Compile Data Set for Download or QSAR
maximum 50k data
Found 33 with Last Name = 'kendall harden' and Initial = 't'
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50390013(CHEMBL2071529)
Affinity DataKi:  6.00E+3nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50390014(CHEMBL2071530)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM59704(1-(3,4-dichlorophenyl)-3-[4-[(3,4-dimethyl-1,2-oxa...)
Affinity DataKi:  1.30E+4nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50390015(CHEMBL2071532)
Affinity DataKi:  2.70E+4nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50390016(CHEMBL2071534)
Affinity DataKi:  4.20E+4nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50390017(CHEMBL2071537)
Affinity DataKi:  4.50E+4nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50390018(CHEMBL2071539)
Affinity DataIC50:  130nMAssay Description:Antagonist activity at human P2Y1R expressed in human 1321N1 cells assessed as inhibition of 2-MeSADP-induced increase in intracellular inositol phos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM59704(1-(3,4-dichlorophenyl)-3-[4-[(3,4-dimethyl-1,2-oxa...)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at human P2Y1R expressed in human 1321N1 cells assessed as inhibition of 2-MeSADP-induced increase in intracellular inositol phos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50366145(CHEMBL1957449)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as stimulation of PLC-induced [3H]inositol phosphate production afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50366146(CHEMBL1957448)
Affinity DataEC50:  4.00E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as stimulation of PLC-induced [3H]inositol phosphate production afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50366147(CHEMBL1957447)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as stimulation of PLC-induced [3H]inositol phosphate production afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50366148(CHEMBL1957446)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as stimulation of PLC-induced [3H]inositol phosphate production afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50366149(CHEMBL1957445)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as stimulation of PLC-induced [3H]inositol phosphate production afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50366150(CHEMBL1957444)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as stimulation of PLC-induced [3H]inositol phosphate production afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50366151(CHEMBL1957443)
Affinity DataEC50:  700nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as stimulation of PLC-induced [3H]inositol phosphate production afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50366152(CHEMBL1957442)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as stimulation of PLC-induced [3H]inositol phosphate production afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50366153(CHEMBL1957441)
Affinity DataEC50:  3.10E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as stimulation of PLC-induced [3H]inositol phosphate production afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50366154(CHEMBL1957440)
Affinity DataEC50:  400nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as stimulation of PLC-induced [3H]inositol phosphate production afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50366155(CHEMBL1957439)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as stimulation of PLC-induced [3H]inositol phosphate production afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50366156(CHEMBL1957438)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as stimulation of PLC-induced [3H]inositol phosphate production afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50258427(CHEMBL522015 | uridine5'-methylene-phosphonate)
Affinity DataEC50:  5.10E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as stimulation of PLC-induced [3H]inositol phosphate production afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50197974(udp-N-acetyl-glucosamine)
Affinity DataEC50:  4.38E+3nMAssay Description:Agonist activity at human P2Y14 receptor expressed in COS7 cells assessed as stimulation of PLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50197975(udp-glucuronic acid)
Affinity DataEC50:  370nMAssay Description:Agonist activity at human P2Y14 receptor expressed in COS7 cells assessed as stimulation of PLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50370674(UDP-GALACTOSE)
Affinity DataEC50:  671nMAssay Description:Agonist activity at human P2Y14 receptor expressed in COS7 cells assessed as stimulation of PLCMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50258291(9-[5'-Deoxy-5'-[(hydroxyphosphoroxy)phosphinyl]-be...)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at human P2Y6 receptor expressed in human 1321N1 cells coexpressing phospholipase C-activating G protein assessed as inositol phosph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50118213(5'-UTP | CHEMBL336296 | H4utp | UTP | uridine 5'-(...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as stimulation of PLC-induced [3H]inositol phosphate production afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50258288(9-[5'-Deoxy-5'-[(hydroxypyrophosphoroxy)phosphinyl...)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells coexpressing phospholipase C-activating G protein assessed as inositol phosph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM2(({[({[(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-...)
Affinity DataEC50:  85nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells coexpressing phospholipase C-activating G protein assessed as inositol phosph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50258289(9-[5'-Deoxy-5'-[(hydroxypyrophosphoroxy)phosphinyl...)
Affinity DataEC50:  8.60E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells coexpressing phospholipase C-activating G protein assessed as inositol phosph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50258427(CHEMBL522015 | uridine5'-methylene-phosphonate)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells coexpressing phospholipase C-activating G protein assessed as inositol phosph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50258291(9-[5'-Deoxy-5'-[(hydroxyphosphoroxy)phosphinyl]-be...)
Affinity DataEC50:  3.40E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells coexpressing phospholipase C-activating G protein assessed as inositol phosph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50423218(5''-Diphosphoglucose | UDPG | URIDINE DIPHOSPHATE ...)
Affinity DataEC50:  354nMAssay Description:Agonist activity at human P2Y14 receptor expressed in COS7 cells assessed as stimulation of PLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50258290(1-[5,6-Dideoxy-6-[(hydroxypyrophosphoroxy)phosphon...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells coexpressing phospholipase C-activating G protein assessed as inositol phosph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed