Affinity DataKi: 0.200nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO-cells (sc)More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO-cells (sc)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO-cells (sc)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of the radioligand [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of the radioligand [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of the radioligand [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of the radioligand [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of the radioligand [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 2.70nMAssay Description:Displacement of the radioligand [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of the radioligand [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT (agonist) as radioligand (sc)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of the radioligand [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 8.40nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 8.70nMAssay Description:Displacement of the radioligand [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 8.70nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT (agonist) as radioligand (sc)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of the radioligand [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 12.6nMAssay Description:Displacement of the radioligand [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of the radioligand [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:In vitro binding affinity against dopamine receptor D2 using [3H]-Raclopride as radioligand in CHO-cells (sc)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:In vitro binding affinity against dopamine receptor D2 using [3H]-Raclopride as radioligand in CHO-cells (sc)More data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Displacement of the radioligand [3H]-spiperone from D2 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 66nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of the radioligand [3H]-spiperone from D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Displacement of the radioligand [3H]-spiperone from D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 145nMAssay Description:Displacement of the radioligand [3H]-spiperone from D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 146nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 146nMAssay Description:Displacement of the radioligand [3H]-spiperone from D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 156nMAssay Description:Displacement of the radioligand [3H]-spiperone from D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 156nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 182nMAssay Description:Displacement of the radioligand [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 190nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Displacement of the radioligand [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Inhibition of human cytochrome P450 2C9More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 317nMAssay Description:Displacement of the radioligand [3H]-spiperone from D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Displacement of the radioligand [3H]-spiperone from D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 382nMAssay Description:Displacement of the radioligand [3H]-spiperone from D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 382nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataKi: 410nMAssay Description:Displacement of the radioligand [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair