Report error Found 565 with Last Name = 'hamacher' and Initial = 'a'
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Human)
Heinrich-Heine-Universit£T D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-Universit£T D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Inhibition of recombinant HDAC3 (unknown origin)/NCOR2 (unknown origin) using acetyl-Lys(Ac)-AMC as substrate preincubated for up to 3 hrs followed b...More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition of HDAC9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human HDAC6 (1 to 1215 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC...More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of C-terminal GST-tagged recombinant human HDAC2 (1 to 488 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC ...More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of recombinant human HDAC6More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Inhibition of recombinant human HDAC6More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human HDAC6 (1 to 1215 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC...More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human HDAC6 (1 to 1215 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC...More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) using acetyl-Lys(Ac)-AMC as substrate preincubated for up to 3 hrs followed by substrate addition an...More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Inhibition of HDAC7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human HDAC6 (1 to 1215 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC...More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibition of recombinant human HDAC6More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Inhibition of recombinant human HDAC2More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Inhibition of recombinant human HDAC6More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Inhibition of C-terminal GST-tagged recombinant human HDAC2 (1 to 488 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC ...More data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Inhibition of HDAC4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition of recombinant human HDAC2More data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Inhibition of recombinant human HDAC2More data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Inhibition of recombinant human HDAC2More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Inhibition of C-terminal GST-tagged recombinant human HDAC2 (1 to 488 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC ...More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human HDAC6 (1 to 1215 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC...More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Inhibition of recombinant human HDAC6More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Inhibition of recombinant human HDAC6More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human HDAC6 (1 to 1215 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC...More data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Inhibition of C-terminal GST-tagged recombinant human HDAC2 (1 to 488 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC ...More data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Inhibition of recombinant human HDAC4More data for this Ligand-Target Pair
Affinity DataKi: 182nMAssay Description:Inhibition of HDAC5 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 189nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Inhibition of recombinant human HDAC2More data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:Inhibition of recombinant human HDAC6More data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Inhibition of recombinant human HDAC6More data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Inhibition of recombinant human HDAC2More data for this Ligand-Target Pair
Affinity DataKi: 420nMAssay Description:Inhibition of recombinant human HDAC6More data for this Ligand-Target Pair
Affinity DataKi: 550nMAssay Description:Inhibition of recombinant human HDAC2More data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Inhibition of recombinant human HDAC6More data for this Ligand-Target Pair
Affinity DataKi: 580nMAssay Description:Inhibition of recombinant human HDAC2More data for this Ligand-Target Pair
Affinity DataKi: 640nMAssay Description:Inhibition of C-terminal His-tagged/N-terminal GST-tagged recombinant human HDAC4 (627 to 1084 residues) expressed in Baculovirus infected insect cel...More data for this Ligand-Target Pair
Affinity DataKi: 750nMAssay Description:Inhibition of C-terminal His-fusion tagged/N-terminal Strep-2 tagged recombinant human HDAC8 (1 to 377 residues) expressed in insect cells using Boc-...More data for this Ligand-Target Pair
Affinity DataKi: 1.25E+3nMAssay Description:Inhibition of C-terminal GST-tagged recombinant human HDAC2 (1 to 488 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC ...More data for this Ligand-Target Pair
Affinity DataKi: 1.33E+3nMAssay Description:Inhibition of recombinant human HDAC2More data for this Ligand-Target Pair
Affinity DataKi: 1.33E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.36E+3nMAssay Description:Inhibition of recombinant human HDAC2More data for this Ligand-Target Pair
Affinity DataKi: 1.57E+3nMAssay Description:Inhibition of recombinant human HDAC2More data for this Ligand-Target Pair
Affinity DataKi: 1.77E+3nMAssay Description:Inhibition of C-terminal His-tagged/N-terminal GST-tagged recombinant human HDAC4 (627 to 1084 residues) expressed in Baculovirus infected insect cel...More data for this Ligand-Target Pair
Affinity DataKi: 2.15E+3nMAssay Description:Inhibition of recombinant human HDAC6More data for this Ligand-Target Pair
Affinity DataKi: 2.81E+3nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.94E+3nMAssay Description:Inhibition of HDAC7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4.21E+3nMAssay Description:Inhibition of C-terminal His-fusion tagged/N-terminal Strep-2 tagged recombinant human HDAC8 (1 to 377 residues) expressed in insect cells using Boc-...More data for this Ligand-Target Pair
Affinity DataKi: 4.44E+3nMAssay Description:Inhibition of recombinant human HDAC8More data for this Ligand-Target Pair
Affinity DataKi: 4.70E+3nMAssay Description:Inhibition of C-terminal His-fusion tagged/N-terminal Strep-2 tagged recombinant human HDAC8 (1 to 377 residues) expressed in insect cells using Boc-...More data for this Ligand-Target Pair