Affinity DataKi: 0.00100nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.00500nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.00700nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.00800nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.00800nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.00900nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.00900nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.0130nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.0150nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:In vitro activity against rabbit FXa.More data for this Ligand-Target Pair
Affinity DataKi: 0.0400nMAssay Description:Binding affinity towards thrombin was tested.More data for this Ligand-Target Pair
Affinity DataKi: 0.0400nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.0400nMAssay Description:Binding affinity to human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.0410nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.0410nMAssay Description:In vitro for inhibition of thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.0450nMAssay Description:Compound was tested in vitro for inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Binding affinity towards thrombin was tested.More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Binding affinity towards thrombin was tested.More data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Binding affinity to human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.0900nMAssay Description:Binding affinity to human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: <0.100nMAssay Description:Binding affinity to human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.110nM ΔG°: -56.3kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Binding affinity to human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:In vitro for inhibition of thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.170nM ΔG°: -55.2kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
Affinity DataKi: 0.180nM ΔG°: -55.1kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Binding affinity to human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Binding affinity to human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.190nM ΔG°: -54.9kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
Affinity DataKi: 0.210nM ΔG°: -54.7kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
Affinity DataKi: 0.220nM ΔG°: -54.6kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Binding affinity to human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Binding affinity to human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:In vitro for inhibition of thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Binding affinity to human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Binding affinity to human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.25nM ΔG°: -54.3kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Binding affinity to human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.270nM ΔG°: -54.1kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Binding affinity towards thrombin was tested.More data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Binding affinity to human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human histamine H3 receptor expressed in CHOK1 cells after 1.5 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding affinity towards thrombin was tested.More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:In vitro activity against rabbit factor XaMore data for this Ligand-Target Pair