Affinity DataKi: 10nMAssay Description:Inhibition of [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Inhibition of [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 569nMAssay Description:Inhibition of [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Ability to inhibit [3H]nitrendipine binding to the L-type calcium channel receptor(CCR) in rat heart homogenate.More data for this Ligand-Target Pair
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Sankyo
Curated by ChEMBL
Sankyo
Curated by ChEMBL
Affinity DataIC50: 12.2nMAssay Description:Inhibitory concentration required against Translocase IMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of Escherichia coli lipopolysaccharide-induced COX2 activity in mouse J774 cells assessed as decrease in PGE2 levels after 24 hrs by RIAMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of Escherichia coli lipopolysaccharide-induced COX2 activity in mouse J774 cells assessed as decrease in PGE2 levels after 24 hrs by RIAMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Ability to inhibit [3H]nitrendipine binding to the L-type calcium channel receptor(CCR) in rat heart homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of Escherichia coli lipopolysaccharide-induced COX2 activity in mouse J774 cells assessed as decrease in PGE2 levels after 24 hrs by RIAMore data for this Ligand-Target Pair
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Sankyo
Curated by ChEMBL
Sankyo
Curated by ChEMBL
Affinity DataIC50: 17.1nMAssay Description:Inhibitory concentration against translocase-IMore data for this Ligand-Target Pair
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Sankyo
Curated by ChEMBL
Sankyo
Curated by ChEMBL
Affinity DataIC50: 17.6nMAssay Description:Inhibitory concentration against translocase-IMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of Escherichia coli lipopolysaccharide-induced COX2 activity in mouse J774 cells assessed as decrease in PGE2 levels after 24 hrs by RIAMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of Escherichia coli lipopolysaccharide-induced COX2 activity in mouse J774 cells assessed as decrease in PGE2 levels after 24 hrs by RIAMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of Escherichia coli lipopolysaccharide-induced COX2 activity in mouse J774 cells assessed as decrease in PGE2 levels after 24 hrs by RIAMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Sankyo
Curated by ChEMBL
Sankyo
Curated by ChEMBL
Affinity DataIC50: 35.9nMAssay Description:Inhibitory concentration required against Translocase IMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Ability to inhibit [3H]nitrendipine binding to the L-type calcium channel receptor(CCR) in rat heart homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Inhibition of Escherichia coli lipopolysaccharide-induced COX2 activity in mouse J774 cells assessed as decrease in PGE2 levels after 24 hrs by RIAMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Ability to inhibit [3H]nitrendipine binding to the L-type calcium channel receptor(CCR) in rat heart homogenate.More data for this Ligand-Target Pair
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Sankyo
Curated by ChEMBL
Sankyo
Curated by ChEMBL
Affinity DataIC50: 58.7nMAssay Description:Inhibitory concentration against translocase-IMore data for this Ligand-Target Pair
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Sankyo
Curated by ChEMBL
Sankyo
Curated by ChEMBL
Affinity DataIC50: 59.9nMAssay Description:Inhibitory concentration required against Translocase IMore data for this Ligand-Target Pair
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Sankyo
Curated by ChEMBL
Sankyo
Curated by ChEMBL
Affinity DataIC50: 63.1nMAssay Description:Inhibitory concentration required against Translocase IMore data for this Ligand-Target Pair
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Sankyo
Curated by ChEMBL
Sankyo
Curated by ChEMBL
Affinity DataIC50: 64.7nMAssay Description:Inhibitory concentration required against Translocase IMore data for this Ligand-Target Pair
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Sankyo
Curated by ChEMBL
Sankyo
Curated by ChEMBL
Affinity DataIC50: 76.5nMAssay Description:Inhibitory concentration required against Translocase IMore data for this Ligand-Target Pair
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Sankyo
Curated by ChEMBL
Sankyo
Curated by ChEMBL
Affinity DataIC50: 80.7nMAssay Description:Inhibitory concentration required against Translocase IMore data for this Ligand-Target Pair
Affinity DataIC50: 89nMAssay Description:Inhibition of Escherichia coli lipopolysaccharide-induced COX2 activity in mouse J774 cells assessed as decrease in PGE2 levels after 24 hrs by RIAMore data for this Ligand-Target Pair
Affinity DataIC50: 139nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Ability to inhibit [3H]nitrendipine binding to the L-type calcium channel receptor(CCR) in rat heart homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Sankyo
Curated by ChEMBL
Sankyo
Curated by ChEMBL
Affinity DataIC50: 182nMAssay Description:Inhibitory concentration required against Translocase IMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of Escherichia coli lipopolysaccharide-induced COX2 activity in mouse J774 cells assessed as decrease in PGE2 levels after 24 hrs by RIAMore data for this Ligand-Target Pair
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Sankyo
Curated by ChEMBL
Sankyo
Curated by ChEMBL
Affinity DataIC50: 215nMAssay Description:Inhibitory concentration required against Translocase IMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Ability to inhibit [3H]nitrendipine binding to the L-type calcium channel receptor(CCR) in rat heart homogenate.More data for this Ligand-Target Pair
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Sankyo
Curated by ChEMBL
Sankyo
Curated by ChEMBL
Affinity DataIC50: 234nMAssay Description:Inhibitory concentration required against Translocase IMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibition of Escherichia coli lipopolysaccharide-induced COX2 activity in mouse J774 cells assessed as decrease in PGE2 levels after 24 hrs by RIAMore data for this Ligand-Target Pair
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Sankyo
Curated by ChEMBL
Sankyo
Curated by ChEMBL
Affinity DataIC50: 253nMAssay Description:Inhibitory concentration against translocase-IMore data for this Ligand-Target Pair
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Sankyo
Curated by ChEMBL
Sankyo
Curated by ChEMBL
Affinity DataIC50: 267nMAssay Description:Inhibitory concentration required against Translocase IMore data for this Ligand-Target Pair
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Sankyo
Curated by ChEMBL
Sankyo
Curated by ChEMBL
Affinity DataIC50: 275nMAssay Description:Inhibitory concentration required against Translocase IMore data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Ability to inhibit [3H]nitrendipine binding to the L-type calcium channel receptor(CCR) in rat heart homogenate.More data for this Ligand-Target Pair
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Sankyo
Curated by ChEMBL
Sankyo
Curated by ChEMBL
Affinity DataIC50: 371nMAssay Description:Inhibitory concentration required against Translocase IMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of COX2 in human whole blood assessed as reduction in LPS-induced PGE2 generation pre-treated prior to LPS-challengeMore data for this Ligand-Target Pair
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