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Found 149 with Last Name = 'grams' and Initial = 'f'
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068485((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  21nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pharmazeutisch-Chemisches Institut Der UniversitäT

Curated by ChEMBL
LigandPNGBDBM50070629(4-[2-(3-Benzenesulfonylamino-5-methyl-phenoxy)-eth...)
Affinity DataKi:  23nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068501((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  26nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068490(CHEMBL146940 | [4-(1-Carbamimidoyl-piperidin-4-ylo...)
Affinity DataKi:  28nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068493((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  30nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068494((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  30nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068488((S)-3-(7-Carbamimidoyl-naphthalen-2-yl)-2-{4-[(S)-...)
Affinity DataKi:  40nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068487(CHEMBL148357 | [4-(1-Carbamimidoyl-piperidin-4-ylo...)
Affinity DataKi:  44nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068506((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  55nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068493((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  80nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068499((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  80nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068502((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  100nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pharmazeutisch-Chemisches Institut Der UniversitäT

Curated by ChEMBL
LigandPNGBDBM50070633(CHEMBL289790 | N-[3-(4-Guanidino-butoxy)-5-methyl-...)
Affinity DataKi:  180nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068485((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  200nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068507((S)-3-{4-[(2-Carbamimidoyl-1,2,3,4-tetrahydro-isoq...)
Affinity DataKi:  200nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068486(CHEMBL147988 | [4-((S)-1-Carbamimidoyl-pyrrolidin-...)
Affinity DataKi:  200nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068487(CHEMBL148357 | [4-(1-Carbamimidoyl-piperidin-4-ylo...)
Affinity DataKi:  200nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068484((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  200nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068490(CHEMBL146940 | [4-(1-Carbamimidoyl-piperidin-4-ylo...)
Affinity DataKi:  200nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068500(CHEMBL344309 | [4-((S)-1-Carbamimidoyl-pyrrolidin-...)
Affinity DataKi:  200nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068491((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  200nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068501((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  200nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50062471(CHEMBL116150 | N-Hydroxy-2-isobutyl-N'-octyl-malon...)
Affinity DataKi:  240nMAssay Description:Inhibition of Matrix metalloproteinase-8 (Human neutrophil collagenase, MMP-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50066047(2-Benzyl-N-hydroxy-2-methyl-N'-(3-phenyl-propyl)-m...)
Affinity DataKi:  240nMAssay Description:Inhibition of human neutrophil collagenase (Matrix metalloproteinase-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pharmazeutisch-Chemisches Institut Der UniversitäT

Curated by ChEMBL
LigandPNGBDBM50070632(4-[2-(3-Benzenesulfonylamino-phenoxy)-ethylamino]-...)
Affinity DataKi:  300nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50066051(CHEMBL105352 | Indan-2,2-dicarboxylic acid hydroxy...)
Affinity DataKi:  300nMAssay Description:Inhibition of human neutrophil collagenase (Matrix metalloproteinase-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50066049(2-Benzyl-N-hydroxy-2-methyl-N'-(4-phenyl-butyl)-ma...)
Affinity DataKi:  380nMAssay Description:Inhibition of human neutrophil collagenase (Matrix metalloproteinase-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068505((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  400nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068494((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  400nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068495(CHEMBL148972 | [4-(1-Acetyl-piperidin-4-yloxy)-phe...)
Affinity DataKi:  400nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50062457(CHEMBL116557 | N-Hydroxy-2-phenethyl-N'-(3-phenyl-...)
Affinity DataKi:  490nMAssay Description:Inhibition of Matrix metalloproteinase-8 (Human neutrophil collagenase, MMP-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50062478(CHEMBL116641 | N-Hydroxy-2-isobutyl-N'-(3-phenyl-p...)
Affinity DataKi:  540nMAssay Description:Inhibition of Matrix metalloproteinase-8 (Human neutrophil collagenase, MMP-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50062453(2-Benzyl-N-hydroxy-N'-(3-phenyl-propyl)-malonamide...)
Affinity DataKi:  560nMAssay Description:Inhibition of Matrix metalloproteinase-8 (Human neutrophil collagenase, MMP-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pharmazeutisch-Chemisches Institut Der UniversitäT

Curated by ChEMBL
LigandPNGBDBM50070622(CHEMBL40704 | N-[3-(3-Guanidino-propoxy)-5-methyl-...)
Affinity DataKi:  630nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068498(CHEMBL342568 | [4-((S)-1-Allyl-pyrrolidin-3-yloxy)...)
Affinity DataKi:  1.00E+3nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068496((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  1.00E+3nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068486(CHEMBL147988 | [4-((S)-1-Carbamimidoyl-pyrrolidin-...)
Affinity DataKi:  1.00E+3nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50066040(2,N-Dibenzyl-N'-hydroxy-2-methyl-malonamide | CHEM...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human neutrophil collagenase (Matrix metalloproteinase-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50062479(CHEMBL119061 | N-Hydroxy-2-isobutyl-N'-[(S)-3-phen...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of Matrix metalloproteinase-8 (Human neutrophil collagenase, MMP-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50066037(CHEMBL100678 | Indan-2,2-dicarboxylic acid benzyla...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of human neutrophil collagenase (Matrix metalloproteinase-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50062456(2,N-Dihydroxy-N'-[(S)-3-phenyl-1-(2-p-tolyl-ethylc...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of Matrix metalloproteinase-8 (Human neutrophil collagenase, MMP-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50062458(2-Benzyl-N-hydroxy-N'-[(S)-3-phenyl-1-(2-p-tolyl-e...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of Matrix metalloproteinase-8 (Human neutrophil collagenase, MMP-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50066043(2,N-Dibenzyl-2,N'-dihydroxy-malonamide | CHEMBL322...)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of human neutrophil collagenase (Matrix metalloproteinase-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50066046(5,7-Dihydro-dibenzo[a,c]cycloheptene-6,6-dicarboxy...)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of human neutrophil collagenase (Matrix metalloproteinase-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068492((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  2.00E+3nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068488((S)-3-(7-Carbamimidoyl-naphthalen-2-yl)-2-{4-[(S)-...)
Affinity DataKi:  2.00E+3nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068506((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  2.00E+3nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068504((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  2.00E+3nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068502((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  2.00E+3nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
Boehringer Mannheim

Curated by ChEMBL
LigandPNGBDBM50068500(CHEMBL344309 | [4-((S)-1-Carbamimidoyl-pyrrolidin-...)
Affinity DataKi:  2.00E+3nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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