Report error Found 2687 with Last Name = 'kai' and Initial = 'm'
Affinity DataKi: 0.00372nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation c...More data for this Ligand-Target Pair
Affinity DataKi: 0.00986nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation c...More data for this Ligand-Target Pair
Affinity DataKi: 0.0128nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation c...More data for this Ligand-Target Pair
Affinity DataKi: 0.0137nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation c...More data for this Ligand-Target Pair
Affinity DataKi: 0.0220nMAssay Description:Inhibition of CYP3A4 in human liver microsomes pre-incubated for 15 mins by LC/MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.0260nMAssay Description:Inhibition of CYP3A4 in human liver microsomes pre-incubated for 15 mins by LC/MS/MS analysisMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.0300nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.0300nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0322nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation c...More data for this Ligand-Target Pair
Affinity DataKi: 0.0405nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation c...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mouse)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.0900nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.165nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation c...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mouse)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.210nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.221nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu opioid receptor expressed in HEK293 cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.274nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu opioid receptor expressed in HEK293 cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 0.296nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation c...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of carbonic anhydrase-2 (unknown origin) incubated for 15 mins prior to testing by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.535nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu opioid receptor expressed in HEK293 cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 0.574nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation c...More data for this Ligand-Target Pair
Affinity DataKi: 0.758nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation c...More data for this Ligand-Target Pair
Affinity DataKi: 0.770nMAssay Description:Inhibition of carbonic anhydrase-2 (unknown origin) incubated for 15 mins prior to testing by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.880nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain using Cbz-Phe-Arg-AMC as substrate by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of human CatL using Cbz-Phe-Arg-AMC as substrate measured over 30 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain using Cbz-Phe-Arg-AMC as substrate by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain using Cbz-Phe-Arg-AMC as substrate by fluorimetric methodMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Rat)
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
Affinity DataKi: 2.30nMAssay Description:Inhibition of human CatL using Cbz-Phe-Arg-AMC as substrate measured over 30 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.32nMAssay Description:Binding affinity to human mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Inhibition of human CatL using Cbz-Phe-Arg-AMC as substrate measured over 30 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain using Cbz-Phe-Arg-AMC as substrate by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibition of human CatL using Cbz-Phe-Arg-AMC as substrate measured over 30 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu opioid receptor expressed in HEK293 cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Inhibition of carbonic anhydrase-2 (unknown origin) incubated for 15 mins prior to testing by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of carbonic anhydrase-2 (unknown origin) incubated for 15 mins prior to testing by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain using Cbz-Phe-Arg-AMC as substrate by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain using Cbz-Phe-Arg-AMC as substrate by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of DPP4 in human plasma using Gly-Pro-AMC as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of human CatL using Cbz-Phe-Arg-AMC as substrate measured over 30 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain using Cbz-Phe-Arg-AMC as substrate by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu opioid receptor expressed in HEK293 cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mouse)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu opioid receptor expressed in HEK293 cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Inhibition of human CatL using Cbz-Phe-Arg-AMC as substrate measured over 30 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibition of carbonic anhydrase-2 (unknown origin) incubated for 15 mins prior to testing by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of human CatL using Cbz-Phe-Arg-AMC as substrate measured over 30 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain using Cbz-Phe-Arg-AMC as substrate by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataKi: 4.55nMAssay Description:Binding affinity to human mu opioid receptorMore data for this Ligand-Target Pair