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Found 213 with Last Name = 'baglini' and Initial = 'e'
TargetTranslocator protein(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50421116(CHEMBL2088374)
Affinity DataKi:  0.280nMAssay Description:Binding affinity to TSPO (unknown origin) relative to controlMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM22041(2-[6-chloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridi...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50588817(CHEMBL5193551)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO receptor in Wistar rat brain without cerebellum incubated for 90 mins by liquid scintillation counter an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50341401(CHEMBL4165351)
Affinity DataKi:  0.730nMAssay Description:Inhibition of recombinant human CA9 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Bos taurus)
Niddk

Curated by ChEMBL
LigandPNGBDBM50019213(1,3-dihydro-7-nitro-5-(2-chlorophenyl)-2H-1,4.benz...)
Affinity DataKi:  0.850nMAssay Description:Binding affinity to bovine brain membrane BzR assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50341404(CHEMBL4169089)
Affinity DataKi:  0.880nMAssay Description:Inhibition of recombinant human CA9 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Bos taurus)
Niddk

Curated by ChEMBL
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to bovine brain membrane BzR assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO receptor in Wistar rat brain without cerebellum incubated for 90 mins by liquid scintillation counter an...More data for this Ligand-Target Pair
TargetCathepsin K(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50601464(CHEMBL5195850)
Affinity DataKi:  1.80nMAssay Description:Inhibition of human Cathepsin K assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50143225(CHEMBL300762 | N,N-Dibutyl-2-[5-chloro-2-(4-chloro...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]-PK11195 from rat kidney mitochondrial membrane TSPO receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50588815(CHEMBL5208364)
Affinity DataKi:  4.90nMAssay Description:Binding affinity to TSPO in Sprague-Dawley rat brainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50341401(CHEMBL4165351)
Affinity DataKi:  5.20nMAssay Description:Inhibition of recombinant human CA2 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50341397(CHEMBL4176953)
Affinity DataKi:  5.20nMAssay Description:Inhibition of recombinant human CA9 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50601465(CHEMBL5204536)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]-PK11195 from rat kidney mitochondrial membrane TSPO receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50143238(2-[5-Chloro-2-(4-chloro-phenyl)-1H-indol-3-yl]-N,N...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]-PK11195 from rat kidney mitochondrial membrane TSPO receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50588814(CHEMBL5181329)
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]-PK11195 from TSPO receptor in Sprague-Dawley rat brain incubated for 30 mins by auto-gamma scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50243007(2-(2-(4-(2-Fluoroethoxy)phenyl)-5,7-dimethylpyrazo...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]-PK11195 from TSPO receptor in Wistar rat Kidney assessed as inhibition constant incubated for 90 mins by liquid scintillation co...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM22041(2-[6-chloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridi...)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO receptor in Wistar rat brain without cerebellum incubated for 90 mins by liquid scintillation counter an...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50341404(CHEMBL4169089)
Affinity DataKi:  8.60nMAssay Description:Inhibition of recombinant human CA2 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataKi:  9.30nMAssay Description:Displacement of [3H]-PK11195 from rat kidney mitochondrial membrane TSPO receptor assessed as inhibition constantMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 4(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50341397(CHEMBL4176953)
Affinity DataKi:  9.5nMAssay Description:Inhibition of recombinant human CA4 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  12nMAssay Description:Inhibition of recombinant human CA2 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50258312(CHEMBL4095528)
Affinity DataKi:  18nMAssay Description:Inhibition of Calpain I (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50588816(CHEMBL5191240)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO receptor in Wistar rat brain without cerebellum incubated for 90 mins by liquid scintillation counter an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM22040(4 -chlorodiazepam | 4' Cl-diazepam | 7-chloro-...)
Affinity DataKi:  23nMAssay Description:Binding affinity rat kidney mitochondrial membrane TSPO receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  26nMAssay Description:Inhibition of recombinant human CA9 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50601464(CHEMBL5195850)
Affinity DataKi:  28nMAssay Description:Inhibition of human Cathepsin B assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50258383(CHEMBL4063636)
Affinity DataKi:  34nMAssay Description:Inhibition of Calpain I (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50341404(CHEMBL4169089)
Affinity DataKi:  40nMAssay Description:Inhibition of recombinant human CA4 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50601464(CHEMBL5195850)
Affinity DataKi:  56nMAssay Description:Inhibition of human Calpain I assessed as dissociation constant using Suc-Leu-Tyr-AMC as substrate preincubated for 15 mins followed by compound addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  74nMAssay Description:Inhibition of recombinant human CA4 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50341397(CHEMBL4176953)
Affinity DataKi:  78nMAssay Description:Inhibition of recombinant human CA2 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50601468(CHEMBL5179024)
Affinity DataKi:  108nMAssay Description:Displacement of [3H] PK11195 from TSPO in human U-87 MGcell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranslocator protein(Bos taurus)
Niddk

Curated by ChEMBL
LigandPNGBDBM50055261(CHEMBL75307 | N-Benzyl-2-(5-nitro-1H-indol-3-yl)-2...)
Affinity DataKi:  117nMAssay Description:Binding affinity to bovine brain membrane BzR assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProcathepsin L(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50601464(CHEMBL5195850)
Affinity DataKi:  137nMAssay Description:Inhibition of human Cathepsin L assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50601467(CHEMBL5169788)
Affinity DataKi:  202nMAssay Description:Displacement of [3H] PK11195 from TSPO (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50341401(CHEMBL4165351)
Affinity DataKi:  214nMAssay Description:Inhibition of recombinant human CA4 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  250nMAssay Description:Inhibition of recombinant human CA1 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50341404(CHEMBL4169089)
Affinity DataKi:  272nMAssay Description:Inhibition of recombinant human CA1 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50341401(CHEMBL4165351)
Affinity DataKi:  296nMAssay Description:Inhibition of recombinant human CA1 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50573533(CHEMBL4873134)
Affinity DataKi:  410nMAssay Description:Inhibition of recombinant human CA2 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50601466(CHEMBL5172740)
Affinity DataKi:  438nMAssay Description:Displacement of [3H] PK11195 from TSPO (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50341397(CHEMBL4176953)
Affinity DataKi:  746nMAssay Description:Inhibition of recombinant human CA1 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50573535(CHEMBL4861393)
Affinity DataKi:  930nMAssay Description:Inhibition of recombinant human CA4 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50573524(CHEMBL4878097)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of recombinant human CA1 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50573534(CHEMBL4872990)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of recombinant human CA2 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50573542(CHEMBL4872434)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of recombinant human CA2 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50601464(CHEMBL5195850)
Affinity DataKi:  3.29E+3nMAssay Description:Inhibition of human Cathepsin S assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50573543(CHEMBL4878111)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition of recombinant human CA2 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50573545(CHEMBL4853204)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of recombinant human CA2 preincubated for 15 mins by phenol red dye-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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