Report error Found 330 with Last Name = 'tsai' and Initial = 'kc'
Affinity DataKi: 0.0360nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +++:highly activeMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +++:highly activeMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +++:highly activeMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +++:highly activeMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +++:highly activeMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +++:highly activeMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +++:highly activeMore data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +++:highly activeMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +++:highly activeMore data for this Ligand-Target Pair
Affinity DataKi: 0.350nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +++:highly activeMore data for this Ligand-Target Pair
Affinity DataKi: 0.360nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +++:highly activeMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +++:highly activeMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +++:highly activeMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +++:highly activeMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +++:highly activeMore data for this Ligand-Target Pair
Affinity DataKi: 0.690nM ΔG°: -53.2kJ/molepH: 4.25 T: 30°CAssay Description:Enzyme inhibition activity assay using 4-methylumbelliferyl N-acetylglucosamine (MUG) as substrate.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nM ΔG°: -51.8kJ/molepH: 4.25 T: 30°CAssay Description:Enzyme inhibition activity assay using 4-methylumbelliferyl N-acetylglucosamine (MUG) as substrate.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nM ΔG°: -50.4kJ/molepH: 4.25 T: 30°CAssay Description:Enzyme inhibition activity assay using 4-methylumbelliferyl N-acetylglucosamine (MUG) as substrate.More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 9.30nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 26.7nM ΔG°: -44.0kJ/molepH: 4.25 T: 30°CAssay Description:Enzyme inhibition activity assay using 4-methylumbelliferyl N-acetylglucosamine (MUG) as substrate.More data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; ++:moderately activeMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +:inactiveMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +:inactiveMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +:inactiveMore data for this Ligand-Target Pair
Affinity DataKi: 420nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +:inactiveMore data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +:inactiveMore data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +:inactiveMore data for this Ligand-Target Pair
Affinity DataKi: 540nM ΔG°: -36.4kJ/molepH: 4.25 T: 30°CAssay Description:Enzyme inhibition activity assay using 4-methylumbelliferyl N-acetylglucosamine (MUG) as substrate.More data for this Ligand-Target Pair
Affinity DataKi: 630nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +:inactiveMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nM ΔG°: -33.5kJ/molepH: 4.25 T: 30°CAssay Description:Enzyme inhibition activity assay using 4-methylumbelliferyl N-acetylglucosamine (MUG) as substrate.More data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +:inactiveMore data for this Ligand-Target Pair