Affinity DataKi: 0.0310nMAssay Description:Binding affinity at Opioid receptor delta 1 using rat brain receptor (P2 synaptosome) assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0350nMAssay Description:Binding affinity at Opioid receptor delta 1 using rat brain receptor (P2 synaptosome) assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0400nMAssay Description:Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by H-Dmt-Tic-OH displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.0420nMAssay Description:Binding affinity at Opioid receptor delta 1 using rat brain receptor (P2 synaptosome) assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0450nMAssay Description:Displacement of [3H]-DPDPE (0.63 nM) from Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 0.0540nMAssay Description:Displacement of [3H]-DPDPE (0.63 nM) from Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 0.0540nMAssay Description:Displacement of [3H]-DPDPE (0.63 nM) from Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 0.0580nMAssay Description:Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by [3H]N,N-(Me)2-Dmt-Tic-OH displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.0660nMAssay Description:Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by [3H]N,N-(Me)2-Dmt-Tic-OH displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.0670nMAssay Description:Binding affinity at Opioid receptor delta 1 using rat brain receptor (P2 synaptosome) assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Tested for inhibition of amplification of electrically induced twitch in guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Binding affinity was determined on delta [3H]-DPDPE site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0730nMAssay Description:Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by [3H]N,N-(Me)2-Dmt-Tic-OH displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.0755nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by H-Dmt-Tic-OH displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by H-Dmt-Tic-OH displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Affinity of the compound was assessed using competitive binding assay labeled with [3H]-DPDPE (6.3 nM) for Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 0.118nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by H-Dmt-Tic-OH displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by H-Dmt-Tic-OH displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Affinity of the compound was assessed using competitive binding assay labeled with [3H]-DPDPE (6.3 nM) for Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Binding affinity against opioid receptor delta in rats by displacing [3H]-DPDPEMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Binding affinity at Opioid receptor delta 1 using rat brain receptor (P2 synaptosome) assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.136nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by H-Dmt-Tic-OH displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Affinity of the compound was assessed using competitive binding assay labeled with [3H]-DPDPE (6.3 nM) for Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Displacement of [3H]-DPDPE (0.63 nM) from Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by [3H]N,N-(Me)2-Dmt-Tic-OH displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Binding affinity for rat brain P2 synaptosome Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Binding affinity for rat brain P2 synaptosome Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity was determined on delta [3H]-DPDPE site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Affinity of the compound was assessed using competitive binding assay labeled with [3H]-DPDPE (6.3 nM) for Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 0.203nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:Binding affinity at Opioid receptor delta 1 using rat brain receptor (P2 synaptosome) assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Binding affinity at Opioid receptor delta 1 using rat brain receptor (P2 synaptosome) assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by [3H]N,N-(Me)2-Dmt-Tic-OH displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Binding affinity against opioid receptor delta in rats by displacing [3H]-DPDPEMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Binding affinity at Opioid receptor mu 1 from rat brain synaptosomal preparations by [3H]-DAGO displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by [3H]N,N-(Me)2-Dmt-Tic-OH displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]-DAGO (1.28 nM) from Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by H-Dmt-Tic-OH displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Binding affinity for rat brain P2 synaptosome Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 0.285nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
Affinity DataKi: 0.285nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Binding affinity was determined on delta [3H]-DPDPE site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Inhibitory concentration against Opioid receptor delta 1 in mouse vas deferens using competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPEMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by [3H]N,N-(Me)2-Dmt-Tic-OH displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Affinity of the compound was assessed using competitive binding assay labeled with [3H]- DAGO (1.28 nM) for Opioid receptor mu 1More data for this Ligand-Target Pair