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Found 140 with Last Name = 'magrioti' and Initial = 'v'
TargetMonoglyceride lipase(Rattus norvegicus (Rat))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50274152((2S,9Z)-octadec-9-ene-1,2-diamine dihydrochloride ...)
Affinity DataKi:  2.18E+4nMAssay Description:Inhibition of Sprague-Dawley rat MGLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Rattus norvegicus (Rat))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50274153((2R,9Z)-octadec-9-ene-1,2-diamine dihydrochloride ...)
Affinity DataKi:  3.90E+4nMAssay Description:Inhibition of Sprague-Dawley rat MGLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Rattus norvegicus (Rat))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50274151(CHEMBL473249 | hexadecane-1,2-diamine dihydrochlor...)
Affinity DataKi:  5.87E+4nMAssay Description:Inhibition of Sprague-Dawley rat MGLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50526358(CHEMBL4476476)
Affinity DataIC50:  1nMAssay Description:Inhibition of human recombinant G6A iPLA2 using arachidonyl-1-14C PAPC and PAPC incubated for 30 mins by HPLC-MS analysis based radioactivity-based g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601034(CHEMBL5191661)
Affinity DataIC50:  6.5nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601033(CHEMBL5209483)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601042(CHEMBL5195885)
Affinity DataIC50:  19nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601035(CHEMBL5194003)
Affinity DataIC50:  150nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601032(CHEMBL5183817)
Affinity DataIC50:  160nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospholipase A2, membrane associated(Mus musculus)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50333788((S)-4-Methyl-2-(2-oxohexadecanamido)pentanoic acid...)
Affinity DataIC50:  180nMAssay Description:Inhibition of mouse group 2A sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601040(CHEMBL5195928)
Affinity DataIC50:  200nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601031(CHEMBL5199194)
Affinity DataIC50:  240nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601042(CHEMBL5195885)
Affinity DataIC50:  250nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601034(CHEMBL5191661)
Affinity DataIC50:  259nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in ovalbumin expressing wild type HEK293S cells assessed as decrease in antigen-mediated IL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601045(CHEMBL5209535)
Affinity DataIC50:  270nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601025(CHEMBL5207828)
Affinity DataIC50:  280nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50023445(CHEMBL3329874)
Affinity DataIC50:  300nMAssay Description:Inhibition of human recombinant GIVA cPLA2 in vitro vesicle assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50333788((S)-4-Methyl-2-(2-oxohexadecanamido)pentanoic acid...)
Affinity DataIC50:  300nMAssay Description:Inhibition of human group 2A sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601057(CHEMBL5171198)
Affinity DataIC50:  330nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601037(CHEMBL5200376)
Affinity DataIC50:  360nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601041(CHEMBL5197001)
Affinity DataIC50:  390nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50333788((S)-4-Methyl-2-(2-oxohexadecanamido)pentanoic acid...)
Affinity DataIC50:  440nMAssay Description:Inhibition of human group 5 sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601040(CHEMBL5195928)
Affinity DataIC50:  460nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601030(CHEMBL5185614)
Affinity DataIC50:  460nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601035(CHEMBL5194003)
Affinity DataIC50:  480nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601029(CHEMBL5194823)
Affinity DataIC50:  510nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601033(CHEMBL5209483)
Affinity DataIC50:  580nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601041(CHEMBL5197001)
Affinity DataIC50:  580nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601033(CHEMBL5209483)
Affinity DataIC50:  590nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601042(CHEMBL5195885)
Affinity DataIC50:  670nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601034(CHEMBL5191661)
Affinity DataIC50:  760nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601036(CHEMBL5184077)
Affinity DataIC50:  820nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601026(CHEMBL5202569)
Affinity DataIC50:  830nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601032(CHEMBL5183817)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601036(CHEMBL5184077)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601034(CHEMBL5191661)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50023444(CHEMBL3329869 | US9597318, Code GK185)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human recombinant GIVA cPLA2 in vitro vesicle assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601029(CHEMBL5194823)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601056(CHEMBL5189714)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of recombinant IRAP (unknown origin) expressed in HEK293S cells using L-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50333789((R)-4-Methyl-2-(2-oxohexadecanamido)pentanoic acid...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human group 5 sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601037(CHEMBL5200376)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601045(CHEMBL5209535)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGroup 10 secretory phospholipase A2(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50333790((S)-4-Methyl-2-palmitamidopentanoic acid | CHEMBL1...)
Affinity DataIC50: >1.66E+3nMAssay Description:Inhibition of human group 10 sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGroup 10 secretory phospholipase A2(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50333791((S)-2-(2-Oxohexadecanamido)-3-phenylpropanoic acid...)
Affinity DataIC50: >1.66E+3nMAssay Description:Inhibition of human group 10 sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGroup 10 secretory phospholipase A2(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50333789((R)-4-Methyl-2-(2-oxohexadecanamido)pentanoic acid...)
Affinity DataIC50: >1.66E+3nMAssay Description:Inhibition of human group 10 sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50333790((S)-4-Methyl-2-palmitamidopentanoic acid | CHEMBL1...)
Affinity DataIC50: >1.66E+3nMAssay Description:Inhibition of human group 5 sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50333791((S)-2-(2-Oxohexadecanamido)-3-phenylpropanoic acid...)
Affinity DataIC50: >1.66E+3nMAssay Description:Inhibition of human group 2A sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50333790((S)-4-Methyl-2-palmitamidopentanoic acid | CHEMBL1...)
Affinity DataIC50: >1.66E+3nMAssay Description:Inhibition of human group 2A sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50333791((S)-2-(2-Oxohexadecanamido)-3-phenylpropanoic acid...)
Affinity DataIC50: >1.66E+3nMAssay Description:Inhibition of human group 5 sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos

Curated by ChEMBL
LigandPNGBDBM50601025(CHEMBL5207828)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate by flourescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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