F)(F)c1ccc(Oc2cc(Cl)ccc2C(=O)Nc2cc[nH]c(=O)c2)cn1
FC(F)(F)c1ccc(C(=O)Nc2cc[nH]c(=O)c2)c(Oc2ccc(nc2)C(F)(F)F)c1
FC(F)(F)c1ccc(C(=O)Nc2ccc(=O)[nH]c2)c(Oc2ccc(nc2)C(F)(F)F)c1
Cc1ccc(Oc2cc(ccc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cn1
Cc1ncccc1Oc1cc(ccc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
Cn1ccc(NC(=O)c2ccc(cc2Oc2ccc(nc2)C(F)(F)F)C(C)(C)C)cc1=O
Cn1cc(NC(=O)c2ccc(cc2Oc2ccc(nc2)C(F)(F)F)C(C)(C)C)ccc1=O
Cc1ncccc1Oc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
Cc1ncccc1Oc1ccc(OC(F)(F)F)cc1C(=O)Nc1cc[nH]c(=O)c1
Fc1ccc(Oc2cc(cc(c2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)C(F)(F)F)c(F)c1
Cc1cc(F)ccc1Oc1cc(cc(c1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F)C(F)(F)F
COc1cc(F)ccc1Oc1cc(cc(c1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F)C(F)(F)F
Fc1ccc(Oc2cc(cc(c2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)C(F)(F)F)cc1
FC(F)(F)c1cc(Oc2ccccc2)c(C(=O)Nc2cc[nH]c(=O)c2)c(c1)C(F)(F)F
OCc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
COc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
Oc1ccc(F)cc1COc1cc(ccc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
Fc1ccc(Oc2ccc(OCCCC(F)(F)F)cc2)c(c1)C(=O)Nc1cc[nH]c(=O)c1
COCCOc1ccc(Oc2cc(CF)ccc2C(=O)Nc2cc[nH]c(=O)c2)cc1
FC(F)(F)c1ccc(Oc2ccc(cc2)C#N)c(c1)C(=O)Nc1cc[nH]c(=O)c1
COc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c(Cl)c1
Cc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c(C)c1
COc1cc(F)ccc1Oc1ccc(Cl)cc1C(=O)Nc1cc[nH]c(=O)c1
FC(F)(F)Oc1ccc(Oc2cc(ccc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1
FC(F)(F)c1ccc(C(=O)Nc2cc[nH]c(=O)c2)c(OCC2CCCO2)c1
CC1(C)CC1COc1ccc(OC(F)(F)F)cc1C(=O)Nc1cc[nH]c(=O)c1
Oc1ccc(F)c(Oc2cc(ccc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c1
NS(=O)(=O)c1cccc(NC(=O)c2nc3ccccc3nc2Oc2ccc(F)cc2)c1
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1cccc(c1)S(N)(=O)=O
NS(=O)(=O)c1cccc(NC(=O)c2nc3ccccc3nc2Oc2ccc(OC(F)(F)F)cc2)c1
COc1ccc(Oc2nc3ccccc3nc2C(=O)Nc2cccc(c2)S(N)(=O)=O)c(Cl)c1
NS(=O)(=O)c1cccc(NC(=O)c2nc3ccccc3nc2Oc2ccc(F)cc2F)c1
NS(=O)(=O)c1cccc(NC(=O)c2nc3ccccc3nc2Oc2ccc(F)cc2Cl)c1
COc1ccc(Oc2nc3ccccc3nc2C(=O)Nc2cccc(c2)S(N)(=O)=O)cc1F
COc1ccc(Oc2nc3ccccc3nc2C(=O)Nc2cccc(c2)S(N)(=O)=O)c(OC)c1
Cc1cc(Cl)ccc1Oc1nc2ccccc2nc1C(=O)Nc1cccc(c1)S(N)(=O)=O
NS(=O)(=O)c1cccc(NC(=O)c2nc3ccccc3nc2Oc2ccccc2OC(F)F)c1
COc1cc(Cl)ccc1Oc1nc2ccccc2nc1C(=O)Nc1cccc(c1)S(N)(=O)=O
COc1ccc(Oc2nc3ccccc3nc2C(=O)Nc2cccc(c2)S(N)(=O)=O)c(F)c1
NS(=O)(=O)c1cccc(NC(=O)c2nc3ccccc3nc2Oc2ccccc2)c1
Cc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1cccc(c1)S(N)(=O)=O
NS(=O)(=O)c1cccc(NC(=O)c2nc3ccccc3nc2Oc2ccc(OCC(F)(F)F)cc2)c1
CNS(=O)(=O)c1cccc(NC(=O)c2nc3ccccc3nc2Oc2ccc(F)cc2OC)c1
OC(=O)c1ccc(NC(=O)c2nc3ccccc3nc2Oc2ccc(OC(F)(F)F)cc2)cc1
OC(=O)c1ccc(NC(=O)c2nc3ccccc3nc2Oc2ccc(F)cc2)cn1
Cc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1ccc(nc1)C(O)=O
OC(=O)c1ccc(NC(=O)c2nc3ccccc3nc2Oc2ccccc2)cn1
COc1ccc(Oc2nc3ccccc3nc2C(=O)Nc2ccc(nc2)C(O)=O)c(F)c1
OC(=O)c1ccc(NC(=O)c2nc3ccccc3nc2Oc2ccc(OCC(F)(F)F)cc2)cn1
COc1cc(Cl)ccc1Oc1nc2ccccc2nc1C(=O)Nc1ccc(nc1)C(O)=O
OC(=O)c1ccc(NC(=O)c2nc3ccccc3nc2Oc2ccccc2OC(F)F)cn1
Cc1cc(Cl)ccc1Oc1nc2ccccc2nc1C(=O)Nc1ccc(nc1)C(O)=O
COc1ccc(Oc2nc3ccccc3nc2C(=O)Nc2ccc(nc2)C(O)=O)c(OC)c1
COc1ccc(Oc2nc3ccccc3nc2C(=O)Nc2ccc(nc2)C(O)=O)cc1F
OC(=O)c1ccc(NC(=O)c2nc3ccccc3nc2Oc2ccc(F)cc2Cl)cn1
OC(=O)c1ccc(NC(=O)c2nc3ccccc3nc2Oc2ccc(F)cc2F)cn1
COc1ccc(Oc2nc3ccccc3nc2C(=O)Nc2ccc(nc2)C(O)=O)c(Cl)c1
OC(=O)c1ccc(NC(=O)c2nc3ccccc3nc2Oc2ccc(OC(F)(F)F)cc2)cn1
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1ccc(nc1)C(O)=O
OC(=O)c1cc(NC(=O)c2nc3ccccc3nc2Oc2ccc(OC(F)(F)F)cc2)ccn1
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1ccnc(c1)C(O)=O
Fc1ccc(Oc2nc3ccccc3nc2C(=O)Nc2cc[nH]c(=O)c2)cc1
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1cccc(c1)C(O)=O
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1nc(cs1)C(O)=O
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1nc[nH]n1
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1nc(co1)C(O)=O
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1cc[nH]n1
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1nnn[nH]1
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1ccc2[nH]nnc2c1
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1cn[nH]c1
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1ccc2[nH]c(CO)nc2c1
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1cccc(c1)-c1nnn[nH]1
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1cccc(c1)S(C)(=O)=O
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1ccc2cn[nH]c2c1
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1ccc2[nH]ncc2c1
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1ccc2nc[nH]c2c1
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1cc(ccn1)C#N
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1ccc(nc1)C#N
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1ccc(cn1)C#N
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1ccncc1
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1cccnc1
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1ccc(cc1)C#N
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1cccc(c1)C#N
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1ccc2[nH]c(=O)[nH]c2c1
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1ccc(cc1)C(N)=O
COc1cc(F)ccc1Oc1nc2ccccc2nc1C(=O)Nc1cccc(c1)C(N)=O
NS(=O)(=O)c1cccc(NC(=O)c2cc3ccccc3nc2Oc2ccc(F)cc2)c1
COc1cc(F)ccc1Oc1nc2ccccc2cc1C(=O)Nc1cccc(c1)S(N)(=O)=O
COc1ccc(Oc2nc3ccccc3cc2C(=O)Nc2cccc(c2)S(N)(=O)=O)cc1F
Cc1cc(F)ccc1Oc1nc2ccccc2cc1C(=O)Nc1cccc(c1)S(N)(=O)=O
NS(=O)(=O)c1cccc(NC(=O)c2cc3ccccc3nc2Oc2ccccc2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc3ccccc3nc2Oc2ccc(F)cc2F)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc3ccccc3nc2Oc2ccc(F)cc2Cl)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc3ccccc3nc2Oc2ccc(OCC(F)(F)F)cc2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc3ccccc3nc2Oc2ccc(OC(F)(F)F)cc2)c1
COc1ccc(Oc2nc3ccccc3cc2C(=O)Nc2cccc(c2)S(N)(=O)=O)c(Cl)c1
COc1ccc(Oc2nc3ccccc3cc2C(=O)Nc2cccc(c2)S(N)(=O)=O)c(F)c1
Cc1cc(Cl)ccc1Oc1nc2ccccc2cc1C(=O)Nc1cccc(c1)S(N)(=O)=O
COc1ccc(Oc2nc3ccccc3cc2C(=O)Nc2cccc(c2)S(N)(=O)=O)c(OC)c1
COc1cc(Cl)ccc1Oc1nc2ccccc2cc1C(=O)Nc1cccc(c1)S(N)(=O)=O
NS(=O)(=O)c1cccc(NC(=O)c2cc3ccccc3nc2Oc2ccccc2OC(F)F)c1
OC(=O)c1ccc(NC(=O)c2cc3ccccc3nc2Oc2ccc(F)cc2F)cc1
Cc1cc(F)ccc1Oc1nc2ccccc2cc1C(=O)Nc1ccc(cc1)C(O)=O
OC(=O)c1ccc(NC(=O)c2cc3ccccc3nc2Oc2ccccc2OC(F)F)cc1
COc1ccc(Oc2nc3ccccc3cc2C(=O)Nc2ccc(cc2)C(O)=O)c(OC)c1
OC(=O)c1ccc(NC(=O)c2cc3ccccc3nc2Oc2ccc(F)cc2Cl)cn1
OC(=O)c1ccc(NC(=O)c2cc3ccccc3nc2Oc2ccc(F)cc2F)cn1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCCC2)C1=O
NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)OC(=O)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)COC(=O)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)CC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@H]1CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@H]1CCN(C1)C(=O)CN1CC(=O)N(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1C(=O)CN(Cc2ccccn2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CC2)C1=O
C[C@H]1CCCN1C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
FC1CCCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2C[C@H]3C[C@@H]2CO3)C1=O |TLB:21:23:28.29:26|
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2cocn2)C1=O
Cc1noc(C)c1CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2ncco2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN([C@@H]2CCOC2)C1=O
CC(N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F)c1nc(C)no1
CCOc1nnc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)s1
Cc1nc(CN2CCCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)oc1C
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2nnc(o2)C2CC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(Cc2nnc(o2)C2CCC2)C1=O
CCS(=O)(=O)N1CC(C1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
O[C@@H]1CCCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@@H]1CCCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@H]1CCCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N[C@@H]2CCOC2)C1=O
Cc1cccc(c1)-n1ncc2c(cccc12)N1CCN(CC(=O)N2CC[C@H](F)C2)C1=O
FC1CCN(CC1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NCC2CCOC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N[C@H]2CCOC2)C1=O
F[C@H]1CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1cccc(OC(F)(F)F)c1
CCN(CC)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CC3(COC3)C2)C1=O
CCC1(O)CN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CCCS(=O)(=O)N1CC(C1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN([C@H]2CCCC[C@@H]2OCc2ccccc2)C1=O
O[C@H]1CCCC[C@@H]1N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CO[C@H]1CCCC[C@@H]1N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)CO[C@H]1CCCC[C@@H]1N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN([C@H]2CCCCC2=O)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C2CN(C2)S(=O)(=O)CC2CC2(Cl)Cl)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C2CN(C2)S(=O)(=O)CC2CC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(C2CN(C2)S(=O)(=O)CC(F)(F)F)C1=O
CC(C)CS(=O)(=O)N1CC(C1)N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)(C)OC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CCOC(=O)C=CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F |w:6.6|
CCOC(=O)\C=C\N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)(C)OC(=O)CCN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
O[C@H]1CCCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
OC1CN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@H]1CCN(C1)C(=O)CCN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCOCC2)C1=O
F[C@H]1CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)C1CCCCC1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCCCC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCCC(F)(F)C2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCC(F)(F)CC2)C1=O
FC1CN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCC(CC2)C(F)(F)F)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCCC(C2)C(F)(F)F)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2C[C@@H]3CC[C@H](C2)O3)C1=O |TLB:21:23:27.26:30|
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCC(=O)C2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCCCCC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NCC(F)(F)F)C1=O
CC(C)(C)CCn1ncc2c(cccc12)N1CCN(CC(=O)N2CCCC2)C1=O
CC(C)(C)n1ncc2c(cccc12)N1CCN(CC(=O)N2CC[C@H](F)C2)C1=O
F[C@H]1CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CC[C@@H](C2)C(F)(F)F)C1=O
CC1(F)CN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CC(F)(F)C2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2[C@H]3CC[C@@H]2CC(=O)C3)C1=O |THB:30:29:23:25.26|
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CC(F)(F)C(F)(F)C2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CCCC(=O)CC2)C1=O
F[C@H]1CCN(C1)C(=O)C=CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F |w:9.10|
CCNC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
OCC1(CCC1)NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@@H]1CCCN(C1)C(=O)CCN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@H]1CCCN(C1)C(=O)CCN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
COC1CN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CCOCC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2COC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CCC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CCCC2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CCCCC2)C1=O
CC(=O)C1CN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CO[C@H]1C[C@@H](C1)NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F |r,wU:2.1,wD:4.6,(4.2,14.09,;5.11,12.85,;4.48,11.44,;5.03,10,;3.6,9.45,;3.04,10.89,;2.97,8.05,;3.88,6.8,;5.41,6.96,;3.25,5.39,;4.15,4.15,;5.69,4.15,;6.17,2.68,;4.92,1.78,;3.68,2.68,;2.21,2.21,;4.92,.24,;6.26,-.53,;6.26,-2.07,;4.92,-2.84,;3.59,-2.07,;2.13,-2.55,;1.22,-1.3,;2.13,-.06,;3.59,-.53,;1.65,-4.01,;2.68,-5.16,;2.2,-6.62,;.7,-6.94,;-.33,-5.8,;.14,-4.33,;-.89,-3.19,)|
CC1(C)CC1NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2CC(C2)C(F)(F)F)C1=O
CC(C)O[C@H]1CCCC[C@@H]1N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
O[C@H]1CCC[C@H]1NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC1(CC1)NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N[C@H]2CCC[C@@H]2OCc2ccccc2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N[C@@H]2CCC[C@H]2OCc2ccccc2)C1=O
CC(C)COC1COCC1N1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)CO[C@H]1CCC[C@H]1NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
F[C@H]1CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccc(Cl)cc1
CC(C)(C)NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CCCC(F)(F)C2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CCC(F)(F)C2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)N2C[C@@H]3CCC[C@@H]3C2)C1=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NCCC(F)(F)F)C1=O
CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
NC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC(C)[C@H](N(C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F)C(C)(C)C)C(N)=O
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CCCC2(F)F)C1=O
F[C@H]1CCN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1cc(Cl)cc(Cl)c1
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2CC(=O)C2)C1=O
OC1CC(C1)NC(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F |(5.11,12.85,;4.48,11.44,;3.04,10.89,;3.6,9.45,;5.03,10,;2.97,8.05,;3.88,6.8,;5.41,6.96,;3.25,5.39,;4.15,4.15,;5.69,4.15,;6.17,2.68,;4.92,1.78,;3.68,2.68,;2.21,2.21,;4.92,.24,;6.26,-.53,;6.26,-2.07,;4.92,-2.84,;3.59,-2.07,;2.13,-2.55,;1.22,-1.3,;2.13,-.06,;3.59,-.53,;1.65,-4.01,;2.68,-5.16,;2.2,-6.62,;.7,-6.94,;-.33,-5.8,;.14,-4.33,;-.89,-3.19,)|
CN(C1CCC1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
CC1CN(C1)C(=O)CN1CCN(C1=O)c1cccc2n(ncc12)-c1ccccc1F
Fc1ccccc1-n1ncc2c(cccc12)N1CCN(CC(=O)NC2(CCC2)C(F)(F)F)C1=O
[#8]\[#7]=[#6]-1/[#6]-[#6](-[#6]-1)-[#7]-[#6](=O)-[#6]-[#7]-1-[#6]-[#6]-[#7](-[#6]-1=O)-c1cccc2n(ncc12)-c1ccccc1F
[#6]-[#8]\[#7]=[#6]-1/[#6]-[#6](-[#6]-1)-[#7]-[#6](=O)-[#6]-[#7]-1-[#6]-[#6]-[#7](-[#6]-1=O)-c1cccc2n(ncc12)-c1ccccc1F
CN(C)CCON=C(C=Cc1ccc(O)cc1)c1ccccc1F |w:6.5,8.7|
NC(SCCCc1cnc[nH]1)=NCCc1ccc(I)cc1 |w:11.12|
S=C(NC1CCCCC1)N1CCC(CC1)c1cnc[nH]1
Cc1nc2C(O)CCCn2c(=O)c1CCN1CCC(CC1)c1noc2cc(F)ccc12
CN1CCN(CC1)C1=c2ccccc2=Nc2ccc(Cl)cc2N1 |c:8,15|
Fc1ccc(cc1)C(CCCN1CCC2(CC1)N(CNC2=O)c1ccccc1)c1ccc(F)cc1
c1cc(ccc1C(=O)CCCN2CCC(CC2)(c3ccc(cc3)Cl)O)F
CN1CCN(CC1)C1=c2cc(C)sc2=Nc2ccccc2N1 |c:8,15|
CN1CC2C(C1)c1cc(Cl)ccc1Oc1ccccc21
c1cc(ccc1C(CCCN2CCC(CC2)(c3ccc(c(c3)C(F)(F)F)Cl)O)c4ccc(cc4)F)F
NC(=O)C1(CCN(CCCC(=O)c2ccc(F)cc2)CC1)N1CCCCC1
OCCOCCN1CCN(CC1)C1=Nc2ccccc2Sc2ccccc12 |t:13|
CC1=C(C(=O)N2CCCCC2=N1)CCN3CCC(CC3)c4c5ccc(cc5on4)F
Fc1ccc(cc1)-n1cc(C2CCN(CCN3CCNC3=O)CC2)c2cc(Cl)ccc12
c1ccc2c(c1)c(ns2)N3CCN(CC3)CCc4cc5c(cc4Cl)NC(=O)C5
CN(C)CCOC1=Cc2ccccc2Sc3c1cc(cc3)Cl
CCN1CCCC1CNC(=O)c1cc(c(N)cc1OC)S(=O)(=O)CC
COCCCN1CCC(CC1)NC(=O)c1cc(Cl)c(N)c2CCOc12
OC(=O)c1ccc(NC(=O)c2ccc(cc2Oc2ccc(F)cc2Cl)C(F)(F)C(F)(F)F)cc1
OC(=O)c1ccc(NC(=O)c2ccc(cc2Oc2ccc(F)cc2F)C(F)(F)C(F)(F)F)cc1
Cc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1ccc(cc1)C(O)=O)C(F)(F)C(F)(F)F
OC(=O)c1ccc(NC(=O)c2ccc(cc2Oc2ccc(F)cc2Cl)C(F)(F)F)cc1
Cc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1ccc(cc1)C(O)=O)C(F)(F)F
OC(=O)c1ccc(NC(=O)c2ccc(cc2Oc2ccc(F)cc2F)C(F)(F)F)cc1
OC(=O)c1ccc(NC(=O)c2ccc(cc2Oc2ccc(OC(F)(F)F)cc2)C(F)(F)F)cc1
OC(=O)c1ccc(NC(=O)c2c(Oc3ccc(F)cc3F)cc(cc2C(F)(F)F)C(F)(F)F)cc1
Cc1cc(F)ccc1Oc1cc(cc(c1C(=O)Nc1ccc(cc1)C(O)=O)C(F)(F)F)C(F)(F)F
COc1cc(F)ccc1Oc1cc(cc(c1C(=O)Nc1ccc(cc1)C(O)=O)C(F)(F)F)C(F)(F)F
OC(=O)c1ccc(NC(=O)c2c(Oc3ccc(F)cc3)cc(cc2C(F)(F)F)C(F)(F)F)cc1
COc1cc(F)ccc1Oc1cc(Cl)c(Cl)cc1C(=O)Nc1ccc(cc1)C(O)=O
OC(=O)c1ccc(NC(=O)c2cc(Cl)c(Cl)cc2Oc2ccc(F)cc2)cc1
Cc1cc(F)ccc1Oc1cc(Cl)c(Cl)cc1C(=O)Nc1ccc(cc1)C(O)=O
OC(=O)c1ccc(NC(=O)c2cc(Cl)c(Cl)cc2Oc2ccccc2)cc1
OCc1ccc(Oc2cc(Cl)c(Cl)cc2C(=O)Nc2ccc(cc2)C(O)=O)c(F)c1
OC(=O)c1ccc(NC(=O)c2cc(Cl)c(Cl)cc2Oc2ccc(OCC(F)(F)F)cc2)cc1
COc1cc(Cl)ccc1Oc1cc(Cl)c(Cl)cc1C(=O)Nc1ccc(cc1)C(O)=O
OC(=O)c1ccc(NC(=O)c2cc(Cl)c(Cl)cc2Oc2ccccc2OC(F)F)cc1
Cc1cc(Cl)ccc1Oc1cc(Cl)c(Cl)cc1C(=O)Nc1ccc(cc1)C(O)=O
COc1cc(CO)ccc1Oc1cc(Cl)c(Cl)cc1C(=O)Nc1ccc(cc1)C(O)=O
OCc1ccc(Oc2cc(Cl)c(Cl)cc2C(=O)Nc2ccc(cc2)C(O)=O)cc1F
OC(=O)c1ccc(NC(=O)c2cc(Cl)c(Cl)cc2Oc2ccc(F)cc2Cl)cc1
OC(=O)c1ccc(NC(=O)c2cc(Cl)c(Cl)cc2Oc2ccc(F)cc2F)cc1
OCc1ccc(Oc2cc(Cl)c(Cl)cc2C(=O)Nc2ccc(cc2)C(O)=O)c(Cl)c1
OC(=O)c1ccc(NC(=O)c2cc(Cl)c(Cl)cc2Oc2ccc(OC(F)(F)F)cc2)cc1
COc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1ccc(cc1)C(O)=O)C(F)(F)C(F)(F)F
Cc1cc(F)ccc1Oc1ccc(cc1C(=O)Nc1ccc(cc1)C(O)=O)C(F)(F)F
OC(=O)c1ccc(NC(=O)c2cc(Cl)c(Cl)cc2Oc2ccc(F)cc2)cn1
CC(C)CCOc1ccc(Oc2cc(Cl)c(Cl)cc2C(=O)Nc2ccc(nc2)C(O)=O)cc1
Cc1cc(F)ccc1Oc1cc(Cl)c(Cl)cc1C(=O)Nc1ccc(nc1)C(O)=O
OC(=O)c1ccc(NC(=O)c2cc(Cl)c(Cl)cc2Oc2ccccc2)cn1
OCc1ccc(Oc2cc(Cl)c(Cl)cc2C(=O)Nc2ccc(nc2)C(O)=O)c(F)c1
OC(=O)c1ccc(NC(=O)c2cc(Cl)c(Cl)cc2Oc2ccc(OCC(F)(F)F)cc2)cn1
COc1cc(Cl)ccc1Oc1cc(Cl)c(Cl)cc1C(=O)Nc1ccc(nc1)C(O)=O
OC(=O)c1ccc(NC(=O)c2cc(Cl)c(Cl)cc2Oc2ccccc2OC(F)F)cn1
Cc1cc(Cl)ccc1Oc1cc(Cl)c(Cl)cc1C(=O)Nc1ccc(nc1)C(O)=O
COc1cc(CO)ccc1Oc1cc(Cl)c(Cl)cc1C(=O)Nc1ccc(nc1)C(O)=O
OCc1ccc(Oc2cc(Cl)c(Cl)cc2C(=O)Nc2ccc(nc2)C(O)=O)cc1F
OC(=O)c1ccc(NC(=O)c2cc(Cl)c(Cl)cc2Oc2ccc(F)cc2Cl)cn1
OC(=O)c1ccc(NC(=O)c2cc(Cl)c(Cl)cc2Oc2ccc(F)cc2F)cn1
OCc1ccc(Oc2cc(Cl)c(Cl)cc2C(=O)Nc2ccc(nc2)C(O)=O)c(Cl)c1
OC(=O)c1ccc(NC(=O)c2cc(Cl)c(Cl)cc2Oc2ccc(OC(F)(F)F)cc2)cn1
COc1ccccc1Oc1cc(cc(c1C(=O)Nc1ccc(nc1)C(O)=O)C(F)(F)F)C(F)(F)F
OCc1ccc(Oc2cc(cc(c2C(=O)Nc2ccc(nc2)C(O)=O)C(F)(F)F)C(F)(F)F)cc1
Cc1cc(F)ccc1Oc1cc(cc(c1C(=O)Nc1ccc(nc1)C(O)=O)C(F)(F)F)C(F)(F)F
COc1cc(F)ccc1Oc1cc(cc(c1C(=O)Nc1ccc(nc1)C(O)=O)C(F)(F)F)C(F)(F)F
COc1cc(CO)ccc1Oc1cc(cc(c1C(=O)Nc1ccc(nc1)C(O)=O)C(F)(F)F)C(F)(F)F
OC(=O)c1ccc(NC(=O)c2c(Oc3ccc(F)cc3)cc(cc2C(F)(F)F)C(F)(F)F)cn1
COc1cc(F)ccc1Oc1cc(Cl)c(Cl)cc1C(=O)Nc1ccc(nc1)C(O)=O
COc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1ccc(nc1)C(O)=O)C(C)(C)C
Cc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1ccc(nc1)C(O)=O)C(C)(C)C
CC(C)(C)c1ccc(C(=O)Nc2ccc(nc2)C(O)=O)c(Oc2ccc(F)cc2)c1
OC(=O)c1ccc(NC(=O)c2ccccc2Oc2ccc(F)cc2)cn1
OC(=O)c1ccc(NC(=O)c2ccc(cc2Oc2ccc(F)cc2)C(F)(F)F)cn1
COc1cc(F)ccc1Oc1ccc(cc1C(=O)Nc1ccc(nc1)C(O)=O)C(F)(F)F
OC(=O)c1ccc(NC(=O)c2cc(ccc2Oc2ccc(F)cc2Cl)C(F)(F)F)cn1
COc1ccc(F)cc1Oc1ccc(cc1C(=O)Nc1ccc(nc1)C(O)=O)C(F)(F)F
OC(=O)c1ccc(NC(=O)c2cc(ccc2Oc2ccccc2OC(F)F)C(F)(F)F)cn1
Cc1cc(Cl)ccc1Oc1ccc(cc1C(=O)Nc1ccc(nc1)C(O)=O)C(F)(F)F
COc1ccccc1Oc1ccc(cc1C(=O)Nc1ccc(nc1)C(O)=O)C(F)(F)F
OC(=O)c1ccc(NC(=O)c2cc(ccc2Oc2ccccc2Cl)C(F)(F)F)cn1
CC(C)Oc1ccccc1Oc1ccc(cc1C(=O)Nc1ccc(nc1)C(O)=O)C(F)(F)F
COc1cc(CO)ccc1Oc1ccc(cc1C(=O)Nc1ccc(nc1)C(O)=O)C(F)(F)F
COc1cc(Cl)ccc1Oc1ccc(cc1C(=O)Nc1ccc(nc1)C(O)=O)C(F)(F)F
Cc1cc(CO)ccc1Oc1ccc(cc1C(=O)Nc1ccc(nc1)C(O)=O)C(F)(F)F
OCc1ccc(Oc2ccc(cc2C(=O)Nc2ccc(nc2)C(O)=O)C(F)(F)F)c(Cl)c1
COc1c(F)cccc1Oc1ccc(cc1C(=O)Nc1ccc(nc1)C(O)=O)C(F)(F)F
OC(=O)c1ccc(NC(=O)c2cc(ccc2Oc2ccccc2)C(F)(F)F)cn1
OC(=O)c1ccc(NC(=O)c2cc(ccc2Oc2ccc(F)cc2)C(F)(F)F)cn1
COc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1ccc(nc1)C(O)=O)C(F)(F)C(F)(F)F
OC(=O)c1ccc(NC(=O)c2ccc(cc2Oc2ccc(F)cc2)C(F)(F)C(F)(F)F)cn1
OC(=O)c1ccc(NC(=O)c2c(Oc3ccc(F)cc3Cl)cccc2C(F)(F)F)cn1
Cc1cc(F)ccc1Oc1ccc(cc1C(=O)Nc1ccc(nc1)C(O)=O)C(F)(F)F
COc1cc(F)ccc1Oc1cc(Cl)c(Cl)cc1C(=O)Nc1ccn(COP(O)(O)=O)c(=O)c1
COc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1ccn(COP(O)(O)=O)c(=O)c1)C(F)(F)C(F)(F)F
Cc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1ccn(COP(O)(O)=O)c(=O)c1)C(F)(F)F
Cc1cc(F)ccc1Oc1ccc(cc1C(=O)Nc1ccn(COP(O)(O)=O)c(=O)c1)C(F)(F)F
Cc1cc(F)ccc1Oc1cc(Cl)ccc1C(=O)Nc1ccn(COP(O)(O)=O)c(=O)c1
OP(O)(=O)OCn1ccc(NC(=O)c2cc(ccc2Oc2ccc(F)cc2)C(F)(F)F)cc1=O
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCS(=O)(=O)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC(C2)N2CCOCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC(CC2)N2CCOCC2)nc1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)nc1
OC1CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)cn1
FC(F)(F)C1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
COCCNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CCC(F)(F)CC2)nc1
FC(F)C1CNCCN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
OCCN1CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
COC[C@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CN(C)C(=O)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
N[C@H]1[C@@H]2CN(C[C@H]12)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC(=O)N2CCCC2)nc1
CCN1CC(CC1=O)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CCN1CC(CC1=O)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN(CC2)C2CCC2)nc1
CC1(COC1)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
N[C@H]1[C@@H]2CN(C[C@H]12)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
F[C@H]1CCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
F[C@@H]1CCN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCN3CC(F)(F)C[C@H]3C2)nc1
CC[C@@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
COCCNC(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
FC(F)Oc1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N[C@H]2CNC(=O)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CC(F)(F)C2)nc1
CCN(C1CCN(CC)C(=O)C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
C[C@@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
COC[C@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
COC[C@@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
CS(=O)(=O)CCCNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
NC1CN(C1)C(=O)c1ccc2cc(Oc3ccc(nc3)C(F)(F)F)ccc2n1
CC1CN(CC(C)N1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
C[C@@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
COC[C@H]1CN(CCN1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)F)ccc2n1
F[C@@H]1CCN(C1)C1CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)[C@@H]1CNCCN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CN1C[C@@H](CC1=O)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CN1C[C@H](CC1=O)NC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
F[C@@H]1CCN(C1)C(=O)c1ccc2cc(Oc3ccc(OC(F)(F)F)cn3)ccc2n1
FC(F)(F)CNC(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC(F)(F)C2)nc1
FC(F)(F)Oc1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCNCC2)nc1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NCC(F)(F)F)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CCC22COC2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N[C@H]2CCNC(=O)C2)nc1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N[C@@H]2CCNC(=O)C2)nc1
CN(C1CCN(C)C(=O)C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)NC2CC(F)(F)C2)nc1
FC(F)[C@H]1CNCCN1C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)COC1CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
C[N+]1(C)CCN(CC1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)CNC1CN(C1)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
CN(CC(F)F)C(=O)c1ccc2cc(Oc3ccc(cn3)C(F)(F)F)ccc2n1
FC(F)(F)c1ccc(Oc2ccc3nc(ccc3c2)C(=O)N2CC3(C2)CCOCC3)nc1
COc1cc(C)ccc1Oc1ccc(OC(F)(F)F)cc1C(=O)Nc1cc[nH]c(=O)c1
CCc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c(Cl)c1
CCCOc1ccc(Oc2ccc(cc2C(=O)NC2=CCNC=C2)C(F)(F)F)cc1 |c:23,t:19|
COc1c(C)cccc1Oc1ccc(cc1C(=O)NC1=CCNC=C1)C(F)(F)F |c:25,t:21|
COc1ccc(Oc2ccc(cc2C(=O)NC2=CCNC=C2)C(F)(F)F)c(F)c1 |c:21,t:17|
CCc1cc(F)cc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c1
COc1ccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)cc1C
FC(F)COc1ccccc1Oc1ccc(cc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
COc1cc(Oc2cc(ccc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)ccc1F
COc1c(C)cccc1Oc1cc(ccc1C(=O)Nc1cc(=O)[nH]cc1C)C(F)(F)F
Fc1cccc(Oc2ccc(cc2C(=O)Nc2cc[nH]c(=O)c2)C(F)(F)F)c1F
COc1ccc(Oc2ccc(F)cc2C(=O)Nc2cc[nH]c(=O)c2)c(C)c1
FC(F)(F)c1ccc(C(=O)Nc2cc[nH]c(=O)c2)c(O[C@@H]2CC3CCC2C3)c1 |THB:19:20:23.24:26|
FC(F)(F)c1ccc(C(=O)Nc2cc[nH]c(=O)c2)c(OCC2CC3CCC2C3)c1
CCc1cc(F)ccc1Oc1cc(cc(c1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F)C(F)(F)F
Cc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1ccn(CCl)c(=O)c1)C(F)(F)F
COc1cc(NC(=O)c2ccc(cc2F)C(F)(F)F)ccn1
NS(=O)(=O)c1cccc(NC(=O)c2ccc(cc2Oc2ccc(F)cc2)C(F)(F)F)c1
NS(=O)(=O)c1cccc(NC(=O)c2ccc(cc2Oc2ccc(F)cc2F)C(F)(F)F)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(ccc2Oc2ccc(F)cc2)C(F)(F)F)c1
NS(=O)(=O)c1cccc(NC(=O)c2ccc(cc2Oc2ccc(F)cc2Cl)C#N)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(Cl)ccc2Oc2ccc(F)cc2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(ccc2Oc2ccc(F)cc2F)C(F)(F)F)c1
Cc1cc(C(=O)Nc2cccc(c2)S(N)(=O)=O)c(Oc2ccc(F)cc2)cc1Cl
NS(=O)(=O)c1cccc(NC(=O)c2ccc(Cl)cc2Oc2ccc(F)cc2Cl)c1
Cc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1cccc(c1)S(N)(=O)=O)C#N
COc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1cccc(c1)S(N)(=O)=O)C#N
NS(=O)(=O)c1cccc(NC(=O)c2cc(ccc2Oc2ccc(F)cc2Cl)C#N)c1
Cc1cc(F)ccc1Oc1cccc(c1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
COc1cc(F)ccc1Oc1cccc(c1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
COc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
COc1cc(F)ccc1Oc1cc(Cl)ccc1C(=O)Nc1cccc(c1)S(N)(=O)=O
COc1cc(F)ccc1Oc1ccc(Cl)cc1C(=O)Nc1cccc(c1)S(N)(=O)=O
NS(=O)(=O)c1cccc(NC(=O)c2cc(Cl)ccc2Oc2ccc(F)cc2Cl)c1
Cc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
Cc1cc(F)ccc1Oc1cc(Cl)ccc1C(=O)Nc1cccc(c1)S(N)(=O)=O
Cc1cc(F)ccc1Oc1ccc(Cl)cc1C(=O)Nc1cccc(c1)S(N)(=O)=O
Cc1cc(F)ccc1Oc1ccc(F)cc1C(=O)Nc1cccc(c1)S(N)(=O)=O
COc1ccc(Oc2ccc(cc2C(=O)Nc2cccc(c2)S(N)(=O)=O)C(F)(F)F)cc1
CCOc1ccc(Oc2ccc(cc2C(=O)Nc2cccc(c2)S(N)(=O)=O)C(F)(F)F)cc1
NS(=O)(=O)c1cccc(NC(=O)c2cc(ccc2Oc2ccc(Cl)cc2)C(F)(F)F)c1
Cc1cc(F)ccc1Oc1ccc(cc1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
NS(=O)(=O)c1cccc(NC(=O)c2cc(ccc2Oc2ccc(F)cc2Cl)C(F)(F)F)c1
COc1cc(F)ccc1Oc1ccc(cc1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
NS(=O)(=O)c1cccc(NC(=O)c2cc(ccc2Oc2ccc(CO)c(F)c2)C(F)(F)F)c1
COc1c(F)cccc1Oc1ccc(cc1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
Cc1cc(Cl)ccc1Oc1ccc(cc1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
COc1ccc(Oc2ccc(cc2C(=O)Nc2cccc(c2)S(N)(=O)=O)C(F)(F)F)c(Cl)c1
Cc1ccccc1Oc1ccc(cc1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
NS(=O)(=O)c1cccc(NC(=O)c2c(Oc3ccc(F)cc3Cl)cccc2C(F)(F)F)c1
COc1ccccc1Oc1ccc(cc1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
COc1cc(Cl)ccc1Oc1ccc(cc1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
COc1ccc(Oc2ccc(cc2C(=O)Nc2cccc(c2)S(N)(=O)=O)C(F)(F)F)c(OC)c1
CC(C)Oc1ccc(Oc2ccc(cc2C(=O)Nc2cccc(c2)S(N)(=O)=O)C(F)(F)F)cc1
Cc1cccc(Oc2ccc(F)cc2Cl)c1C(=O)Nc1cccc(c1)S(N)(=O)=O
NS(=O)(=O)c1cccc(NC(=O)c2cc(ccc2Oc2ccc(OC(F)(F)F)cc2)C(F)(F)F)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(ccc2Oc2ccc(F)cc2Cl)C(F)F)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(ccc2Oc2ccc(OC(F)F)cc2)C(F)(F)F)c1
COc1cc(Cl)ccc1Oc1cc(ccc1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
COc1ccc(Oc2cc(ccc2C(=O)Nc2cccc(c2)S(N)(=O)=O)C(F)(F)F)cc1F
COc1ccccc1Oc1cc(ccc1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
CCOc1ccc(Oc2cc(ccc2C(=O)Nc2cccc(c2)S(N)(=O)=O)C(F)(F)F)cc1
CCCOc1ccccc1Oc1cc(ccc1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
NS(=O)(=O)c1cccc(NC(=O)c2ccc(cc2Oc2ccccc2C(F)(F)F)C(F)(F)F)c1
COc1ccc(Oc2cc(ccc2C(=O)Nc2cccc(c2)S(N)(=O)=O)C(F)(F)F)c(Cl)c1
COc1ccc(Oc2cc(ccc2C(=O)Nc2cccc(c2)S(N)(=O)=O)C(F)(F)F)c(C)c1
COc1ccc(Oc2cc(ccc2C(=O)Nc2cccc(c2)S(N)(=O)=O)C(F)(F)F)c(OC)c1
NS(=O)(=O)c1cccc(NC(=O)c2ccc(cc2Oc2ccc(OC(F)(F)F)cc2)C(F)(F)F)c1
COc1c(F)cccc1Oc1cc(ccc1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
CC(C)Oc1ccc(Oc2cc(ccc2C(=O)Nc2cccc(c2)S(N)(=O)=O)C(F)(F)F)cc1
COc1cc(F)ccc1Oc1cc(OC(F)(F)F)ccc1C(=O)Nc1cccc(c1)S(N)(=O)=O
NS(=O)(=O)c1cccc(NC(=O)c2ccc(OC(F)(F)F)cc2Oc2ccc(F)cc2)c1
NS(=O)(=O)c1cccc(NC(=O)c2ccc(OC(F)(F)F)cc2Oc2ccc(F)cc2Cl)c1
COc1ccccc1Oc1cccc(c1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
Cc1cc(Cl)ccc1Oc1cccc(c1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
Cc1c(F)cccc1Oc1cccc(c1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
NS(=O)(=O)c1cccc(NC(=O)c2c(Oc3ccc(OC(F)(F)F)cc3)cccc2C(F)(F)F)c1
COc1ccc(Oc2cccc(c2C(=O)Nc2cccc(c2)S(N)(=O)=O)C(F)(F)F)cc1F
COc1ccc(Oc2cc(OC(F)(F)F)ccc2C(=O)Nc2cccc(c2)S(N)(=O)=O)c(Cl)c1
NS(=O)(=O)c1cccc(NC(=O)c2ccc(OC(F)(F)F)cc2Oc2ccccc2Cl)c1
NS(=O)(=O)c1cccc(NC(=O)c2ccc(OC(F)(F)F)cc2Oc2ccccc2OC(F)F)c1
COc1cc(Cl)ccc1Oc1cc(OC(F)(F)F)ccc1C(=O)Nc1cccc(c1)S(N)(=O)=O
COc1c(Cl)cccc1Oc1cc(OC(F)(F)F)ccc1C(=O)Nc1cccc(c1)S(N)(=O)=O
COc1ccc(Oc2cc(ccc2C(=O)Nc2cccc(c2)S(N)(=O)=O)C(F)(F)F)cc1Cl
COc1c(Cl)cccc1Oc1cc(ccc1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F
NS(=O)(=O)c1cccc(NC(=O)c2ccc(cc2Oc2ccc(F)cc2)C(F)(F)C(F)(F)F)c1
COc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)C(F)(F)F
COc1cc(Cl)ccc1Oc1cc(ccc1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)C(F)(F)F
NS(=O)(=O)c1cccc(NC(=O)c2ccc(cc2Oc2ccc(CO)cc2Cl)C(F)(F)C(F)(F)F)c1
NS(=O)(=O)c1cccc(NC(=O)c2ccc(cc2Oc2ccccc2Cl)C(F)(F)F)c1
NS(=O)(=O)c1cccc(NC(=O)c2c(Oc3ccccc3Cl)cccc2C(F)(F)F)c1
COc1ccc(Oc2cccc(c2C(=O)Nc2cccc(c2)S(N)(=O)=O)C(F)(F)F)c(Cl)c1
COc1ccc(Oc2cc(Cl)c(Cl)cc2C(=O)Nc2cccc(c2)S(N)(=O)=O)c(OC)c1
COc1cc(F)ccc1Oc1cc(Cl)c(Cl)cc1C(=O)Nc1cccc(c1)S(N)(=O)=O
NS(=O)(=O)c1cccc(NC(=O)c2cc(Cl)c(Cl)cc2Oc2ccc(F)cc2)c1
COc1ccc(Oc2cc(Cl)c(Cl)cc2C(=O)Nc2cccc(c2)S(N)(=O)=O)cc1F
COc1cc(Cl)ccc1Oc1cc(Cl)c(Cl)cc1C(=O)Nc1cccc(c1)S(N)(=O)=O
COc1ccc(Oc2cc(Cl)c(Cl)cc2C(=O)Nc2cccc(c2)S(N)(=O)=O)c(F)c1
COc1ccc(Oc2cc(Cl)c(Cl)cc2C(=O)Nc2cccc(c2)S(N)(=O)=O)c(Cl)c1
Cc1cc(F)ccc1Oc1cc(Cl)c(Cl)cc1C(=O)Nc1cccc(c1)S(N)(=O)=O
COc1ccc(Oc2cc(Cl)ccc2C(=O)Nc2cccc(c2)S(N)(=O)=O)c(OC)c1
COc1cc(Cl)ccc1Oc1cc(Cl)ccc1C(=O)Nc1cccc(c1)S(N)(=O)=O
COc1ccc(Oc2cc(Cl)ccc2C(=O)Nc2cccc(c2)S(N)(=O)=O)c(Cl)c1
CC(C)Oc1ccc(Oc2cc(Cl)ccc2C(=O)Nc2cccc(c2)S(N)(=O)=O)cc1
NS(=O)(=O)c1cccc(NC(=O)c2c(Oc3ccc(F)cc3)cc(cc2C(F)(F)F)C(F)(F)F)c1
COc1cc(F)ccc1Oc1cc(cc(c1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F)C(F)(F)F
COc1ccc(Oc2cc(cc(c2C(=O)Nc2cccc(c2)S(N)(=O)=O)C(F)(F)F)C(F)(F)F)cc1F
COc1ccc(Oc2cc(cc(c2C(=O)Nc2cccc(c2)S(N)(=O)=O)C(F)(F)F)C(F)(F)F)c(F)c1
COc1ccc(F)cc1Oc1cc(cc(c1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F)C(F)(F)F
Cc1cc(F)ccc1Oc1cc(cc(c1C(=O)Nc1cccc(c1)S(N)(=O)=O)C(F)(F)F)C(F)(F)F
NS(=O)(=O)c1cccc(NC(=O)c2c(Cl)cc(Cl)cc2Oc2ccc(F)cc2)c1
COc1cc(F)ccc1Oc1cc(Cl)cc(Cl)c1C(=O)Nc1cccc(c1)S(N)(=O)=O
Cc1cc(F)ccc1Oc1cc(Cl)cc(Cl)c1C(=O)Nc1cccc(c1)S(N)(=O)=O
NS(=O)(=O)c1cccc(NC(=O)c2c(Cl)cc(Cl)cc2Oc2ccc(OC(F)(F)F)cc2)c1
COc1cc(Cl)ccc1Oc1cc(Cl)cc(Cl)c1C(=O)Nc1cccc(c1)S(N)(=O)=O
COc1ccc(Oc2cc(Cl)cc(Cl)c2C(=O)Nc2cccc(c2)S(N)(=O)=O)c(F)c1
COc1ccc(Oc2cc(cc(C3CC3)c2C(=O)Nc2cccc(c2)S(N)(=O)=O)C(F)(F)F)cc1F
NS(=O)(=O)c1cncc(NC(=O)c2cc(cnc2N2CCC(F)(F)CC2)C(F)(F)F)n1
COc1ccnc(NC(=O)c2cc(cnc2N2CCC(F)(F)CC2)C(F)(F)F)n1
OC(=O)c1ccc(NC(=O)c2cc(cnc2N2CCC(F)(F)CC2)C(F)(F)F)cn1
OC(=O)c1cc(NC(=O)c2cc(cnc2N2CCC(F)(F)CC2)C(F)(F)F)ccn1
FC(F)(F)c1cnc(N2CCC(F)(F)CC2)c(c1)C(=O)Nc1ccc(nc1)C#N
CS(=O)(=O)c1cncc(NC(=O)c2cc(cnc2N2CCCCCC2)C(F)(F)F)c1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCCC(CO)C2)C(F)(F)F)ccn1
NC(=O)c1cncc(NC(=O)c2cc(cnc2N2CCCCCC2)C(F)(F)F)c1
Cc1ccc(C(=O)Nc2cncc(c2)S(N)(=O)=O)c(n1)N1CCC(F)(F)CC1
NS(=O)(=O)c1cncc(NC(=O)c2cc(Cl)cnc2N2CCC(F)(F)CC2)c1
Cc1cc(Cl)nc(N2CCC(F)(F)CC2)c1C(=O)Nc1cncc(c1)S(N)(=O)=O
NS(=O)(=O)c1cc(NC(=O)c2cc(C3CC3)c(nc2N2CCC(F)(F)CC2)C2CC2)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCCC(F)(F)CC2)C(F)(F)F)ccn1
Cc1nc(N2CCC(F)(F)CC2)c(cc1C1CC1)C(=O)Nc1ccnc(c1)S(N)(=O)=O
Cc1nc(N2CCC(F)(F)CC2)c(cc1C1CCC1)C(=O)Nc1ccnc(c1)S(N)(=O)=O
Cc1nc(N2CCC(F)(F)CC2)c(cc1C#CC1CC1)C(=O)Nc1ccnc(c1)S(N)(=O)=O
Cc1ccc(C(=O)Nc2ccnc(c2)S(N)(=O)=O)c(n1)N1CCCC(F)(F)CC1
NS(=O)(=O)c1cc(NC(=O)c2ccc(CC3CC3)nc2N2CCCC(F)(F)CC2)ccn1
Cc1cc(C(=O)Nc2ccnc(c2)S(N)(=O)=O)c(nc1C)N1CCCC(F)(F)CC1
NS(=O)(=O)c1cc(NC(=O)c2cc(C3CC3)c(OCC(F)(F)F)nc2N2CCC(F)(F)CC2)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(Cl)c(nc2N2CCCC(F)(F)CC2)C2CC2)ccn1
NS(=O)(=O)c1cc(NC(=O)c2ccc(nc2N2CCCC(F)(F)CC2)C2CC2)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(Cl)c(nc2N2CCCC(F)(F)CC2)C2CCC2)ccn1
NS(=O)(=O)c1cc(NC(=O)c2ccc(nc2N2CCCC(F)(F)CC2)C2CCC2)ccn1
Cc1nc(N2CCCC(F)(F)CC2)c(cc1C#N)C(=O)Nc1ccnc(c1)S(N)(=O)=O
NS(=O)(=O)c1cc(NC(=O)c2cccnc2N2CCC(F)(F)CC2)ccn1
FC1(F)CCCN(CC1)c1nc(C2CC2)c(Cl)cc1C(=O)Nc1cc[nH]c(=O)c1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCC(F)(F)CCC2=O)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCC(Cl)(Cl)CC2)C(F)(F)F)ccn1
CS(=O)(=O)n1cc(NC(=O)c2cc(cnc2N2CCCC(F)(F)CC2)C(F)(F)F)c2cccnc12
Cc1nc(N2CCCC(F)(F)CC2)c(cc1Cl)C(=O)Nc1cnn(c1)S(C)(=O)=O
Cc1nc(N2CCCC(F)(F)CC2)c(C(=O)Nc2cnn(c2)S(C)(=O)=O)c(C)c1Cl
Cc1nc(N2CCCC(F)(F)CC2)c(cc1Cl)C(=O)Nc1cnn(c1)S(=O)(=O)CCN
CS(=O)(=O)n1nc(NC(=O)c2cc(cnc2N2CCCC(F)(F)CC2)C(F)(F)F)c2ccccc12
CS(=O)(=O)n1cc(NC(=O)c2cc(cnc2N2CCCC(F)(F)CC2)C(F)(F)F)c2cnccc12
FC(F)(F)c1cnc(N2CCCC(F)(F)CC2)c(c1)C(=O)Nc1cnn(c1)S(=O)(=O)C1CC1
CS(=O)(=O)n1ncc(NC(=O)c2cc(cnc2N2CCCC(F)(F)CC2)C(F)(F)F)c1C1CC1
NS(=O)(=O)c1cc(NC(=O)c2cnc(nc2N2CCCC(F)(F)CC2)C2CC2)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(nnc2N2CCCC(F)(F)CC2)C2CC2)ccn1
Cc1ccc(C(=O)Nc2ccnc(c2)S(N)(=O)=O)c(n1)N1CCCC(F)(F)C(F)C1
COc1nc(N2CCCC(F)(F)CC2)c(cc1Cl)C(=O)Nc1ccnc(c1)S(N)(=O)=O
COc1nc(N2CCCC(F)(F)CC2)c(cc1Cl)C(=O)Nc1ccnc(c1)S(=O)(=O)NC(C)(C)C
NS(=O)(=O)c1cc(NC(=O)c2cc(C#N)c(nc2N2CCC(F)(F)CC2)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(C#CC3CC3)c(nc2N2CCC(F)(F)CC2)C(F)(F)F)ccn1
FC(F)(F)c1cnc(N2CCCCCC2)c(c1)C(=O)Nc1nc(no1)C#N
NS(=O)(=O)c1cc(NC(=O)c2cc(CC3CC3)cnc2N2CCCC(F)(F)CC2)ccn1
CC1CN(CCC1(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
C[C@H]1CN(CCC1(Cl)Cl)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
C[C@@H]1CN(CCC1(Cl)Cl)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCCC(Cl)(Cl)CC2)C(F)(F)F)ccn1
C[C@H]1CN(C[C@@H](C)C1(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
C[C@H]1CN(C[C@@H](C)C1(F)F)c1nc(C)c(Cl)cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O
C[C@@H]1CN(CCC1(F)F)c1nc(C)c(Cl)cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O
C[C@H]1CN(CCC1(F)F)c1nc(C)c(Cl)cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O
C[C@@H]1CCCN(C1)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
C[C@H]1CCCN(C1)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2C[C@H]3CC[C@]3(C2)C(F)(F)F)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2C[C@H]3CC[C@@]3(C2)C(F)(F)F)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2C[C@H]3[C@@H](C2)C(F)(F)C3(F)F)C(F)(F)F)ccn1
C[C@]12CCN(C[C@H]1C2(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
C[C@@]12CCN(C[C@@H]1C2(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2C[C@@H]3CC[C@H](C2)C3(F)F)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2C[C@@H]3CC(F)(F)[C@@H]3C2)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCC[C@]3(CC3(F)F)C2)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2C[C@@H]3CC[C@@H]3C2)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CC[C@H]3[C@@H](C2)C3(F)F)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CC[C@@H]3[C@H](C2)C3(F)F)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2C[C@H]3C[C@@H]2CC3(F)F)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2C[C@@H]3C[C@H]2CC3(F)F)C(F)(F)F)ccn1
CC1CC(F)(F)CCN1c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
C[C@H]1CN(C[C@@H](C)[C@@]1(C)O)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F |r|
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2C[C@@H]3C[C@H](C2)C3(F)F)C(F)(F)F)ccn1
C[C@H]1CN(CC[C@@H]1O)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
CC1CN(CC(C)C1O)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCc3sccc3C2)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCCC(C2)C(F)(F)F)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCCC(C2)c2cc(F)cc(F)c2)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCC(CC2)C(F)(F)F)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCCC(Cc3ccc(cc3)C(F)(F)F)C2)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCSCC2)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCC(C2)c2ccc(cc2)C(F)(F)F)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCn3c(Cc4ccccc4)cnc3C2)C(F)(F)F)ccn1
CC1(C)CN(CCN1CC(F)(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
CC1(C)CN(CCO1)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCc3cccc(c3C2)C(F)(F)F)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2Cc3cccc(OC(F)(F)F)c3C2)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCOC(C2)c2ccc(cc2)C(F)(F)F)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CC(F)(F)C(F)(F)C2)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CC(C2)C(F)(F)F)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCC(C2)n2cccn2)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCCCC2c2ccc(F)cc2)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCC3OCCC23)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CC(C2)Oc2ccc(cc2)C(F)(F)F)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCC(CC2)Oc2cccc(c2)C(F)(F)F)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCN(CC3CC3)C(=O)C2)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCN(CC(F)(F)F)CC2)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(Cl)cnc2N2CCCC(F)(F)CC2)ccn1
C[C@@H]1CN(C[C@H](O1)C(F)(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
C[C@H]1CN(C[C@@H](O1)C(F)(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCCO[C@@H](C2)C(F)(F)F)C(F)(F)F)ccn1 |r|
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCCO[C@H](C2)C(F)(F)F)C(F)(F)F)ccn1 |r|
CC1(C)CO[C@H](CN(C1)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F)C(F)(F)F |r|
CC1(C)CN(CCCO1)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
C[C@H]1CCN(CCO1)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
CC(C)(C)NS(=O)(=O)c1cc(NC(=O)c2cc(Cl)cnc2N2CCCC(F)(F)CC2)ccn1
C[C@H]1CN(CCO1)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
C[C@@H]1CN(CCCO1)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
CC1(O)CCCN(C1)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
CC1(C)N(Cc2ccc(F)cc12)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
Cc1sc(cc1NC(=O)c1cc(cnc1N1CCCCCC1)C(F)(F)F)S(N)(=O)=O
CC1CCN(CCC1(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
Cc1nc(N2CCO[C@H](CC2)C(F)F)c(cc1Cl)C(=O)Nc1ccnc(c1)S(N)(=O)=O
Cc1nc(N2CCO[C@@H](CC2)C(F)F)c(cc1Cl)C(=O)Nc1ccnc(c1)S(N)(=O)=O
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCO[C@@H](CC2)C(F)(F)F)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCO[C@H](CC2)C(F)(F)F)C(F)(F)F)ccn1
C[C@H]1CN(CC[C@@H](O1)C(F)(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
CC1CN(CCC(O1)C(F)(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
CC1CN(CCC(O1)C(F)(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F |$;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;C;;;$|
Cc1nc(N2CCO[C@@H](C2)C(F)F)c(cc1Cl)C(=O)Nc1ccnc(c1)S(N)(=O)=O
Cc1nc(N2CCO[C@H](C2)C(F)F)c(cc1Cl)C(=O)Nc1ccnc(c1)S(N)(=O)=O
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCC[C@H]2C(F)(F)F)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCC[C@@H]2C(F)(F)F)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCC(C2)C(F)(F)F)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CC[C@H](C2)C#N)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CC[C@@H](C2)C#N)C(F)(F)F)ccn1
CC1CN(CCCC1(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
NS(=O)(=O)c1cc(NC(=O)c2ccc(nc2N2CCCC(F)(F)CC2)C(F)(F)F)ccn1
CC[C@@H]1CN(C[C@H](O1)C(F)(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
CCC1CN(CC(O1)C(F)(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
CC1(C)CN(C[C@@H](O1)C(F)(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F |r|
CC1(C)CN(C[C@H](O1)C(F)(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F |r|
NC(=O)c1cc(NC(=O)c2cc(cnc2N2CCCC(F)(F)CC2)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2ccc(Cl)nc2N2CCCC(F)(F)CC2)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCCCCC2)C(F)(F)F)ccn1
CS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCCCCC2)C(F)(F)F)ccn1
NS(=O)(=O)c1cccc(NC(=O)c2cc(cnc2N2CCCCCC2)C(F)(F)F)n1
COc1ccc(C(=O)Nc2ccnc(c2)S(N)(=O)=O)c(n1)N1CCCC(F)(F)CC1
COc1cc(NC(=O)c2cc(cnc2N2CCC3(CC3)CC2)C(F)(F)F)ccn1
NS(=O)(=O)c1cncc(NC(=O)c2cc(cnc2N2CCCC(F)(F)CC2)C(F)(F)F)c1
NS(=O)(=O)c1cncc(NC(=O)c2cc(cnc2N2CCCCCC2)C(F)(F)F)c1
COc1cc(NC(=O)c2cc(cnc2N2CCCC(F)(F)CC2)C(F)(F)F)ccn1
CC1CN(CC(C)C1(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(C)(=O)=O)C(F)(F)F
C[C@@H]1CN(CCC1(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(C)(=O)=O)C(F)(F)F
C[C@H]1CN(CCC1(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)S(C)(=O)=O)C(F)(F)F
C[C@H]1CN(C[C@@H](C)C1(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)C#N)C(F)(F)F
CS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2C[C@H]3[C@@H](C2)C(F)(F)C3(F)F)C(F)(F)F)ccn1
CS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2C[C@@H]3CC[C@@H]3C2)C(F)(F)F)ccn1
FC(F)(F)c1cnc(N2C[C@@H]3CC[C@@H]3C2)c(c1)C(=O)Nc1ccnc(c1)C#N
C[C@@H]1CN(CCC1(F)F)c1nc(ccc1C(=O)Nc1ccnc(c1)C#N)C(F)(F)F
C[C@H]1CN(CCC1(F)F)c1nc(ccc1C(=O)Nc1ccnc(c1)C#N)C(F)(F)F
CC1CN(CC(C)C1(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)C(N)=O)C(F)(F)F
C[C@H]1CN(CCC1(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)C(N)=O)C(F)(F)F
C[C@@H]1CN(CCC1(F)F)c1ncc(cc1C(=O)Nc1ccnc(c1)C(N)=O)C(F)(F)F
COc1ccnc(N2CCC(F)(F)CC2)c1C(=O)Nc1ccnc(c1)S(N)(=O)=O
CC1CN(CC(O1)C(F)(F)F)c1nc(C2CCC2)c(Cl)cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O
CC1CN(CCC1(F)F)c1nc(ccc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
CC1CN(CCC1(F)F)c1nc(c(Cl)cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C(F)(F)F
CC1CN(CC(C)C1(F)F)c1nc(ccc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C1CCC1
CC1CN(CC(O1)C(F)(F)F)c1nc(ccc1C(=O)Nc1ccnc(c1)S(N)(=O)=O)C1CCC1
CC1CN(CC(C)C1(F)F)c1nc(C2CCC2)c(Cl)cc1C(=O)Nc1ccnc(c1)S(N)(=O)=O
Cc1cc(Cl)nc(N2CCC(F)(F)CC2)c1C(=O)Nc1ccnc(c1)S(N)(=O)=O
NS(=O)(=O)c1cc(NC(=O)c2cc(OC(F)F)cnc2N2CCCC(F)(F)CC2)ccn1
Cc1nc(N2CCCC(F)(F)CC2)c(cc1Cl)C(=O)Nc1ccnc(c1)S(N)(=O)=O
Cc1ncc(C(=O)Nc2ccnc(c2)S(N)(=O)=O)c(n1)N1CCCC(F)(F)CC1
NS(=O)(=O)c1cc(NC(=O)c2ccc(nc2N2CCCC(F)(F)CC2)C(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCC(F)(F)CC2)C(F)(F)F)ccn1
OS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCC(F)(F)CC2)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(OC(F)(F)F)cnc2N2CCCC(F)(F)CC2)ccn1
Cc1nc(N2CCC(F)(F)CC2)c(cc1F)C(=O)Nc1ccnc(c1)S(N)(=O)=O
NS(=O)(=O)c1cc(NC(=O)c2cc(nnc2N2CCCC(F)(F)CC2)C(F)(F)F)ccn1
Cc1nc(N2CCC(F)(F)CC2)c(cc1C(C)(C)C)C(=O)Nc1ccnc(c1)S(N)(=O)=O
NS(=O)(=O)c1cc(NC(=O)c2cc(C3CC3)c(nc2N2CCC(F)(F)CC2)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(C3CC3)c(OC(F)(F)F)nc2N2CCC(F)(F)CC2)ccn1
Cc1nc(N2CCC(F)(F)CC2)c(cc1OCC(F)(F)F)C(=O)Nc1ccnc(c1)S(N)(=O)=O
Cc1nc(N2CCCC(F)(F)CC2)c(cc1C(F)(F)F)C(=O)Nc1ccnc(c1)S(N)(=O)=O
NS(=O)(=O)c1cc(NC(=O)c2cc(c(nc2N2CCCC(F)(F)CC2)C2CC2)C(F)(F)F)ccn1
Fc1cc(NC(=O)c2cc(cnc2N2CCCCCC2)C(F)(F)F)ccn1
COc1cc(NC(=O)c2c(C)c(Cl)c(C)nc2N2CCCCCC2)ccn1
Cc1nc(N2CCCCCC2)c(C(=O)Nc2cncc(c2)S(N)(=O)=O)c(C)c1Cl
Cc1nc(N2CCC(F)(F)CC2)c(C(=O)Nc2cncc(c2)S(N)(=O)=O)c(C)c1Cl
Cc1nc(N2CCC3(CC3)CC2)c(C(=O)Nc2cncc(c2)S(N)(=O)=O)c(C)c1Cl
Cc1nc(N2CCCCC2)c(C(=O)Nc2cncc(c2)S(N)(=O)=O)c(C)c1Cl
COc1ccc(C(=O)Nc2cncc(c2)S(N)(=O)=O)c(n1)N1CCCC(F)(F)CC1
FC(F)(F)c1cnc(N2CCCCCC2)c(c1)C(=O)Nc1cncc(c1)C#N
COc1cncc(NC(=O)c2cc(cnc2N2CCCCCC2)C(F)(F)F)c1
Cc1cncc(NC(=O)c2cc(cnc2N2CCCCCC2)C(F)(F)F)c1
OCc1cncc(NC(=O)c2cc(cnc2N2CCCCCC2)C(F)(F)F)c1
FC(F)(F)c1cnc(N2CCCCCC2)c(c1)C(=O)Nc1ccnc(c1)C#N
CCS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCCCCC2)C(F)(F)F)ccn1
FC(F)(F)c1cnc(N2CCCCCC2)c(c1)C(=O)Nc1ccc2ncc(Br)n2c1
FC(F)(F)c1cncc(NC(=O)c2cc(cnc2N2CCCCCC2)C(F)(F)F)c1
Cc1nc(N2CCCCCC2)c(C(=O)Nc2ccnc(c2)S(N)(=O)=O)c(C)c1Cl
Cc1nc(N2CCC3(CC3)CC2)c(C(=O)Nc2ccnc(c2)S(N)(=O)=O)c(C)c1Cl
NC(=O)c1cc(NC(=O)c2cc(cnc2N2CCCCCC2)C(F)(F)F)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(Br)cnc2N2CCC(F)(F)CC2)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCC(F)(F)CC2)-c2ccccc2)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCC(F)(F)CC2)N2CCCCC2)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc(cnc2N2CCC(F)(F)CC2)-n2cccn2)ccn1
FC(F)(F)c1cnc(N2CCC3(CC3)CC2)c(c1)C(=O)Nc1cc[nH]c(=O)c1
Cc1nc(N2CCC3(CC3)CC2)c(C(=O)Nc2cc[nH]c(=O)c2)c(C)c1Cl
FC(F)(F)c1cnc(N2CCCC(F)(F)CC2)c(c1)C(=O)Nc1cc[nH]c(=O)c1
Cc1nc(N2CCCCC2)c(C(=O)Nc2cc[nH]c(=O)c2)c(C)c1Cl
FC(F)(F)c1cnc(N2CCCCCC2)c(c1)C(=O)Nc1cc[nH]c(=O)c1
Cc1nc(N2CCCCCC2)c(C(=O)Nc2cc[nH]c(=O)c2)c(C)c1Cl
CN(C(=O)c1c(C)c(Cl)c(C)nc1N1CCCC(F)(F)CC1)c1ccnc(c1)S(N)(=O)=O
CC1CCC(CC1)c1nc(C)c(Cl)c(C)c1C(=O)Nc1ccnc(c1)S(N)(=O)=O |(2.67,-3.85,;1.33,-3.08,;,-3.85,;-1.33,-3.08,;-1.33,-1.54,;,-.77,;1.33,-1.54,;-2.67,-.77,;-4,-1.54,;-5.33,-.77,;-6.67,-1.54,;-5.33,.77,;-6.67,1.54,;-4,1.54,;-4,3.08,;-2.67,.77,;-1.33,1.54,;-1.33,3.08,;,.77,;1.33,1.54,;1.33,3.08,;2.67,3.85,;4,3.08,;4,1.54,;2.67,.77,;5.33,.77,;6.67,1.54,;4.56,-.56,;6.1,-.56,)|
NS(=O)(=O)c1cc(NC(=O)c2ncc(Cl)nc2N2CCCC(F)(F)CC2)ccn1
Cc1nc(C2CCCCCC2)c(C(=O)Nc2ccnc(c2)S(N)(=O)=O)c(C)c1Cl
Cc1nc(C2CCC(F)(F)CC2)c(C(=O)Nc2ccnc(c2)S(N)(=O)=O)c(C)c1Cl
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(OCC(F)(F)F)nc1)c1ccc(F)c(Cl)c1F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(OCC(F)(F)F)nc1)c1ccc(F)c(Cl)c1F |r|
Fc1ccc(cc1Cl)[C@@H](NC(=O)N1CCNC(=O)C1)c1ccc(OCC(F)(F)F)nc1 |r|
Fc1ccc(cc1Cl)[C@H](NC(=O)N1CCNC(=O)C1)c1ccc(OCC(F)(F)F)nc1 |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(OCC(F)(F)F)nc1)c1ccc(F)c(Cl)c1
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(OCC(F)(F)F)nc1)c1ccc(F)c(Cl)c1
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(OC(F)(F)F)nc1)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(OC(F)(F)F)nc1)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(Cl)cc1)c1ccc(OCC(F)(F)F)nc1
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(Cl)cc1)c1ccc(OCC(F)(F)F)nc1
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(OCC(F)(F)F)nc1)c1ccc(F)c(F)c1
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(OCC(F)(F)F)nc1)c1ccc(F)c(F)c1
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(OCC(F)(F)F)nc1)c1cc(F)c(F)c(Cl)c1
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(OCC(F)(F)F)nc1)c1cc(F)c(F)c(Cl)c1
Fc1ccc([C@@H](NC(=O)N2CCNC(=O)C2)c2ccc(OCC(F)(F)F)nc2)c(F)c1Cl |r|
Fc1ccc([C@H](NC(=O)N2CCNC(=O)C2)c2ccc(OCC(F)(F)F)nc2)c(F)c1Cl |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(Cl)cc1)c1cccc(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(Cl)cc1)c1cccc(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1cnc(OCC(F)(F)F)c(F)c1)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1cnc(OCC(F)(F)F)c(F)c1)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(F)c(Cl)c1)c1ccc2nc(cn2c1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)NC(c1ccc(F)c(Cl)c1)c1ccc2nc(cn2c1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1cnc(OCC(F)(F)F)nc1)c1ccc(F)c(Cl)c1F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1cnc(OCC(F)(F)F)nc1)c1ccc(F)c(Cl)c1F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1cnc(OCC(F)(F)F)s1)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1cnc(OCC(F)(F)F)s1)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1cnc(OC(F)F)s1)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1cnc(OC(F)F)s1)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(nc1)C(F)(F)F)c1ccc(F)c(Cl)c1F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(nc1)C(F)(F)F)c1ccc(F)c(Cl)c1F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(nc1)C(F)(F)F)c1ccc(F)c(Cl)c1
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(nc1)C(F)(F)F)c1ccc(F)c(Cl)c1
C[C@H]1N(CCNC1=O)C(=O)NC(c1ccc(Cl)cc1)c1ccc(nc1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(Cl)cc1)c1ccc(nc1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(nc1)C(F)(F)F)c1ccc(Cl)c(Cl)c1
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(nc1)C(F)(F)F)c1ccc(Cl)c(Cl)c1
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(nc1)C(F)(F)F)c1ccc(F)c(OC(F)(F)F)c1
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(nc1)C(F)(F)F)c1ccc(F)c(OC(F)(F)F)c1
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(OC(F)(F)F)cc1)c1cnc(c(Cl)c1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(OC(F)(F)F)cc1)c1cnc(c(Cl)c1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(OC(F)(F)F)c(F)c1)c1cnc(c(Cl)c1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(OC(F)(F)F)c(F)c1)c1cnc(c(Cl)c1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(OC(F)(F)F)c(Cl)c1)c1cnc(c(Cl)c1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(OC(F)(F)F)c(Cl)c1)c1cnc(c(Cl)c1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(Cl)c(c1)C#N)c1cnc(c(Cl)c1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(Cl)c(c1)C#N)c1cnc(c(Cl)c1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(C#N)c(Cl)c1)c1cnc(c(Cl)c1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(C#N)c(Cl)c1)c1cnc(c(Cl)c1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(OC2CC2)c(F)c1)c1cnc(c(Cl)c1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(OC2CC2)c(F)c1)c1cnc(c(Cl)c1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(F)c(Cl)c1)c1cnc(c(Cl)c1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(F)c(Cl)c1)c1cnc(c(Cl)c1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1cnc(C2CC2)c(Cl)c1)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1cnc(C2CC2)c(Cl)c1)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(Cl)c(Cl)c1)c1cnc(nc1)C(F)(F)F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(Cl)c(Cl)c1)c1cnc(nc1)C(F)(F)F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(nc1)C(F)(F)F)c1ccc(Cl)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(nc1)C(F)(F)F)c1ccc(Cl)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1cnc(nc1)C(F)(F)F)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1cnc(nc1)C(F)(F)F)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(OC(F)F)nc1)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(OC(F)F)nc1)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(nc1)C(F)F)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(nc1)C(F)F)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(nc1)C1CC1)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(nc1)C1CC1)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1cnc(c(F)c1)C(F)(F)F)c1ccc(F)c(Cl)c1F |r|
C[C@H]1N(CCNC1=O)C(=O)NC(c1cnc(c(Cl)c1)C(F)(F)F)c1ccc(F)c(Cl)c1F
Fc1ccc(C(NC(=O)N2CCNC(=O)C2)c2cnc(c(Cl)c2)C(F)(F)F)c(F)c1Cl
Fc1ccc([C@H](NC(=O)N2CCNC(=O)[C@@H]2C2CC2)c2cnc(c(F)c2)C(F)(F)F)c(F)c1Cl
Fc1ccc([C@@H](NC(=O)N2CCNC(=O)[C@@H]2C2CC2)c2cnc(c(F)c2)C(F)(F)F)c(F)c1Cl
Fc1ccc([C@@H](NC(=O)N2CCNC(=O)[C@H]2C2CC2)c2ccc(nc2)C(F)(F)F)c(F)c1Cl |r|
Fc1ccc([C@H](NC(=O)N2CCNC(=O)[C@@H]2C2CC2)c2ccc(nc2)C(F)(F)F)c(F)c1Cl |r|
CC(C)[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(nc1)C(F)(F)F)c1ccc(F)c(Cl)c1F
CC(C)[C@@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(nc1)C(F)(F)F)c1ccc(F)c(Cl)c1F
CC[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(nc1)C(F)(F)F)c1ccc(F)c(Cl)c1F
CC[C@@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(nc1)C(F)(F)F)c1ccc(F)c(Cl)c1F
Fc1ccc([C@H](NC(=O)N2CCNC(=O)[C@H]2C2CC2)c2cnc(nc2)C(F)(F)F)c(F)c1Cl
Fc1ccc([C@H](NC(=O)N2CCNC(=O)[C@@H]2C2CC2)c2cnc(nc2)C(F)(F)F)c(F)c1Cl
Fc1ccc(cc1Cl)C(NC(=O)N1CCNC(=O)C1)c1cccc(n1)C(F)(F)F
CC1(C)N(CCNC1=O)C(=O)NC(c1ccc(F)c(Cl)c1)c1cccc(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)NC(c1ccc(F)c(Cl)c1)c1cccc(n1)C(F)(F)F
C[C@@H]1N(CCNC1=O)C(=O)NC(c1ccc(F)c(Cl)c1)c1cccc(n1)C(F)(F)F
C[C@H]1CN(CC(=O)N1)C(=O)N[C@@H](c1ccc(F)c(Cl)c1)c1cccc(n1)C(F)(F)F
FC[C@H]1CNC(=O)CN1C(=O)N[C@H](c1ccc(F)c(Cl)c1)c1cccc(n1)C(F)(F)F
FC[C@H]1CNC(=O)CN1C(=O)N[C@@H](c1ccc(F)c(Cl)c1)c1cccc(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1cnc(OCC(F)(F)F)c(F)c1)c1ccc(F)c(n1)C(F)(F)F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1cnc(OCC(F)(F)F)c(F)c1)c1ccc(F)c(n1)C(F)(F)F |r|
C[C@H]1N(CCNC1=O)C(=O)NC(c1ccc(F)c(F)c1)c1ccc(F)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(F)c(F)c1)c1ccc(F)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(OCC(F)(F)F)nc1)c1ccc(F)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(OCC(F)(F)F)nc1)c1ccc(F)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(OC(F)(F)F)nc1)c1ccc(F)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(OC(F)(F)F)nc1)c1ccc(F)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(Cl)c(c1)C#N)c1ccc(F)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(Cl)c(c1)C#N)c1ccc(F)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(Cl)c(F)c1)c1ccc(F)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(Cl)c(F)c1)c1ccc(F)c(n1)C(F)(F)F
Fc1cc(ccc1Cl)[C@H](NC(=O)N1CCNC(=O)C1)c1ccc(F)c(n1)C(F)(F)F |r|
Fc1cc(ccc1Cl)[C@@H](NC(=O)N1CCNC(=O)C1)c1ccc(F)c(n1)C(F)(F)F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(OC(F)(F)F)cc1)c1ccc(F)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(OC(F)(F)F)cc1)c1ccc(F)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(OC(F)(F)F)c(F)c1)c1ccc(F)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(OC(F)(F)F)c(F)c1)c1ccc(F)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)NC(c1ccc(OCC(F)(F)F)cc1)c1ccc(F)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1cccc(OC(F)(F)F)c1)c1ccc(F)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(OC2CC2)c(F)c1)c1ccc(F)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(OC2CC2)c(F)c1)c1ccc(F)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(F)c(n1)C(F)(F)F)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(F)c(n1)C(F)(F)F)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(OC(F)(F)F)c(F)c1)c1ccc(C#N)c(n1)C(F)(F)F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(OC(F)(F)F)c(F)c1)c1ccc(C#N)c(n1)C(F)(F)F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1cnc(s1)C(F)(F)F)c1ccc(F)c(Cl)c1F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1cnc(s1)C(F)(F)F)c1ccc(F)c(Cl)c1F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1cnn(c1)C(F)(F)F)c1ccc(OC(F)(F)F)c(Cl)c1
C[C@H]1N(CCNC1=O)C(=O)NC(c1cnn(c1)C(F)(F)F)c1ccc(OC(F)(F)F)c(Cl)c1
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1coc(n1)C(F)(F)F)c1ccc(OC(F)(F)F)c(Cl)c1
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1coc(n1)C(F)(F)F)c1ccc(OC(F)(F)F)c(Cl)c1
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1cnn(c1)-c1ccc(F)cc1)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1cnn(c1)-c1ccc(F)cc1)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccn(n1)C(F)F)c1ccc(F)c(Cl)c1 |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccn(n1)C(F)F)c1ccc(F)c(Cl)c1 |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1cnn(CC(F)(F)F)c1)c1ccc(F)c(Cl)c1
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C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1cnc(nc1)C(F)(F)F)c1ccc(F)c(Cl)c1
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C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(F)c(Cl)c1)c1cccc(OC(F)F)n1 |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(OC(F)F)nc1)c1ccc(F)c(Cl)c1
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C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1cnc(OC(F)F)nc1)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1cnc(OC(F)F)nc1)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(nc1)C(C)(F)F)c1ccc(F)c(Cl)c1F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(nc1)C(C)(F)F)c1ccc(F)c(Cl)c1F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(cc1)C#N)c1ccc(Cl)c(n1)C(F)(F)F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(cc1)C#N)c1ccc(Cl)c(n1)C(F)(F)F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1ccc(Cl)c(n1)C(F)(F)F)c1ccc(F)c(Cl)c1F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(Cl)c(n1)C(F)(F)F)c1ccc(F)c(Cl)c1F
Fc1ccc([C@@H](NC(=O)N2CCNC(=O)C2)c2ccc(Cl)c(n2)C(F)(F)F)c(F)c1Cl |r|
Fc1ccc([C@H](NC(=O)N2CCNC(=O)C2)c2ccc(Cl)c(n2)C(F)(F)F)c(F)c1Cl |r|
C[C@H]1N(CCNC1=O)C(=O)NC(c1ccc(F)c(Cl)c1)c1ccc(Cl)c(n1)C(F)(F)F
Fc1ccc(cc1Cl)C(NC(=O)N1CCNC(=O)C1)c1ccc(Cl)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)NC(c1ccc(nc1)C(F)(F)F)c1ccc(Cl)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1ccc(nc1)C(F)(F)F)c1ccc(Cl)c(n1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1cnc(c(Cl)c1)C(F)(F)F)c1ccc(F)c(n1)C(F)(F)F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1cnc(c(Cl)c1)C(F)(F)F)c1ccc(F)c(n1)C(F)(F)F |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1csc(n1)C(F)(F)F)c1cnc(c(Cl)c1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1csc(n1)C(F)(F)F)c1cnc(c(Cl)c1)C(F)(F)F
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1cc(n[nH]1)C(F)(F)F)c1ccc(F)c(Cl)c1 |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1cc(n[nH]1)C(F)(F)F)c1ccc(F)c(Cl)c1 |r|
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1cc(nn1C)C(F)(F)F)c1ccc(F)c(Cl)c1
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1cc(nn1C)C(F)(F)F)c1ccc(F)c(Cl)c1
C[C@H]1N(CCNC1=O)C(=O)N[C@H](c1cc(n[nH]1)C(F)(F)F)c1ccc(OC(F)(F)F)cc1
C[C@H]1N(CCNC1=O)C(=O)N[C@@H](c1cc(n[nH]1)C(F)(F)F)c1ccc(OC(F)(F)F)cc1
O=C(Nc1ccc[n+]([O-])c1)c1nc2ccccc2nc1N1CCCC(F)(F)CC1
NC(=O)c1cc(NC(=O)c2nc3ccccc3nc2N2CCCC(F)(F)CC2)ccc1F
O=C(Nc1cc[nH]c(=O)c1)c1nc2ccccc2nc1N1CCCC(F)(F)CC1
O=C(Nc1cn[nH]c(=O)c1)c1nc2ccccc2nc1N1CCCC(F)(F)CC1
NC(=O)c1cc(NC(=O)c2nc3ccccc3nc2N2CCCC(F)(F)CC2)ccn1
NS(=O)(=O)c1cc(NC(=O)c2nc3ccccc3nc2N2CCCC(F)(F)CC2)ccn1
NC(=O)c1cccc(NC(=O)c2nc3ccccc3nc2N2CCCC(F)(F)CC2)c1
NC(=O)c1cc(NC(=O)c2cc3ccccc3nc2N2CCCC(F)(F)CC2)ccn1
NC(=O)c1cc(NC(=O)c2cc3ccccc3nc2N2CCCC(F)(F)CC2)ccc1F
NC(=O)c1cc(NC(=O)c2cc3cc(F)c(F)cc3nc2N2CCCC(F)(F)CC2)ccn1
NS(=O)(=O)c1cc(NC(=O)c2cc3ccccc3nc2N2CCCC(F)(F)CC2)ccn1
NS(=O)(=O)c1cccc(NC(=O)c2cc3cc(F)c(F)cc3nc2N2CCCC(F)(F)CC2)c1
NS(=O)(=O)c1cc(NC(=O)c2cc3cc(F)c(F)cc3nc2N2CCCC(F)(F)CC2)ccn1
NC(=O)c1cc(NC(=O)c2cc3cc(F)c(F)cc3nc2N2CCCC(F)(F)CC2)ccc1F
Cc1ccc2cc(C(=O)Nc3ccnc(C(N)=O)c3)c(N3CCCC(F)(F)CC3)nc2c1
COc1cc2cc(C(=O)Nc3ccnc(C(N)=O)c3)c(N3CCCC(F)(F)CC3)nc2cc1OC
COc1ccc2nc(N3CCCC(F)(F)CC3)c(C(=O)Nc3ccnc(C(N)=O)c3)cc2c1
CS(=N)(=O)c1cc(NC(=O)c2cc3ccccc3nc2N2CCCC(F)(F)CC2)ccn1
CNS(=O)(=O)c1cc(NC(=O)c2cc3ccccc3nc2N2CCCC(F)(F)CC2)ccn1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCC(F)(F)CC2)c1
Cc1nc(N2CCCCCC2)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)c(C)c1Cl
Cc1c(F)c(Cl)nc(N2CCCCCC2)c1C(=O)Nc1cccc(S(N)(=O)=O)c1
Cc1cc(C)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)c(N2CCCCCC2)n1
Cc1nc(N2CCC(F)(F)C2)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)c(C)c1Cl
NS(=O)(=O)c1cccc(NC(=O)c2cc(F)cnc2N2CCCCC2)c1
Cc1nc(N2CCCCCC2)c(C(=O)Nc2cccc(S(C)(=O)=O)c2)c(C)c1Cl
Cc1cc(Cl)nc(N2CCCC(F)(F)CC2)c1C(=O)Nc1cccc(S(C)(=O)=O)c1
CS(=O)(=O)c1cccc(NC(=O)c2ccc(Cl)nc2N2CCCC(F)(F)CC2)c1
Cc1ccc(C(=O)Nc2cccc(S(C)(=O)=O)c2)c(N2CCCC(F)(F)CC2)n1
COc1ccc(C(=O)Nc2cccc(S(C)(=O)=O)c2)c(N2CCCC(F)(F)CC2)n1
Cc1nc(N2CCCCC2)c(C(=O)Nc2cccc(S(C)(=O)=O)c2)c(C)c1Cl
Cc1nc(N2CCC3(CC2)CC3)c(C(=O)Nc2cccc(C(N)=O)c2)c(C)c1Cl
NC(=O)c1cccc(NC(=O)c2ccc(Cl)nc2N2CCCC(F)(F)CC2)c1
NC(=O)c1cccc(NC(=O)c2cc(Cl)cnc2N2CCCC(F)(F)CC2)c1
Cc1nc(N2CCC(F)(F)CC2)c(C(=O)Nc2cccc(C(N)=O)c2)c(C)c1Cl
Cc1cc(Cl)nc(N2CCCC(F)(F)CC2)c1C(=O)Nc1cccc(C(N)=O)c1
COc1ccc(C(=O)Nc2cccc(C(N)=O)c2)c(N2CCCC(F)(F)CC2)n1
Cc1nc(N2CCCCC2)c(C(=O)Nc2cccc(C(N)=O)c2)c(C)c1Cl
Cc1nc(N2CCC(F)(F)CC2)c(C(=O)Nc2cccc(C#N)c2)c(C)c1Cl
N#Cc1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCCCC2)c1
N#Cc1ccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCCCC2)cc1
Cc1cnc(N2CCCCCC2)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)c1
O=C(Nc1cccc(S(=O)(=O)N2CCCC2)c1)c1cc(C(F)(F)F)cnc1N1CCCCCC1
NS(=O)(=O)c1ccc(O)c(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCCCC2)c1
Cc1nc(N2CCCCCC2)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)cc1Cl
Cc1ccc(-c2cnc(N3CCCCC3)c(C(=O)Nc3cccc(S(N)(=O)=O)c3)c2)cc1
NS(=O)(=O)c1c(F)ccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCC(F)(F)CC2)c1F
Cc1cc(Cl)nc(N2CCCCCC2)c1C(=O)Nc1cccc(S(N)(=O)=O)c1
Cc1cc(C(=O)Nc2cccc(S(N)(=O)=O)c2)c(N2CCCCCC2)nc1C
NS(=O)(=O)c1cccc(NC(=O)c2cc(Cl)cnc2N2CCCCCC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(Br)cnc2N2CCCCCC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2c(Br)ccnc2N2CCCCCC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(-c3cccnc3)cnc2N2CCCCCC2)c1
CS(=O)(=O)c1cccc(NC(=O)c2cc(Br)cnc2N2CCCCCC2)c1
Cc1cc(C(=O)Nc2cccc(S(C)(=O)=O)c2)c(N2CCCCCC2)nc1C
Cc1cc(C(=O)Nc2cccc(C(N)=O)c2)c(N2CCCCCC2)nc1C
NC(=O)c1cccc(NC(=O)c2cc(Br)cnc2N2CCCCCC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(OC(F)(F)F)cnc2N2CCCC(F)(F)CC2)c1
CC(C)(C)c1nc(N2CCCCC2)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)cc1Cl
CC(C)(C)c1ccc(C(=O)Nc2cccc(S(C)(=O)=O)c2)c(N2CCCCC2)n1
CC(C)(C)c1ccc(C(=O)Nc2cccc(S(N)(=O)=O)c2)c(N2CCCCC2)n1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCC3(CC2)CC3)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCCCC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC3CCC(C3)C2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC3CC4CC(C3)CC2C4)c1
CC1CCN(c2ncc(C(F)(F)F)cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)CC(C)(C)C1
COC(=O)C1CCCN(c2ncc(C(F)(F)F)cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)CC1
COC1CCCN(c2ncc(C(F)(F)F)cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)CC1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCC(C(F)F)CC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCC(F)(F)C2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC3CCC(C2)O3)c1
CC1(O)CCCN(c2ncc(C(F)(F)F)cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)CC1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCC[C@H](F)C2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCc3scnc3C2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCOCC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC3CCC(C2)O3)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC(C(F)(F)F)C2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC3CCCC32)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCC(F)(F)C2)c1
COC(=O)C1CCN(c2ncc(C(F)(F)F)cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)CC1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCC(F)C2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC3COC(C3)C2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCC(O)CC2)c1
COC1CCN(c2ncc(C(F)(F)F)cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)CC1
COC(=O)C1CCCCN(c2ncc(C(F)(F)F)cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)C1
CC(C)CC1CCCCCN1c1ncc(C(F)(F)F)cc1C(=O)Nc1cccc(S(N)(=O)=O)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCOCC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCS(=O)(=O)CC2)c1
CN1C2CCC1CN(c1ncc(C(F)(F)F)cc1C(=O)Nc1cccc(S(N)(=O)=O)c1)C2
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCC3(CCCO3)CC2)c1
Cc1nc2c(o1)CCN(c1ncc(C(F)(F)F)cc1C(=O)Nc1cccc(S(N)(=O)=O)c1)C2
COC(=O)N1CCN(c2ncc(C(F)(F)F)cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)CC1
Cc1ccc(C(=O)Nc2cccc(C(N)=O)c2)c(N2CCCC(F)(F)CC2)n1
Cc1nc(N2CCC3(CC2)CC3)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)c(C)c1Cl
NS(=O)(=O)c1cccc(NC(=O)c2ccc(C(F)(F)F)nc2N2CCCCC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCC(F)(F)CC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCC3(CC2)CC3)c1
CC1(C)CCCN(c2ncc(C(F)(F)F)cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)CC1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC3(CCOCC3)C2)c1
CS(=O)(=O)c1cccc(NC(=O)c2ccc(C(F)(F)F)nc2N2CCCCCC2)c1
NC(=O)c1cccc(NC(=O)c2ccc(C(F)(F)F)nc2N2CCC3(CC2)CC3)c1
NS(=O)(=O)c1cccc(NC(=O)c2ccc(OC(F)(F)F)nc2N2CCCCC2)c1
C[Si](C)(C)c1cc(C(=O)Nc2cccc(S(N)(=O)=O)c2)c(N2CCCCCC2)nc1OC(F)(F)F
C[Si](C)(C)c1cnc(N2CCCCCC2)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)c1
C[Si](C)(C)c1cnc(N2CCC3(CC2)COC3)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCCCCC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2ccc(Cl)nc2N2CCCCCC2)c1
Cc1ccc(C(=O)Nc2cccc(S(N)(=O)=O)c2)c(N2CCCCCC2)n1
COc1ccc(C(=O)Nc2cccc(S(N)(=O)=O)c2)c(N2CCCCCC2)n1
NS(=O)(=O)c1cccc(NC(=O)c2cc(F)c(Cl)nc2N2CCCCCC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2ccc(F)nc2N2CCCCCC2)c1
CS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCC(F)(F)CC2)c1
CS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCCCCC2)c1
CS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC3CCC(F)(F)C3C2)c1
CS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2C[C@H]3CCCC[C@H]3C2)c1
CS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCc3ccccc3C2)c1
CS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCC3(CC2)CC3)c1
CS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCC(F)CC2)c1
CS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCC3(CC3)C(F)(F)C2)c1
CS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCC(F)(F)C2)c1
CS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2Cc3ccccc3C2)c1
CS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCC3OCCC32)c1
CS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCC(c3ccccc3)CC2)c1
NC(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCC(F)(F)CC2)c1
NC(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCCCCC2)c1
NC(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC3CCC(F)(F)C3C2)c1
NC(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCC3(CC3)C(F)(F)C2)c1
NC(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCC(F)(F)C2)c1
CC1CN(c2ncc(C(F)(F)F)cc2C(=O)Nc2ccc3c(c2)S(=O)(=O)NC3)CC(C)C1(F)F
CC1CN(c2ncc(C(F)(F)F)cc2C(=O)Nc2ccc3c(c2)S(=O)(=O)NC3)CCC1(F)F
CC1CN(c2ncc(C(F)(F)F)cc2C(=O)Nc2ccc3c(c2)S(=O)(=O)NC3)CCC1(F)F
NS(=O)(=O)c1cc(F)cc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCCC2)c1
NS(=O)(=O)c1cc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCCC2)ccc1F
NS(=O)(=O)c1ccc(F)c(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCCC2)c1
CC(C)S(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCCCC2)c1
O=C(Nc1ccc2c(c1)S(=O)(=O)C=C2)c1cc(C(F)(F)F)cnc1N1CCCCCC1
CC(C)CS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCCCC2)c1
O=C(Nc1cccc(S(=O)(=O)C2CCCC2)c1)c1cc(C(F)(F)F)cnc1N1CCCCCC1
O=C(Nc1ccc2c(c1)S(=O)(=O)NC2)c1cc(C(F)(F)F)cnc1N1CCCCCC1
CN1Cc2ccc(NC(=O)c3cc(C(F)(F)F)cnc3N3CCCCCC3)cc2S1(=O)=O
C[C@H]1CN(c2ncc(C(F)(F)F)cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1(F)F
C[C@@H]1CN(c2ncc(C(F)(F)F)cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1(F)F
CC1CN(c2ncc(C(F)(F)F)cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)CC(C)C1(F)F
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCC3(C2)CC3(F)F)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCC3(C2)CC3(F)F)c1
CC12CCN(c3ncc(C(F)(F)F)cc3C(=O)Nc3cccc(S(N)(=O)=O)c3)CC1C2(F)F
CC12CCN(c3ncc(C(F)(F)F)cc3C(=O)Nc3cccc(S(N)(=O)=O)c3)CC1C2(F)F
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC3CCC3(C(F)(F)F)C2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC3CCC3(C(F)(F)F)C2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC3CC(C2)C3(F)F)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC3C(C2)C(F)(F)C3(F)F)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC3CCC3C2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC3CC(F)(F)C3C2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC3CC(F)(F)C3C2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC3CC2CC3(F)F)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CC3CC2CC3(F)F)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2C3CCC2CC3)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCO[C@H](C(F)(F)F)C2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCO[C@@H](C(F)(F)F)C2)c1
C[C@@H]1CN(c2ncc(C(F)(F)F)cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)C[C@H](C(F)(F)F)O1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCNC(C(F)(F)F)C2)c1
NS(=O)(=O)c3cccc(NC(=O)c1cc(C(F)(F)F)cnc1N2CCCO[C@@H](C(F)(F)F)C2)c3
C[C@H]1CN(c2ncc(C(F)(F)F)cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)C[C@H](C(F)(F)F)O1
C[C@@H]1CN(c2ncc(C(F)(F)F)cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)C[C@@H](C(F)(F)F)O1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCO[C@H](C(F)(F)F)C2)c1
C[C@H]1CN(c2ncc(C(F)(F)F)cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)C[C@@H](C(F)(F)F)O1
CC1CN(c2ncc(C(F)(F)F)cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)CC(C)O1
CC1CN(c2ncc(C(F)(F)F)cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)CC(C)O1
O=C(Nc1cccc(S(=O)(=O)Nc2ccncn2)c1)c1cc(C(F)(F)F)cnc1N1CCCCCC1
CS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCC(F)(F)CC2)c1
CC(C)Cc1cnc(N2CCCCC2)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C3CCCC3)cnc2N2CCCCC2)c1
COc1nc(N2CCCCCC2)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)cc1C
COc1nc(N2CCCCCC2)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)cc1Br
Cc1nc(N2CCCCCC2)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)cc1C#N
Cc1cc(Cl)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)c(N2CCCCCC2)n1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C3CCC3)cnc2N2CCCC(F)(F)CC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C3COC3)cnc2N2CCCC(F)(F)CC2)c1
C=CCCc1cnc(N2CCCC(F)(F)CC2)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)c1
CC(C)c1cnc(N2CCCC(F)(F)CC2)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C3CC3)cnc2N2CCCC(F)(F)CC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)C(F)(F)F)cnc2N2CCCCCC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2ccc(C(F)(F)C(F)(F)F)nc2N2CCCCC2)c1
CS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)C(F)(F)F)cnc2N2CCCCCC2)c1
NC(=O)c1cccc(NC(=O)c2cc(C(F)(F)C(F)(F)F)cnc2N2CCCCCC2)c1
Cc1nc(N2CCCCCC2)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)cc1C(F)(F)F
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)c(CO)nc2N2CCCCCC2)c1
NS(=O)(=O)c3cccc(NC(=O)c1cc(C(F)(F)F)cnc1N2CCC(F)(F)CC2)c3F
NS(=O)(=O)c1cc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCC(F)(F)CC2)cc(F)c1F
NS(=O)(=O)c1cccc(NC(=O)c2cc(OC(F)F)cnc2N2CCCC(F)(F)CC2)c1
CS(=O)(=O)c1cccc(NC(=O)c2cc(Cl)cnc2N2CCCC(F)(F)CC2)c1
Cc1c(Cl)nc(N2CCCCCC2)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)c1C
Cc1ccnc(N2CCCCCC2)c1C(=O)Nc1cccc(S(N)(=O)=O)c1
Cc1nc(N2CCCC(F)(F)CC2)c(C(=O)Nc2cccc(S(C)(=O)=O)c2)cc1C#N
Cc1nc(N2CCCC(F)(F)CC2)c(C(=O)Nc2cccc(C(N)=O)c2)cc1C#N
Cc1nc(N2CCCCCC2)c(C(=O)Nc2cccc(C(N)=O)c2)cc1C#N
Cc1nc(N2CCCC(F)(F)CC2)c(C(=O)N(C)c2cccc(S(N)(=O)=O)c2)c(C)c1Cl
NS(=O)(=O)c1cccc(NC(=O)c2cnc(C3CC3)nc2N2CCCC(F)(F)CC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)nnc2N2CCCC(F)(F)CC2)c1
COc1c([C@@H]2[C@H](c3nc4cc(C(=O)NO)c(F)cc4[nH]3)O[C@@](C)(C(F)(F)F)[C@H]2C)ccc(F)c1F
COc1c([C@H]2[C@H](c3nc4c(C(=N)N)c(F)ccc4[nH]3)O[C@@](C)(C(F)(F)F)[C@H]2C)ccc(F)c1F
COc1c([C@H]2[C@H](C3Nc4cc[n+]([O-])cc4N3)O[C@@](C)(C(F)(F)F)[C@H]2C)ccc(F)c1F
COc1c([C@H]2[C@H](c3nc4c(C(N)=O)nccc4[nH]3)O[C@@](C)(C(F)(F)F)[C@H]2C)ccc(F)c1F
COc1c([C@H]2[C@H](c3nc4c(C(=N)N)nccc4[nH]3)O[C@@](C)(C(F)(F)F)[C@H]2C)ccc(F)c1F
COc1c([C@H]2[C@H](C3Nc4ccnc(N)c4N3)O[C@@](C)(C(F)(F)F)[C@H]2C)ccc(F)c1F
COc1c([C@H]2[C@H](C3Nc4ccnc(NC(N)=O)c4N3)O[C@@](C)(C(F)(F)F)[C@H]2C)ccc(F)c1F
COc1c([C@H]2[C@H](c3nc4c(C(O)CO)nccc4[nH]3)O[C@@](C)(C(F)(F)F)[C@H]2C)ccc(F)c1F
COc1c([C@H]2[C@H](c3nc4c(C(N)=O)[n+]([O-])ccc4[nH]3)O[C@@](C)(C(F)(F)F)[C@H]2C)ccc(F)c1F
COc1c([C@H]2[C@H](C(=O)Nc3cc(NC(=O)CCN)nc(C(N)=O)c3)O[C@@](C)(C(F)(F)F)[C@H]2C)ccc(F)c1F
COc1c([C@@H]2[C@@H](C(=O)Nc3ccnc4c(=O)[nH]cnc34)O[C@](C)(C(F)(F)F)[C@@H]2C)ccc(F)c1F
COc1c([C@H]2[C@H](C(=O)NC3C=[N+]([O-])C=CC3)O[C@@](C)(C(F)(F)F)[C@H]2C)ccc(F)c1F
Cc1cc(F)ccc1N1CN(c2ccc(=O)n(COP(=O)(O)O)c2C)C(=O)c2cc(C(F)(F)F)ccc21
Cc1cc(F)ccc1N1CN(c2ccc(=O)[nH]c2C)C(=O)c2cc(C(F)(F)F)ccc21
Cc1cc(F)ccc1N1CN(c2ccc(=O)n(COP(=O)(O)O)c2C)C(=O)c2ccc(C(F)(F)F)cc21
Cc1cc(F)ccc1N1CN(c2ccc(=O)[nH]c2C)C(=O)c2ccc(C(F)(F)F)cc21
Cc1cc(F)ccc1N1CN(c2ccc(=O)n(COP(=O)(O)O)c2C)C(=O)c2cc(Cl)ccc21
Cc1cc(F)ccc1N1CN(c2ccc(=O)[nH]c2C)C(=O)c2cc(Cl)ccc21
Cc1cc(OC(F)(F)F)ccc1N1CN(c2ccc(=O)n(COP(=O)(O)O)c2C)C(=O)c2cc(C(F)(F)F)cnc21
Cc1cc(OC(F)(F)F)ccc1N1CN(c2ccc(=O)[nH]c2C)C(=O)c2cc(C(F)(F)F)cnc21
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1ncns1
Fc1cc(Oc2ccc(cc2-c2ccnnc2)C(F)(F)F)c(Cl)cc1S(=O)(=O)Nc1nncs1
Nc1[nH]ncc1-c1cc(Cl)ccc1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
CCN1CC(C1)n1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1C#N)S(=O)(=O)Nc1cscn1
Cn1nccc1-c1cc(Cl)ccc1Oc1ccc(cc1F)S(=O)(=O)Nc1ncns1
Fc1cc2N(CCOc2cc1S(=O)(=O)Nc1nccs1)c1ccc(cc1C#N)C(F)(F)F
CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccc(Br)cc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](CC#C)NC(=O)[C@@H](N)CCC(O)=O |r|
CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CC#C |r|
CCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](Cc4c[nH]c5ccc(Br)cc45)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](Cc4c[nH]c5ccccc45)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(N)=O)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)CC#C |r|
NC1(Cc2nc(c[nH]2)-c2ccc(OC(F)(F)F)cc2)CCCOC1
CC(C)CC[C@H](N)c1nc2cc(ccc2[nH]1)C(C)(C)C |r|
C[C@@H](N1CC[C@H](C1)n1nc(C)c2cc(C(=O)NS(=O)(=O)C3CC3)c(F)cc12)c1cc(Cl)cc(Cl)c1 |r|
FC(F)(F)c1ccc(CN2C(=O)[C@@]3(COc4cc5OCOc5cc34)c3ccccc23)o1
c1ccc(c(c1)COc2ccc(cc2)[C@H]3CC[C@H](N3)C(=O)N)F
C([C@@]1([C@H]2[C@@H]3[C@H](N=C(N[C@@]34[C@@H]([C@@H]1O[C@]([C@H]4O)(O2)O)O)N)O)O)O
NC(=O)OC[C@@H]1NC(=N)N2CCC(O)(O)[C@@]22NC(=N)N[C@@H]12 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(ccc3Cl)C(F)(F)F)CC2)cc1F
FC(F)(F)c1cccc(c1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnc(CNCCC2CCNCC2)c1
CSCC[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]2CSSC[C@@H]3NC(=O)[C@H](CC(O)=O)NC(=O)CNC(=O)[C@H](Cc4ccccc4)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc4ccc(O)cc4)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](Cc4ccc(O)cc4)NC(=O)[C@H](CCCCN)NC1=O)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1c[nH]c4ccccc14)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H]([C@@H](C)O)C(O)=O)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(O)=O)NC3=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N2)NC(=O)[C@@H](N)CC(O)=O |r|
CC(C)(C)c1ccc2[nH]c(nc2c1)C(C)(C)N
CC1(CC1)c1ccc2[nH]c(nc2c1)[C@@H](N)CO |r|
CC(C)(C)c1ccc2[nH]c(nc2c1)[C@@](C)(N)CO |r|
CCCC(O)c1nc2cc(ccc2[nH]1)C(C)(C)C
CC(C)(C)c1ccc2nc(cnc2c1)[C@@H](N)CO
CC(C)(C)c1ccc2ncc(nc2c1)[C@H](N)CO
CC(C)(C)c1ccc2ncc(nc2c1)[C@@H](N)CO |r|
C[C@H](O)[C@@H](N)c1nc2cc(ccc2[nH]1)-c1ccc(cc1)C#N |r|
CO[C@H](C)[C@H](N)c1nc2cc(ccc2[nH]1)-c1ccc(cc1F)C#N |r|
C[C@@H](O)[C@H](N)c1nc2cc(ccc2[nH]1)C(F)(F)F |r|
C[C@@H](O)[C@H](N)c1nc2cc(ccc2[nH]1)C(C)(C)C#N |r|
CC(C)c1ccc2[nH]c(nc2c1)[C@@H](N)[C@@H](C)O |r|
CC(C)[C@@H](O)[C@H](N)c1nc2cc(ccc2[nH]1)C(C)(C)C |r|
CC(C)(C)c1ccc2[nH]c(nc2c1)[C@@H](N)CO |r|
CO[C@H](C)[C@H](N)c1nc2cc(ccc2[nH]1)C(C)(C)C |r|
CC(C)(C)c1ccc2[nH]c(nc2c1)[C@@H](N)C(C)(C)C(N)=O |r|
CN[C@@H](CC(N)=O)c1nc2cc(ccc2[nH]1)C(C)(C)C |r|
CC(C)(C)c1ccc2[nH]c(nc2c1)[C@H]1C[C@@H](O)CN1 |r|
CC(C)(C)c1ccc2[nH]c(nc2c1)[C@H]1CCCN1 |r|
CCC[C@H](N)c1nc2cc(ccc2[nH]1)C(C)(C)C |r|
CC(C)(C)c1ccc2nc(cnc2c1)[C@H](N)CO
CO[C@H](C)[C@H](N)c1nc2cc(ccc2[nH]1)-c1ccc(nc1)C#N |r|
CCC(C)c1ccc2[nH]c(nc2c1)[C@@H](N)CO |r|
CO[C@H](C)[C@H](N)c1nc2cc(OC(F)(F)F)ccc2[nH]1 |r|
C[C@@H](O)[C@H](N)c1nc2cc(ccc2[nH]1)C(C)(C)C |r|
C[C@H]([C@H](N)c1nc2ccc(cc2[nH]1)C(C)(C)C)C(N)=O
C[C@H]([C@H](N)c1cn2cc(ccc2n1)C(C)(C)C)C(N)=O |r|
C[C@@H](O)[C@H](N)c1nc2cc(ccc2[nH]1)S(F)(F)(F)(F)F |r|
CC(C)(C)c1ccc2[nH]c(nc2c1)[C@H](N)CC(N)=O |r|
COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(Oc2cc(F)ccc2F)c(Cl)c1
Cn1nccc1[C@H]1CCCC[C@@H]1Oc1cc(F)c(cc1Cl)S(=O)(=O)Nc1ccncn1 |r|
COc1c(Oc2ccc(c(C)c2C(=O)Nc2ccnc(c2)C(N)=O)C(F)(F)F)ccc(OC(F)(F)F)c1F
COc1cc(OC(F)(F)F)ccc1Oc1ccc(c(C)c1C(=O)Nc1ccnc(c1)C(N)=O)C(F)(F)F
COc1cc(OC(F)(F)F)ccc1Oc1ccc(c(Cl)c1C(=O)Nc1ccnc(c1)C(N)=O)C(F)(F)F
COc1cc(OC(F)(F)F)ccc1Oc1ccc(c(Br)c1C(=O)Nc1ccnc(c1)C(N)=O)C(F)(F)F
COc1c(F)c(OC(F)(F)F)ccc1Oc1ccc(Cl)c(F)c1C(=O)Nc1ccnc(c1)C(N)=O
COc1c(F)c(OC(F)(F)F)ccc1Oc1cc(Cl)c(C)c(F)c1C(=O)Nc1ccnc(c1)C(N)=O
COc1cc(Oc2ccc(OC(F)(F)F)c(F)c2OC)c(C(=O)Nc2ccnc(c2)C(N)=O)c(F)c1C(F)(F)F
COc1c(Oc2cc(c(C)c(F)c2C(=O)Nc2ccnc(c2)C(N)=O)C(F)(F)F)ccc(OC(F)(F)F)c1F
COc1cc(Oc2ccc(OC(F)(F)F)c(F)c2OC)c(C(=O)Nc2ccnc(c2)C(N)=O)c(F)c1Cl
COc1c(Oc2cc(c(OC)c(F)c2C(=O)Nc2ccnc(c2)C(N)=O)C(F)(F)F)ccc(OC(F)(F)F)c1F
COc1c(Cl)cc(Oc2ccc(OC(F)(F)F)c(F)c2OC)c(C(=O)Nc2ccnc(c2)C(N)=O)c1F
COc1cc(OC(F)(F)F)ccc1Oc1cc(OC)c(c(F)c1C(=O)Nc1ccnc(c1)C(N)=O)C(F)(F)F
FC(F)(F)Oc1ccc(cc1)-c1ccc2OCCN(Cc3ncccn3)C(=O)c2c1
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CCC(F)(F)CC1
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CCC2(CC2)CC1
Cc1nc(N2CCCC(F)(F)CC2)c(cc1Cl)C(=O)Nc1ccc2CNC(=O)c2c1
COc1cc(NC(=O)c2ccc(o2)-c2ccc(Cl)cc2)cc(OC)c1
COc1ccc(Cl)c(c1)-c1ccc(NC(=O)c2ccnn2C)nc1N
CN(Cc1ccc(cc1)-c1ccccc1S(N)(=O)=O)C(=O)[C@@H]1CCC[C@H]1C(=O)NCc1ccc(OC(F)(F)F)cc1
FC(F)(F)C1CCN(CC1)c1cc(ccc1C(=O)Nc1cc[nH]c(=O)c1)C(F)(F)F
CCN(CC)CCOC(=O)Oc1c(C(C)C)cccc1C(C)C
NS(=O)(=O)c1cccc(NC(=O)c2nc3ccccc3nc2N2CCCCC2)c1
CN1CCN(c2nc3ccccc3nc2C(=O)Nc2cccc(S(N)(=O)=O)c2)CC1
CN1CCN(c2nc3ccccc3cc2C(=O)Nc2cccc(S(N)(=O)=O)c2)CC1
NS(=O)(=O)c1cccc(NC(=O)c2cc3ccccc3nc2N2CCOCC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc3ccccc3nc2N2CCCCC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cccnc2N2CCCCC2)c1
Cc1ccnc(N2CCCCC2)c1C(=O)Nc1cccc(S(N)(=O)=O)c1
Cc1cnc(N2CCCCC2)c(C(=O)Nc2cccc(S(N)(=O)=O)c2)c1
Cc1ccc(C(=O)Nc2cccc(S(N)(=O)=O)c2)c(N2CCCCC2)n1
Cc1cc(C(=O)Nc2cccc(S(N)(=O)=O)c2)c(N2CCCCC2)nc1C
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCCC2)c1
NS(=O)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2N2CCCC3(CC3)C2)c1
CC(C)(C)c1cc(C(=O)Nc2cccc(S(N)(=O)=O)c2)n(Cc2ccccc2)n1
COc1ccccc1NC(=O)c1nc2ccccc2nc1N1CCCCC1
C[C@@H](NC(=O)c1ccc(o1)-c1ccc(Cl)cc1)C(=O)N1CCN(CCCOc2ccc(cc2)C(=O)C2CC2)CC1 |r|
Clc1ccc(cc1)-c1ccc(o1)C(=O)N1CCNCC1
CN(C)C1CCN(CC1)C(=O)c1ccc(o1)-c1ccc(Cl)cc1
Clc1ccc(cc1)-c1ccc(o1)C(=O)NCCCN1CCCCC1
CN(C)CC(C)(C)CNC(=O)c1ccc(o1)-c1ccc(Cl)cc1
CN1CCC(CC1)NC(=O)c1ccc(o1)-c1ccc(Cl)cc1
Clc1ccc(cc1)-c1ccc(o1)C(=O)NCCN1CCCCC1
FC(F)(F)c1cccc(c1)N1CCN(CC1)C(=O)c1ccc(o1)-c1ccc(Cl)cc1
Clc1ccc(cc1)-c1ccc(o1)C(=O)N1CCOCC1
CN1CCN(CC1)C(=O)c1ccc(o1)-c1ccc(Cl)cc1
Clc1ccc(cc1)-c1ccc(o1)C(=O)N1CCN(CC1)C1CCCCC1
Nc1nnc(c(N)n1)-c1cccc(Cl)c1Cl
Cc1cccc(c1OC[C@@H](C)N)C
CC(C)(C)c1ccc(cc1)-c1ccc(o1)C(=O)N1CCN(CC1)C1CCCCC1
Cc1ccccc1CNC(=O)c1cncc(c1)-c1ccc(Cl)cc1
Clc1ccc(cc1)-c1cncc(c1)C(=O)NCc1ccccc1N1CCCCC1
Clc1ccc(cc1)-c1cncc(c1)C(=O)NCc1cccnc1N1CCOCC1
Clc1ccc(cc1)-c1cncc(c1)C(=O)NCc1cccnc1N1CCCCC1
FC(F)(F)COc1ncccc1CNC(=O)c1cncc(c1)-c1ccc(Cl)cc1
CCOc1ncccc1CNC(=O)c1cncc(c1)-c1ccc(Cl)cc1
Clc1ccc(cc1)-c1cncc(c1)C(=O)NCc1cccnc1Cl
Clc1ccc(cc1)-c1cncc(c1)C(=O)NCc1ccccc1N1CCOCC1
Clc1ccc(cc1)-c1cncc(c1)C(=O)NCc1ccccc1Cl
Clc1ccc(cc1)-c1cncc(c1)C(=O)NCc1ccccc1
Cc1cc(C)cc(NC(=O)c2cncc(c2)-c2ccc(Cl)cc2)c1
Cc1cc(C)cc(NC(=O)c2cncc(c2)-c2ccc(F)cc2)c1
Cc1cc(C)cc(NC(=O)c2cncc(c2)-c2ccc(cc2)C#N)c1
Cc1cc(C)cc(NC(=O)c2cncc(c2)-c2ccc(OC(F)(F)F)cc2)c1
Cc1cc(C)cc(NC(=O)c2cccc(n2)-c2ccc(OC(F)(F)F)cc2)c1
Cc1cc(C)cc(NC(=O)c2cncc(n2)-c2ccc(OC(F)(F)F)cc2)c1
Cc1cc(C)cc(NC(=O)c2nsc(n2)-c2ccc(OC(F)(F)F)cc2)c1
Cc1cc(C)cc(NC(=O)c2csc(n2)-c2ccc(OC(F)(F)F)cc2)c1
Cc1cc(C)cc(NC(=O)c2nc(no2)-c2ccc(OC(F)(F)F)cc2)c1
Cc1cc(C)cc(NC(=O)c2coc(n2)-c2ccc(OC(F)(F)F)cc2)c1
Cc1cc(C)cc(NC(=O)c2cnc(o2)-c2ccc(OC(F)(F)F)cc2)c1
Cc1cc(C)cc(NC(=O)c2ccc(o2)-c2ccc(OC(F)(F)F)cc2)c1
Cc1cc(C)cc(NC(=O)c2ccnc(c2)-c2ccc(OC(F)(F)F)cc2)c1
Clc1ccc(cc1)-c1cncc(c1)C(=O)NCc1cccnc1
Cc1ncccc1CNC(=O)c1cncc(c1)-c1ccc(Cl)cc1
FC(F)(F)Oc1ccc(cc1)-c1cncc(n1)C(=O)NCc1cccnc1N1CCOCC1
Cc1cc(C)cc(NC(=O)c2cncc(n2)-c2ccc(Cl)cc2)c1
Clc1ccc(cc1)-c1cncc(n1)C(=O)NCc1cccnc1N1CCCC1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)Nc1cccc(C)c1
CC(C)Oc1cccc(NC(=O)c2cncc(n2)-c2ccc(cc2)C#N)c1
Cc1cccc(NC(=O)c2cncc(n2)-c2ccc(Cl)cc2)c1
FC(F)(F)Oc1ccc(cc1)-c1cncc(n1)C(=O)NCc1cccnc1Cl
COc1cc(NC(=O)c2cncc(n2)-c2ccc(Cl)cc2)cc(OC)c1
Cc1ccccc1CNC(=O)c1cncc(n1)-c1ccc(Cl)cc1
Clc1ccc(cc1)-c1cncc(n1)C(=O)NCc1cccnc1N1CCOCC1
Clc1ccc(CCNC(=O)c2cncc(n2)-c2ccc(Cl)cc2)cc1
Clc1ccc(cc1)-c1cncc(n1)C(=O)NCc1ccncc1N1CCOCC1
Cc1ccccc1CNC(=O)c1cncc(n1)-c1ccc(cc1)C#N
CCOc1ccc(cc1)-c1cncc(n1)C(=O)NCc1ccccc1C
Cc1ccccc1CNC(=O)c1cncc(n1)-c1ccc(OC(F)(F)F)cc1
Cc1cc(C)cc(NC(=O)c2cncc(n2)-c2ccc(cc2)C#N)c1
CCOc1ccc(cc1)-c1cncc(n1)C(=O)Nc1cc(C)cc(C)c1
Cc1cccc(NC(=O)c2cncc(n2)-c2ccc(OC(F)(F)F)cc2)c1
Clc1ccc(cc1)-c1cncc(n1)C(=O)NCc1cccnc1
Clc1ccc(cc1)-c1cncc(n1)C(=O)Nc1cccnc1
Clc1ccc(cc1)-c1cncc(n1)C(=O)NCc1cnccc1N1CCOCC1
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1cccc(OC(F)(F)F)c1F
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1c(F)cccc1OC(F)(F)F
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1cc(ccc1OC(F)(F)F)C(F)(F)F
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1cc(F)ccc1OCC(F)(F)C(F)(F)F
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1cccc(OC(F)(F)F)c1OCC(F)(F)C(F)(F)F
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1cccc(c1OCC(F)(F)C(F)(F)F)C(F)(F)F
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1ccccc1OC(F)(F)F
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1ccccc1C(F)(F)F
NC(=O)c1cc(C(N)=O)n(n1)-c1cccc(c1)-c1cc(ccc1C(F)(F)F)C(F)(F)F
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccc(OC(F)(F)F)cc2)c1C
CC(C)CCC[C@@](C)(O)[C@H]1CC[C@H]2[C@@H]3C[C@H](O[C@@H]4O[C@H](C)[C@@H](O)[C@H](O[C@@H]5OC[C@@H](O[C@@H]6O[C@H](C)[C@@H](O[C@@H]7OC[C@H](O)[C@H](O)[C@H]7O)[C@H](O)[C@H]6O[C@@H]6O[C@H](C)[C@H](O)[C@H](O)[C@H]6O)[C@H](O)[C@H]5O[C@@H]5O[C@H](C)[C@@H](O)[C@H](O)[C@H]5O)[C@H]4O)[C@H]4C[C@H](CC[C@]4(C)C3=CC[C@]12C)OS([O-])(=O)=O |c:90|
Clc1ccc(cc1)-c1ccc(o1)C(=O)Nc1ccc2ncccc2c1
Cc1ccnc(NC(=O)c2ccc(o2)-c2ccc(Cl)cc2)c1
Clc1ccc(cc1)-c1ccc(o1)C(=O)Nc1cccc(c1)N1CCOCC1
Cc1cccc(NC(=O)c2ccc(o2)-c2ccc(cc2)C#N)c1
Clc1ccc(cc1)-c1ccc(o1)C(=O)Nc1ccc2cc[nH]c2c1
CN1CCCc2cc(NC(=O)c3ccc(o3)-c3ccc(Cl)cc3)ccc12
Clc1ccc(cc1)-c1ccc(o1)C(=O)NCCc1ccccc1Cl
CN(C(=O)c1ccc(o1)-c1ccc(Cl)cc1)c1cccc(C)c1
Cc1cccc(NC(=O)c2ccc(o2)-c2ccc(Cl)cc2)c1
Cc1cccc(NC(=O)c2ccc(o2)-c2ccc(OC(F)(F)F)cc2)c1
Cc1cc(NC(=O)c2ccc(o2)-c2ccc(Cl)cc2)ccn1
Cc1cccc(NC(=O)c2ccc(o2)-c2cccc(c2)C(F)(F)F)c1
Cc1cccc(c1)N=C(NC#N)c1ccc(o1)-c1ccc(Cl)cc1 |w:7.7|
CN1CCOc2cc(NC(=O)c3ccc(o3)-c3ccc(Cl)cc3)ccc12
Cc1cccc(c1)N=C(N)c1ccc(o1)-c1ccc(Cl)cc1 |w:7.7|
Cc1cccc(NC(=O)c2ccc(o2)-c2ccc(cc2)S(C)(=O)=O)c1
Cc1cccc(NC(=O)c2coc(c2)-c2ccc(Cl)cc2)c1
Cc1cccc(NC(=O)c2cc(co2)-c2ccc(Cl)cc2)c1
Clc1ccc(cc1)-c1ccc(o1)C(=O)Nc1cccc(c1)C1=NCCO1 |t:24|
CN1CCc2ccc(NC(=O)c3ccc(o3)-c3ccc(Cl)cc3)cc12
Cc1cccc(NC(=O)c2ccc(o2)-c2cccc(c2)C#N)c1
Clc1ccc(cc1)-c1ccc(o1)C(=O)Nc1cccc(CC#N)c1
Cc1ccccc1CNC(=O)c1ccc(o1)-c1ccc(Cl)cc1
CCOc1ccc(cc1)-c1ccc(o1)C(=O)Nc1cccc(C)c1
CC(C)(C)CC(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1Cc1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1c(F)ccc(F)c1F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1OC(F)(F)F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
FC(F)(F)Oc1ccccc1C(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1Cc1ccccc1
CC1(CC1)C(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1cccc(F)c1C(F)(F)F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1Cc1ccccc1
FC(F)(F)c1ccccc1C[C@@H](NC(=O)c1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1Cc1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)C(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1Cc1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1cc(F)ccc1Cl)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
FC(F)(F)Oc1ccccc1C(=O)N[C@H](Cc1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1c(F)cccc1F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
Fc1cccc(F)c1C[C@@H](NC(=O)C1(CC1)C(F)(F)F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)OC(=O)N[C@H](Cc1ccc(F)cc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
Fc1ccc(F)c(C[C@@H](NC(=O)C2(CC2)C(F)(F)F)C(=O)NCc2nc3cccnc3n2C2(CC2)c2ccccc2)c1F
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1Cl)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
FC(F)(F)c1ccccc1C[C@@H](NC(=O)C1(CC1)C(F)(F)F)C(=O)NCc1nc2cccnc2n1C1(CC1)c1ccccc1
CC(C)(C)C(=O)ON[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCc2ccccc2N(CC(F)(F)F)C1=O |r|
CC(=O)N[C@H](COC)C(=O)NCc1ccccc1
FC(F)(F)Oc1cccc(c1)C(=O)NCc1noc(n1)-c1n(CCn2ccnc2)nc2ccccc12
O=C(NCc1noc(n1)-c1nn(CCn2ccnc2)c2ccccc12)c1ccccc1
[H][C@@]12CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@]1([H])CSSC[C@H](NC(=O)[C@@H](N)CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](Cc3ccccc3)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@]3([H])CSSC[C@]([H])(NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC2=O)C(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@]([H])([C@@H](C)O)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc2c[nH]c4ccccc24)C(=O)N[C@@H](CSSC[C@]([H])(NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(O)=O)NC(=O)[C@]2([H])CCCN2C(=O)[C@@]([H])(NC3=O)[C@@H](C)CC)C(=O)N1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(N)=O |r|
CNC(=O)c1ccc(c(N)n1)-c1cc(Cl)cc(Cl)c1Cl
Cc1nocc1C(=O)Nc1ccc(c(N)n1)-c1ccccc1OC(F)(F)F
CNC(=O)c1cnc(N)c(c1)-c1cc(Cl)cc(Cl)c1Cl
CC(=O)Nc1ccc(c(N)n1)-c1cc(Cl)cc(Cl)c1Cl
CNC(=O)c1ccc(c(N)n1)-c1ccccc1Cl
CNC(=O)c1ccc(c(N)n1)-c1cccc(Cl)c1
CNC(=O)c1ccc(c(N)n1)-c1ccc(Cl)cc1
CNC(=O)c1ccc(c(N)n1)-c1cc(Cl)ccc1Cl
CNC(=O)c1ccc(c(N)n1)-c1cc(Cl)cc(Cl)c1
Cn1nccc1C(=O)Nc1ccc(c(N)n1)-c1cc(Cl)cc(Cl)c1Cl
Cc1nocc1C(=O)Nc1ccc(c(N)n1)-c1cc(Cl)cc(Cl)c1Cl
Cn1nccc1C(=O)Nc1ccc(c(N)n1)-c1cc(Cl)ccc1Cl
COc1ccc(Cl)c(c1)-c1ccc(NC(=O)c2conc2C)nc1N
COc1ccc(Cl)cc1-c1ccc(NC(=O)c2ccnn2C)nc1N
Cn1nccc1C(=O)Nc1ccc(c(N)n1)-c1ccccc1Cl
COc1ccc(Cl)c(c1)-c1ccc(NC(=O)C(C)C)nc1N
Cn1nccc1C(=O)Nc1ccc(c(N)n1)-c1ccccc1OC(F)(F)F
Cn1nncc1C(=O)Nc1ccc(c(N)n1)-c1ccccc1OC(F)(F)F
Nc1nc(NC(=O)c2ccccc2)ccc1-c1ccccc1OC(F)(F)F
Cn1nccc1C(=O)Nc1ccc(c(N)n1)-c1ccc(F)cc1Cl
CO[C@H](C)[C@H](N)c1nc2cc(ccc2[nH]1)-c1ccc(C#N)c(F)c1 |r|
Cc1nocc1C(=O)Nc1cnc(c(N)n1)-c1cc(Cl)cc(Cl)c1Cl
c1ccc(cc1)C(c2ccccc2)C(=O)Nc3ccc(cc3)S(=O)(=O)Nc4nccs4
Nc1nc2cc(ccc2[nH]1)-c1cc(Cl)ccc1Oc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
COc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F