Affinity DataKi: 0.0480nMAssay Description:Inhibitory activity against human adenosine A2A receptor expressed in HEK-293 cells by displacement of [3H]-SCH-58,261More data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Binding affinity for rat dopamine D3 receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibitory activity against Dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibitory activity against adenosine A2A receptor in rat striatal membranes by displacement of [3H]-SCH-58,261More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity for rat dopamine D3 receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity for rat dopamine D3 receptor using [11C]-GR-218,231More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Inhibitory activity against Dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) of Neisseria gonorrhoeaMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) from rat liverMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
University Of Milano/Bicocca
Curated by ChEMBL
University Of Milano/Bicocca
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Binding affinity for rat Alpha-1A adrenergic receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Binding affinity for rat Opioid receptor sigma 1 using [11C] radiotracerMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of Milano/Bicocca
Curated by ChEMBL
University Of Milano/Bicocca
Curated by ChEMBL
Affinity DataKi: 184nMAssay Description:Binding affinity for rat 5-Hydroxytryptamine receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: 342nMAssay Description:Binding affinity for rat Opioid receptor sigma 1 using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: 373nMAssay Description:Binding affinity for rat dopamine D4 receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of Milano/Bicocca
Curated by ChEMBL
University Of Milano/Bicocca
Curated by ChEMBL
Affinity DataKi: 575nMAssay Description:Binding affinity for rat 5-Hydroxytryptamine receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: 720nMAssay Description:Binding affinity towards rat dopamine D2 receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: 720nMAssay Description:Binding affinity towards rat dopamine D2 receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: 830nMAssay Description:Binding affinity for rat dopamine D4 receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: 1.11E+3nMAssay Description:Inhibitory activity against human adenosine A1 receptor expressed in CHO cells by displacement of [3H]-DPCPXMore data for this Ligand-Target Pair
Affinity DataKi: 1.82E+3nMAssay Description:Displacement of [3H]-DPCPX from adenosine A1 receptor in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
University Of Milano/Bicocca
Curated by ChEMBL
University Of Milano/Bicocca
Curated by ChEMBL
Affinity DataKi: 5.10E+3nMAssay Description:Binding affinity for rat Alpha-1A adrenergic receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]-AB-MECA from human adenosine A3 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against rat adenosine A3 receptor expressed in HEK-293 cells by displacement of [125I]-AB-MECAMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against human adenosine A2B receptor expressed in HEK-293 cells by displacement of [3H]-DPCPXMore data for this Ligand-Target Pair
Affinity DataIC50: 0.000100nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.00170nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0100nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0110nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0300nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0750nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibitory activity against Dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibitory activity against Dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibitory activity against Dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibition of rat liver Dihydrofolate reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibition of rat liver Dihydrofolate reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Evaluated for the inhibition of chicken liver Dihydrofolate reductase by using standard enzyme assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Inhibition of rat liver Dihydrofolate reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) of Plasmodium bergheiMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40nMAssay Description:Compound was tested for inhibitory activity against Dihydrofolate Reductase(DHFR) of rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 8.40nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
Affinity DataIC50: 8.70nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Inhibitory activity against Dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:Evaluated for the inhibition of chicken liver Dihydrofolate reductase by using standard enzyme assayMore data for this Ligand-Target Pair