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Found 125 with Last Name = 'pégurier' and Initial = 'c'
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214136(4-(((4-nitrophenethyl)(1-(2,6-difluorobenzoyl)pipe...)
Affinity DataIC50:  6.30nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214142(4-(((4-nitrophenethyl)(1-picolinoylpiperidin-4-yl)...)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214124(4-(((4-nitrophenethyl)(1-(2,4-dimethylnicotinoyl)p...)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214121(4-(((4-chlorophenethyl)(1-(2,6-difluorobenzoyl)pip...)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at human CCR3 receptor assessed as inhibition of eotaxin-induced eosinophil shape changeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214121(4-(((4-chlorophenethyl)(1-(2,6-difluorobenzoyl)pip...)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at human CCR3 receptor assessed as inhibition of calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214121(4-(((4-chlorophenethyl)(1-(2,6-difluorobenzoyl)pip...)
Affinity DataIC50:  20nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214127(4-(((4-chlorophenethyl)(1-(2,6-difluorobenzoyl)pip...)
Affinity DataIC50:  25nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423088(CHEMBL396031)
Affinity DataIC50:  32nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214123(4-(((4-chlorophenethyl)(1-(2,6-difluorobenzoyl)pip...)
Affinity DataIC50:  32nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214140(4-(((4-chlorophenethyl)(1-(2,6-difluorobenzoyl)pip...)
Affinity DataIC50:  40nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423097(CHEMBL438129)
Affinity DataIC50:  50nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 12 member 5(Rattus norvegicus)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50315368(CHEMBL1090182 | benzyl 1-acetyl-2-(4-methoxy-3-(tr...)
Affinity DataIC50:  50nMAssay Description:Antagonist activity of rat KCC2 transporter expressed in human SK-Hep cells assessed as inhibition of N-ethylmaleimide-mediated Rb+ influx after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 12 member 5(Rattus norvegicus)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50315367(CHEMBL1089847 | benzyl 1-acetyl-2-(4-fluoro-3-(tri...)
Affinity DataIC50:  60nMAssay Description:Antagonist activity of rat KCC2 transporter expressed in human SK-Hep cells assessed as inhibition of N-ethylmaleimide-mediated Rb+ influx after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214130(4-(((4-chlorophenethyl)(1-(2,6-difluorobenzoyl)pip...)
Affinity DataIC50:  63nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423077(CHEMBL232031)
Affinity DataIC50:  79nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214133(4-(((4-chlorophenethyl)(1-(2,6-difluorobenzoyl)pip...)
Affinity DataIC50:  79nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 12 member 5(Rattus norvegicus)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50315366(CHEMBL1092661 | benzyl 1-acetyl-2-(3-(trifluoromet...)
Affinity DataIC50:  80nMAssay Description:Antagonist activity of rat KCC2 transporter expressed in human SK-Hep cells assessed as inhibition of N-ethylmaleimide-mediated Rb+ influx after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423101(CHEMBL396030)
Affinity DataIC50:  100nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214137(4-(((4-chlorophenethyl)(1-(2,6-difluorobenzoyl)pip...)
Affinity DataIC50:  100nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214129(4-(((4-chlorophenethyl)(1-(2,6-difluorobenzoyl)pip...)
Affinity DataIC50:  100nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214132(4-(((4-chlorophenethyl)(1-(2,6-difluorobenzoyl)pip...)
Affinity DataIC50:  100nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214131(4-(((4-chlorophenethyl)(1-(2,6-difluorobenzoyl)pip...)
Affinity DataIC50:  100nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214134(4-(((4-chlorophenethyl)(1-(2,6-difluorobenzoyl)pip...)
Affinity DataIC50:  100nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214146(4-(((4-chlorophenethyl)(1-(2,6-difluorobenzoyl)pip...)
Affinity DataIC50:  100nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214141(4-(((4-chlorophenethyl)(1-(2,6-difluorobenzoyl)pip...)
Affinity DataIC50:  100nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423098(CHEMBL233671)
Affinity DataIC50:  126nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214145(4-(((1-(1-naphthoyl)piperidin-4-yl)(4-phenylbutyl)...)
Affinity DataIC50:  158nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423076(CHEMBL234101)
Affinity DataIC50:  158nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214122(4-(4-(((4-chlorophenethyl)(1-(2,6-difluorobenzoyl)...)
Affinity DataIC50:  158nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 12 member 5(Rattus norvegicus)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50315362(CHEMBL1092325 | benzyl 1-acetyl-2-(4-cyanobenzyl)p...)
Affinity DataIC50:  160nMAssay Description:Antagonist activity of rat KCC2 transporter expressed in human SK-Hep cells assessed as inhibition of N-ethylmaleimide-mediated Rb+ influx after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423084(CHEMBL233675)
Affinity DataIC50:  200nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423067(CHEMBL234005)
Affinity DataIC50:  200nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 12 member 5(Rattus norvegicus)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50384302(CHEMBL2030663)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat KCC2 expressed in human Sk-Hep cells assessed as induction off Rb+ flux by atomic absorption spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 12 member 5(Rattus norvegicus)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50384300(CHEMBL2030661)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat KCC2 expressed in human Sk-Hep cells assessed as induction off Rb+ flux by atomic absorption spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 12 member 5(Rattus norvegicus)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50315359(CHEMBL1092255 | benzyl 1-acetyl-2-(4-fluorobenzyl)...)
Affinity DataIC50:  200nMAssay Description:Antagonist activity of rat KCC2 transporter expressed in human SK-Hep cells assessed as inhibition of N-ethylmaleimide-mediated Rb+ influx after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214143(4-({[2-(4-chloro-phenyl)-ethyl]-[1-(1-oxy-pyridine...)
Affinity DataIC50:  200nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214135(4-(((4-fluorophenethyl)(1-(2,6-difluorobenzoyl)pip...)
Affinity DataIC50:  200nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214125(4-(((4-chlorophenethyl)(1-(2,6-difluorobenzoyl)pip...)
Affinity DataIC50:  250nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 12 member 5(Rattus norvegicus)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50315365(CHEMBL1092338 | benzyl 1-acetyl-2-(3-(methylsulfon...)
Affinity DataIC50:  250nMAssay Description:Antagonist activity of rat KCC2 transporter expressed in human SK-Hep cells assessed as inhibition of N-ethylmaleimide-mediated Rb+ influx after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 12 member 5(Rattus norvegicus)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50384298(CHEMBL2030659)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat KCC2 expressed in human Sk-Hep cells assessed as induction off Rb+ flux by atomic absorption spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 12 member 5(Rattus norvegicus)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50384301(CHEMBL2030662)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat KCC2 expressed in human Sk-Hep cells assessed as induction off Rb+ flux by atomic absorption spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423085(CHEMBL390036 | CHEMBL535624 | CHEMBL535625)
Affinity DataIC50:  316nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423074(CHEMBL234304)
Affinity DataIC50:  316nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 12 member 5(Rattus norvegicus)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50315376(CHEMBL1093303 | benzyl 2-benzyl-1-(cyclopropanecar...)
Affinity DataIC50:  320nMAssay Description:Antagonist activity of rat KCC2 transporter expressed in human SK-Hep cells assessed as inhibition of N-ethylmaleimide-mediated Rb+ influx after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 12 member 5(Rattus norvegicus)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50315363(CHEMBL1092336 | benzyl 1-acetyl-2-(3-cyanobenzyl)p...)
Affinity DataIC50:  320nMAssay Description:Antagonist activity of rat KCC2 transporter expressed in human SK-Hep cells assessed as inhibition of N-ethylmaleimide-mediated Rb+ influx after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 12 member 5(Rattus norvegicus)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50315360(CHEMBL1092256 | benzyl 1-acetyl-2-(4-chlorobenzyl)...)
Affinity DataIC50:  320nMAssay Description:Antagonist activity of rat KCC2 transporter expressed in human SK-Hep cells assessed as inhibition of N-ethylmaleimide-mediated Rb+ influx after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 12 member 5(Rattus norvegicus)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50315350((+)-benzyl 1-acetyl-2-benzylpyrrolidine-2-carboxyl...)
Affinity DataIC50:  320nMAssay Description:Antagonist activity of rat KCC2 transporter expressed in human SK-Hep cells assessed as inhibition of N-ethylmaleimide-mediated Rb+ influx after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 12 member 5(Rattus norvegicus)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50315361((+)-benzyl 1-acetyl-2-(4-(methylsulfonyl)benzyl)py...)
Affinity DataIC50:  400nMAssay Description:Antagonist activity of rat KCC2 transporter expressed in human SK-Hep cells assessed as inhibition of N-ethylmaleimide-mediated Rb+ influx after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50214147(CHEMBL392405 | N-(4-(4-(((4-chlorophenethyl)(1-(2,...)
Affinity DataIC50:  400nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 12 member 5(Rattus norvegicus)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50315373(2-benzyl 1-methyl 2-benzylpyrrolidine-1,2-dicarbox...)
Affinity DataIC50:  400nMAssay Description:Antagonist activity of rat KCC2 transporter expressed in human SK-Hep cells assessed as inhibition of N-ethylmaleimide-mediated Rb+ influx after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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