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Found 104 with Last Name = 'iegre' and Initial = 'j'
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of CLK2 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  15nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) using RRRADDSDDDD substrate incubated for 40 min...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50252622(CHEMBL4070389)
Affinity DataIC50:  370nMAssay Description:Inhibition of CK2alpha (unknown origin) using RRRADDSDDDD as substrate after 40 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461938(CHEMBL459510 | NSC-7223)
Affinity DataIC50:  400nMAssay Description:Inhibition of GST-tagged human recombinant CK2alpha (1 to 335 residues) expressed in Escherichia coli BL21 by radiometric kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50252622(CHEMBL4070389)
Affinity DataIC50:  670nMAssay Description:Binding affinity to CK2alpha/beta (unknown origin) expressed in Escherichia coli BL21(DE3) by ITCMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590137(CHEMBL5198078)
Affinity DataIC50:  5.00E+3nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590138(CHEMBL5201730)
Affinity DataIC50:  6.00E+3nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50428449(CHEMBL449451)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of GLUT1 in human H1299 cells assessed as inhibition of 2-deoxy-D-[3H]-glucose uptake incubated for 15 mins prior to 2-deoxy-D-[3H]-glucos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50428447(CHEMBL479638)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibition of GLUT1 in human H1299 cells assessed as inhibition of 2-deoxy-D-[3H]-glucose uptake incubated for 15 mins prior to 2-deoxy-D-[3H]-glucos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50444088(CHEMBL3092944)
Affinity DataIC50:  1.09E+4nMAssay Description:Inhibition of GLUT1 in human H1299 cells assessed as inhibition of 2-deoxy-D-[3H]-glucose uptake incubated for 15 mins prior to 2-deoxy-D-[3H]-glucos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590134(CHEMBL5180335)
Affinity DataIC50:  1.10E+4nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50444086(CHEMBL479837)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of GLUT1 in human H1299 cells assessed as inhibition of 2-deoxy-D-[3H]-glucose uptake incubated for 15 mins prior to 2-deoxy-D-[3H]-glucos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590135(CHEMBL5180822)
Affinity DataIC50:  1.60E+4nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590136(CHEMBL5203610)
Affinity DataIC50:  1.90E+4nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461999(CHEMBL4227052)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of [35S]methionine-labelled human recombinant His6-tagged CK2alpha/MBP-tagged CK2beta (unknown origin) interaction incubated for 1 hr by s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM23446(3-(4-hydroxyphenyl)-1-(2,4,6-trihydroxyphenyl)prop...)
Affinity DataIC50:  2.14E+4nMAssay Description:Inhibition of GLUT1 in human H1299 cells assessed as inhibition of 2-deoxy-D-[3H]-glucose uptake incubated for 15 mins prior to 2-deoxy-D-[3H]-glucos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50444087(CHEMBL480612)
Affinity DataIC50:  2.34E+4nMAssay Description:Inhibition of GLUT1 in human H1299 cells assessed as inhibition of 2-deoxy-D-[3H]-glucose uptake incubated for 15 mins prior to 2-deoxy-D-[3H]-glucos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461948(CHEMBL4227516)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590133(CHEMBL5184713)
Affinity DataIC50:  8.60E+4nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461942(CHEMBL4225845)
Affinity DataIC50:  1.50E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461942(CHEMBL4225845)
Affinity DataIC50:  1.50E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461965(CHEMBL4224990)
Affinity DataIC50:  1.60E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461945(CHEMBL4225193)
Affinity DataIC50:  2.05E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461945(CHEMBL4225193)
Affinity DataIC50:  2.05E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461946(CHEMBL4227626)
Affinity DataIC50:  2.08E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461946(CHEMBL4227626)
Affinity DataIC50:  2.08E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50462000(CHEMBL4227296)
Affinity DataIC50:  2.70E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461982(CHEMBL4226034)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590132(CHEMBL5202453)
Affinity DataIC50:  3.33E+5nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50099398(5-Bromo-1H-indazole | CHEMBL16425 | cid_761929)
Affinity DataIC50:  4.10E+5nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461947(CHEMBL4225463)
Affinity DataIC50:  4.93E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461947(CHEMBL4225463)
Affinity DataIC50:  4.93E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461937(CHEMBL4226507)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461966(CHEMBL4117419)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461967(CHEMBL4228752)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461968(CHEMBL4228350)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461971(CHEMBL4226330)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461972(CHEMBL4224921)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461981(CHEMBL4225723)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461985(CHEMBL4229078)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461994(CHEMBL4225769)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50029105(2-(3,4,-dichlorophenyl)ethylamine | 2-(3,4-Dichlor...)
Affinity DataIC50:  7.00E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461988(CHEMBL1178112)
Affinity DataIC50:  7.50E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461954(CHEMBL4227171)
Affinity DataIC50:  8.30E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM93339(Integrase inhibitor, R1{1})
Affinity DataIC50:  9.00E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461975(CHEMBL4229161)
Affinity DataIC50:  9.00E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461955(CHEMBL4225265)
Affinity DataIC50:  9.00E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461995(3,4-Dichlorobenzylalcohol | CHEMBL2323843)
Affinity DataIC50:  9.80E+5nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461939(CHEMBL4225945)
Affinity DataIC50:  1.01E+6nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50461956(CHEMBL4226065)
Affinity DataIC50:  1.02E+6nMAssay Description:Inhibition of CK2alpha (unknown origin) (2 to 329 residues) expressed in Escherichia coli BL21 (DE3) interaction with CK2beta (unknown origin) using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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