TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.350nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity to rat pituitary GnRH receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity to human recombinant GnRH receptorMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.570nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Competitive inhibition of GnRH-stimulated extracellular acidification in cells expressing recombinant rat GnRH receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.5nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.30nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:In vitro binding affinity towards rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:In vitro binding affinity to human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:In vitro binding affinity towards human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:In vitro binding affinity to human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair