Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rattus norvegicus)
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 0.0700nMAssay Description:Inhibition of recombinant Steroid 5-alpha-reductase type I was evaluated as binding affinity (in vitro)More data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rattus norvegicus)
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Inhibition of recombinant Steroid 5-alpha-reductase type I was evaluated as binding affinity of the compoundMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rattus norvegicus)
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 0.120nMAssay Description:Inhibitory activity was measured on rat Steroid 5-alpha-reductase type 2More data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Binding affinity to recombinant human Steroid 5-alpha-reductase type I was evaluatedMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rattus norvegicus)
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 0.170nMAssay Description:Inhibitory activity was measured on rat Steroid 5-alpha-reductase type 2More data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rattus norvegicus)
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Inhibition of recombinant Steroid 5-alpha-reductase type I was evaluated as binding affinity of the compoundMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Inhibition of wild type fully glycosylated human recombinant CD38-catalyzed NAD hydrolysisMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:In vitro inhibitory activity against human type 1 5-alpha reductaseMore data for this Ligand-Target Pair
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Inhibition of wild type fully glycosylated human recombinant CD38-catalyzed NAD hydrolysisMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Inhibition of wild type fully glycosylated human recombinant CD38-catalyzed NAD hydrolysisMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:In vitro inhibitory activity against human type 1 5-alpha reductaseMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:In vitro inhibitory activity against human type 1 5-alpha reductaseMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rattus norvegicus)
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Inhibitory activity was measured on rat Steroid 5-alpha-reductase type 2More data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:In vitro inhibitory activity against human type 1 5-alpha reductaseMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:In vitro inhibitory activity against human type 1 5-alpha reductaseMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 3.60nMAssay Description:In vitro inhibitory activity against human type 1 5-alpha reductaseMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 3.60nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:In vitro inhibitory activity against human type 1 5-alpha reductaseMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 4.20nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:In vitro inhibitory activity against human type 1 5-alpha reductaseMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:In vitro inhibitory activity against human type 1 5-alpha reductaseMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:In vitro inhibitory activity against human type 1 5-alpha reductaseMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 6.40nMAssay Description:In vitro inhibitory activity against human type 1 5-alpha reductaseMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 6.70nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 6.80nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rattus norvegicus)
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 6.80nMAssay Description:Inhibition of recombinant Steroid 5-alpha-reductase type I was evaluated as binding affinity (in vitro)More data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 6.90nMAssay Description:In vitro inhibitory activity against human type 1 5-alpha reductaseMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 6.90nMAssay Description:Inhibition of recombinant human 5-alpha reductase-1 at a concentration of 5 microL after preincubation for 10 minutesMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 7.5nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Inhibition of recombinant steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 8.20nMAssay Description:Inhibition of recombinant human 5-alpha reductase-1 at a concentration of 5 microL after preincubation for 10 minutesMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by ChEMBL
Glaxo Inc. Research Institute
Curated by ChEMBL
Affinity DataKi: 8.20nMAssay Description:In vitro inhibitory activity against human type 1 5-alpha reductaseMore data for this Ligand-Target Pair