Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 7nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 10nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of human CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]E1 from human placental 17beta-HSD1 after 10 mins by fluid scintillation countingMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 20nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 20nMAssay Description:Inhibition of human placental 17beta-HSD1 assessed as conversion of [3H]estrone to [3H]17beta-estradiolMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 20nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 20nMAssay Description:Displacement of [3H]E1 from human placental 17beta-HSD1 after 10 mins by fluid scintillation countingMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 23nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 26nMAssay Description:Displacement of [3H]E1 from human placental 17beta-HSD1 after 10 mins by fluid scintillation countingMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 30nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 33nMAssay Description:Displacement of [3H]E1 from human placental 17beta-HSD1 after 10 mins by fluid scintillation countingMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 36nMAssay Description:Displacement of [3H]E1 from human placental 17beta-HSD1 after 10 mins by fluid scintillation countingMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 39nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 40nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 40nMAssay Description:Inhibition of human placental 17beta-HSD1 assessed as conversion of [3H]estrone to [3H]17beta-estradiolMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 50nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 50nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 52nMAssay Description:Inhibition of human placental 17beta-HSD1More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 53nMAssay Description:Displacement of [3H]E1 from human placental 17beta-HSD1 after 10 mins by fluid scintillation countingMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 60nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 64nMAssay Description:Displacement of [3H]E1 from human placental 17beta-HSD1 after 10 mins by fluid scintillation countingMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 70nMAssay Description:Displacement of [3H]E1 from human placental 17beta-HSD1 after 10 mins by fluid scintillation countingMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 70nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 71nMAssay Description:Displacement of [3H]E1 from 17beta-HSD1 in human T47D cells after 10 mins by fluid scintillation countingMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 90nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 114nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 115nMAssay Description:Displacement of [3H]E1 from 17beta-HSD1 in human T47D cells after 10 mins by fluid scintillation countingMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 116nMAssay Description:Inhibition of human placental 17beta-HSD1More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 116nMAssay Description:Inhibition of human placental 17beta-HSD1 assessed as conversion of [3H]estrone to [3H]17beta-estradiolMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 116nMAssay Description:Displacement of [3H]E1 from human placental 17beta-HSD1 after 10 mins by fluid scintillation countingMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 140nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 165nMAssay Description:Displacement of [3H]E1 from 17beta-HSD1 in human T47D cells after 10 mins by fluid scintillation countingMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 195nMAssay Description:The determination of IC50 values was performed with enzyme isolated from human placenta (Luu-The, V. et al., J. Steroid Biochem. Mol. Biol., 55:581-5...More data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 221nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
Affinity DataIC50: 224nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Universitaet Des Saarlandes
US Patent
Universitaet Des Saarlandes
US Patent
Affinity DataIC50: 229nMAssay Description:Displacement of [3H]E1 from 17beta-HSD1 in human T47D cells after 10 mins by fluid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
Affinity DataIC50: 259nMAssay Description:Inhibition assay using P450 CYP enzymes.More data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair