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Found 102 with Last Name = 'severin' and Initial = 'c'
TargetMu-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073519((S)-1-[(S)-2-[2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hy...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]-DAGO from Opioid receptor mu 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50001468((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]-NLT from Opioid receptor delta 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50059841((S)-1-[(S)-2-[2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hy...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-DAGO from Opioid receptor mu 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073517((S)-1-[(S)-2-[2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hy...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]-DAGO from Opioid receptor mu 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073522(2-({1-[2-(2-{2-[2-(2-Amino-2-(4-hydroxy-phenyl)-ac...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]-DAGO from Opioid receptor mu 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073523(2-({1-[2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-DAGO from Opioid receptor mu 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073518(2-({1-[2-(2-{2-[2-(2-Amino-2-[4-hydroxy-phenyl]-ac...)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]-DAGO from Opioid receptor mu 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073525(2-({1-[2-(2-{2-[2-(2-Amino-2-[4-hydroxy-phenyl]-ac...)
Affinity DataKi:  11.2nMAssay Description:Displacement of [3H]-DAGO from Opioid receptor mu 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073515(CHEMBL405663 | N-(1-{1-[1-(3-Acetoxy-4,5,6-trihydr...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-NLT from Opioid receptor delta 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073521(CHEMBL429717 | N-(1-{1-[1-(3-Acetoxy-4,5,6-trihydr...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]-NLT from Opioid receptor delta 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073524((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]-NLT from Opioid receptor delta 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073520((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]-NLT from Opioid receptor delta 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073516(CHEMBL268625 | N-(1-{1-[1-(3-Acetoxy-4,5,6-trihydr...)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]-NLT from Opioid receptor delta 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073526(3-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylami...)
Affinity DataKi:  176nMAssay Description:Displacement of [3H]-NLT from Opioid receptor delta 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073515(CHEMBL405663 | N-(1-{1-[1-(3-Acetoxy-4,5,6-trihydr...)
Affinity DataKi:  879nMAssay Description:Displacement of [3H]-DAGO from Opioid receptor mu 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50059841((S)-1-[(S)-2-[2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hy...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]-NLT from Opioid receptor delta 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073524((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]-DAGO from Opioid receptor mu 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073517((S)-1-[(S)-2-[2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hy...)
Affinity DataKi:  1.11E+3nMAssay Description:Displacement of [3H]-NLT from Opioid receptor delta 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073522(2-({1-[2-(2-{2-[2-(2-Amino-2-(4-hydroxy-phenyl)-ac...)
Affinity DataKi:  1.25E+3nMAssay Description:Displacement of [3H]-NLT from Opioid receptor delta 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073518(2-({1-[2-(2-{2-[2-(2-Amino-2-[4-hydroxy-phenyl]-ac...)
Affinity DataKi:  1.32E+3nMAssay Description:Displacement of [3H]-NLT from Opioid receptor delta 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073519((S)-1-[(S)-2-[2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hy...)
Affinity DataKi:  1.41E+3nMAssay Description:Displacement of [3H]-NLT from Opioid receptor delta 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073526(3-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylami...)
Affinity DataKi:  1.59E+3nMAssay Description:Displacement of [3H]-DAGO from Opioid receptor mu 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073520((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]-DAGO from Opioid receptor mu 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073521(CHEMBL429717 | N-(1-{1-[1-(3-Acetoxy-4,5,6-trihydr...)
Affinity DataKi:  1.92E+3nMAssay Description:Displacement of [3H]-DAGO from Opioid receptor mu 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50001468((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  1.98E+3nMAssay Description:Displacement of [3H]-DAGO from Opioid receptor mu 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073516(CHEMBL268625 | N-(1-{1-[1-(3-Acetoxy-4,5,6-trihydr...)
Affinity DataKi:  2.83E+3nMAssay Description:Displacement of [3H]-DAGO from Opioid receptor mu 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073523(2-({1-[2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  2.85E+3nMAssay Description:Displacement of [3H]-NLT from Opioid receptor delta 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50073525(2-({1-[2-(2-{2-[2-(2-Amino-2-[4-hydroxy-phenyl]-ac...)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-NLT from Opioid receptor delta 1 of adult male mouse brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM283216(4-[2-(4-amino-piperidin-1-yl)-5- (3-fluoro-4-metho...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of LSD1 (unknown origin) using H3K4me1 substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM501809(4-[6-(4-amino-piperidin-1-yl)-4- methyl-5-oxo-3-p...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of LSD1 (unknown origin) using H3K4me1 substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM283129(4-[2-(4-amino-piperidin-1-yl)-5- (4-methoxyphenyl)...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of LSD1 (unknown origin) using H3K4me1 substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM50503504(CHEMBL4444902 | US10626103, Example 54)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM283200(4-[2-(4-amino-piperidin-1-yl)-5-(4- methoxyphenyl)...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of LSD1 (unknown origin) using H3K4me1 substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM50503514(CHEMBL4522607 | US10626103, Example 55)
Affinity DataIC50:  1nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM283128(4-(2-(4-aminopiperidin-1-yl)- 1-methyl-6-oxo-5-p-t...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of LSD1 (unknown origin) using H3K4me1 substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM501778(4-[6-(4-aminopiperidin-1-yl)-4- methyl-3-(4-methy...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of LSD1 (unknown origin) using H3K4me1 substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM50554230(CHEMBL4748670)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of LSD1 (unknown origin) using H3K4me1 substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM50503507(CHEMBL4451607 | US10626103, Example 53)
Affinity DataIC50:  2nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM50554231(CHEMBL4796870)
Affinity DataIC50:  2nMAssay Description:Inhibition of LSD1 (unknown origin) using H3K4me1 substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM301089(4-[2-(4-aminopiperidin-1-yl)-5-(4- methylphenyl)py...)
Affinity DataIC50:  3nMAssay Description:Inhibition of LSD1 (unknown origin) using H3K4me1 substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM50503493(CHEMBL4448358 | US10626103, Example 23)
Affinity DataIC50:  3nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM50503503(CHEMBL4548929 | US10626103, Example 22)
Affinity DataIC50:  3nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM50503505(CHEMBL4516248 | US10626103, Example 49)
Affinity DataIC50:  4nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM50503516(CHEMBL4447527 | US10626103, Example 12)
Affinity DataIC50:  4nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM50503499(CHEMBL4454128 | US10626103, Example 18)
Affinity DataIC50:  4nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM50503500(CHEMBL4451430 | US10626103, Example 62)
Affinity DataIC50:  5nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM50503509(CHEMBL4440004 | US10626103, Example 16)
Affinity DataIC50:  7nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM50503495(CHEMBL4514358 | US10626103, Example 94)
Affinity DataIC50:  7nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM283216(4-[2-(4-amino-piperidin-1-yl)-5- (3-fluoro-4-metho...)
Affinity DataIC50:  7nMAssay Description:Inhibition of LSD1 in human THP1 cells assessed as induction of cell differentiation by measuring CD11b expression incubated for 96 hrs by FACS assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Fount Therapeutics

Curated by ChEMBL
LigandPNGBDBM50503508(CHEMBL4569059 | US10626103, Example 11)
Affinity DataIC50:  8nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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