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TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191756(4'-fluoro-biphenyl-4-carboxylic acid methyl-(3-pip...)
Affinity DataKi:  31nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191752(6-(4-chlorophenyl)-3-((3-((4-hydroxypiperidin-1-yl...)
Affinity DataKi:  51nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191768(6-(4-chlorophenyl)-3-((3-(pyrrolidin-1-ylmethyl)qu...)
Affinity DataKi:  91nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191765(4'-fluoro-biphenyl-4-carboxylic acid (3-diethylami...)
Affinity DataKi:  102nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191753(6-(4-chlorophenyl)-3-((3-((4-methylpiperazin-1-yl)...)
Affinity DataKi:  110nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191766(6-(4-chlorophenyl)-3-((3-((diethylamino)methyl)qui...)
Affinity DataKi:  126nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191755(2-(((8-((6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyri...)
Affinity DataKi:  136nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191764(4'-fluoro-biphenyl-4-carboxylic acid [3-((S)-3-hyd...)
Affinity DataKi:  142nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191761(4'-fluoro-biphenyl-4-carboxylic acid [3-(4-hydroxy...)
Affinity DataKi:  195nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191762(6-(4-chlorophenyl)-3-((3-((dimethylamino)methyl)qu...)
Affinity DataKi:  197nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191754(CHEMBL213817 | N-(3-diethylaminomethyl-quinolin-8-...)
Affinity DataKi:  310nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191767(4'-fluoro-biphenyl-4-carboxylic acid [3-(4-methane...)
Affinity DataKi:  310nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191760(CHEMBL216038 | N-(3-dimethylaminomethyl-quinolin-8...)
Affinity DataKi:  414nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191759(6-(4-chlorophenyl)-3-((3-((4-(methylsulfonyl)piper...)
Affinity DataKi:  773nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191750(6-(4-fluoro-phenyl)-N-[3-(4-hydroxy-piperidin-1-yl...)
Affinity DataKi:  803nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191763(6-(4-fluoro-phenyl)-N-[3-((S)-3-hydroxy-pyrrolidin...)
Affinity DataKi:  1.15E+3nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191758(4'-fluoro-biphenyl-4-carboxylic acid (3-morpholin-...)
Affinity DataKi:  1.41E+3nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191751(6-(4-fluoro-phenyl)-N-[3-(4-methyl-piperazin-1-ylm...)
Affinity DataKi:  3.54E+3nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191757(6-(4-fluoro-phenyl)-N-(3-morpholin-4-ylmethyl-quin...)
Affinity DataKi:  2.01E+4nMAssay Description:Binding affinity to MCHR1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189360((1S,10S)-9-[(Isoquinoline-1-carbonyl)-amino]-6,10-...)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189365(CHEMBL212345 | N'-(2-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  30nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189375(CHEMBL212981 | N-[(3S)-2-hydroxy-5-oxotetrahydrofu...)
Affinity DataIC50:  40nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189370(CHEMBL212870 | N'-(2-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  40nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-8(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189360((1S,10S)-9-[(Isoquinoline-1-carbonyl)-amino]-6,10-...)
Affinity DataIC50:  40nMAssay Description:Inhibition of caspase8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189371(CHEMBL209626 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  50nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189376(CHEMBL213952 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  50nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-8(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189371(CHEMBL209626 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  70nMAssay Description:Inhibition of caspase8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189364(CHEMBL211512 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  90nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-8(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189375(CHEMBL212981 | N-[(3S)-2-hydroxy-5-oxotetrahydrofu...)
Affinity DataIC50:  90nMAssay Description:Inhibition of caspase8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-8(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189376(CHEMBL213952 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  130nMAssay Description:Inhibition of caspase8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189363(CHEMBL213784 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  150nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189362(CHEMBL214166 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  150nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189372(CHEMBL379764 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  200nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-8(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189359(CHEMBL210114 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  230nMAssay Description:Inhibition of caspase8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189374(CHEMBL210118 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  240nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189368(CHEMBL214215 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  240nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189369(CHEMBL386240 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  260nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-8(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189366(CHEMBL214044 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  300nMAssay Description:Inhibition of caspase8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-8(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189367(CHEMBL213408 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  310nMAssay Description:Inhibition of caspase8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189367(CHEMBL213408 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  310nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-8(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189370(CHEMBL212870 | N'-(2-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  420nMAssay Description:Inhibition of caspase8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189361(CHEMBL213965 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  430nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189358(2-(carbamoyl)-N'-(3-methylbenzoyl)-2,3-dihydro-1H-...)
Affinity DataIC50:  430nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189377(CHEMBL210023 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  490nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189378(CHEMBL213553 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  580nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189366(CHEMBL214044 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  700nMAssay Description:Inhibition of ICEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-8(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189372(CHEMBL379764 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of caspase8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-8(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189377(CHEMBL210023 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of caspase8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50191762(6-(4-chlorophenyl)-3-((3-((dimethylamino)methyl)qu...)
Affinity DataIC50:  1.31E+3nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-8(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189368(CHEMBL214215 | N'-(1-(((3S)-2-hydroxy-5-oxo-tetrah...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of caspase8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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