Compile Data Set for Download or QSAR
maximum 50k data
Found 208 with Last Name = 'thull' and Initial = 'u'
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM19183(3-(3-nitrophenyl)-4aH,9H,9aH-indeno[1,2-e][1,2,4]t...)
Affinity DataIC50:  80nMAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031048(3-(4-(trifluoromethyl)phenyl)-5H-indeno[1,2-c]pyri...)
Affinity DataIC50:  89nMAssay Description:Inhibitory activity against Monoamine oxidase B from rat brain mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031048(3-(4-(trifluoromethyl)phenyl)-5H-indeno[1,2-c]pyri...)
Affinity DataIC50:  90nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031036(3-(3-(trifluoromethyl)phenyl)-5H-indeno[1,2-c]pyri...)
Affinity DataIC50:  280nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031028(3-(3-Nitro-phenyl)-indeno[1,2-c]pyridazin-5-one | ...)
Affinity DataIC50: >500nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031047(3-(4-Nitro-phenyl)-indeno[1,2-c]pyridazin-5-one | ...)
Affinity DataIC50:  500nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031047(3-(4-Nitro-phenyl)-indeno[1,2-c]pyridazin-5-one | ...)
Affinity DataIC50:  501nMAssay Description:Inhibitory activity against Monoamine oxidase B from rat brain mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031028(3-(3-Nitro-phenyl)-indeno[1,2-c]pyridazin-5-one | ...)
Affinity DataIC50:  631nMAssay Description:Inhibitory activity against Monoamine oxidase B from rat brain mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031044(3-(3-Bromo-phenyl)-indeno[1,2-c]pyridazin-5-one | ...)
Affinity DataIC50:  660nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031069(3-(3,5-Dichloro-phenyl)-indeno[1,2-c]pyridazin-5-o...)
Affinity DataIC50:  710nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031045(3-(3-Chloro-phenyl)-indeno[1,2-c]pyridazin-5-one |...)
Affinity DataIC50:  900nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031034(3-(4-Fluoro-phenyl)-indeno[1,2-c]pyridazin-5-one |...)
Affinity DataIC50:  912nMAssay Description:Inhibitory activity against Monoamine oxidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031020(3-(4-Chloro-phenyl)-indeno[1,2-c]pyridazin-5-one |...)
Affinity DataIC50:  912nMAssay Description:Inhibitory activity against Monoamine oxidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM19184(3-(3-nitrophenyl)-4aH,5H,9bH-indeno[2,1-e][1,2,4]t...)
Affinity DataIC50:  912nMAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031034(3-(4-Fluoro-phenyl)-indeno[1,2-c]pyridazin-5-one |...)
Affinity DataIC50:  920nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031053(3-(3,4-Difluoro-phenyl)-indeno[1,2-c]pyridazin-5-o...)
Affinity DataIC50:  920nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031020(3-(4-Chloro-phenyl)-indeno[1,2-c]pyridazin-5-one |...)
Affinity DataIC50:  920nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031046(CHEMBL127717 | Indeno[1,2-c]cinnolin-11-one)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50031035(3-((E)-Styryl)-indeno[1,2-c]pyridazin-5-one | CHEM...)
Affinity DataIC50: >1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase A enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50031030(3-(3-Hydroxy-phenyl)-indeno[1,2-c]pyridazin-5-one ...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase A enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031026(3-Thiophen-2-yl-indeno[1,2-c]pyridazin-5-one | CHE...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50031054(3-(4-Piperidin-1-yl-phenyl)-indeno[1,2-c]pyridazin...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase A enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031067(3-(2-Hydroxy-phenyl)-indeno[1,2-c]pyridazin-5-one ...)
Affinity DataIC50: >1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031054(3-(4-Piperidin-1-yl-phenyl)-indeno[1,2-c]pyridazin...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50031072(3-(3,4-Dimethoxy-phenyl)-indeno[1,2-c]pyridazin-5-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase A enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031030(3-(3-Hydroxy-phenyl)-indeno[1,2-c]pyridazin-5-one ...)
Affinity DataIC50: >1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50031071(3-(4-Bromo-phenyl)-indeno[1,2-c]pyridazin-5-one | ...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase A enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50031026(3-Thiophen-2-yl-indeno[1,2-c]pyridazin-5-one | CHE...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase A enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50031028(3-(3-Nitro-phenyl)-indeno[1,2-c]pyridazin-5-one | ...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase A enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031072(3-(3,4-Dimethoxy-phenyl)-indeno[1,2-c]pyridazin-5-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50031044(3-(3-Bromo-phenyl)-indeno[1,2-c]pyridazin-5-one | ...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase A enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50031067(3-(2-Hydroxy-phenyl)-indeno[1,2-c]pyridazin-5-one ...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase A enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50031070(3-(3,5-Bis-trifluoromethyl-phenyl)-indeno[1,2-c]py...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase A enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50031069(3-(3,5-Dichloro-phenyl)-indeno[1,2-c]pyridazin-5-o...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase A enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50031053(3-(3,4-Difluoro-phenyl)-indeno[1,2-c]pyridazin-5-o...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase A enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50031048(3-(4-(trifluoromethyl)phenyl)-5H-indeno[1,2-c]pyri...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase A enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50031046(CHEMBL127717 | Indeno[1,2-c]cinnolin-11-one)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase A enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031058(3-(3-trifluoromethyl)phenyl-7-methoxy-5H-indeno[1,...)
Affinity DataIC50:  1.31E+3nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031071(3-(4-Bromo-phenyl)-indeno[1,2-c]pyridazin-5-one | ...)
Affinity DataIC50:  1.33E+3nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031035(3-((E)-Styryl)-indeno[1,2-c]pyridazin-5-one | CHEM...)
Affinity DataIC50:  1.50E+3nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031055(3-(3-Methoxy-phenyl)-indeno[1,2-c]pyridazin-5-one ...)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibitory activity against Monoamine oxidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031055(3-(3-Methoxy-phenyl)-indeno[1,2-c]pyridazin-5-one ...)
Affinity DataIC50:  1.60E+3nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031027(3-(4-Acetyl-phenyl)-indeno[1,2-c]pyridazin-5-one |...)
Affinity DataIC50:  1.78E+3nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM19168(3-(4-fluorophenoxymethyl)-5H-indeno[1,2-c]pyridazi...)
Affinity DataIC50:  1.90E+3nMAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031070(3-(3,5-Bis-trifluoromethyl-phenyl)-indeno[1,2-c]py...)
Affinity DataIC50: >2.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031061(3-(naphthalen-2-yl)-5H-indeno[1,2-c]pyridazin-5-on...)
Affinity DataIC50:  2.18E+3nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM50031018(4-(5-Oxo-5H-indeno[1,2-c]pyridazin-3-yl)-benzonitr...)
Affinity DataIC50:  2.20E+3nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM19175(2-phenyl-9H-indeno[2,1-d]pyrimidin-9-one | Aza-het...)
Affinity DataIC50:  2.37E+3nMAssay Description:Inhibitory activity against Monoamine oxidase A from rat brain mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM19175(2-phenyl-9H-indeno[2,1-d]pyrimidin-9-one | Aza-het...)
Affinity DataIC50:  2.37E+3nMpH: 7.4 T: 2°CAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Bari

LigandPNGBDBM19167(3-(phenoxymethyl)-5H-indeno[1,2-c]pyridazin-5-one ...)
Affinity DataIC50:  2.51E+3nMAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 208 total ) | Next | Last >>
Jump to: