Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 105 hits in this display   

TargetD(2) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetD(2) dopamine receptor(Rattus norvegicus (rat))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(3) dopamine receptor(BOVINE)
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  2.90nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]N-methyl-spiperone from D2R (unknown origin) assessed as inhibition constant by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
In DepthDetails ArticlePubMedDrugBank

TargetD(3) dopamine receptor(Homo sapiens)
Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]N-methyl-spiperone from D3R (unknown origin) assessed as inhibition constant by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  3.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  3.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  11.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) assessed as inhibition constant by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]spiperone from human dopamine D2 receptor short form expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]RX 821002 from adrenergic alpha-2 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  136nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  316nMAssay Description:Displacement of [3H]DOI from 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  631nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  1.11E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  1.34E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  1.54E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(RAT)
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  1.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  1.74E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  2.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  2.37E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  4.15E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  7.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  8.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAP-2 complex subunit sigma(RAT)
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine 1D receptor(Bos taurus (Bovine))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(PIG)
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A(RAT)
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetType-1 angiotensin II receptor(RABBIT)
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetType-2 angiotensin II receptor(RAT)
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(1A) dopamine receptor(RAT)
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlutamate receptor 3(RAT)
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlutamate receptor 3(RAT)
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlycine amidinotransferase, mitochondrial(RAT)
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlycine receptor subunit alpha-1(RAT)
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNischarin(RAT)
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium channel protein type 10 subunit alpha(Rattus norvegicus (Rat))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataIC50:  1.5nMAssay Description:The ability of Compound 102 to bind dopamine D2 receptors was measured in a cell-based assay. Dopamine D2 receptor cells were seeded in a half a blac...More data for this Ligand-Target Pair
In DepthDetails US PatentDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataIC50:  1.5nMAssay Description:The ability of Compound 102 to bind dopamine D2 receptors was measured in a cell-based assay. Dopamine D2 receptor cells were seeded in a half a blac...More data for this Ligand-Target Pair
In DepthDetails US PatentDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataIC50:  3nMAssay Description:Antagonistic activity at D2 receptor (unknown origin) expressed in CHOK1 cells co-expressing G-alpha 15 assessed as inhibition of dopamine-induced ca...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataIC50:  8.5nMAssay Description:The ability of Compound 102 to bind the dopamine D2 receptor in a membrane preparation was examined. Medium was removed from dopamine D2 receptor cel...More data for this Ligand-Target Pair
In DepthDetails US PatentDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataIC50:  8.5nMAssay Description:The ability of Compound 102 to bind the dopamine D2 receptor in a membrane preparation was examined. Medium was removed from dopamine D2 receptor cel...More data for this Ligand-Target Pair
In DepthDetails US PatentDrugBank

TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataIC50: >1.33E+5nMAssay Description:Inhibition of human MRP2 overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ATP and...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 4(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataIC50: >1.33E+5nMAssay Description:Inhibition of human MRP4 overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ATP and...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataIC50: >1.33E+5nMAssay Description:Inhibition of human BSEP overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-taurocholate in presence of ATP measured after 15 to ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataIC50: >1.33E+5nMAssay Description:Inhibition of human MRP3 overexpressed in Sf9 insect cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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