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Found 124 with Last Name = 'ryan' and Initial = 'p'
TargetRelaxin-3 receptor 1(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50382993(CHEMBL2030702)
Affinity DataKi:  110nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin-3 receptor 1(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50382991(CHEMBL2030700)
Affinity DataKi:  112nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin-3 receptor 1(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50382992(CHEMBL2030701)
Affinity DataKi:  112nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin-3 receptor 1(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50383000(CHEMBL2030696)
Affinity DataKi:  741nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin-3 receptor 1(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50382999(CHEMBL2030698)
Affinity DataKi:  2.09E+3nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin-3 receptor 1(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50383002(CHEMBL2030699)
Affinity DataKi:  2.57E+3nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin-3 receptor 1(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50382994(CHEMBL2030691)
Affinity DataKi:  2.95E+3nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin-3 receptor 1(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50382998(CHEMBL2030697)
Affinity DataKi:  3.39E+3nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin receptor 1(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50382991(CHEMBL2030700)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of europium-labelled H2 relaxin from RXFP1 expressed in HEK-293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin receptor 1(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50382993(CHEMBL2030702)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of europium-labelled H2 relaxin from RXFP1 expressed in HEK-293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin-3 receptor 1(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50382995(CHEMBL2030693)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin-3 receptor 1(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50382996(CHEMBL2030694)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin-3 receptor 1(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50382997(CHEMBL2030695)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin receptor 1(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50382992(CHEMBL2030701)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of europium-labelled H2 relaxin from RXFP1 expressed in HEK-293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin-3 receptor 1(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50383001(CHEMBL2030692)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50323697((3AR,5R,6S,7R,7AR)-2-(ETHYLAMINO)-5-(HYDROXYMETHYL...)
Affinity DataIC50:  0.410nMAssay Description:Inhibition of human O-GlcNAcaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046401(CHEMBL432806 | N-{1-Benzyl-2,3-dihydroxy-4-[3-meth...)
Affinity DataIC50:  1nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046439(2N-[1-[1-benzyl-2-hydroxy-3-[1-(1H-2-indolylcarbox...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046435(1N-[1-[1-benzyl-2,3-dihydroxy-4-[2-methyl-1-(4-phe...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046422(CHEMBL324916 | N-{1-Benzyl-2,3-dihydroxy-4-[3-meth...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046428(CHEMBL112930 | N-{1-Benzyl-2,3-dihydroxy-4-[3-meth...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046385(CHEMBL331363 | N-{1-Benzyl-2,3-dihydroxy-4-[3-meth...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046392(2N-[1-[1-benzyl-2-hydroxy-3-[2-methyl-1-(2-quinoly...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046384(CHEMBL113575 | N-{1-Benzyl-2,3-dihydroxy-4-[3-meth...)
Affinity DataIC50:  1.66nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046408((1-{1-Benzyl-2,3-dihydroxy-4-[3-methyl-2-(pyridin-...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046412(CHEMBL113626 | N-{1-Benzyl-2-hydroxy-3-[3-methyl-2...)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046390((1-{1-Benzyl-2,3-dihydroxy-4-[3-methyl-2-(pyridin-...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Staphylococcus aureus (strain MRSA252))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50526643(CHEMBL4475677)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of MraY in Staphylococcus aureusMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50014147(A-74704 | CHEMBL430891 | {(S)-1-[(1S,3S)-1-Benzyl-...)
Affinity DataIC50:  3nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046378(CHEMBL109371 | {1-[1-Benzyl-3-(2-benzyloxycarbonyl...)
Affinity DataIC50:  3nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin-3 receptor 2(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50382993(CHEMBL2030702)
Affinity DataIC50:  3.47nMAssay Description:Agonist activity at RXFP4 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 6 hrs by beta galactosidase r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046407(CHEMBL113627 | {1-[1-Benzyl-3-(2-benzyloxycarbonyl...)
Affinity DataIC50:  4nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin-3 receptor 1(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50382991(CHEMBL2030700)
Affinity DataIC50:  4.27nMAssay Description:Agonist activity at RXFP3 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 6 hrs by beta galactosidase r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046414((1-{1-Benzyl-2-hydroxy-3-[3-methyl-2-(pyridin-2-yl...)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin-3 receptor 1(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50382992(CHEMBL2030701)
Affinity DataIC50:  5.13nMAssay Description:Agonist activity at RXFP3 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 6 hrs by beta galactosidase r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046416(CHEMBL323955 | N-(1-Benzyl-2,3-dihydroxy-4-{3-meth...)
Affinity DataIC50:  5.20nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046429(CHEMBL111957 | N-{1-Benzyl-2,3-dihydroxy-4-[3-meth...)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046386(CHEMBL112578 | N-{1-Benzyl-2,3-dihydroxy-4-[3-meth...)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046433((1-{1-Benzyl-2-hydroxy-3-[3-methyl-2-(pyridin-3-yl...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046380(CHEMBL112546 | {1-[1-Benzyl-3-(2-benzyloxycarbonyl...)
Affinity DataIC50:  7nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046417(3N-[1-[1-benzyl-2-hydroxy-3-[2-methyl-1-(1,2,3,4-t...)
Affinity DataIC50:  7.10nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046421(CHEMBL112846 | N-{1-Benzyl-2,3-dihydroxy-4-[3-meth...)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046381(1N-[1-[1-benzyl-4-[1-(4-benzylhexahydro-1-pyraziny...)
Affinity DataIC50:  7.80nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM205424(US9243020, 19 | US9815861, Example 19)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of human O-GlcNAcaseMore data for this Ligand-Target Pair
TargetRelaxin-3 receptor 2(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50382992(CHEMBL2030701)
Affinity DataIC50:  7.94nMAssay Description:Agonist activity at RXFP4 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 6 hrs by beta galactosidase r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046387((1-{1-Benzyl-2-hydroxy-3-[3-methyl-2-(2-morpholin-...)
Affinity DataIC50:  9nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046447(1N-[1-[1-benzyl-4-[1-(4-benzylhexahydro-1-pyraziny...)
Affinity DataIC50:  9nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046419(CHEMBL114192 | N-{1-Benzyl-2-hydroxy-3-[3-methyl-2...)
Affinity DataIC50:  10nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50046383(CHEMBL331829 | N-{1-Benzyl-2-hydroxy-3-[3-methyl-2...)
Affinity DataIC50:  12nMAssay Description:Inhibition of purified recombinant HIV-1 protease in a fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin-3 receptor 1(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50382993(CHEMBL2030702)
Affinity DataIC50:  12.6nMAssay Description:Agonist activity at RXFP3 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 6 hrs by beta galactosidase r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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