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Found 90 with Last Name = 'pinna' and Initial = 'la'
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34046(iodinated benzimidazole, 9a)
Affinity DataKi:  19nM ΔG°:  -45.8kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)
Affinity DataKi:  23nM ΔG°:  -45.4kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34044(iodinated benzimidazole, 7a)
Affinity DataKi:  24nM ΔG°:  -45.2kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34051(iodinated benzimidazole, 14)
Affinity DataKi:  27nM ΔG°:  -44.9kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34054(iodinated benzimidazole, 17)
Affinity DataKi:  50nM ΔG°:  -43.3kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34052(iodinated benzimidazole, 15)
Affinity DataKi:  50nM ΔG°:  -43.3kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34053(iodinated benzimidazole, 16)
Affinity DataKi:  54nM ΔG°:  -43.2kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34048(iodinated benzimidazole, 11a)
Affinity DataKi:  70nM ΔG°:  -42.5kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34043(iodinated benzimidazole, 6a)
Affinity DataKi:  75nM ΔG°:  -42.3kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34050(iodinated benzimidazole, 13a)
Affinity DataKi:  90nM ΔG°:  -41.8kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34040(iodinated benzimidazole, 3a)
Affinity DataKi:  100nM ΔG°:  -41.6kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34049(iodinated benzimidazole, 12a)
Affinity DataKi:  120nM ΔG°:  -41.1kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34047(iodinated benzimidazole, 10a)
Affinity DataKi:  120nM ΔG°:  -41.1kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34056(iodinated benzimidazole, 23)
Affinity DataKi:  130nM ΔG°:  -40.9kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34055(iodinated benzimidazole, 21)
Affinity DataKi:  140nM ΔG°:  -40.7kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34058(iodinated benzimidazole, 27)
Affinity DataKi:  160nM ΔG°:  -40.3kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34039(iodinated benzimidazole, 2a)
Affinity DataKi:  160nM ΔG°:  -40.3kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM11319((5-oxo-5,6-dihydroindolo[1,2-a]quinazolin-7-yl)ace...)
Affinity DataKi:  170nM ΔG°:  -38.2kJ/mole IC50:  390nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34057(iodinated benzimidazole, 25)
Affinity DataKi:  180nM ΔG°:  -40.0kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34045(iodinated benzimidazole, 8a)
Affinity DataKi:  330nM ΔG°:  -38.5kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
University of Padova

LigandPNGBDBM11315(1,4-diamino-5,8-dihydroxy-9,10-dihydroanthracene-9...)
Affinity DataKi:  350nM ΔG°:  -36.5kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM11323(4,5,6,7-tetrabromo-1H-1,2,3-benzotriazole | 4,5,6,...)
Affinity DataKi:  400nM ΔG°:  -36.2kJ/mole IC50:  500nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34041(iodinated benzimidazole, 4a)
Affinity DataKi:  460nM ΔG°:  -37.6kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34042(iodinated benzimidazole, 5a)
Affinity DataKi:  590nM ΔG°:  -37.0kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM7458(5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataKi:  740nM ΔG°:  -34.6kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Zea mays (Maize))
University of Padova

LigandPNGBDBM11313(1,8-dihydroxy-4-nitro-anthraquinone | 4,5-dihydrox...)
Affinity DataKi:  780nM ΔG°:  -34.5kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Zea mays (Maize))
University of Padova

LigandPNGBDBM11314(1,8-dihydroxy-4-nitro-9H-xanthen-9-one | 1,8-dihyd...)
Affinity DataKi:  800nM ΔG°:  -34.4kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataKi:  1.18E+3nM ΔG°:  -33.5kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34059(brominated benzimidazole, 20)
Affinity DataKi:  1.34E+3nM ΔG°:  -34.9kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34060(brominated benzimidazole, 22)
Affinity DataKi:  1.45E+3nM ΔG°:  -34.7kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34062(brominated benzimidazole, 26)
Affinity DataKi:  1.51E+3nM ΔG°:  -34.6kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
Affinity DataKi:  1.85E+3nM ΔG°:  -32.4kJ/mole IC50:  890nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Zea mays (Maize))
University of Padova

LigandPNGBDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
Affinity DataKi:  1.85E+3nM ΔG°:  -32.4kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34061(brominated benzimidazole, 24)
Affinity DataKi:  1.91E+3nM ΔG°:  -34.0kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM11324((2R,3R,4S,5R)-2-(5,6-dichloro-1H-1,3-benzodiazol-1...)
Affinity DataKi:  4.50E+3nM ΔG°:  -30.2kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Zea mays (Maize))
University of Padova

LigandPNGBDBM11317(1,8-dihydroxy-9H-xanthen-9-one | Xanthenone-relate...)
Affinity DataKi: >4.00E+4nM ΔG°: >-24.8kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
University of Padova

LigandPNGBDBM11316(1,8-dihydroxy-9,10-dihydroanthracene-9,10-dione | ...)
Affinity DataKi: >4.00E+4nM ΔG°: >-24.8kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM92757(CX-5279)
Affinity DataIC50:  0.910nMAssay Description:Phosphorylation assay using casein kinase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM92755(CX-4945)
Affinity DataIC50:  1.5nMAssay Description:Phosphorylation assay using casein kinase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM92756(CX-5011)
Affinity DataIC50:  2.07nMAssay Description:Phosphorylation assay using casein kinase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM92756(CX-5011)
Affinity DataIC50:  2.30nMAssay Description:Phosphorylation assay using casein kinase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM92756(CX-5011)
Affinity DataIC50:  2.32nMAssay Description:Phosphorylation assay using casein kinase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM92756(CX-5011)
Affinity DataIC50:  2.5nMAssay Description:Phosphorylation assay using casein kinase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM92755(CX-4945)
Affinity DataIC50:  3.51nMAssay Description:Phosphorylation assay using casein kinase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM92757(CX-5279)
Affinity DataIC50:  12.5nMAssay Description:Phosphorylation assay using casein kinase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM92755(CX-4945)
Affinity DataIC50:  13.5nMAssay Description:Phosphorylation assay using casein kinase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM92757(CX-5279)
Affinity DataIC50:  13.8nMAssay Description:Phosphorylation assay using casein kinase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM92755(CX-4945)
Affinity DataIC50:  15nMAssay Description:Phosphorylation assay using casein kinase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University of Padova

LigandPNGBDBM92757(CX-5279)
Affinity DataIC50:  23.4nMAssay Description:Phosphorylation assay using casein kinase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50156670(2-(dimethylamino)-4,5,6,7-tetrabromo-1H-benzimidaz...)
Affinity DataIC50:  120nMAssay Description:Inhibition of DYRK1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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