Affinity DataKi: 4nMAssay Description:Binding affinity to wild type FKBP51 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity to wild type FKBP51 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 7.5nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity to FKBP52 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity to wild type FKBP51 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity to wild type FKBP51 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Binding affinity to FKBP51 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 306nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 447nMAssay Description:Binding affinity to FKBP51 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 936nMAssay Description:Binding affinity to FKBP52 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 958nMAssay Description:Binding affinity to FKBP51 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.18E+3nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity to CypA (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.69E+3nMAssay Description:Binding affinity to FKBP52 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity to CypD (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nMAssay Description:Binding affinity to CypB (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Binding affinity to CypA (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Binding affinity to CypD (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Binding affinity to CypD (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Binding affinity to CypA (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.40E+3nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to FKBP52 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to FKBP51 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+4nMAssay Description:Binding affinity to CypA (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2.30E+4nMAssay Description:Binding affinity to wild type FKBP51 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to FKBP52 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to FKBP52 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to FKBP52 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to FKBP52 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.10E+4nMAssay Description:Binding affinity to wild type FKBP51 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.30E+4nMAssay Description:Binding affinity to CypB (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to FKBP52 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to FKBP52 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of CypA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of CypA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of CypA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 520nMAssay Description:Inhibition of CypA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.42E+3nMAssay Description:Inhibition of CypD (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 6.28E+3nMAssay Description:Inhibition of CypD (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of CypB (unknown origin)More data for this Ligand-Target Pair
TargetHeat shock factor protein 1(Homo sapiens (Human))
University of California At San Francisco
Curated by ChEMBL
University of California At San Francisco
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of recombinant human HSF1 expressed in Escherichia coli BL21 (DE3) assessed as reduction in HSF1 trimer-5-fluorescein labeled HSE interact...More data for this Ligand-Target Pair
TargetHeat shock factor protein 1(Homo sapiens (Human))
University of California At San Francisco
Curated by ChEMBL
University of California At San Francisco
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of recombinant human HSF1 expressed in Escherichia coli BL21 (DE3) assessed as reduction in HSF1 trimer-5-fluorescein labeled HSE interact...More data for this Ligand-Target Pair