Affinity DataKi: 2.18E+4nMAssay Description:Inhibition of Sprague-Dawley rat MGLMore data for this Ligand-Target Pair
Affinity DataKi: 3.90E+4nMAssay Description:Inhibition of Sprague-Dawley rat MGLMore data for this Ligand-Target Pair
Affinity DataKi: 5.87E+4nMAssay Description:Inhibition of Sprague-Dawley rat MGLMore data for this Ligand-Target Pair
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
National and Kapodistrian University of Athens
Curated by ChEMBL
National and Kapodistrian University of Athens
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of human recombinant G6A iPLA2 using arachidonyl-1-14C PAPC and PAPC incubated for 30 mins by HPLC-MS analysis based radioactivity-based g...More data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 6.5nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of mouse group 2A sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 259nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in ovalbumin expressing wild type HEK293S cells assessed as decrease in antigen-mediated IL...More data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of human recombinant GIVA cPLA2 in vitro vesicle assayMore data for this Ligand-Target Pair
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
University Of Athens
Curated by ChEMBL
University Of Athens
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of human group 2A sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 390nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibition of human group 5 sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 460nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 460nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 760nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 820nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 830nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant GIVA cPLA2 in vitro vesicle assayMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human group 5 sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
TargetGroup 10 secretory phospholipase A2(Homo sapiens (Human))
University Of Athens
Curated by ChEMBL
University Of Athens
Curated by ChEMBL
Affinity DataIC50: >1.66E+3nMAssay Description:Inhibition of human group 10 sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
TargetGroup 10 secretory phospholipase A2(Homo sapiens (Human))
University Of Athens
Curated by ChEMBL
University Of Athens
Curated by ChEMBL
Affinity DataIC50: >1.66E+3nMAssay Description:Inhibition of human group 10 sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
TargetGroup 10 secretory phospholipase A2(Homo sapiens (Human))
University Of Athens
Curated by ChEMBL
University Of Athens
Curated by ChEMBL
Affinity DataIC50: >1.66E+3nMAssay Description:Inhibition of human group 10 sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.66E+3nMAssay Description:Inhibition of human group 5 sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
University Of Athens
Curated by ChEMBL
University Of Athens
Curated by ChEMBL
Affinity DataIC50: >1.66E+3nMAssay Description:Inhibition of human group 2A sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
University Of Athens
Curated by ChEMBL
University Of Athens
Curated by ChEMBL
Affinity DataIC50: >1.66E+3nMAssay Description:Inhibition of human group 2A sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.66E+3nMAssay Description:Inhibition of human group 5 sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
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