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Found 17 with Last Name = 'delouvroy' and Initial = 'f'
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Tibotec

Curated by ChEMBL
LigandPNGBDBM50204832(4-(2-(5-bromo-2-fluorophenyl)pteridin-4-ylamino)-N...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Tibotec

Curated by ChEMBL
LigandPNGBDBM50204832(4-(2-(5-bromo-2-fluorophenyl)pteridin-4-ylamino)-N...)
Affinity DataIC50:  37nMAssay Description:Inhibition of human JNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Tibotec

Curated by ChEMBL
LigandPNGBDBM50204832(4-(2-(5-bromo-2-fluorophenyl)pteridin-4-ylamino)-N...)
Affinity DataIC50:  47nMAssay Description:Inhibition of human VEGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Tibotec

Curated by ChEMBL
LigandPNGBDBM50204834(2-(5-chloro-2-fluorophenyl)-N-(pyridin-4-yl)pterid...)
Affinity DataIC50:  53nMAssay Description:Inhibition of TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Tibotec

Curated by ChEMBL
LigandPNGBDBM50204832(4-(2-(5-bromo-2-fluorophenyl)pteridin-4-ylamino)-N...)
Affinity DataIC50:  59nMAssay Description:Inhibition of human JNK3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Tibotec

Curated by ChEMBL
LigandPNGBDBM50204832(4-(2-(5-bromo-2-fluorophenyl)pteridin-4-ylamino)-N...)
Affinity DataIC50:  123nMAssay Description:Inhibition of human VEGFR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Tibotec

Curated by ChEMBL
LigandPNGBDBM50204832(4-(2-(5-bromo-2-fluorophenyl)pteridin-4-ylamino)-N...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Tibotec

Curated by ChEMBL
LigandPNGBDBM50336504((2R,3aR,10Z,11aS,12aR,14aR)-N-(cyclopropylsulfonyl...)
Affinity DataIC50:  800nMAssay Description:Inhibition of human cathepsin S in human JY cells assessed as p10 accumulation by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Tibotec

Curated by ChEMBL
LigandPNGBDBM50204832(4-(2-(5-bromo-2-fluorophenyl)pteridin-4-ylamino)-N...)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibition of JNK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase subunit gamma-1(Homo sapiens (Human))
Tibotec

Curated by ChEMBL
LigandPNGBDBM50336503(10-acetyl-11-(3-(benzyloxy)-4-methoxyphenyl)-3,3-d...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human DNA polymerase gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase subunit gamma-1(Homo sapiens (Human))
Tibotec

Curated by ChEMBL
LigandPNGBDBM50336502(10-acetyl-11-(2,4-dichlorophenyl)-3,3-dimethyl-2,3...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human DNA polymerase gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha catalytic subunit(Homo sapiens (Human))
Tibotec

Curated by ChEMBL
LigandPNGBDBM50336502(10-acetyl-11-(2,4-dichlorophenyl)-3,3-dimethyl-2,3...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha catalytic subunit(Homo sapiens (Human))
Tibotec

Curated by ChEMBL
LigandPNGBDBM50336503(10-acetyl-11-(3-(benzyloxy)-4-methoxyphenyl)-3,3-d...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Homo sapiens (Human))
Tibotec

Curated by ChEMBL
LigandPNGBDBM50336502(10-acetyl-11-(2,4-dichlorophenyl)-3,3-dimethyl-2,3...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human DNA polymerase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Homo sapiens (Human))
Tibotec

Curated by ChEMBL
LigandPNGBDBM50336503(10-acetyl-11-(3-(benzyloxy)-4-methoxyphenyl)-3,3-d...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human DNA polymerase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Tibotec

Curated by ChEMBL
LigandPNGBDBM50336501(10-acetyl-11-(4-(benzyloxy)-2-chlorophenyl)-6-hydr...)
Affinity DataIC50: >3.00E+7nMAssay Description:Inhibition of peripheral benzodiazepine BZD receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Tibotec

Curated by ChEMBL
LigandPNGBDBM50336501(10-acetyl-11-(4-(benzyloxy)-2-chlorophenyl)-6-hydr...)
Affinity DataIC50: >3.00E+7nMAssay Description:Inhibition of peripheral benzodiazepine BZD receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed