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Found 98 with Last Name = 'kongsted' and Initial = 'j'
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50505279(CHEMBL4436207)
Affinity DataKi:  0.00100nMAssay Description:Inhibition of HIV1 protease using RE(Edans)SGIFLETSK(Dabcyl)R as substrate by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Shandong University

Curated by ChEMBL
LigandPNGBDBM8125((3R,3aS,6aR)-hexahydrofuro[2,3-b]furan-3-yl N-[(2S...)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of HIV1 protease using RE(Edans)SGIFLETSK(Dabcyl)R as substrate by fluorescence methodMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50163737(CHEMBL3799941)
Affinity DataKi:  1.70nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataKi:  2.90nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50163750(CHEMBL3797292)
Affinity DataKi:  4nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50505281(CHEMBL2315948)
Affinity DataKi:  8.10nMAssay Description:Inhibition of NO711 binding to mouse GAT1 receptor expressed in HEK293 cell membranes incubated for 1 hr by LC-ESI-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50163750(CHEMBL3797292)
Affinity DataKi:  9.70nMAssay Description:Inhibition of HIV1 protease G48V mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50163737(CHEMBL3799941)
Affinity DataKi:  10nMAssay Description:Inhibition of HIV1 protease V82F mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50163750(CHEMBL3797292)
Affinity DataKi:  13nMAssay Description:Inhibition of HIV1 protease V82F mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50163737(CHEMBL3799941)
Affinity DataKi:  22nMAssay Description:Inhibition of HIV1 protease G48V mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50163737(CHEMBL3799941)
Affinity DataKi:  27nMAssay Description:Inhibition of HIV1 protease V82A mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50163750(CHEMBL3797292)
Affinity DataKi:  30nMAssay Description:Inhibition of HIV1 protease V82A mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50505274(CHEMBL2315639)
Affinity DataKi:  117nMAssay Description:Inhibition of NO711 binding to mouse GAT1 receptor expressed in HEK293 cell membranes incubated for 1 hr by LC-ESI-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50163737(CHEMBL3799941)
Affinity DataIC50:  6nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50137113(CHEMBL3753096)
Affinity DataIC50:  6nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50137112(CHEMBL309896)
Affinity DataIC50:  12nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50163750(CHEMBL3797292)
Affinity DataIC50:  13nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50163750(CHEMBL3797292)
Affinity DataIC50:  17nMAssay Description:Inhibition of HIV1 protease G48V mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50163737(CHEMBL3799941)
Affinity DataIC50:  19nMAssay Description:Inhibition of HIV1 protease V82F mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM3107(3,4-Dihydroquinazolinon 4a | 6-Chloro-4-cyclopyrop...)
Affinity DataIC50:  23nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50163750(CHEMBL3797292)
Affinity DataIC50:  24nMAssay Description:Inhibition of HIV1 protease V82F mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50121209(CHEMBL3622376)
Affinity DataIC50:  35nMAssay Description:Inhibition of human JAK3 using GGEEEEYFELVKKKK substrate preincubated for 20 mis followed by addition of ATP and measured after 120 mins in presence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM1517(2-ethyl-7-methyl-2,4,9,15-tetraazatricyclo[9.4.0.0...)
Affinity DataIC50:  35nMAssay Description:Inhibition of HIV1 reverse transcriptase derived from HIV patient plasma by LC/MS/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataIC50:  38nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50163737(CHEMBL3799941)
Affinity DataIC50:  39nMAssay Description:Inhibition of HIV1 protease G48V mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50163737(CHEMBL3799941)
Affinity DataIC50:  46nMAssay Description:Inhibition of HIV1 protease V82A mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50524092(CHEMBL4436313)
Affinity DataIC50:  46nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50163750(CHEMBL3797292)
Affinity DataIC50:  52nMAssay Description:Inhibition of HIV1 protease V82A mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50524088(CHEMBL4483481)
Affinity DataIC50:  56nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50524089(CHEMBL4529500)
Affinity DataIC50:  82nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Rajiv Gandhi Proudyogiki Vishwavidyalaya

Curated by ChEMBL
LigandPNGBDBM7401((2 Z,3 E)-6-Bromoindirubin-3 -oxime | (3E)-6-bromo...)
Affinity DataIC50:  83nMAssay Description:inhibition of human recombinant CDK5/p25 using histone H1 as substrate by scintillation counting in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataIC50:  84nMAssay Description:Inhibition of HIV1 reverse transcriptase derived from HIV patient plasma by LC/MS/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM1518(2-ethyl-9-methyl-2,4,9,15-tetraazatricyclo[9.4.0.0...)
Affinity DataIC50:  125nMAssay Description:Inhibition of HIV1 reverse transcriptase derived from HIV patient plasma by LC/MS/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50505275(CHEMBL4573432)
Affinity DataIC50:  130nMAssay Description:Inhibition of HIV1 JRFL gp120 assessed as reduction in CD4/gp 120 complex formation incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50121210(CHEMBL3622374)
Affinity DataIC50:  240nMAssay Description:Inhibition of recombinant human HDAC3/GST-tagged NCOR1 DAD (397 to 503 residues) expressed in baculovirus expression system using Fluor de Lys as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM1944(BHAP deriv. | CHEMBL593 | DELAVIRDINE MESYLATE | D...)
Affinity DataIC50:  260nMAssay Description:Inhibition of wild type recombinant HIV1 reverse transcriptase using poly(rA)-oligo(dT) as template/primerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50121211(CHEMBL3622375)
Affinity DataIC50:  260nMAssay Description:Inhibition of recombinant human HDAC3/GST-tagged NCOR1 DAD (397 to 503 residues) expressed in baculovirus expression system using Fluor de Lys as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50505276(CHEMBL4540823)
Affinity DataIC50:  330nMAssay Description:Inhibition of HIV1 JRFL gp120 assessed as reduction in CD4/gp 120 complex formation incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM1633(2-ethyl-10-methyl-2,4,10-triazatricyclo[9.4.0.0^{3...)
Affinity DataIC50:  350nMAssay Description:Inhibition of HIV1 reverse transcriptase derived from HIV patient plasma by LC/MS/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Rajiv Gandhi Proudyogiki Vishwavidyalaya

Curated by ChEMBL
LigandPNGBDBM7401((2 Z,3 E)-6-Bromoindirubin-3 -oxime | (3E)-6-bromo...)
Affinity DataIC50:  520nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate by scintillation counting in presence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50137120(CHEMBL3753006)
Affinity DataIC50:  800nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50137115(CHEMBL3754170)
Affinity DataIC50:  950nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Rajiv Gandhi Proudyogiki Vishwavidyalaya

Curated by ChEMBL
LigandPNGBDBM50290835((3,4-Dimethoxy-phenyl)-(6,7-dimethoxy-quinazolin-4...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human recombinant GST-fused CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Rajiv Gandhi Proudyogiki Vishwavidyalaya

Curated by ChEMBL
LigandPNGBDBM7401((2 Z,3 E)-6-Bromoindirubin-3 -oxime | (3E)-6-bromo...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human recombinant GST-fused CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM1437(5-methoxyindole-2-carboxylic acid [N -[3-(aminoeth...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of wild type recombinant HIV1 reverse transcriptase using poly(rA)-oligo(dT) as template/primerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50121209(CHEMBL3622376)
Affinity DataIC50:  2.45E+3nMAssay Description:Inhibition of human JAK2 using poly[Glu:Tyr] (4:1) substrate preincubated for 20 mis followed by addition of ATP and measured after 120 mins in prese...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50121209(CHEMBL3622376)
Affinity DataIC50:  2.73E+3nMAssay Description:Inhibition of human JAK1 using poly[Glu:Tyr] (4:1) substrate preincubated for 20 mis followed by addition of ATP and measured after 120 mins in prese...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50121209(CHEMBL3622376)
Affinity DataIC50:  5.62E+3nMAssay Description:Inhibition of human TYK2 using KKSRGDYMTMQIG] substrate preincubated for 20 mis followed by addition of ATP and measured after 120 mins in presence o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50524091(CHEMBL307792)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase derived from HIV patient plasma by LC/MS/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Rajiv Gandhi Proudyogiki Vishwavidyalaya

Curated by ChEMBL
LigandPNGBDBM4626(Anilinoquinazoline deriv. 9 | CHEMBL301018 | N-(3-...)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of human recombinant GST-fused CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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